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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S,4S)-2-[(1-ethoxy-ethoxy)-(5-methyl-[1,2,4]oxadiazole-3-yl)-methyl]-4-fluoro-pyrrolidine-1-carboxylic acid tert-butyl ester 851029-36-2 C17H28FN3O5
(2S,4S)-2-[(1-ethoxy-ethoxy)-(5-methyl-[1,2,4]oxadiazole-3-yl)-methyl]-4-fluoro-pyrrolidine-1-carboxylic acid tert-butyl ester
—— tert-butyl 4-({[3-benzoyl-7-(cyclopropylmethyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}carbonyl)piperidine-1-carboxylate 851748-94-2 C29H33N3O5S
tert-butyl 4-({[3-benzoyl-7-(cyclopropylmethyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}carbonyl)piperidine-1-carboxylate
—— tert-butyl [2-[3'-(cyclohexyloxy)-4'-[[[(2-hydroxyethyl)sulfonyl]amino]carbonyl]-4-biphenylyl]-ethyl][(2R)-2-hydroxy-2-phenylethyl]carbamate 881408-31-7 C36H46N2O8S
tert-butyl [2-[3'-(cyclohexyloxy)-4'-[[[(2-hydroxyethyl)sulfonyl]amino]carbonyl]-4-biphenylyl]-ethyl][(2R)-2-hydroxy-2-phenylethyl]carbamate
—— tert-butyl (1R,3R,4S)-4-benzyloxycarbonylamino-3-((pyridin-3-yloxy)methyl)cyclohexylcarbamate 847957-10-2 C25H33N3O5
tert-butyl (1R,3R,4S)-4-benzyloxycarbonylamino-3-((pyridin-3-yloxy)methyl)cyclohexylcarbamate
—— tert-butyl 4-(3-(pyrrolidin-1-yl)-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazin-2-yl)-1,4-diazepane-1-carboxylate 894808-54-9 C25H33N7O2
tert-butyl 4-(3-(pyrrolidin-1-yl)-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazin-2-yl)-1,4-diazepane-1-carboxylate
—— 1H-imidazole-4-carboxylic acid {3-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide 882983-49-5 C26H20N8O2
1H-imidazole-4-carboxylic acid {3-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide
—— tert-butyl [2-[3'-(cyclohexyloxy)-4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-4-biphenylyl]ethyl]-[(2R)-2-hydroxy-2-(4-nitrophenyl)ethyl]carbamate 881407-61-0 C37H47N3O10S
tert-butyl [2-[3'-(cyclohexyloxy)-4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-4-biphenylyl]ethyl]-[(2R)-2-hydroxy-2-(4-nitrophenyl)ethyl]carbamate
—— tert-butyl [2-(4-{3-[2-(acetylamino)-1,3-thiazol-4-yl]propyl}phenyl)ethyl]carbamate 874901-08-3 C21H29N3O3S
tert-butyl [2-(4-{3-[2-(acetylamino)-1,3-thiazol-4-yl]propyl}phenyl)ethyl]carbamate
—— florbetaben 878052-27-8 C21H26FNO3
florbetaben
—— tert-butyl 3-{[3-benzoyl-7-(2,6-difluorophenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate 851749-82-1 C28H25F2N3O4S
tert-butyl 3-{[3-benzoyl-7-(2,6-difluorophenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate
—— 1-(4-fluoro-5-{2-[4-(5-fluoro-benzo[d]isoxazol-3-yl)-piperazin-1-yl]-ethyl}-2,3-dihydro-indol-1-yl)-ethanone 860023-32-1 C23H24F2N4O2
