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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]heptanamide —— C28H45N5O
N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]heptanamide
—— [4-[4-[4-(2-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperazin-1-yl]-[(2S)-oxolan-2-yl]methanone —— C28H31FN6O3
[4-[4-[4-(2-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperazin-1-yl]-[(2S)-oxolan-2-yl]methanone
—— N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-fluorobenzamide —— C28H36FN5O
N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-fluorobenzamide
—— (2S)-2-chloro-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(2-methylpropyl)propanamide —— C26H39ClFN5O
(2S)-2-chloro-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(2-methylpropyl)propanamide
—— (2R)-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-methylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(furan-2-ylmethyl)butan-2-amine —— C26H36FN5O
(2R)-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-methylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(furan-2-ylmethyl)butan-2-amine
—— N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methylbutanamide —— C26H41N5O
N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methylbutanamide
—— (2S)-2-chloro-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-propylpropanamide —— C25H37ClFN5O
(2S)-2-chloro-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-propylpropanamide
—— (2S)-2-chloro-N-cyclopropyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]propanamide —— C23H31ClFN5O
(2S)-2-chloro-N-cyclopropyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]propanamide
—— N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3,5-dimethoxybenzamide —— C30H41N5O3
N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3,5-dimethoxybenzamide
—— N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-(4-fluorophenyl)acetamide —— C29H38FN5O
N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-(4-fluorophenyl)acetamide
—— N-[(2R)-butan-2-yl]-4-[4-(3-methoxyphenyl)piperazin-1-yl]phthalazine-1-carboxamide —— C24H29N5O2
N-[(2R)-butan-2-yl]-4-[4-(3-methoxyphenyl)piperazin-1-yl]phthalazine-1-carboxamide
—— (1S,2R)-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-2-phenyl-N-propylcyclopropane-1-carboxamide —— C32H42FN5O
(1S,2R)-N-[[3-ethyl-1-(4-fluorophenyl)-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-2-phenyl-N-propylcyclopropane-1-carboxamide
—— 4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]phthalazine-1-carboxamide —— C25H28ClN5O3
4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]phthalazine-1-carboxamide
—— (1S,2R)-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-methylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(3-methoxypropyl)-2-phenylcyclopropane-1-carboxamide —— C30H38FN5O2
(1S,2R)-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-methylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-(3-methoxypropyl)-2-phenylcyclopropane-1-carboxamide
—— N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-(trifluoromethyl)benzamide —— C29H36F3N5O
N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-(trifluoromethyl)benzamide
—— (2S)-N-[(2S)-butan-2-yl]-2-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]hexanamide —— C29H47N5O
(2S)-N-[(2S)-butan-2-yl]-2-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]hexanamide
—— (2S)-2-ethyl-N-[[3-methyl-5-(4-methylpiperazin-1-yl)-1-phenylpyrazol-4-yl]methyl]-N-(2-methylpropyl)hexanamide —— C28H45N5O
(2S)-2-ethyl-N-[[3-methyl-5-(4-methylpiperazin-1-yl)-1-phenylpyrazol-4-yl]methyl]-N-(2-methylpropyl)hexanamide
—— (2R)-N-[(2-chlorophenyl)methyl]-N-[[5-(4-ethylpiperazin-1-yl)-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methyl]butan-2-amine —— C28H37ClFN5
(2R)-N-[(2-chlorophenyl)methyl]-N-[[5-(4-ethylpiperazin-1-yl)-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methyl]butan-2-amine
—— (2R)-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-2-phenyl-N-propan-2-ylbutanamide —— C31H42FN5O
(2R)-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-2-phenyl-N-propan-2-ylbutanamide
—— ethyl (3S)-1-[2-[4-[2-(4-fluoroanilino)-1,3-thiazole-4-carbonyl]piperazin-1-yl]acetyl]piperidine-3-carboxylate —— C24H30FN5O4S
ethyl (3S)-1-[2-[4-[2-(4-fluoroanilino)-1,3-thiazole-4-carbonyl]piperazin-1-yl]acetyl]piperidine-3-carboxylate
—— N-[(2R)-butan-2-yl]-3-chloro-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide —— C28H36ClN5O
N-[(2R)-butan-2-yl]-3-chloro-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide
—— N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]-2-(4-methoxyphenyl)acetamide —— C30H40FN5O2
N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]-2-(4-methoxyphenyl)acetamide
—— N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxybenzenesulfonamide —— C28H39N5O3S
N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxybenzenesulfonamide
—— (1R,2R)-N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-phenylcyclopropane-1-carboxamide —— C31H41N5O
(1R,2R)-N-[(2R)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-2-phenylcyclopropane-1-carboxamide
—— 4-[4-(2-chlorophenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide —— C27H26ClN5O
