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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(2-methylsulfanylethylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide 1033244-32-4 C21H24F2N6OS
2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(2-methylsulfanylethylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide
—— 4-{7-[(4-ethylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]benzothiazol-2-yl}aniline 1191251-78-1 C22H25N5S
4-{7-[(4-ethylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]benzothiazol-2-yl}aniline
—— methyl-{4-[7-(3-morpholin-4-yl-propyl)-benzo[d]imidazo[2,1-b]thiazol-2-yl]-phenyl}-amine 950770-35-1 C23H26N4OS
methyl-{4-[7-(3-morpholin-4-yl-propyl)-benzo[d]imidazo[2,1-b]thiazol-2-yl]-phenyl}-amine
—— 7-[3-(4-methanesulfonyl-piperazin-1-yl)-propoxy]-2-(4-aminophenyl)-imidazo[2,1-b][1,3]benzothiazole 1191251-65-6 C23H27N5O3S2
7-[3-(4-methanesulfonyl-piperazin-1-yl)-propoxy]-2-(4-aminophenyl)-imidazo[2,1-b][1,3]benzothiazole
—— 2-(4-aminophenyl)-5-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazole 1191251-71-4 C21H22N4O2S
2-(4-aminophenyl)-5-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazole
—— 4-[6-(butylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1330075-45-0 C22H26F2N6O
4-[6-(butylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 3-{4-[(3-fluoro-6-methylpyridin-2-yl)amino]phenyl}-N-(1-methylpiperidin-4-yl)imidazo[1,2-b]pyridazin-6-amine 1400873-60-0 C24H26FN7
3-{4-[(3-fluoro-6-methylpyridin-2-yl)amino]phenyl}-N-(1-methylpiperidin-4-yl)imidazo[1,2-b]pyridazin-6-amine
—— 7-(2-chloroethoxy)-2-(4-aminophenyl)imidazo[2,1-b]benzothiazolel 1225542-43-7 C17H14ClN3OS
7-(2-chloroethoxy)-2-(4-aminophenyl)imidazo[2,1-b]benzothiazolel
—— 2-(4-Amino-phenyl)-imidazo[1,2-b]pyridazine 104691-63-6 C12H10N4
2-(4-Amino-phenyl)-imidazo[1,2-b]pyridazine
—— 2-(dimethylamino)-1-(4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-1-yl)ethanone 1361951-26-9 C23H27F3N6O2
2-(dimethylamino)-1-(4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-1-yl)ethanone
—— 2-fluoro-4-[6-(5-fluoropentylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1033244-34-6 C23H27F3N6O
2-fluoro-4-[6-(5-fluoropentylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 3-methyl-1-phenylpyrazolo[4',3':5,6]pyrano[3,2-c]pyridin-4(1H)-one 929569-03-9 C16H11N3O2
3-methyl-1-phenylpyrazolo[4',3':5,6]pyrano[3,2-c]pyridin-4(1H)-one
—— ethyl 3-[2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-yl]propanoate 950769-87-6 C20H19N3O2S
ethyl 3-[2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-yl]propanoate
—— Ethyl 2-amino-4-(2-bromophenyl)-1,3-thiazole-5-carboxylate 899354-41-7 C12H11BrN2O2S
Ethyl 2-amino-4-(2-bromophenyl)-1,3-thiazole-5-carboxylate
—— ethyl 2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-carboxylate 950769-92-3 C18H15N3O2S
ethyl 2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-carboxylate
—— N-(3-methylbutyl)-4-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide 1330594-15-4 C24H32N6O
N-(3-methylbutyl)-4-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide
—— ethyl[2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-yl]acetate 950769-81-0 C19H17N3O2S
ethyl[2-(4-aminophenyl)imidazo[2,1-b][1,3]benzothiazol-7-yl]acetate
—— {3-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}carbamic acid methyl ester 1330594-45-0 C20H24N6O2
{3-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}carbamic acid methyl ester
—— N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(4-methylsulfonylphenyl)-1,2,4-triazole-3-carboxamide trifluoroacetate 1613021-36-5 C2HF3O2*C20H20N8O3S
N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(4-methylsulfonylphenyl)-1,2,4-triazole-3-carboxamide trifluoroacetate
—— 4-[6-(cyclopentylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1330075-48-3 C23H26F2N6O
4-[6-(cyclopentylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 2-fluoro-4-[6-(4-fluorobutylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1033244-26-6 C22H25F3N6O
2-fluoro-4-[6-(4-fluorobutylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(pentylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide 1330075-46-1 C23H28F2N6O
2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(pentylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide
—— 3-(6-((3S)-2-(3-fluorophenyl)-3-hydroxypyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile 1196546-35-6 C23H18FN5O
3-(6-((3S)-2-(3-fluorophenyl)-3-hydroxypyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile
—— N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(p-tolyl)-1,2,4-triazole-3-carboxamide trifluoroacetate salt 1613021-38-7 C2HF3O2*C20H20N8O
N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(p-tolyl)-1,2,4-triazole-3-carboxamide trifluoroacetate salt
