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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C36H45N5O8
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C34H41N5O8
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C40H46N6O7
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C34H40N4O8
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 2-(2-methoxyethylsulfanyl)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]acetamide —— C19H31N3O2S
2-(2-methoxyethylsulfanyl)-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]acetamide
—— 1-[4-(2-Fluorophenyl)piperazin-1-yl]-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propan-1-one —— C20H20FN5O2
1-[4-(2-Fluorophenyl)piperazin-1-yl]-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propan-1-one
—— 1-[4-(4-Methoxyphenyl)piperazin-1-yl]-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propan-1-one —— C21H23N5O3
1-[4-(4-Methoxyphenyl)piperazin-1-yl]-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propan-1-one
—— [4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone —— C24H30FN3O2
[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone
—— [4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone —— C24H30FN3O2
[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone
—— 5-[(1R)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C21H21N5OS
5-[(1R)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanediamide —— C39H47N7O5
N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanediamide
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C34H44N6O6
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— [(1S,2S)-2-methylcyclopropyl]-[4-(4-methylpiperazin-1-yl)sulfonylpiperazin-1-yl]methanone —— C14H26N4O3S
[(1S,2S)-2-methylcyclopropyl]-[4-(4-methylpiperazin-1-yl)sulfonylpiperazin-1-yl]methanone
—— N'-hydroxy-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanediamide —— C33H42N6O6
N'-hydroxy-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanediamide
—— N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]-6-pyrazol-1-ylpyridine-3-carboxamide —— C23H28N6O
N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]-6-pyrazol-1-ylpyridine-3-carboxamide
—— 2,4,5-trimethyl-N-[3-[(2S)-4-methyl-2-phenylpiperazin-1-yl]propyl]furan-3-carboxamide —— C22H31N3O2
2,4,5-trimethyl-N-[3-[(2S)-4-methyl-2-phenylpiperazin-1-yl]propyl]furan-3-carboxamide
—— N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]cyclopropanecarboxamide —— C18H27N3O
N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]cyclopropanecarboxamide
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C33H41N5O6
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C38H45N7O5
N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— 3-cyano-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]benzamide —— C22H26N4O
3-cyano-N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]benzamide
—— (2S)-1-(2,5-dimethylphenoxy)-3-[4-(4-fluorophenyl)piperazin-1-yl]propan-2-ol —— C21H27FN2O2
(2S)-1-(2,5-dimethylphenoxy)-3-[4-(4-fluorophenyl)piperazin-1-yl]propan-2-ol
—— N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]-3-[(2S)-oxolan-2-yl]propanamide —— C21H33N3O2
N-[3-[(2R)-4-methyl-2-phenylpiperazin-1-yl]propyl]-3-[(2S)-oxolan-2-yl]propanamide
—— (2S)-1-[(2-fluorophenyl)methoxy]-3-[4-(2-fluorophenyl)piperazin-1-yl]propan-2-ol —— C20H24F2N2O2
(2S)-1-[(2-fluorophenyl)methoxy]-3-[4-(2-fluorophenyl)piperazin-1-yl]propan-2-ol
—— (2R)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[(2-fluorophenyl)methoxy]propan-2-ol —— C20H24ClFN2O2
(2R)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[(2-fluorophenyl)methoxy]propan-2-ol
—— 4-[(3-methyl-1,2-oxazol-5-yl)methyl]-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]piperazine-1-carboxamide —— C18H31N5O2
4-[(3-methyl-1,2-oxazol-5-yl)methyl]-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]piperazine-1-carboxamide
—— (2R)-1-[(2-fluorophenyl)methoxy]-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-ol —— C18H23FN4O2
(2R)-1-[(2-fluorophenyl)methoxy]-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-ol
—— (2S)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[(2-fluorophenyl)methoxy]propan-2-ol —— C20H24ClFN2O2
(2S)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[(2-fluorophenyl)methoxy]propan-2-ol
—— (E)-1-[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-3-(5-methylthiophen-2-yl)prop-2-en-1-one —— C18H27N3O4S2
(E)-1-[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-3-(5-methylthiophen-2-yl)prop-2-en-1-one
—— (2S)-1-[(2-fluorophenyl)methoxy]-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-ol —— C18H23FN4O2
(2S)-1-[(2-fluorophenyl)methoxy]-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-ol
—— N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C40H49N7O5
N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C38H45N7O5
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C32H40N6O6
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C31H38N6O6
N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide
—— 5-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid —— C32H39N5O6
5-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-5-oxopentanoic acid
—— N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide —— C32H40N6O6
N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanediamide
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C31H38N6O6
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide
—— N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C37H43N7O5
N'-(2-aminophenyl)-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide
—— 8-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid —— C34H43N5O6
8-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid
—— 5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C31H37N5O6
5-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C32H39N5O6
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C33H42N6O6
N'-hydroxy-N-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— 4-benzyl-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]piperazine-1-carboxamide —— C20H32N4O
4-benzyl-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]piperazine-1-carboxamide
—— N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C33H42N6O6
N'-hydroxy-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— 7-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-7-oxoheptanoic acid —— C34H43N5O6
7-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-7-oxoheptanoic acid
—— 5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C31H37N5O6
5-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— 8-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid —— C35H45N5O6
8-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide —— C39H47N7O5
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]heptanediamide
—— N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide —— C40H49N7O5
N'-(2-aminophenyl)-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]heptanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide —— C40H49N7O5
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]octanediamide
—— N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide —— C37H43N7O5
N'-(2-aminophenyl)-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]pentanediamide