1-(4-fluoro-5-{2-[4-(5-fluoro-benzo[d]isoxazol-3-yl)-piperazin-1-yl]-ethyl}-2,3-dihydro-indol-1-yl)-ethanone
—— tert-butyl (1R)-1-((4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperazinyl)carbonyl)-3-(methylthio)propylcarbamate 856417-88-4 C20H32N6O4S
tert-butyl (1R)-1-((4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperazinyl)carbonyl)-3-(methylthio)propylcarbamate
—— 2-(4-benzyloxy-phenoxy)-2,N-dimethyl-propionamide 872167-40-3 C18H21NO3
2-(4-benzyloxy-phenoxy)-2,N-dimethyl-propionamide
—— tert-butyl 4-(6-(1H-indazol-5-yl)-3-(pyrrolidin-1-yl)pyrazin-2-yl)-1,4-diazepane-1-carboxylate 894808-55-0 C25H33N7O2
tert-butyl 4-(6-(1H-indazol-5-yl)-3-(pyrrolidin-1-yl)pyrazin-2-yl)-1,4-diazepane-1-carboxylate
—— phenyl {1-(3-{[tert-butyl(dimethyl)silyl]oxy}phenyl)-3-[1-methyl-1-(methylthio)ethyl]-1H-pyrazol-5-yl}carbamate 876300-24-2 C26H35N3O3SSi
phenyl {1-(3-{[tert-butyl(dimethyl)silyl]oxy}phenyl)-3-[1-methyl-1-(methylthio)ethyl]-1H-pyrazol-5-yl}carbamate
—— 3-(R)-dimethylamino-2-(R)-phenyl-piperidine-1-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 815630-19-4 C24H27F6N3O
3-(R)-dimethylamino-2-(R)-phenyl-piperidine-1-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide
—— tert-butyl [2-[4'-[(butyrylamino)sulfonyl]-3'-(cyclohexyloxy)-4-biphenylyl]ethyl][(2R)-2-hydroxy-2-phenylethyl]carbamate 855479-27-5 C37H48N2O7S
tert-butyl [2-[4'-[(butyrylamino)sulfonyl]-3'-(cyclohexyloxy)-4-biphenylyl]ethyl][(2R)-2-hydroxy-2-phenylethyl]carbamate
—— 2-(R)-(4-fluoro-2-methyl-phenyl)-3-(S)-[(2,2.2-trifluoro-ethylamino)-methyl]-pyrrolidine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 815626-77-8 C26H27F10N3O
2-(R)-(4-fluoro-2-methyl-phenyl)-3-(S)-[(2,2.2-trifluoro-ethylamino)-methyl]-pyrrolidine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide
—— 3-benzyloxy-4-methoxy-6-bromo-pyridine-2-carboxylic acid (4-fluoro-benzyl)-(2-hydroxy-ethyl)amide 895134-27-7 C23H22BrFN2O4
3-benzyloxy-4-methoxy-6-bromo-pyridine-2-carboxylic acid (4-fluoro-benzyl)-(2-hydroxy-ethyl)amide
—— methyl({[(2,3-dichlorophenyl)(methyl)amino]carbonyl}thio)acetate 882871-02-5 C11H11Cl2NO3S
methyl({[(2,3-dichlorophenyl)(methyl)amino]carbonyl}thio)acetate
—— tert-butyl 3-{[3-benzoyl-7-(4-methylphenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate 851749-94-5 C29H29N3O4S
tert-butyl 3-{[3-benzoyl-7-(4-methylphenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate
—— 1-[4-(4-azido-2-fluoro-phenyl)-piperazin-1-yl]-2-hydroxy-propan-1-one 864147-47-7 C13H16FN5O2
1-[4-(4-azido-2-fluoro-phenyl)-piperazin-1-yl]-2-hydroxy-propan-1-one
