中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
5-[(3R)-1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]pyrrolidin-3-yl]-3-ethyl-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C20H25N5O2S |
|
—— |
5-[(3S)-1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]pyrrolidin-3-yl]-3-ethyl-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C20H25N5O2S |
|
—— |
5-(1-propan-2-ylpiperidin-4-yl)-2-[(2S)-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H28N6O2S |
|
—— |
2-[(2R)-1-(6-methylpyridine-3-carbonyl)pyrrolidin-2-yl]-5-(1-propan-2-ylpiperidin-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C25H32N6O2 |
|
—— |
5-(1-propan-2-ylpiperidin-4-yl)-2-[(2R)-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H28N6O2S |
|
—— |
2-[(3S)-1-[2,2-dimethyl-3-(4-methylpiperidin-1-yl)propyl]pyrrolidin-3-yl]-5-ethyl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C23H37N5O |
|
—— |
5-(1-propan-2-ylpiperidin-4-yl)-2-[(2R)-1-(2-pyridin-2-ylacetyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C25H32N6O2 |
|
—— |
5-ethyl-2-[(2S)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H26N4O5 |
|
—— |
2-[(2R)-1-(1-ethyl-5-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dimethyl-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C19H24N6O2 |
|
—— |
5,6-dimethyl-2-[(2S)-1-[3-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C17H21N7O2 |
|
—— |
6-ethyl-5-methyl-2-[(2S)-1-[4-(1,2,4-triazol-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C19H25N7O2 |
|
—— |
5-ethyl-2-[(2R)-1-(3,4,5-trimethoxybenzoyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H26N4O5 |
|
—— |
6-ethyl-5-methyl-2-[(2R)-1-[4-(1,2,4-triazol-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C19H25N7O2 |
|
—— |
(1R,5R)-8-[5,6-dimethyl-2-(5-methyl-1,2-oxazol-3-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-(1-methylimidazol-2-yl)-8-azabicyclo[3.2.1]octan-3-ol |
—— |
C23H27N7O2 |
|
—— |
5,6-dimethyl-2-[(2R)-1-[3-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C17H21N7O2 |
|
—— |
(13R)-5,11-diamino-3-hydroxy-6,6-dimethyl-13-pyridin-3-yl-10-oxa-5,7,8-triazatricyclo[7.4.0.02,7]trideca-1,3,8,11-tetraene-12-carbonitrile |
—— |
C17H17N7O2 |
|
—— |
(13S)-5,11-diamino-3-hydroxy-6,6-dimethyl-13-pyridin-3-yl-10-oxa-5,7,8-triazatricyclo[7.4.0.02,7]trideca-1,3,8,11-tetraene-12-carbonitrile |
—— |
C17H17N7O2 |
|
—— |
3-[4-[[(6-Methylpyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]methyl]cyclohexyl]thieno[2,3-b]pyridine-2-carboxamide |
—— |
C23H24N6O2S |
|
—— |
2-[(3S)-1-butanoylpyrrolidin-3-yl]-5-methyl-6-(3-oxo-3-piperidin-1-ylpropyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C23H33N5O3 |
|
—— |
5-methyl-6-(3-oxo-3-piperidin-1-ylpropyl)-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H33N5O2 |
|
—— |
2-[(3R)-1-butanoylpyrrolidin-3-yl]-5-methyl-6-(3-oxo-3-piperidin-1-ylpropyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C23H33N5O3 |
|
—— |
5-methyl-6-(3-oxo-3-piperidin-1-ylpropyl)-2-[(3S)-1-propan-2-ylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C22H33N5O2 |
|
—— |
5-[2-(3-chlorophenyl)ethyl]-3-(piperazin-1-ylmethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C19H22ClN5O |
|
—— |
5-(2-phenylethyl)-3-(piperazin-1-ylmethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C19H23N5O |
|
—— |
6-[3-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-3-oxopropyl]-5-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C24H35N5O3 |
|
—— |
6-[3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-oxopropyl]-5-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C24H35N5O3 |
|
—— |
6-[3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-oxopropyl]-5-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C24H35N5O3 |
|
—— |
6-[3-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-3-oxopropyl]-5-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one |
—— |
C24H35N5O3 |
|
—— |
N-[[4-(2-carbamoyl-1-benzothiophen-3-yl)cyclohexyl]methyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
—— |
C24H25N5O2S |
|
—— |
[5-(furan-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4O2 |
|
—— |
[5-(furan-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4O2 |
|
—— |
[(5S,7R)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C25H31F3N4O2 |
|
—— |
[(5S,7R)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C25H31F3N4O2 |
|
—— |
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4OS |
|
—— |
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4OS |
|
—— |
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4OS |
|
—— |
[5-thiophen-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H23F3N4OS |
|
—— |
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H27F3N4OS |
|
—— |
[(5S,7R)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone |
—— |
C22H27F3N4OS |
|
—— |
3-[5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-4-(2-methylpropyl)-1H-1,2,4-triazole-5-thione |
—— |
C20H23F3N6OS |
|
—— |
ethyl (1S,5S)-3-[3-(1H-indazol-4-yl)-2-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-7-yl]-8-azabicyclo[3.2.1]octane-8-carboxylate |
—— |
C28H27N7O2 |
|
—— |
4-[1-(1,4-dioxaspiro[4.5]decan-8-yl)-4-[(1R,5R)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl]pyrazolo[3,4-d]pyrimidin-6-yl]aniline |
—— |
C25H30N6O3 |
|
—— |
ethyl (1R,5R)-3-[3-(1H-indazol-4-yl)-2-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-7-yl]-8-azabicyclo[3.2.1]octane-8-carboxylate |
—— |
C28H27N7O2 |
|
—— |
4-[1-(1,4-dioxaspiro[4.5]decan-8-yl)-4-[(1S,5S)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl]pyrazolo[3,4-d]pyrimidin-6-yl]aniline |
—— |
C25H30N6O3 |
|
—— |
(6R)-2,6-dimethyl-1H-pyrazolo[1,5-a]pyrimidine-5,7-dione |
—— |
C8H9N3O2 |
|
—— |
5-(1-adamantyl)-7-(difluoromethyl)-2-methyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine |
—— |
C18H25F2N3 |
|
—— |
3-[(2S)-nonan-2-yl]-2H-pyrazolo[3,4-d]pyrimidin-4-amine |
—— |
C14H23N5 |
|
—— |
6-[(E)-2-phenylethenyl]-1,5-dihydropyrazolo[3,4-d]pyrimidin-4-one |
—— |
C13H10N4O |
|
—— |
tert-butyl (2S)-2-(7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)piperidine-1-carboxylate |
—— |
C16H22N4O3 |
|
—— |
tert-butyl (3S)-3-(7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)piperidine-1-carboxylate |
—— |
C16H22N4O3 |
|