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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C27H29BrN2O5
tert-butyl N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C27H26BrF3N2O5
butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— methyl (3S)-3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C22H19BrN2O4
methyl (3S)-3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— N-[(3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide —— C32H27F3N6O3
N-[(3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide
—— Methyl 3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate;2,2,2-trifluoroacetic acid —— C24H20BrF3N2O6
Methyl 3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate;2,2,2-trifluoroacetic acid
—— Methyl 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C28H29BrN2O7
Methyl 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— tert-butyl N-(9-bromo-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl)carbamate —— C14H17BrN2O4
tert-butyl N-(9-bromo-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl)carbamate
—— [(3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-methylcarbamic acid —— C28H21N5O4
[(3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-methylcarbamic acid
—— [(2S,3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamic acid —— C28H21N5O4
[(2S,3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamic acid
—— [(2S,3S)-2,8-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C12H14N2O4
[(2S,3S)-2,8-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid
—— (10bR)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidin-1-ium] —— C25H32N3O2+
(10bR)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidin-1-ium]
—— 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-3,4-dihydro-2H-1,5-benzoxazepin-3-amine —— C22H23BrN2O2
5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-3,4-dihydro-2H-1,5-benzoxazepin-3-amine
—— 3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-3,5-dihydro-2H-1,5-benzoxazepine-9-carboxylic acid —— C15H18N2O6
3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-3,5-dihydro-2H-1,5-benzoxazepine-9-carboxylic acid
—— (10bS)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine] —— C25H31N3O2
(10bS)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine]
—— (S)-methyl 3-amino-5-((4-bromonaphthalen-1-yl)methyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-9-carboxylate trifluoroacetate 1562189-04-1 C2HF3O2*C22H19BrN2O4
(S)-methyl 3-amino-5-((4-bromonaphthalen-1-yl)methyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-9-carboxylate trifluoroacetate
—— 3-Amino-5-[(2-methylnaphthalen-1-yl)methyl]-2,3-dihydro-1,5-benzoxazepin-4-one —— C21H20N2O2
3-Amino-5-[(2-methylnaphthalen-1-yl)methyl]-2,3-dihydro-1,5-benzoxazepin-4-one
—— N-[(3S)-5-[[6-bromo-1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide —— C30H26BrF3N6O3
N-[(3S)-5-[[6-bromo-1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide
—— N-[(2S)-3-[(3S)-8-bromo-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-3-yl]-2-(methylamino)propyl]-2,2,2-trifluoroacetamide —— C34H32BrF3N6O4
N-[(2S)-3-[(3S)-8-bromo-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-3-yl]-2-(methylamino)propyl]-2,2,2-trifluoroacetamide
—— (10bS)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidin-1-ium] —— C25H32N3O2+
(10bS)-2-(4-methoxyphenyl)-9-methyl-1'-propan-2-ylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidin-1-ium]
—— 3-cyano-4-[3-[[(2S,3S)-2-methyl-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl]methyl]indazol-1-yl]benzoic acid —— C35H38N6O6
3-cyano-4-[3-[[(2S,3S)-2-methyl-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl]methyl]indazol-1-yl]benzoic acid
—— methyl 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C32H38BrN3O7
methyl 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— [5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-3,5-dihydro-2H-1,4-benzoxazepin-4-ium-3-yl]carbamic acid —— C22H20BrN2O5+
[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-3,5-dihydro-2H-1,4-benzoxazepin-4-ium-3-yl]carbamic acid
—— [5-[(6-Bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamic acid —— C22H19BrN2O5
[5-[(6-Bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamic acid
—— 2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]indazol-1-yl]benzonitrile —— C24H19N5O2
2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]indazol-1-yl]benzonitrile
—— [(2S,3S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C11H12N2O4
[(2S,3S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid
—— [(2S)-1-[[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid —— C26H26BrN3O6
[(2S)-1-[[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid
—— methyl (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C32H38BrN3O7
methyl (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— tert-butyl N-[9-bromo-5-[(2-methylnaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C26H27BrN2O4
tert-butyl N-[9-bromo-5-[(2-methylnaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— 1-[(10bR)-2-(4-methoxyphenyl)-9-methylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine]-1'-yl]ethanone —— C24H27N3O3
1-[(10bR)-2-(4-methoxyphenyl)-9-methylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine]-1'-yl]ethanone
—— methyl-[(3S)-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C11H12N2O4
methyl-[(3S)-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid
—— (S)-tert-butyl 5-(benzo[d]isoxazol-3-ylmethyl)-4-oxo-9-(trifluoromethyl)-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-ylcarbamate 1562201-33-5 C23H22F3N3O5
(S)-tert-butyl 5-(benzo[d]isoxazol-3-ylmethyl)-4-oxo-9-(trifluoromethyl)-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-ylcarbamate
—— [(1S)-1-[[(2S,3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid —— C33H30N6O5
[(1S)-1-[[(2S,3S)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid
—— (3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid —— C27H27BrF3N3O6
(3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid
—— (2,2,2-trifluoroacetyl) (3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C27H25BrF3N3O5
(2,2,2-trifluoroacetyl) (3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— (3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C25H26BrN3O4
(3S)-5-[(4-bromonaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— 1-[(10bS)-2-(4-methoxyphenyl)-9-methylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine]-1'-yl]ethanone —— C24H27N3O3
1-[(10bS)-2-(4-methoxyphenyl)-9-methylspiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-piperidine]-1'-yl]ethanone
—— [[(3S)-5-[[2-chloro-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate —— C30H26ClN5O5
[[(3S)-5-[[2-chloro-1-(2-cyanophenyl)indol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate
—— [(2R,3S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C11H12N2O4
[(2R,3S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid
—— (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid —— C28H29BrF3N3O7
(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid
—— Methyl 5-[(4-bromonaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C27H27BrN2O6
Methyl 5-[(4-bromonaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— 2,2,2-trifluoro-N-[6-methoxy-5-[[(3S)-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-5-yl]methyl]naphthalen-1-yl]-N-methylsulfonylacetamide —— C32H37F3N4O7S
2,2,2-trifluoro-N-[6-methoxy-5-[[(3S)-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-5-yl]methyl]naphthalen-1-yl]-N-methylsulfonylacetamide
—— 2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]-6-fluoroindazol-1-yl]benzonitrile —— C24H18FN5O2
2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]-6-fluoroindazol-1-yl]benzonitrile
—— (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C26H28BrN3O5
(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— [(1S)-1-[[(3S)-5-[[1-(2-cyanophenyl)-6-fluoroindazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid —— C30H27FN6O5
[(1S)-1-[[(3S)-5-[[1-(2-cyanophenyl)-6-fluoroindazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid
—— methyl 5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C32H39N3O7
methyl 5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— tert-butyl N-[5-(1,2-benzoxazol-3-ylmethyl)-4-oxo-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C23H22F3N3O5
tert-butyl N-[5-(1,2-benzoxazol-3-ylmethyl)-4-oxo-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— N-[(2S,3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-2,8-dimethyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide —— C29H31BrF3N3O4
N-[(2S,3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-2,8-dimethyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide
—— 5-[(6-Bromo-2-methoxynaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C27H27BrN2O7
5-[(6-Bromo-2-methoxynaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(2-hydroxyethylamino)butyl]acetamide —— C29H31BrF3N3O5
N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(2-hydroxyethylamino)butyl]acetamide
—— (3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C31H37N3O7
(3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid