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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4E)(3S)-4-methyl-5-(2-methyl(1,3-thiazol-4-yl))-3-(1,1,2,2-tetramethyl-1-silapropoxy)pent-4-enylidene]butane-1,4-diol 1089733-16-3 C20H35NO3SSi
2-[(4E)(3S)-4-methyl-5-(2-methyl(1,3-thiazol-4-yl))-3-(1,1,2,2-tetramethyl-1-silapropoxy)pent-4-enylidene]butane-1,4-diol
—— 1-(4-Methylpyridin-2-yl)-3-(5-pyridin-3-yl-1,3,4-thiadiazol-2-yl)urea 1140522-64-0 C14H12N6OS
1-(4-Methylpyridin-2-yl)-3-(5-pyridin-3-yl-1,3,4-thiadiazol-2-yl)urea
—— methyl 2-(4-aminoazepan-1-yl)-1,3-thiazole-5-carboxylate hydrochloride 1007585-28-5 C11H17N3O2S*ClH
methyl 2-(4-aminoazepan-1-yl)-1,3-thiazole-5-carboxylate hydrochloride
—— (3E,7E)(6S)-3-(chloromethyl)-7-methyl-8-(2-methyl(1,3-thiazol-4-yl))-6-(1,1,2,2-tetramethyl-1-silapropoxy)octa-3,7-dien-1-ol 1089733-18-5 C20H34ClNO2SSi
(3E,7E)(6S)-3-(chloromethyl)-7-methyl-8-(2-methyl(1,3-thiazol-4-yl))-6-(1,1,2,2-tetramethyl-1-silapropoxy)octa-3,7-dien-1-ol
—— (3E,7E)(6S)-1,6-bis(1,1,2,2-tetramethyl-1-silapropoxy)-3-(chloromethyl)-7-methyl-8-(2-methyl(1,3-thiazol-4-yl))octa-3,7-diene 1089733-19-6 C26H48ClNO2SSi2
(3E,7E)(6S)-1,6-bis(1,1,2,2-tetramethyl-1-silapropoxy)-3-(chloromethyl)-7-methyl-8-(2-methyl(1,3-thiazol-4-yl))octa-3,7-diene
—— 1-(3-piperidin-1-yl-propyl)-4-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-b]pyridazin-7-yl]-1H-pyridin-2-one 1107655-20-8 C28H29N7O
1-(3-piperidin-1-yl-propyl)-4-[3-(3-pyrazol-1-yl-phenyl)-imidazo[1,2-b]pyridazin-7-yl]-1H-pyridin-2-one
—— N-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)(4-fluorophenyl)methyl]propionamide 1104872-54-9 C21H22FN3O
N-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)(4-fluorophenyl)methyl]propionamide
—— benzyl P-[2-(anilinocarbonyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-N,N-diisopropylphosphonamidate 1120366-01-9 C24H31N4O4P
benzyl P-[2-(anilinocarbonyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-N,N-diisopropylphosphonamidate
—— 1-[(2E)(1S)-2-methyl-3-(2-methyl(1,3-thiazol-4-yl))-1-(2-(3-2,4,5-trihydrofurylidene)ethyl)prop-2-enyloxy]-1,1,2,2-tetramethyl-1-silapropane 1089733-21-0 C20H33NO2SSi
1-[(2E)(1S)-2-methyl-3-(2-methyl(1,3-thiazol-4-yl))-1-(2-(3-2,4,5-trihydrofurylidene)ethyl)prop-2-enyloxy]-1,1,2,2-tetramethyl-1-silapropane
—— (S)-tert-butyl 3-(6-(1-(5-fluoropyridin-2-yl)ethylamino)pyrazin-2-ylamino)-5-isopropoxy-1H-pyrazole-1-carboxylate 1065267-80-2 C22H28FN7O3
(S)-tert-butyl 3-(6-(1-(5-fluoropyridin-2-yl)ethylamino)pyrazin-2-ylamino)-5-isopropoxy-1H-pyrazole-1-carboxylate
—— 4-(7-sec-butyl-5-cyano-1,3-benzoxazol-2-yl)-N-({1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}methyl)benzamide 1093397-42-2 C30H29F3N6O2
4-(7-sec-butyl-5-cyano-1,3-benzoxazol-2-yl)-N-({1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}methyl)benzamide
—— 5-(4-methoxyphenyl)-4-phenyl-1-methyl-1H-imidazole 1111266-62-6 C17H16N2O
5-(4-methoxyphenyl)-4-phenyl-1-methyl-1H-imidazole
—— 3-[4-(4-fluorophenyl)-1-methyl-1H-imidazol-5-yl]pyridine 1111267-20-9 C15H12FN3
3-[4-(4-fluorophenyl)-1-methyl-1H-imidazol-5-yl]pyridine
—— 4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(6-(trifluoromethyl)pyridin-2-yl)piperidin-4-yl)methyl)benzamide 1292821-38-5 C30H28F3N5O2
4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(6-(trifluoromethyl)pyridin-2-yl)piperidin-4-yl)methyl)benzamide
—— 5-({[3-(2,6-dichlorophenyl)-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1-{[4-(1H-tetrazol-5-yl)phenyl]methyl}-1H-indole 1097777-96-2 C29H24Cl2N6O2
5-({[3-(2,6-dichlorophenyl)-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1-{[4-(1H-tetrazol-5-yl)phenyl]methyl}-1H-indole
—— 6-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-2-N-[(1R)-1-phenylethyl]pyridine-2,6-dicarboxamide 1022892-99-4 C32H30N8O4
