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—— 3-(S)-[(cyclopropylmethyl-amino)-methyl]-2-(R)-(4-fluoro-2-methyl-phenyl)-pyrrolidine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 815631-52-8 C28H32F7N3O
3-(S)-[(cyclopropylmethyl-amino)-methyl]-2-(R)-(4-fluoro-2-methyl-phenyl)-pyrrolidine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide
—— dimethyl 5-(4-tert-butoxycarbonylaminopiperidin-1-yl)terephthalate 848499-86-5 C20H28N2O6
dimethyl 5-(4-tert-butoxycarbonylaminopiperidin-1-yl)terephthalate
—— tert-Butyl 2-(benzamido)-4-(3-(trifluoromethoxy)phenoxy)benzoate 890315-18-1 C25H22F3NO5
tert-Butyl 2-(benzamido)-4-(3-(trifluoromethoxy)phenoxy)benzoate
—— tert-Butyl 2-(3-acetylbenzamido)-4-phenoxybenzoate 890314-69-9 C26H25NO5
tert-Butyl 2-(3-acetylbenzamido)-4-phenoxybenzoate
—— tert-Butyl {1-[5-(2-chloro-5-fluorobenzyl)-1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl]piperidin-3-yl}carbamate 894794-77-5 C25H31ClFN5O4
tert-Butyl {1-[5-(2-chloro-5-fluorobenzyl)-1,3-dimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl]piperidin-3-yl}carbamate
—— 3-(R)-amino-2-(S)-o-tolyl-pyrrolidine-1-(R)-carboxylic acid [1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 815630-29-6 C23H25F6N3O
3-(R)-amino-2-(S)-o-tolyl-pyrrolidine-1-(R)-carboxylic acid [1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide
—— 1-[4-(4-azido-2,6-difluoro-phenyl)-piperazin-1-yl]-2-bromo-ethanone 864147-28-4 C12H12BrF2N5O
1-[4-(4-azido-2,6-difluoro-phenyl)-piperazin-1-yl]-2-bromo-ethanone
—— naphthalene-2-carboxylic acid {3-[4-(3,4-dimethoxy-phenyl)-pyrimidin-2-ylamino]-phenyl}-amide 881676-83-1 C29H24N4O3
naphthalene-2-carboxylic acid {3-[4-(3,4-dimethoxy-phenyl)-pyrimidin-2-ylamino]-phenyl}-amide
—— tert-butyl 3-{[(3-benzoyl-6-oxo-7-phenyl-6,7-dihydrothieno[2,3-b]pyridin-2-yl)amino]methyl}azetidine-1-carboxylate 851749-30-9 C29H29N3O4S
tert-butyl 3-{[(3-benzoyl-6-oxo-7-phenyl-6,7-dihydrothieno[2,3-b]pyridin-2-yl)amino]methyl}azetidine-1-carboxylate
—— 3-[[2-[[3-[[(aminoacetyl)amino]methyl]phenyl]amino]-5-cyano-4-pyrimidinyl]]amino-benzoic acid 892414-18-5 C21H19N7O3
3-[[2-[[3-[[(aminoacetyl)amino]methyl]phenyl]amino]-5-cyano-4-pyrimidinyl]]amino-benzoic acid
—— tert-butyl [4-chloro-2-(2-methoxyethyl)-6,7-dimethyl-1H-imidazo[4,5-c]pyridin-1-yl]carbamate 878492-84-3 C16H23ClN4O3
tert-butyl [4-chloro-2-(2-methoxyethyl)-6,7-dimethyl-1H-imidazo[4,5-c]pyridin-1-yl]carbamate
—— methyl (2S)-2-{[4-methoxy-6-(1H-pyrazol-5-yl)pyridin-3-yl]oxy}propanoate 871836-43-0 C13H15N3O4
methyl (2S)-2-{[4-methoxy-6-(1H-pyrazol-5-yl)pyridin-3-yl]oxy}propanoate
—— (2S)-6-bromo-5-oxo-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]hexanoic acid 815619-01-3 C17H21BrN2O6