—— N-[2-[[2-(3-chlorophenyl)-5-phenylpyrazol-3-yl]amino]phenyl]-2,2,2-trifluoroacetamide 881303-62-4 C23H16ClF3N4O
N-[2-[[2-(3-chlorophenyl)-5-phenylpyrazol-3-yl]amino]phenyl]-2,2,2-trifluoroacetamide
—— 3-[2-(3-methoxypropoxy)phenyl]-2-oxo-4-phenyl-1H-imidazole-5-carboxylic acid 1041399-12-5 C20H20N2O5
3-[2-(3-methoxypropoxy)phenyl]-2-oxo-4-phenyl-1H-imidazole-5-carboxylic acid
—— 4-(pyrrol-2-yl)-2-aminothiazole 189011-25-4 C7H7N3S
4-(pyrrol-2-yl)-2-aminothiazole
—— 2-fluoro-4-[6-(3-fluoropropylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1033244-28-8 C21H23F3N6O
2-fluoro-4-[6-(3-fluoropropylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(3-methylsulfanylpropylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide 1033244-29-9 C22H26F2N6OS
2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]-4-[6-(3-methylsulfanylpropylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide
—— 5-(6-(2-(2,5-dimethylphenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-2-fluorobenzonitrile 1196546-36-7 C25H22FN5
5-(6-(2-(2,5-dimethylphenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-2-fluorobenzonitrile
—— 2-(4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-1-yl)ethanol 1361951-12-3 C21H24F3N5O2
2-(4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-1-yl)ethanol
—— 6-((tetrahydro-2H-pyran-4-yl)methoxy)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazine 1418142-61-6 C19H18F3N3O3
6-((tetrahydro-2H-pyran-4-yl)methoxy)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazine
—— (S)-1-(3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)piperidin-3-amine 1418142-64-9 C17H18ClN5
(S)-1-(3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)piperidin-3-amine
—— N-((4,4-difluorocyclohexyl)methyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine 1361951-02-1 C20H19F5N4O
N-((4,4-difluorocyclohexyl)methyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine
—— Ethyl 2-(4-nitrophenyl)-1H-imidazole-5-carboxylate 951626-92-9 C12H11N3O4
Ethyl 2-(4-nitrophenyl)-1H-imidazole-5-carboxylate
—— N1-(3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)cyclohexane-1,3-diamine 1418142-63-8 C18H20ClN5
N1-(3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)cyclohexane-1,3-diamine
—— 4-(6-{[(3-fluorophenyl)methyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzonitrile 1022981-78-7 C20H14FN5
4-(6-{[(3-fluorophenyl)methyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzonitrile
—— 1-methyl-4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-4-ol 1361951-07-6 C20H22F3N5O2
1-methyl-4-(((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)methyl)piperidin-4-ol
—— N-(2-morpholinoethyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine 1361951-25-8 C19H20F3N5O2
N-(2-morpholinoethyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine
—— 4-((3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)amino)cyclohexane-1-sulfonamide 1418142-73-0 C18H20ClN5O2S
4-((3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl)amino)cyclohexane-1-sulfonamide
—— 4-(5-amino-4-cyano-1H-pyrazol-1-yl)-benzoic acid 882233-04-7 C11H8N4O2
4-(5-amino-4-cyano-1H-pyrazol-1-yl)-benzoic acid
—— 5-Thiazolecarboxylic acid, 4-methyl-2-[[[5-(1-methylethyl)-1-(tetrahydro-1,1-dioxido-3-thienyl)-1H-pyrazol-3-yl]carbonyl]amino]-, 1-methylethyl ester 1795488-86-6 C19H26N4O5S2
5-Thiazolecarboxylic acid, 4-methyl-2-[[[5-(1-methylethyl)-1-(tetrahydro-1,1-dioxido-3-thienyl)-1H-pyrazol-3-yl]carbonyl]amino]-, 1-methylethyl ester
—— 2-methyl-4-((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)butan-2-ol 1361950-89-1 C18H19F3N4O2
2-methyl-4-((3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)butan-2-ol
—— 1-(6-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)pyridin-2-yl)piperidin-4-ol 1196546-70-9 C29H29F2N7O
1-(6-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)pyridin-2-yl)piperidin-4-ol
—— (S)-4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile 1196546-48-1 C23H17F2N5
(S)-4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile
—— 3-phenylimidazo[1,2-b]pyridazine 54248-71-4 C12H9N3
3-phenylimidazo[1,2-b]pyridazine
—— (R)-4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile 1196546-38-9 C23H17F2N5
(R)-4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)benzonitrile
—— tert-butyl 4-(2-oxo-1,5-diphenyl-2,3-dihydro-1H-imidazole-4-carbonyl)piperazine-1-carboxylate 1041399-17-0 C25H28N4O4
tert-butyl 4-(2-oxo-1,5-diphenyl-2,3-dihydro-1H-imidazole-4-carbonyl)piperazine-1-carboxylate
—— 4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-2-fluorobenzonitrile 1196546-61-8 C23H16F3N5
4-(6-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)-2-fluorobenzonitrile
—— 2-(4-Ethyl-benzyl)-4-(4-methylaminomethyl-phenyl)-2,4-dihydro-[1,2,4]triazol-3-one 887139-66-4 C19H22N4O
2-(4-Ethyl-benzyl)-4-(4-methylaminomethyl-phenyl)-2,4-dihydro-[1,2,4]triazol-3-one