6-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-2-N-[(1R)-1-phenylethyl]pyridine-2,6-dicarboxamide
—— 1-(4-aminosulfonylphenyl)-3-trifluoromethyl-5-[4-(1-hydroxy-1,2-dihydro)pyrid-2-one]-1H-pyrazole 1095371-82-6 C15H11F3N4O4S
1-(4-aminosulfonylphenyl)-3-trifluoromethyl-5-[4-(1-hydroxy-1,2-dihydro)pyrid-2-one]-1H-pyrazole
—— 4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-({1-[2-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}methyl)benzamide 1093395-90-4 C30H33N7O2
4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-({1-[2-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}methyl)benzamide
—— N-methylsulfonyl-S-methyl-S-[(2-chloro-1,3-thiazol-5-yl)methyl] sulfoximine 1092391-12-2 C6H9ClN2O3S3
N-methylsulfonyl-S-methyl-S-[(2-chloro-1,3-thiazol-5-yl)methyl] sulfoximine
—— 2-chloro-5-(S-methylsulfonimidoylmethyl)thiazole 1092391-10-0 C5H7ClN2OS2
2-chloro-5-(S-methylsulfonimidoylmethyl)thiazole
—— 4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[1-(2-isopropylpyrimidin-4-yl)piperidin-4-yl]methyl}benzamide 1093395-92-6 C31H34N6O2
4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[1-(2-isopropylpyrimidin-4-yl)piperidin-4-yl]methyl}benzamide
—— 6-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxo-2-N-(2-phenylpropan-2-yl)-1H-pyridine-2,6-dicarboxamide 1022893-04-4 C33H32N8O5
6-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxo-2-N-(2-phenylpropan-2-yl)-1H-pyridine-2,6-dicarboxamide
—— 2-amino-4,6-dichloro-N-((S)-1-{[1-(4-fluorophenyl)-1H-indazol-5-ylamino]methyl}propyl)benzenesulfonamide 1070341-67-1 C23H22Cl2FN5O2S
2-amino-4,6-dichloro-N-((S)-1-{[1-(4-fluorophenyl)-1H-indazol-5-ylamino]methyl}propyl)benzenesulfonamide
—— [2-[[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]carbamoyl]-6-(2-phenylpropan-2-ylcarbamoyl)pyridin-4-yl] methanesulfonate 1022893-03-3 C34H34N8O7S
[2-[[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]carbamoyl]-6-(2-phenylpropan-2-ylcarbamoyl)pyridin-4-yl] methanesulfonate
—— 2-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxo-6-N-[(1R)-1-phenylethyl]pyran-2,6-dicarboxamide 1022893-01-1 C32H29N7O6
2-N-[(2S,3S)-3-hydroxy-4-oxo-1-phenyl-4-[3-(2H-tetrazol-5-yl)anilino]butan-2-yl]-4-oxo-6-N-[(1R)-1-phenylethyl]pyran-2,6-dicarboxamide
—— 1-(4-methylsulfonylphenyl)-3-trifluoromethyl-5-[4-(1-hydroxy-1,2-dihydro)pyrid-2-one]-1H-pyrazole 1095371-77-9 C16H12F3N3O4S
1-(4-methylsulfonylphenyl)-3-trifluoromethyl-5-[4-(1-hydroxy-1,2-dihydro)pyrid-2-one]-1H-pyrazole
—— KMI-1036 1022893-07-7 C34H32N8O8S
KMI-1036
—— 2-[5-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonyl-3,6-dihydro-2H-pyridin-4-yl]acetic acid 647002-93-5 C32H30N2O6
2-[5-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonyl-3,6-dihydro-2H-pyridin-4-yl]acetic acid
—— KMI-1030 1022893-08-8 C33H30N8O6
KMI-1030
—— 4-(4-chlorophenyl)-3-[4-[4-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione 156525-77-8 C22H14Cl2N6S2
4-(4-chlorophenyl)-3-[4-[4-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione
—— (3E)-5-hydroxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one 1087343-95-0 C22H17N3O2S
(3E)-5-hydroxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one
—— 5-(4-methoxyphenyl)oxazole-4-carboxaldehyde 1166384-52-6 C11H9NO3
5-(4-methoxyphenyl)oxazole-4-carboxaldehyde
—— (3E)-5-methoxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one 1087343-92-7 C23H19N3O2S
(3E)-5-methoxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one
—— 5-(2-methyl-2H-pyrazol-3-yl)-2-(2,4,6-trimethylphenylamino)-benzamide 1085386-27-1 C20H22N4O
5-(2-methyl-2H-pyrazol-3-yl)-2-(2,4,6-trimethylphenylamino)-benzamide
—— [5-(6-Amino-pyridin-3-yl)-3-cyclopropyl-2-(4-trifluoromethoxy-phenyl)-3H-imidazol-4-yl]-(4-pyrrolidin-1-yl-piperidin-1-yl)-methanone 1097068-65-9 C28H31F3N6O2