(2S)-6-bromo-5-oxo-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]hexanoic acid
—— N-(3,4-dichlorophenyl)-3-phenylbutanamide 86886-79-5 C16H15Cl2NO
N-(3,4-dichlorophenyl)-3-phenylbutanamide
—— tert-butyl [3-[3'-cyclopentyl-4'-[[(methylsulfonyl)amino]carbonyl]-4-biphenylyl]propyl][(2R)-2-hydroxy-2-phenylethyl]carbamate 855479-80-0 C35H44N2O6S
tert-butyl [3-[3'-cyclopentyl-4'-[[(methylsulfonyl)amino]carbonyl]-4-biphenylyl]propyl][(2R)-2-hydroxy-2-phenylethyl]carbamate
—— 1-(5-chloro-2-fluoro-4-nitro-phenyl)-4-methyl-piperidine 864838-41-5 C18H26FN3O2
1-(5-chloro-2-fluoro-4-nitro-phenyl)-4-methyl-piperidine
—— tert-butyl [2-[[3'-(cyclohexyloxy)-4'-[[[(3-hydroxy-propyl)sulfonyl]amino]carbonyl]-4-biphenylyl]oxy]-ethyl][(2R)-2-hydroxy-2-(4-nitrophenyl)ethyl]-carbamate 881407-64-3 C37H47N3O11S
tert-butyl [2-[[3'-(cyclohexyloxy)-4'-[[[(3-hydroxy-propyl)sulfonyl]amino]carbonyl]-4-biphenylyl]oxy]-ethyl][(2R)-2-hydroxy-2-(4-nitrophenyl)ethyl]-carbamate
—— 3-chloro-N-[5-(diethylsulfamoyl)-2-methoxyphenyl]benzamide 847471-69-6 C18H21ClN2O4S
3-chloro-N-[5-(diethylsulfamoyl)-2-methoxyphenyl]benzamide
—— tert-butyl [(2R)-2-(3-chlorophenyl)-2-hydroxy-ethyl][3-[4'-[[[(3-hydroxypropyl)sulfonyl]amino]-carbonyl]-3'-isopropoxy-4-biphenylyl]propyl]carbamate 881407-75-6 C35H45ClN2O8S
tert-butyl [(2R)-2-(3-chlorophenyl)-2-hydroxy-ethyl][3-[4'-[[[(3-hydroxypropyl)sulfonyl]amino]-carbonyl]-3'-isopropoxy-4-biphenylyl]propyl]carbamate
—— 1-[4-(4-azido-2,6-difluoro-phenyl)-piperazin-1-yl]-2-pyridin-3-yl-ethanone 864147-20-6 C17H16F2N6O
1-[4-(4-azido-2,6-difluoro-phenyl)-piperazin-1-yl]-2-pyridin-3-yl-ethanone
—— tert-butyl (7S)-7-[(tert-butoxycarbonyl)amino]-7-[5-(2-naphthyl)-1,3,4-oxadiazol-2-yl]heptanoate 891270-06-7 C28H37N3O5
tert-butyl (7S)-7-[(tert-butoxycarbonyl)amino]-7-[5-(2-naphthyl)-1,3,4-oxadiazol-2-yl]heptanoate
—— 4-([1,4]oxazepane-4-carbonyl)-1H-pyrrole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide 863483-96-9 C19H30N4O3
4-([1,4]oxazepane-4-carbonyl)-1H-pyrrole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
—— tert-butyl [(2R)-2-(4-aminophenyl)-2-hydroxyethyl][2-[[3'-(cyclohexyloxy)-4'-[[[(3-hydroxypropyl)-sulfonyl]amino]carbonyl]-4-biphenylyl]oxy]ethyl]-carbamate 881408-14-6 C37H49N3O9S
tert-butyl [(2R)-2-(4-aminophenyl)-2-hydroxyethyl][2-[[3'-(cyclohexyloxy)-4'-[[[(3-hydroxypropyl)-sulfonyl]amino]carbonyl]-4-biphenylyl]oxy]ethyl]-carbamate
—— 4-(Hydroxyphenylmethylene)-1-[3-(1H-imidazol-1-yl)propyl]-5-(3-pyridinyl)-2,3-pyrrolidinedione 898796-78-6 C22H20N4O3
4-(Hydroxyphenylmethylene)-1-[3-(1H-imidazol-1-yl)propyl]-5-(3-pyridinyl)-2,3-pyrrolidinedione