—— tert-butyl [(2R)-2-(4-aminophenyl)-2-hydroxyethyl][2-[[3 '-cyclopentyl-4'-[[[(3-hydroxypropyl)sulfonyl]-amino]carbonyl]-4-biphenylyl]oxy]ethyl]carbamate 881408-15-7 C36H47N3O8S
tert-butyl [(2R)-2-(4-aminophenyl)-2-hydroxyethyl][2-[[3 '-cyclopentyl-4'-[[[(3-hydroxypropyl)sulfonyl]-amino]carbonyl]-4-biphenylyl]oxy]ethyl]carbamate
—— [3-(2,4-dichloro-benzyl)-2-oxo-2,3-dihydro-benzoxazol-4-yloxy]-acetic acid tert-butyl ester 883000-04-2 C20H19Cl2NO5
[3-(2,4-dichloro-benzyl)-2-oxo-2,3-dihydro-benzoxazol-4-yloxy]-acetic acid tert-butyl ester
—— tert-butyl (1R)-1-cyclohexyl-2-(4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperazinyl)-2-oxoethylcarbamate 856417-86-2 C23H36N6O4
tert-butyl (1R)-1-cyclohexyl-2-(4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperazinyl)-2-oxoethylcarbamate
—— (5S)-3-[3-fluoro-4-(4-(5-methylene-1,3-thiazolidine-2,4-dione)phenylpiperazin-1-yl)phenyl]-1,3-oxazolidin-2-one-5-methyl carbamate 864665-20-3 C26H26FN5O6S
(5S)-3-[3-fluoro-4-(4-(5-methylene-1,3-thiazolidine-2,4-dione)phenylpiperazin-1-yl)phenyl]-1,3-oxazolidin-2-one-5-methyl carbamate
—— 7-[N-[(2-methylsulfonyl)phenyl]-N-propylamino]-3-(4-methoxybenzyl)-1-methyl-1,3-dihydro-2H-benzimidazol-2-one 851889-20-8 C26H29N3O4S
7-[N-[(2-methylsulfonyl)phenyl]-N-propylamino]-3-(4-methoxybenzyl)-1-methyl-1,3-dihydro-2H-benzimidazol-2-one
—— tert-butyl N-[3-(6-dibenzofuran-4-ylpyrimidin-4-ylamino)phenyl]carbamate 872602-64-7 C27H24N4O3
tert-butyl N-[3-(6-dibenzofuran-4-ylpyrimidin-4-ylamino)phenyl]carbamate
—— 2,9-Dibenzoyl-6-chloro-3,4-dihydropyrido[3,4-b]indol-1-one 889444-70-6 C25H17ClN2O3
2,9-Dibenzoyl-6-chloro-3,4-dihydropyrido[3,4-b]indol-1-one
—— 2-ethoxy-4-methoxy-6-[(3R)-tetrahydro-3-furanyloxy]-5-pyrimidinecarbaldehyde 811802-28-5 C12H16N2O5
2-ethoxy-4-methoxy-6-[(3R)-tetrahydro-3-furanyloxy]-5-pyrimidinecarbaldehyde
—— N-(Diphenylaminocarbonylmethyl)pyridinium 85691-17-4 C19H17N2O
N-(Diphenylaminocarbonylmethyl)pyridinium
—— 6-methyl-2-oxo-N-(pyridin-3-ylmethyl)chromene-3-carboxamide 878441-45-3 C17H14N2O3
6-methyl-2-oxo-N-(pyridin-3-ylmethyl)chromene-3-carboxamide
—— tert-butyl {(1R,2R)-1-[(morpholin-4-ylsulfinyl)methyl]-2,3-dihydro-1H-inden-2-yl}carbamate 845269-59-2 C19H28N2O4S
tert-butyl {(1R,2R)-1-[(morpholin-4-ylsulfinyl)methyl]-2,3-dihydro-1H-inden-2-yl}carbamate
—— (3-Chloro-4-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]phenyl)amine 878441-21-5 C15H22ClN3O
(3-Chloro-4-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]phenyl)amine
—— 1-(1,3-benzothiazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol 890593-68-7 C12H11N3OS
1-(1,3-benzothiazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol
