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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-ethyl-8-[1-(4-ethylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C26H29NO4S
5-ethyl-8-[1-(4-ethylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— 8-[1-(3,4-dichlorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C24H23Cl2NO4S
8-[1-(3,4-dichlorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— 5-ethyl-8-(1-((4-ethylphenyl)sulfonyl)cyclopentyl)-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563205-79-7 C26H33NO4S
5-ethyl-8-(1-((4-ethylphenyl)sulfonyl)cyclopentyl)-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-(1-((4-chlorophenyl)sulfonyl)cyclohexyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-16-5 C25H30ClNO4S
8-(1-((4-chlorophenyl)sulfonyl)cyclohexyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 5-ethyl-3,3-dimethyl-8-[1-(4-propan-2-ylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one —— C27H31NO4S
5-ethyl-3,3-dimethyl-8-[1-(4-propan-2-ylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one
—— 5-Ethyl-3,3-dimethyl-8-[1-(4-methylphenyl)sulfonylcyclopentyl]-2,4-dihydro-1,5-benzoxazepine —— C25H33NO3S
5-Ethyl-3,3-dimethyl-8-[1-(4-methylphenyl)sulfonylcyclopentyl]-2,4-dihydro-1,5-benzoxazepine
—— 5-ethyl-3,3-dimethyl-8-(5-((4-(trifluoromethyl)phenyl)sulfonyl)spiro[2.3]hexan-5-yl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563205-86-6 C26H28F3NO4S
5-ethyl-3,3-dimethyl-8-(5-((4-(trifluoromethyl)phenyl)sulfonyl)spiro[2.3]hexan-5-yl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 5-ethyl-3,3-dimethyl-8-[1-(3-propan-2-yloxyphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one —— C27H31NO5S
5-ethyl-3,3-dimethyl-8-[1-(3-propan-2-yloxyphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one
—— 5-ethyl-8-(1-((4-isopropylphenyl)sulfonyl)cyclopentyl)-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563205-98-0 C27H35NO4S
5-ethyl-8-(1-((4-isopropylphenyl)sulfonyl)cyclopentyl)-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-(4-((4-chlorophenyl)sulfonyl)tetrahydro-2H-pyran-4-yl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-24-5 C24H26F3NO4S
8-(4-((4-chlorophenyl)sulfonyl)tetrahydro-2H-pyran-4-yl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 5-ethyl-8-[1-(4-fluoro-3-methylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C25H26FNO4S
5-ethyl-8-[1-(4-fluoro-3-methylphenyl)sulfonylcyclopenta-2,4-dien-1-yl]-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— tert-butyl N-[5-[[1-(2-cyanophenyl)-6-fluoroindazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C29H26FN5O4
tert-butyl N-[5-[[1-(2-cyanophenyl)-6-fluoroindazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— 5-ethyl-3,3-dimethyl-8-[1-[3-(trifluoromethyl)phenyl]sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one —— C25H24F3NO4S
5-ethyl-3,3-dimethyl-8-[1-[3-(trifluoromethyl)phenyl]sulfonylcyclopenta-2,4-dien-1-yl]-2H-1,5-benzoxazepin-4-one
—— (2,2,7-trifluoro-3-oxo-4H-1,4-benzoxazin-6-yl)carbamic acid —— C9H5F3N2O4
(2,2,7-trifluoro-3-oxo-4H-1,4-benzoxazin-6-yl)carbamic acid
—— (S)-2-(3-((3-amino-4-oxo-3,4-dihydrobenzo[b][1,4]oxazepin-5(2H)-yl)methyl)-6-bromo-1H-indazol-1-yl)benzonitrile 1562199-68-1 C24H18BrN5O2
(S)-2-(3-((3-amino-4-oxo-3,4-dihydrobenzo[b][1,4]oxazepin-5(2H)-yl)methyl)-6-bromo-1H-indazol-1-yl)benzonitrile
—— 2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]-6-bromoindazol-1-yl]benzonitrile —— C24H18BrN5O2
2-[3-[(3-Amino-4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)methyl]-6-bromoindazol-1-yl]benzonitrile
—— N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,3'-oxetane]-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide —— C29H29BrF3N3O5
N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,3'-oxetane]-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide
—— 5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C31H36BrN3O7
5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— N-[(2S,3S)-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-N-[(2S)-2-(ethylamino)propyl]-2,2,2-trifluoroacetamide —— C32H31F3N6O3
N-[(2S,3S)-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-2-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-N-[(2S)-2-(ethylamino)propyl]-2,2,2-trifluoroacetamide
—— tert-butyl N-[5-[[6-bromo-1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C29H26BrN5O4
tert-butyl N-[5-[[6-bromo-1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— (3S)-3-amino-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-2,3-dihydro-1,5-benzoxazepin-4-one —— C22H21BrN2O3
(3S)-3-amino-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-2,3-dihydro-1,5-benzoxazepin-4-one
—— 3-Amino-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-2,3-dihydro-1,5-benzoxazepin-4-one —— C22H21BrN2O3
3-Amino-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-2,3-dihydro-1,5-benzoxazepin-4-one
—— (3S)-3-amino-5-(1,2-benzoxazol-3-ylmethyl)-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-4-one —— C18H14F3N3O3
(3S)-3-amino-5-(1,2-benzoxazol-3-ylmethyl)-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-4-one
—— (2,2,2-trifluoroacetyl) (3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C28H28F3N3O6
(2,2,2-trifluoroacetyl) (3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— (S)-3-amino-5-(benzo[d]isoxazol-3-ylmethyl)-9-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetate 1562201-36-8 C2HF3O2*C18H14F3N3O3