—— tert-butyl [(2R)-2-[[tert-butyl(dimethyl)silyl]oxy]-2-(3-chlorophenyl)ethyl][2-[4'-[[[(cyanomethyl)sulfonyl]-amino]carbonyl]-3'-(cyclohexyloxy)-4-biphenylyl]ethyl]-carbamate 881408-89-5 C42H56ClN3O7SSi
tert-butyl [(2R)-2-[[tert-butyl(dimethyl)silyl]oxy]-2-(3-chlorophenyl)ethyl][2-[4'-[[[(cyanomethyl)sulfonyl]-amino]carbonyl]-3'-(cyclohexyloxy)-4-biphenylyl]ethyl]-carbamate
—— tert-butyl 4-[({5-[2-(2-acetylaminothiazol-4-yl)ethyl]-2-thienyl}acetyl)amino]-1-piperidinecarboxylate 878629-05-1 C23H32N4O4S2
tert-butyl 4-[({5-[2-(2-acetylaminothiazol-4-yl)ethyl]-2-thienyl}acetyl)amino]-1-piperidinecarboxylate
—— tert-butyl 3-{[3-(4-fluoro-3-methylbenzoyl)-7-(4-methylphenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate 851750-07-7 C30H30FN3O4S
tert-butyl 3-{[3-(4-fluoro-3-methylbenzoyl)-7-(4-methylphenyl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridin-2-yl]amino}azetidine-1-carboxylate
—— 2-amino-5-[N-(2-dimethylaminoethyl)-N-methylamino]-7-methylthiazolo[5,4-b]pyridine 850172-58-6 C12H19N5S
2-amino-5-[N-(2-dimethylaminoethyl)-N-methylamino]-7-methylthiazolo[5,4-b]pyridine
—— 12b,12c-Dihydroacenaphthyleno[1,2-b]quinoxaline 864718-12-7 C18H12N2
12b,12c-Dihydroacenaphthyleno[1,2-b]quinoxaline
—— N2-[2-(3azidomethyl-phenyl)-1-methyl-ethyl]-N4-methyl-N4-(7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-pyrimidine-2,4-diamine 872059-08-0 C26H25N11
N2-[2-(3azidomethyl-phenyl)-1-methyl-ethyl]-N4-methyl-N4-(7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-pyrimidine-2,4-diamine
—— 3-{2,6-difluoro-4-[4,5-dihydro-6-(3-isopropyloxypropyl)-naphtho[1,2-d]thiazol-2-ylcarbamoyl]-phenyl}-2-methylacrylic acid 844843-95-4 C28H28F2N2O4S
3-{2,6-difluoro-4-[4,5-dihydro-6-(3-isopropyloxypropyl)-naphtho[1,2-d]thiazol-2-ylcarbamoyl]-phenyl}-2-methylacrylic acid
—— benzo[b]thiophene-2-carboxylic acid [4-(1H-benzoimidazol-2-yl)-3-fluoro-phenyl]-amide 849508-06-1 C22H14FN3OS
benzo[b]thiophene-2-carboxylic acid [4-(1H-benzoimidazol-2-yl)-3-fluoro-phenyl]-amide
—— 5-pyridin-3-yl-thiophene-2-carboxylic acid [4-(1H-benzoimidazol-2-yl)-phenyl]-amide 849509-04-2 C23H16N4OS
5-pyridin-3-yl-thiophene-2-carboxylic acid [4-(1H-benzoimidazol-2-yl)-phenyl]-amide
—— N5,2,2-trimethyl-N8-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydropyrimido[4',5':4,5]thieno[2,3-c]isoquinoline-5,8-diamine 890024-79-0 C22H24N6S
N5,2,2-trimethyl-N8-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydropyrimido[4',5':4,5]thieno[2,3-c]isoquinoline-5,8-diamine
—— methyl {[2-(2,2-dimethylpropyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}acetate 886049-83-8 C21H30N2O5S
methyl {[2-(2,2-dimethylpropyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}acetate
—— 1-Methyl-3-hydroxy-2-oxo-3-(3-nitrophenacyl)-indolin 853-12-3 C17H14N2O5