[5-(6-Amino-pyridin-3-yl)-3-cyclopropyl-2-(4-trifluoromethoxy-phenyl)-3H-imidazol-4-yl]-(4-pyrrolidin-1-yl-piperidin-1-yl)-methanone
—— 3-phenyl-5-(dec-9-enyl)-1H-1,2,4-triazole 1107003-57-5 C18H25N3
3-phenyl-5-(dec-9-enyl)-1H-1,2,4-triazole
—— 2-(2-aminophenyl)-benzoxazole-4-carboxylic acid methyl ester 1086562-03-9 C15H12N2O3
2-(2-aminophenyl)-benzoxazole-4-carboxylic acid methyl ester
—— N-(1-amino-1,2-dioxoheptan-3-yl)-2-(4-phenyl-1H-imidazol-1-yl)nicotinamide 1037826-40-6 C22H23N5O3
N-(1-amino-1,2-dioxoheptan-3-yl)-2-(4-phenyl-1H-imidazol-1-yl)nicotinamide
—— 1-(4-phenyl-5-thioxo-1,2,4-triazol-3-yl)methyl-4-amino-3-p-methoxybenzyl-5-oxo-4,5-dihydro-1,2,4-triazole 1161426-89-6 C19H19N7O2S
1-(4-phenyl-5-thioxo-1,2,4-triazol-3-yl)methyl-4-amino-3-p-methoxybenzyl-5-oxo-4,5-dihydro-1,2,4-triazole
—— 4-(3-methylphenyl)-3-[4-[4-(3-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione 1174172-04-3 C24H20N6S2
4-(3-methylphenyl)-3-[4-[4-(3-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione
—— N-(4-(1H-pyrazol-4-yl)phenyl)chroman-3-carboxamide 1093961-37-5 C19H17N3O2
N-(4-(1H-pyrazol-4-yl)phenyl)chroman-3-carboxamide
—— 5-{(E)-2-[1-(3,5-bis-trifluoromethyl-phenyl)-3-(3-chlorophenyl)-1H-pyrazol-4-yl]-vinyl}-1H-tetrazole 1097120-39-2 C20H11ClF6N6
5-{(E)-2-[1-(3,5-bis-trifluoromethyl-phenyl)-3-(3-chlorophenyl)-1H-pyrazol-4-yl]-vinyl}-1H-tetrazole
—— 4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[(4R,5R)-4-(3,4-difluorophenyl)-3-methyl-2-oxo-1,3-oxazolidin-5-yl]methyl}-N-methylbenzamide 1093753-56-0 C30H26F2N4O4
4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[(4R,5R)-4-(3,4-difluorophenyl)-3-methyl-2-oxo-1,3-oxazolidin-5-yl]methyl}-N-methylbenzamide
—— N-{[(3S)-1-(5-bromopyridin-2-yl)pyrrolidin-3-yl]methyl}-4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzamide 1093753-50-4 C28H26BrN5O2
N-{[(3S)-1-(5-bromopyridin-2-yl)pyrrolidin-3-yl]methyl}-4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzamide
—— 4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[5-methyl-3-(5-nitropyridin-2-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl}benzamide 1093753-04-8 C28H24N6O6
4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)-N-{[5-methyl-3-(5-nitropyridin-2-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl}benzamide
—— 3-[2,4-bis(trifluoromethyl)phenyl]-5-methyl-7-[3-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]-2-(trifluoromethyl)-3H-imidazo[4,5-b]pyridine 1075253-34-7 C22H11F9N6S
3-[2,4-bis(trifluoromethyl)phenyl]-5-methyl-7-[3-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]-2-(trifluoromethyl)-3H-imidazo[4,5-b]pyridine
—— N-{[(3R)-1-(5-bromopyridin-2-yl)pyrrolidin-3-yl]methyl}-4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzamide 1093753-49-1 C28H26BrN5O2
N-{[(3R)-1-(5-bromopyridin-2-yl)pyrrolidin-3-yl]methyl}-4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzamide
—— 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N'-(2-methylhexanoyl)pyrazole-3-carbohydrazide 1020797-88-9 C24H25Cl3N4O2
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N'-(2-methylhexanoyl)pyrazole-3-carbohydrazide
—— 3-(2-{[(1,1-dimethylethyl)(dimethyl)silyl]oxy}ethyl)-6-methyl-N-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4-[3-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]-2-pyridinamine 727993-19-3 C30H37N7OSSi
3-(2-{[(1,1-dimethylethyl)(dimethyl)silyl]oxy}ethyl)-6-methyl-N-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4-[3-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]-2-pyridinamine
—— 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N'-hexanoyl-4-methylpyrazole-3-carbohydrazide 1020796-92-2 C23H23Cl3N4O2
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N'-hexanoyl-4-methylpyrazole-3-carbohydrazide