(S)-3-amino-5-(benzo[d]isoxazol-3-ylmethyl)-9-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetate
—— tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-[2-hydroxyethyl(methyl)carbamoyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C30H34BrN3O7
tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-[2-hydroxyethyl(methyl)carbamoyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— (3S)-3-amino-9-bromo-5-[(2-methylnaphthalen-1-yl)methyl]-2,3-dihydro-1,5-benzoxazepin-4-one —— C21H19BrN2O2
(3S)-3-amino-9-bromo-5-[(2-methylnaphthalen-1-yl)methyl]-2,3-dihydro-1,5-benzoxazepin-4-one
—— (3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid —— C28H30F3N3O7
(3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid;2,2,2-trifluoroacetic acid
—— butyl N-[5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C29H27N5O4
butyl N-[5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-7-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide —— C28H26BrF6N3O4
N-[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-4-oxo-7-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-3-yl]-2,2,2-trifluoro-N-[(2S)-2-(methylamino)propyl]acetamide
—— [(2S)-1-[[(3S)-5-[(2-chlorophenyl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid —— C21H22ClN3O5
[(2S)-1-[[(3S)-5-[(2-chlorophenyl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid
—— (S)-3-amino-5-((2-methylnaphthalen-1-yl)methyl)-9-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetate 1562201-27-7 C2HF3O2*C22H19F3N2O2
(S)-3-amino-5-((2-methylnaphthalen-1-yl)methyl)-9-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetate
—— (2,2,2-trifluoroacetyl) (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C28H27BrF3N3O6
(2,2,2-trifluoroacetyl) (3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— 5-[(4-Bromonaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C26H25BrN2O6
5-[(4-Bromonaphthalen-1-yl)methyl]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— (3S)-3-amino-5-[(2-methylnaphthalen-1-yl)methyl]-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-4-one —— C22H19F3N2O2
(3S)-3-amino-5-[(2-methylnaphthalen-1-yl)methyl]-9-(trifluoromethyl)-2,3-dihydro-1,5-benzoxazepin-4-one
—— tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C27H29BrN2O5
tert-butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— [[(3S)-5-[(2-chlorophenyl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate —— C21H22ClN3O5
[[(3S)-5-[(2-chlorophenyl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate
—— (2S,3S)-2,8-dimethyl-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-amine —— C11H16N2O
(2S,3S)-2,8-dimethyl-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-amine
—— [(2S,3S)-4-[[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-8-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamic acid —— C27H28BrN3O7
[(2S,3S)-4-[[(3S)-5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-8-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamic acid
—— [[(3S)-5-[(1-ethylindol-4-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate —— C25H28N4O5
[[(3S)-5-[(1-ethylindol-4-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate
—— methyl 3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-3,5-dihydro-2H-1,5-benzoxazepine-9-carboxylate —— C16H20N2O6
methyl 3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxo-3,5-dihydro-2H-1,5-benzoxazepine-9-carboxylate
—— (3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid —— C26H29N3O5
(3S)-5-[(2-methoxynaphthalen-1-yl)methyl]-3-[[(2S)-2-(methylamino)propyl]amino]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylic acid
—— N-[(2S)-3-[(3S)-8-cyano-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-3-yl]-2-(methylamino)propyl]-2,2,2-trifluoroacetamide —— C35H32F3N7O4
N-[(2S)-3-[(3S)-8-cyano-5-[[1-(2-cyanophenyl)indazol-3-yl]methyl]-4-oxospiro[3H-1,5-benzoxazepine-2,4'-oxane]-3-yl]-2-(methylamino)propyl]-2,2,2-trifluoroacetamide
—— [4-oxo-9-(trifluoromethyl)-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C11H9F3N2O4
[4-oxo-9-(trifluoromethyl)-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid
—— tert-butyl N-[5-[(2-methylnaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C26H28N2O4
tert-butyl N-[5-[(2-methylnaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— [(2S)-1-[[(3S)-5-[(6-cyclopropyl-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid —— C29H31N3O6
[(2S)-1-[[(3S)-5-[(6-cyclopropyl-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino]-3-oxopropan-2-yl]-methylcarbamic acid
—— Methyl 3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate —— C22H19BrN2O4
Methyl 3-amino-5-[(4-bromonaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepine-9-carboxylate
—— [[(3S)-5-[(6-cyclopropyl-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate —— C29H31N3O6
[[(3S)-5-[(6-cyclopropyl-2-methoxynaphthalen-1-yl)methyl]-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate
—— butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate —— C27H29BrN2O5
butyl N-[5-[(6-bromo-2-methoxynaphthalen-1-yl)methyl]-9-methyl-4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]carbamate
—— methyl-[(3S)-8-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid —— C12H14N2O4
methyl-[(3S)-8-methyl-4-oxo-3,5-dihydro-2H-1,5-benzoxazepin-3-yl]carbamic acid