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中文名称 英文名称 CAS号 化学式 结构式图片
—— US9656955, Example 661 —— C23H22F4N4O4S
US9656955, Example 661
—— 4-[(3R,4S)-3-[(2,4-dichlorophenoxy)methyl]-4-(4-fluorophenyl)pyrrolidin-1-yl]sulfonyl-1-methylimidazole —— C21H20Cl2FN3O3S
4-[(3R,4S)-3-[(2,4-dichlorophenoxy)methyl]-4-(4-fluorophenyl)pyrrolidin-1-yl]sulfonyl-1-methylimidazole
—— US9656955, Example 562 —— C18H20ClN5O2S2
US9656955, Example 562
—— N-({trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)-4-(trifluoromethyl)aniline —— C22H22F4N4O2S
N-({trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)-4-(trifluoromethyl)aniline
—— 2-[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]oxy-N-propylacetamide —— C19H25FN4O4S
2-[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]oxy-N-propylacetamide
—— 2-[(3R,4S)-3-(4-fluoroanilino)-4-phenylpyrrolidin-1-yl]sulfonylbenzonitrile —— C23H20FN3O2S
2-[(3R,4S)-3-(4-fluoroanilino)-4-phenylpyrrolidin-1-yl]sulfonylbenzonitrile
—— rac-(3R,4S)-4-(4-fluorophenyl)pyrrolidin-3-ol —— C10H12FNO
rac-(3R,4S)-4-(4-fluorophenyl)pyrrolidin-3-ol
—— (3R,4S)-N-[2-fluoro-5-(trifluoromethyl)phenyl]-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-amine —— C21H20F4N4O2S
(3R,4S)-N-[2-fluoro-5-(trifluoromethyl)phenyl]-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-amine
—— 3-chloro-N-({trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)aniline —— C21H22ClFN4O2S
3-chloro-N-({trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)aniline
—— (3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-phenyl-N-(3-phenylmethoxypropyl)pyrrolidin-3-amine —— C24H30N4O3S
(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-phenyl-N-(3-phenylmethoxypropyl)pyrrolidin-3-amine
—— (3R,4S)-4-(3-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-amine —— C14H17FN4O2S
(3R,4S)-4-(3-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-amine
—— (3S,4R)-N-(2-ethoxyethyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-3-carboxamide —— C19H25FN4O4S
(3S,4R)-N-(2-ethoxyethyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-3-carboxamide
—— trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine —— C21H21F3N4O3S
trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine
—— US9656955, Example 233 —— C20H20F2N4O2S
US9656955, Example 233
—— (3R,4S)-N-[2-chloro-4-(trifluoromethyl)benzyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4yl)sulfonyl]pyrrolidin-3-amine —— C22H21ClF4N4O2S
(3R,4S)-N-[2-chloro-4-(trifluoromethyl)benzyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4yl)sulfonyl]pyrrolidin-3-amine
—— US9656955, Example 355 —— C23H25F3N4O2S
US9656955, Example 355
—— trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-(2,3,4-trifluorophenyl)pyrrolidin-3-amine —— C20H19F3N4O2S
trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-(2,3,4-trifluorophenyl)pyrrolidin-3-amine
—— trans-N-(2,4-difluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-amine —— C20H20F2N4O2S
trans-N-(2,4-difluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-amine
—— (3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-N,4-diphenylpyrrolidin-3-amine —— C20H22N4O2S
(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-N,4-diphenylpyrrolidin-3-amine
—— US9656955, Example 332 —— C22H21ClF4N4O2S
US9656955, Example 332
—— US9656955, Example 478 —— C26H25F2N3O3S
US9656955, Example 478
—— US9656955, Example 698 —— C19H22F4N4O3S
US9656955, Example 698
—— (3R,4S)-N-[[2-chloro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-amine —— C23H24ClF3N4O2S
(3R,4S)-N-[[2-chloro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-amine
—— US9656955, Example 221 —— C24H30N4O2S
US9656955, Example 221
—— US9656955, Example 716 —— C21H25FN6O3S
US9656955, Example 716