1-Methyl-3-hydroxy-2-oxo-3-(3-nitrophenacyl)-indolin
—— 3-(3-amino-1H-indazol-5-yl)-N-[(1S)-1-(3-hydroxyphenyl)ethyl]prop-2-enamide 871709-60-3 C18H18N4O2
3-(3-amino-1H-indazol-5-yl)-N-[(1S)-1-(3-hydroxyphenyl)ethyl]prop-2-enamide
—— ethyl {4-(2-[amino(hydroxyimino)methyl]-8-[4-(4-phenylbutoxy)styryl]-2,3-dihydro-4H-1,4-benzoxazin-4-yl)}butanoate 847657-86-7 C33H39N3O5
ethyl {4-(2-[amino(hydroxyimino)methyl]-8-[4-(4-phenylbutoxy)styryl]-2,3-dihydro-4H-1,4-benzoxazin-4-yl)}butanoate
—— 2-{4-[(1E)-2-nitroethenyl]phenoxy}propanoic acid 86636-43-3 C11H11NO5
2-{4-[(1E)-2-nitroethenyl]phenoxy}propanoic acid
—— 2-bromo-1-{(S)-2-[5-(2-methoxy-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-pyrrolidin e-1-yl}-ethanone 851029-79-3 C16H16BrN3O4
2-bromo-1-{(S)-2-[5-(2-methoxy-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-pyrrolidin e-1-yl}-ethanone
—— 6-{[2-(azidomethyl)phenyl]thio}-3-[2-(benzyloxy)phenyl][1,2,4]triazolo[4,3-a]pyridine 876299-57-9 C26H20N6OS
6-{[2-(azidomethyl)phenyl]thio}-3-[2-(benzyloxy)phenyl][1,2,4]triazolo[4,3-a]pyridine
—— N-(1-adamantyl)-2-chloro-5-nitrobenzamide 85469-95-0 C17H19ClN2O3
N-(1-adamantyl)-2-chloro-5-nitrobenzamide
—— 6-{[2-(azidomethyl)phenyl]thio}-3-(2-chloro-3-methoxyphenyl)[1,2,4]triazolo[4,3-a]pyridine 876301-04-1 C20H15ClN6OS
6-{[2-(azidomethyl)phenyl]thio}-3-(2-chloro-3-methoxyphenyl)[1,2,4]triazolo[4,3-a]pyridine
—— 4-(Dimethylamino)-1,1-diphenylbutan-1-ol hydrochloride 894-19-9 C18H24ClNO
4-(Dimethylamino)-1,1-diphenylbutan-1-ol hydrochloride
—— 3-[6-({[1-(4-chlorobenzyl)-5-oxo-3-pyrrolidinyl]carbonyl}amino)-1H-benzimidazol-1-yl]-3-phenylpropanoic acid 887272-99-3 C28H25ClN4O4
3-[6-({[1-(4-chlorobenzyl)-5-oxo-3-pyrrolidinyl]carbonyl}amino)-1H-benzimidazol-1-yl]-3-phenylpropanoic acid
—— tert-Butyl 4-phenyl-2-(6-(1H-pyrrol-1-yl)pyridine-3-carboxamido)benzoate 890314-56-4 C27H25N3O3
tert-Butyl 4-phenyl-2-(6-(1H-pyrrol-1-yl)pyridine-3-carboxamido)benzoate
—— tert-butyl [1-(6-methoxy-3-nitropyridin-2-yl)piperidin-4-yl]carbamate 848500-04-9 C16H24N4O5
tert-butyl [1-(6-methoxy-3-nitropyridin-2-yl)piperidin-4-yl]carbamate
—— (2R,4S)-2-bromo-1-[4-fluoro-2-(5-tert-butyl-[1,3,4]oxadiazole-2-carbonyl)-pyrrolidine-1-yl]-ethanone 851029-11-3 C13H17BrFN3O3
(2R,4S)-2-bromo-1-[4-fluoro-2-(5-tert-butyl-[1,3,4]oxadiazole-2-carbonyl)-pyrrolidine-1-yl]-ethanone
—— 1,1-dimethylethyl {3-[1-({[5-(2-amino-4-pyrimidinyl)-2-thienyl]carbonyl}amino)ethyl]phenyl}carbamate 862698-72-4 C22H25N5O3S
1,1-dimethylethyl {3-[1-({[5-(2-amino-4-pyrimidinyl)-2-thienyl]carbonyl}amino)ethyl]phenyl}carbamate
—— 5-bromo-3-hydroxy-3-[2-oxo-2-(thiophen-2-yl)ethyl]indolin-2-one 83393-69-5 C14H10BrNO3S
5-bromo-3-hydroxy-3-[2-oxo-2-(thiophen-2-yl)ethyl]indolin-2-one