4-[4-(2-chlorophenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide
—— 1-[(2R)-butan-2-yl]-1-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-(2-methylphenyl)urea —— C29H40N6O
1-[(2R)-butan-2-yl]-1-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-(2-methylphenyl)urea
—— 4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide —— C28H28ClN5O2
4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide
—— 4-[4-(4-fluorophenyl)piperazin-1-yl]-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]phthalazine-1-carboxamide —— C26H31FN6O
4-[4-(4-fluorophenyl)piperazin-1-yl]-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]phthalazine-1-carboxamide
—— (2R)-2-chloro-N-cyclopropyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]propanamide —— C23H31ClFN5O
(2R)-2-chloro-N-cyclopropyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]propanamide
—— N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3,5-dimethoxybenzamide —— C30H41N5O3
N-[(2S)-butan-2-yl]-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3,5-dimethoxybenzamide
—— ethyl 4-[[(2S)-butan-2-yl]-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-4-oxobutanoate —— C27H41N5O3
ethyl 4-[[(2S)-butan-2-yl]-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-4-oxobutanoate
—— N-[(2S)-butan-2-yl]-4-[4-(2-chlorophenyl)piperazin-1-yl]phthalazine-1-carboxamide —— C23H26ClN5O
N-[(2S)-butan-2-yl]-4-[4-(2-chlorophenyl)piperazin-1-yl]phthalazine-1-carboxamide
—— [(6R)-6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl]-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]methanone —— C25H25F3N4O
[(6R)-6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl]-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]methanone
—— 4-[4-(4-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide —— C28H29N5O2
4-[4-(4-methoxyphenyl)piperazin-1-yl]-N-[(1S)-1-phenylethyl]phthalazine-1-carboxamide
—— (2R)-2-chloro-N-(3-methoxypropyl)-N-[[3-methyl-5-(4-methylpiperazin-1-yl)-1-phenylpyrazol-4-yl]methyl]propanamide —— C23H34ClN5O2
(2R)-2-chloro-N-(3-methoxypropyl)-N-[[3-methyl-5-(4-methylpiperazin-1-yl)-1-phenylpyrazol-4-yl]methyl]propanamide
—— 4-[4-(2-fluorophenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]phthalazine-1-carboxamide —— C24H26FN5O2
4-[4-(2-fluorophenyl)piperazin-1-yl]-N-[[(2R)-oxolan-2-yl]methyl]phthalazine-1-carboxamide
—— (1S,2R)-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-(3-methoxypropyl)-2-phenylcyclopropane-1-carboxamide —— C31H41N5O2
(1S,2R)-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-(3-methoxypropyl)-2-phenylcyclopropane-1-carboxamide
—— N-[(2R)-butan-2-yl]-3-cyclopentyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]propanamide —— C29H45N5O
N-[(2R)-butan-2-yl]-3-cyclopentyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]propanamide
—— 4-[4-(2-fluorophenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]phthalazine-1-carboxamide —— C24H26FN5O2
4-[4-(2-fluorophenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]phthalazine-1-carboxamide
—— N-[(2S)-butan-2-yl]-3-chloro-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide —— C28H36ClN5O
N-[(2S)-butan-2-yl]-3-chloro-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide
—— N-[(2R)-butan-2-yl]-4-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide —— C30H41N5O
N-[(2R)-butan-2-yl]-4-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]benzamide
—— ethyl (3S)-1-[4-[4-(2-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperidine-3-carboxylate —— C27H30FN5O3
ethyl (3S)-1-[4-[4-(2-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperidine-3-carboxylate
—— 4-[4-[(1S)-1-(ethylamino)ethyl]-2-fluorophenyl]piperazin-2-one —— C14H20FN3O
4-[4-[(1S)-1-(ethylamino)ethyl]-2-fluorophenyl]piperazin-2-one
—— [4-(2-methoxyphenyl)piperazin-1-yl]-[(6R)-6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl]methanone —— C25H28N4O2
[4-(2-methoxyphenyl)piperazin-1-yl]-[(6R)-6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-2-yl]methanone
—— (2R)-2-ethyl-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-propan-2-ylhexanamide —— C29H46FN5O
(2R)-2-ethyl-N-[[1-(3-fluorophenyl)-3-methyl-5-(4-propan-2-ylpiperazin-1-yl)pyrazol-4-yl]methyl]-N-propan-2-ylhexanamide
—— 1-[(2S)-butan-2-yl]-3-cyclohexyl-1-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]urea —— C28H44N6O
1-[(2S)-butan-2-yl]-3-cyclohexyl-1-[[5-(4-ethylpiperazin-1-yl)-3-methyl-1-phenylpyrazol-4-yl]methyl]urea
—— ethyl (3R)-1-[4-[4-(4-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperidine-3-carboxylate —— C27H30FN5O3
ethyl (3R)-1-[4-[4-(4-fluorophenyl)piperazin-1-yl]phthalazine-1-carbonyl]piperidine-3-carboxylate
—— 4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]phthalazine-1-carboxamide —— C25H28ClN5O3
4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]phthalazine-1-carboxamide
—— (1R,2R)-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]-2-phenyl-N-propylcyclopropane-1-carboxamide —— C30H38FN5O
(1R,2R)-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]-2-phenyl-N-propylcyclopropane-1-carboxamide
—— (2S)-N-cyclopropyl-2-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]hexanamide —— C28H42FN5O
(2S)-N-cyclopropyl-2-ethyl-N-[[5-(4-ethylpiperazin-1-yl)-1-(3-fluorophenyl)-3-methylpyrazol-4-yl]methyl]hexanamide