中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-[2-(Triazol-2-yl)phenyl]-2-[[4-(trifluoromethyl)pyridin-2-yl]amino]-7-azabicyclo[2.2.1]heptane-7-carbaldehyde |
—— |
C21H19F3N6O |
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—— |
(+/-)-Tert-butyl-2-((6-(trifluoromethyl)pyridin-2-yl)amino)-7-azabicyclo[2.2.1]heptane-7-carboxylate |
—— |
C17H22F3N3O2 |
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—— |
6-[[1-[(2R)-2-hydroxy-2-(4-methyl-1-oxo-3H-2-benzofuran-5-yl)ethyl]-3-phenylpyrrolidin-3-yl]-methylamino]pyridine-3-carbonitrile |
—— |
C28H28N4O3 |
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—— |
racemic cis-2-{1-[4-(3,3-Difluoropyrrolidin-1-yl)benzyl]-6-[(5-methylpyridin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid |
—— |
C32H34F2N4O3 |
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—— |
N-[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-yl]-3-(2,2,2-trifluoroethoxy)pyridin-2-amine |
—— |
C21H22F3N5O3S |
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—— |
(E)-4-[[(3S)-1-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-[(4-methoxyphenyl)methyl]amino]-4-oxobut-2-enoate |
—— |
C23H21N2O7- |
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—— |
(E)-4-[[(3R)-1-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-[(4-methoxyphenyl)methyl]amino]-4-oxobut-2-enoate |
—— |
C23H21N2O7- |
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—— |
6-fluoro-N-[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]pyridin-2-amine |
—— |
C19H19F2N5O2S |
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—— |
4-((trans-3-(2,2-dibromovinyl)-4-(4-fluorophenyl)pyrrolidin-1-yl)sulfonyl)-1-methyl-1H-imidazole |
—— |
C16H16Br2FN3O2S |
|
—— |
7-(1-Methylimidazol-4-yl)sulfonyl-9-phenyl-1-(2,2,2-trifluoro-1-phenylethyl)-3-oxa-1,7-diazaspiro[4.4]nonan-2-one |
—— |
C24H23F3N4O4S |
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—— |
2-[[(1R,4R)-4-(4-fluorophenyl)-1-(1H-imidazol-5-ylsulfonyl)-1-methylpyrrolidin-1-ium-3-yl]methoxy]-4-(trifluoromethyl)pyridine |
—— |
C21H21F4N4O3S+ |
|
—— |
1-[[(3R,4S)-1-(1-methylimidazol-4-yl)sulfonyl-4-phenylpyrrolidin-3-yl]amino]pentan-2-ol |
—— |
C19H28N4O3S |
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—— |
US9656955, Example 656 |
—— |
C22H20F6N4O2S |
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—— |
4-Phenyl-3-((4-(trifluoromethyl)pyridin-2-yl)methyl)pyrrolidin-2-one |
—— |
C17H15F3N2O |
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—— |
US9656955, Example 162 |
—— |
C20H19ClF2N4O2S |
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—— |
US9656955, Example 174 |
—— |
C20H19ClF2N4O2S |
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—— |
3-methoxy-N-{trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}benzamide |
—— |
C22H24N4O4S |
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—— |
3-fluoro-5-({trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-yl}amino)benzonitrile |
—— |
C21H20FN5O2S |
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—— |
4-(4-Fluorophenyl)-3-[4-fluoro-3-(trifluoromethoxy)anilino]-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-2-one |
—— |
C21H17F5N4O4S |
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—— |
N-{trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}-4-(trifluoromethyl)benzamide |
—— |
C22H20F4N4O3S |
|
—— |
N-{trans-4-(2-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}-2-(trifluoromethyl)pyridin-4-amine |
—— |
C20H19F4N5O2S |
|
—— |
trans-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine |
—— |
C21H19F5N4O2S |
|
—— |
2-[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]oxyacetic acid |
—— |
C16H18FN3O5S |
|
—— |
N-[4-chloro-2-[[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]amino]phenyl]acetamide |
—— |
C22H23ClFN5O3S |
|
—— |
tert-butyl-[(3S,4R)-4-(4-fluorophenyl)pyrrolidin-3-yl]carbamic acid |
—— |
C15H21FN2O2 |
|
—— |
trans-N-(2-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-amine |
—— |
C20H21FN4O2S |
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—— |
US9656955, Example 101 |
—— |
C22H23N5O2S |
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—— |
US9656955, Example 55 |
—— |
C22H19ClF4N4O3S |
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—— |
US9656955, Example 470 |
—— |
C21H32N4O2S |
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—— |
US9656955, Example 595 |
—— |
C19H27FN4O2S |
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—— |
trans-N-(2-fluorobenzyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine |
—— |
C21H22F2N4O2S |
|
—— |
(3R,4S)-N-(4-chloro-3-fluorophenyl)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-amine |
—— |
C20H19ClF2N4O2S |
|
—— |
US9656955, Example 525 |
—— |
C23H19F3N4O2S |
|
—— |
trans-N-(4-chloro-3-fluorophenyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine |
—— |
C20H19ClF2N4O2S |
|
—— |
US9656955, Example 440 |
—— |
C23H23ClN4O2S2 |
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—— |
US9656955, Example 299 |
—— |
C21H20ClF3N4O3S |
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—— |
trans-N-(2,3-difluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenylpyrrolidin-3-amine |
—— |
C20H20F2N4O2S |
|
—— |
US9656955, Example 502 |
—— |
C20H20F2N4O2S |
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—— |
2-chloro-N-[(3R,4S)-1-(6-methoxypyridin-3-yl)sulfonyl-4-phenylpyrrolidin-3-yl]-3-(trifluoromethyl)benzamide |
—— |
C24H21ClF3N3O4S |
|
—— |
[(3R,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl] N-butylcarbamate |
—— |
C19H25FN4O4S |
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—— |
6-fluoro-N-{trans-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}pyridin-2-amine |
—— |
C19H19F2N5O2S |
|
—— |
N-[[(3S,4S)-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidin-3-yl]methyl]-1-methoxypropan-2-amine |
—— |
C19H27FN4O3S |
|
—— |
Tert-butyl 2-hydroxyethyl((3R,4S)-1-(1-methyl-1H-imidazol-4-ylsulfonyl)-4-phenylpyrrolidin-3-yl)carbamate |
—— |
C21H30N4O5S |
|
—— |
(3R,4S)-3-(benzenesulfonyl)-1-benzyl-4-phenylpyrrolidine |
—— |
C23H23NO2S |
|
—— |
US9656955, Example 142 |
—— |
C24H19Cl2F3N2O3S |
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—— |
trans-N-(3,4-difluorophenyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine |
—— |
C20H19F3N4O2S |
|
—— |
trans-N-(3-chloro-5-fluorophenyl)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-amine |
—— |
C20H19ClF2N4O2S |
|
—— |
US9656955, Example 21 |
—— |
C22H24N4O4S |
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—— |
US9656955, Example 624 |
—— |
C22H28N6O3S |
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—— |
(3R,4S)-N-[4-chloro-3-(trifluoromethoxy)phenyl]-4-(4-fluorophenyl)-1-(1-methylimidazol-4-yl)sulfonylpyrrolidine-3-carboxamide |
—— |
C22H19ClF4N4O4S |
|