—— 2-({5-[(4-methylphenoxy)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)-N-[4-(morpholin-4-yl)phenyl]acetamide 878427-68-0 C22H24N4O4S
2-({5-[(4-methylphenoxy)methyl]-1,3,4-oxadiazol-2-yl}sulfanyl)-N-[4-(morpholin-4-yl)phenyl]acetamide
—— 7-(furan-2-yl)-5-hydroxy-2-methyl-N-(6-methylpyridin-2-yl)-4-phenyl-4,6,7,8-tetrahydroquinoline-3-carboxamide 878427-73-7 C27H25N3O3
7-(furan-2-yl)-5-hydroxy-2-methyl-N-(6-methylpyridin-2-yl)-4-phenyl-4,6,7,8-tetrahydroquinoline-3-carboxamide
—— 2-{[4-ethyl-5-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-[4-(morpholin-4-yl)phenyl]acetamide 878437-61-7 C24H29N5O3S
2-{[4-ethyl-5-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-[4-(morpholin-4-yl)phenyl]acetamide
—— 2-{[5-(4-chlorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide 878426-97-2 C16H15ClN6OS2
2-{[5-(4-chlorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide
—— 2-{[5-(4-methoxybenzyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide 878437-58-2 C16H18N6O2S2
2-{[5-(4-methoxybenzyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide
—— N-[2-(1-propylbenzimidazol-2-yl)ethyl]furan-2-carboxamide 877287-92-8 C17H19N3O2
N-[2-(1-propylbenzimidazol-2-yl)ethyl]furan-2-carboxamide
—— N-[2-(1-ethylbenzimidazol-2-yl)ethyl]furan-2-carboxamide 871547-25-0 C16H17N3O2
N-[2-(1-ethylbenzimidazol-2-yl)ethyl]furan-2-carboxamide
—— 8-(4-(2-fluorobenzyl)piperazin-1-yl)-3-methyl-7-(2-methylallyl)-1H-purine-2,6(3H,7H)-dione 878430-56-9 C21H25FN6O2
8-(4-(2-fluorobenzyl)piperazin-1-yl)-3-methyl-7-(2-methylallyl)-1H-purine-2,6(3H,7H)-dione
—— 2-(9-benzyl-1-methyl-2,4-dioxo-7,8-dihydro-6H-purino[7,8-a]pyrimidin-3-yl)acetic acid 878423-55-3 C18H19N5O4
2-(9-benzyl-1-methyl-2,4-dioxo-7,8-dihydro-6H-purino[7,8-a]pyrimidin-3-yl)acetic acid
—— 3-((4-morpholinophenyl)amino)-1,2,4-triazin-5(4H)-one 857492-04-7 C13H15N5O2
3-((4-morpholinophenyl)amino)-1,2,4-triazin-5(4H)-one
—— N-(3-Morpholin-4-yl-propyl)-3-(2-oxo-benzooxazol-3-yl)-propionamide 853751-91-4 C17H23N3O4
N-(3-Morpholin-4-yl-propyl)-3-(2-oxo-benzooxazol-3-yl)-propionamide
—— 3-(2-isopropoxybenzyl)benzo[d]oxazol-2(3H)-one 871673-03-9 C17H17NO3
3-(2-isopropoxybenzyl)benzo[d]oxazol-2(3H)-one
—— 3-(2-Oxo-benzooxazol-3-yl)-N-m-tolyl-propionamide 851989-08-7 C17H16N2O3
3-(2-Oxo-benzooxazol-3-yl)-N-m-tolyl-propionamide
—— N-(4-methylbenzyl)-3-(2-oxo-1,3-benzoxazol-3(2H)-yl)propanamide 851988-89-1 C18H18N2O3
N-(4-methylbenzyl)-3-(2-oxo-1,3-benzoxazol-3(2H)-yl)propanamide
—— N-(2-{[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methoxy}phenyl)acetamide 853752-01-9 C17H14ClN3O3
N-(2-{[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methoxy}phenyl)acetamide