—— trans-4-(3-fluorophenyl)-1-(1-methyl-1H-imidazol-4-ylsulfonyl)pyrrolidin-3-amine —— C14H17FN4O2S
trans-4-(3-fluorophenyl)-1-(1-methyl-1H-imidazol-4-ylsulfonyl)pyrrolidin-3-amine
—— 2-[4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]oxy-N-propylacetamide —— C19H25FN4O4S
2-[4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]oxy-N-propylacetamide
—— US9656955, Example 75 —— C20H21ClN4O2S
US9656955, Example 75
—— US9656955, Example 356 —— C23H24ClF3N4O2S
US9656955, Example 356
—— US9656955, Example 588 —— C18H26N4O3S
US9656955, Example 588
—— trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[4-(trifluoromethyl)phenyl]pyrrolidin-3-amine —— C21H21F3N4O2S
trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[4-(trifluoromethyl)phenyl]pyrrolidin-3-amine
—— 4-Butyl-1-[1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-yl]triazole —— C20H26N6O2S
4-Butyl-1-[1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-yl]triazole
—— trans-N-[3-chloro-4-(trifluoromethyl)phenyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-3-carboxamide —— C22H19ClF4N4O3S
trans-N-[3-chloro-4-(trifluoromethyl)phenyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-3-carboxamide
—— US9656955, Example 431 —— C19H23N5O2S2
US9656955, Example 431
—— N-{trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}quinolin-7-amine —— C23H23N5O2S
N-{trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}quinolin-7-amine
—— trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[3-(propan-2-yl)phenyl]pyrrolidin-3-amine —— C23H28N4O2S
trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-N-[3-(propan-2-yl)phenyl]pyrrolidin-3-amine
—— US9656955, Example 333 —— C21H22ClFN4O2S
US9656955, Example 333
—— US9656955, Example 276 —— C22H19ClF4N4O3S
US9656955, Example 276
—— trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-N-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine —— C21H20F4N4O3S
trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-N-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine
—— 3,5-dichloro-N-{trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}benzamide —— C21H20Cl2N4O3S
3,5-dichloro-N-{trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}benzamide
—— US9656955, Example 627 —— C21H29FN4O3S
US9656955, Example 627
—— trans-N-[4-chloro-3-(trifluoromethoxy)phenyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine —— C21H19ClF4N4O3S
trans-N-[4-chloro-3-(trifluoromethoxy)phenyl]-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine
—— 2-chloro-N-[[4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]methyl]-4-(trifluoromethyl)aniline —— C22H21ClF4N4O2S
2-chloro-N-[[4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]methyl]-4-(trifluoromethyl)aniline
—— N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}-4-(2,2,2-trifluoroethoxy)pyridin-2-amine —— C21H21F4N5O3S
N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}-4-(2,2,2-trifluoroethoxy)pyridin-2-amine
—— US9656955, Example 735 —— C20H25F3N4O3S
US9656955, Example 735
—— tert-butyl N-benzyl-N-[(3R,4S)-1-benzyl-2,5-dioxo-4-phenylpyrrolidin-3-yl]carbamate —— C29H30N2O4
tert-butyl N-benzyl-N-[(3R,4S)-1-benzyl-2,5-dioxo-4-phenylpyrrolidin-3-yl]carbamate
—— US9656955, Example 394 —— C22H22ClF3N4O2S
US9656955, Example 394
—— US9656955, Example 674 —— C21H32N4O3S
US9656955, Example 674
—— Trans-1-benzyl-4-phenyl-3-((1-propyl-1H-1,2,3-triazol-4-yl)methyl)pyrrolidin-2-one —— C23H26N4O
Trans-1-benzyl-4-phenyl-3-((1-propyl-1H-1,2,3-triazol-4-yl)methyl)pyrrolidin-2-one
—— trans-N-(3-chloro-4-fluorophenyl)-4-(3-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine —— C20H19ClF2N4O2S
trans-N-(3-chloro-4-fluorophenyl)-4-(3-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine