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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-acetyl-piperidine-4-carboxylic acid {3-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide 882983-59-7 C30H29N7O3
1-acetyl-piperidine-4-carboxylic acid {3-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide
—— 8-benzyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-ene 842110-09-2 C21H23N
8-benzyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-ene
—— 4-[(2-Chloro-6-fluorophenyl)methyl]thieno[3,2-b]pyrrole-5-carboxylic acid 842110-71-8 C14H9ClFNO2S
4-[(2-Chloro-6-fluorophenyl)methyl]thieno[3,2-b]pyrrole-5-carboxylic acid
—— 2,3-dihydro-benzo[1,4]dioxine-6-carboxylic acid [4-(5-pyridin-4-yl-1H-benzoimidazol-2-yl)-phenyl]-amide 849509-00-8 C27H20N4O3
2,3-dihydro-benzo[1,4]dioxine-6-carboxylic acid [4-(5-pyridin-4-yl-1H-benzoimidazol-2-yl)-phenyl]-amide
—— [1-(furan-2-ylmethylamino)-1-oxopropan-2-yl] 2H-chromene-3-carboxylate 841282-23-3 C18H17NO5
[1-(furan-2-ylmethylamino)-1-oxopropan-2-yl] 2H-chromene-3-carboxylate
—— N4,N4-dibenzyl-6-chloro-2-(ethoxymethyl)-N1-isopropyl-7-methyl-1H-imidazo[4,5-c]pyridine-1,4-diamine 878491-73-7 C27H32ClN5O
N4,N4-dibenzyl-6-chloro-2-(ethoxymethyl)-N1-isopropyl-7-methyl-1H-imidazo[4,5-c]pyridine-1,4-diamine
—— tert-butyl {1-[(3-chlorophenyl)(cyclopentyl)acetyl]piperidin-4-yl}carbamate 850618-00-7 C23H33ClN2O3
tert-butyl {1-[(3-chlorophenyl)(cyclopentyl)acetyl]piperidin-4-yl}carbamate
—— 3-(3-amino-1H-indazol-5-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]prop-2-enamide 871709-76-1 C19H20N4O2
3-(3-amino-1H-indazol-5-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]prop-2-enamide
—— (5,6-Dihydro-4H-[1,3]thiazin-2-yl)-(3-methoxy-phenyl)-amine 841223-61-8 C11H14N2OS
(5,6-Dihydro-4H-[1,3]thiazin-2-yl)-(3-methoxy-phenyl)-amine
—— methyl({[(2,5-dichlorophenyl)(methyl)amino]carbonyl}thio)acetate 882871-00-3 C11H11Cl2NO3S
methyl({[(2,5-dichlorophenyl)(methyl)amino]carbonyl}thio)acetate
—— 5-pyridin-2-yl-thiopene-2-carboxylix acid [4-(5-fluoro-1H-benzimidazol-2-yl)-phenyl]-amide 849507-53-5 C23H15FN4OS
5-pyridin-2-yl-thiopene-2-carboxylix acid [4-(5-fluoro-1H-benzimidazol-2-yl)-phenyl]-amide
—— N-(6-Chloro-3-pyridazinyl)hexahydro-1H-azepine-1-ethanamine 845736-80-3 C12H19ClN4
N-(6-Chloro-3-pyridazinyl)hexahydro-1H-azepine-1-ethanamine
—— 6-chloro-N-(cyclohexylmethyl)pyridazin-3-amine 845736-79-0 C11H16ClN3
6-chloro-N-(cyclohexylmethyl)pyridazin-3-amine
—— 2-(3-hydroxypropylamino)-N-naphthalen-1-ylacetamide 838090-78-1 C15H18N2O2
2-(3-hydroxypropylamino)-N-naphthalen-1-ylacetamide
—— 1-[6-chloro-9-[2-(trifluoromethoxy)benzoyl]-3,4-dihydro-1H-pyrido[3,4-b]indol-2-yl]-2,2,2-trifluoroethanone 889444-86-4 C21H13ClF6N2O3
1-[6-chloro-9-[2-(trifluoromethoxy)benzoyl]-3,4-dihydro-1H-pyrido[3,4-b]indol-2-yl]-2,2,2-trifluoroethanone
—— (2R,4S)-2-[(1-ethoxy-ethoxy)-(N-hydroxycarbamimidoyl)-methyl]-4-fluoro-pyrrolidine-1-carboxylic acid tert-butyl ester 851029-21-5 C15H28FN3O5
(2R,4S)-2-[(1-ethoxy-ethoxy)-(N-hydroxycarbamimidoyl)-methyl]-4-fluoro-pyrrolidine-1-carboxylic acid tert-butyl ester
—— 3-(1H-benzo[d]imidazol-2-yl)-N-(biphenyl-2-yl)piperidine-1-carboxamide 837389-93-2 C25H24N4O
3-(1H-benzo[d]imidazol-2-yl)-N-(biphenyl-2-yl)piperidine-1-carboxamide
—— 3-(1H-benzo[d]imidazol-2-yl)-N-(4-chloro-3-(trifluoromethyl)phenyl)piperidine-1-carboxamide 837389-88-5 C20H18ClF3N4O
3-(1H-benzo[d]imidazol-2-yl)-N-(4-chloro-3-(trifluoromethyl)phenyl)piperidine-1-carboxamide
—— isoquinoline-5-sulfonic acid {3-[4-(3,4-dimethoxy-phenyl)-pyrimidin-2-ylamino]-4-methyl-phenyl}-amide 881676-95-5 C28H25N5O4S
isoquinoline-5-sulfonic acid {3-[4-(3,4-dimethoxy-phenyl)-pyrimidin-2-ylamino]-4-methyl-phenyl}-amide
—— tert-butyl 3-(3-(azepan-1-yl)-6-bromopyrazin-2-ylamino)piperidine-1-carboxylate 894808-69-6 C20H32BrN5O2
tert-butyl 3-(3-(azepan-1-yl)-6-bromopyrazin-2-ylamino)piperidine-1-carboxylate
—— thiophene-2-sulfonic acid [4-(4-pyridin-4-yl-pyrimidin-2-ylamino)-phenyl]-amide 881675-99-6 C19H15N5O2S2
thiophene-2-sulfonic acid [4-(4-pyridin-4-yl-pyrimidin-2-ylamino)-phenyl]-amide
—— 1-(1-(3-chloro-2-methylphenylsulfonyl)piperidin-4-yl)-3-adamantylurea 836682-16-7 C23H32ClN3O3S
1-(1-(3-chloro-2-methylphenylsulfonyl)piperidin-4-yl)-3-adamantylurea
—— 1-adamantyl-3-(1-(phenylsulfonyl)piperidin-4-yl)urea 836681-64-2 C22H31N3O3S
1-adamantyl-3-(1-(phenylsulfonyl)piperidin-4-yl)urea
—— N-[1-(Benzylcarbamoyl-methyl)-piperidin-4-yl]-4-ethoxy-benzamide 836679-21-1 C23H29N3O3
N-[1-(Benzylcarbamoyl-methyl)-piperidin-4-yl]-4-ethoxy-benzamide
—— (S,S)-2-methyl-propane-2-sulfinic acid [2-methyl-1-(2-piperazin-1-yl-5-trifluoromethyl-phenyl)-propyl]-amide 851753-80-5 C19H30F3N3OS
(S,S)-2-methyl-propane-2-sulfinic acid [2-methyl-1-(2-piperazin-1-yl-5-trifluoromethyl-phenyl)-propyl]-amide
—— 4-(4-azido-2,6-difluoro-phenyl)-1,2,3,6-tetrahydro-pyridine 864147-09-1 C11H10F2N4
4-(4-azido-2,6-difluoro-phenyl)-1,2,3,6-tetrahydro-pyridine
—— N-[(3-Methoxy)propyl] 6-ethoxy-4-oxo-1,4-dihydro-quinoline-3-carboxamide 835924-73-7 C16H20N2O4
N-[(3-Methoxy)propyl] 6-ethoxy-4-oxo-1,4-dihydro-quinoline-3-carboxamide
—— tert-butyl 2-(4-cyanobenzoyl)-3-oxobutanoate 873326-76-2 C16H17NO4
tert-butyl 2-(4-cyanobenzoyl)-3-oxobutanoate
—— tert-butyl (R)-2-[[(R)-3-methylpiperidin-1-yl]carbonyl]-indoline-1-carboxylate 899825-49-1 C20H28N2O3
tert-butyl (R)-2-[[(R)-3-methylpiperidin-1-yl]carbonyl]-indoline-1-carboxylate
—— cyclopropanecarboxylic acid {3-[3-(2-trifluoromethyl-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide 882984-19-2 C26H19F3N6O
cyclopropanecarboxylic acid {3-[3-(2-trifluoromethyl-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide
—— cyclohexanecarboxylic acid {4-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide 882983-26-8 C29H28N6O2
cyclohexanecarboxylic acid {4-[3-(4-methoxy-phenyl)-[1,2,4]triazolo[3,4-a]phthalazin-6-ylamino]-phenyl}-amide
—— tert-butyl (2S)-2-(4-amino-2-chlorophenoxymethyl)pyrrolidine-1-carboxylate 884342-76-1 C16H23ClN2O3
tert-butyl (2S)-2-(4-amino-2-chlorophenoxymethyl)pyrrolidine-1-carboxylate
—— tert-butyl [(2R)-2-hydroxy-2-phenylethyl][3-[4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-3'-isopropoxy-4-biphenylyl]propyl]carbamate 881407-70-1 C35H46N2O8S
tert-butyl [(2R)-2-hydroxy-2-phenylethyl][3-[4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-3'-isopropoxy-4-biphenylyl]propyl]carbamate
—— tert-butyl 3-(6-bromo-3-(methylamino)pyrazin-2-ylamino)piperidine-1-carboxylate 894808-30-1 C15H24BrN5O2
tert-butyl 3-(6-bromo-3-(methylamino)pyrazin-2-ylamino)piperidine-1-carboxylate
—— 1,1-dimethylethyl (2S)-2-[[5-chloro-3'-fluoro-4'-(methylsulfonyl)[1,1'-biphenyl]-2-yl]oxy]propanoate 877383-53-4 C20H22ClFO5S
1,1-dimethylethyl (2S)-2-[[5-chloro-3'-fluoro-4'-(methylsulfonyl)[1,1'-biphenyl]-2-yl]oxy]propanoate
—— tert-butyl [(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]-[2-[[4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-3'-isopropoxy-4-biphenylyl]oxy]ethyl]carbamate 881407-58-5 C34H43ClN2O9S
tert-butyl [(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]-[2-[[4'-[[[(3-hydroxypropyl)sulfonyl]amino]carbonyl]-3'-isopropoxy-4-biphenylyl]oxy]ethyl]carbamate
—— 9-(3-dimethylamino-propyl)-2,3,4,9-tetrahydro-β-carbolin-1-one 894-58-6 C16H21N3O
9-(3-dimethylamino-propyl)-2,3,4,9-tetrahydro-β-carbolin-1-one
—— [4-fluoro-2-[[4-[(phenylmethyl)sulfonyl]-1-piperazinyl]methyl]phenoxy]-acetic acid, 1,1-dimethylethyl ester 888972-86-9 C24H31FN2O5S
[4-fluoro-2-[[4-[(phenylmethyl)sulfonyl]-1-piperazinyl]methyl]phenoxy]-acetic acid, 1,1-dimethylethyl ester
—— tert-butyl (1-{4-[2-(2-acetylaminothiazol-4-yl)ethyl]benzyl}-3-pyrrolidinyl)carbamate 878629-33-5 C23H32N4O3S
tert-butyl (1-{4-[2-(2-acetylaminothiazol-4-yl)ethyl]benzyl}-3-pyrrolidinyl)carbamate
—— 2-(R)-(4-fluoro-2-methyl-phenyl)-3-(S)-(4-methyl-piperidin-1-ylmethyl)-pyrrolidine-1-carboxylic acid [1-(R)-(3.5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 815626-69-8 C30H36F7N3O
2-(R)-(4-fluoro-2-methyl-phenyl)-3-(S)-(4-methyl-piperidin-1-ylmethyl)-pyrrolidine-1-carboxylic acid [1-(R)-(3.5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide
—— tert-butyl (1R)-1-benzyl-2-(4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperidinyl)-2-oxoethylcarbamate 856417-22-6 C25H33N5O4
tert-butyl (1R)-1-benzyl-2-(4-(5-methyl-3-oxo-1H-imidazo[1,5-c]imidazol-2(3H)-yl)-1-piperidinyl)-2-oxoethylcarbamate
—— tert-butyl (S)-2-(4-(2-(4-phenyl-3-fluorophenyl)propoxy)phenylcarbamoyl)-1-hydroxypropan-2-ylcarbamate 876915-54-7 C30H35FN2O5
tert-butyl (S)-2-(4-(2-(4-phenyl-3-fluorophenyl)propoxy)phenylcarbamoyl)-1-hydroxypropan-2-ylcarbamate
—— tert-butyl (S)-2-[[(R)-3-methylpiperidin-1-yl]carbonyl]-indoline-1-carboxylate 899825-35-5 C20H28N2O3
tert-butyl (S)-2-[[(R)-3-methylpiperidin-1-yl]carbonyl]-indoline-1-carboxylate
—— tert-butyl {[2-isobutyl-6-methyl-4-(4-methylphenyl)-5-({[4-(methylsulfonyl)phenyl]sulfonyl}methyl)pyridin-3-yl]methyl}carbamate 851579-60-7 C31H40N2O6S2
tert-butyl {[2-isobutyl-6-methyl-4-(4-methylphenyl)-5-({[4-(methylsulfonyl)phenyl]sulfonyl}methyl)pyridin-3-yl]methyl}carbamate
—— tert-butyl (4-chloro-2-{[4-(methylsulfonyl)phenyl]sulfonyl}phenoxy)acetate 847148-31-6 C19H21ClO7S2
tert-butyl (4-chloro-2-{[4-(methylsulfonyl)phenyl]sulfonyl}phenoxy)acetate
—— [2-(5,6-difluoro-pyridin-3-yl)-4-fluoro-benzyl]-carbamic acid tert-butyl ester 870063-09-5 C17H17F3N2O2
[2-(5,6-difluoro-pyridin-3-yl)-4-fluoro-benzyl]-carbamic acid tert-butyl ester
—— 1-phenyl-hexahydro-pyrrolo[3,4-c]pyrrole-2-carboxylic acid [1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide 815630-96-7 C24H25F6N3O
1-phenyl-hexahydro-pyrrolo[3,4-c]pyrrole-2-carboxylic acid [1-(3,5-bis-trifluoromethyl-phenyl)-ethyl]-methyl-amide
—— 2-(3-amino-3-{4-[2-(4-methoxy-phenyl)-quinolin-4-ylmethoxy]-phenyl}-2-oxo-pyrrolidin-l-yl)-propionic acid methyl ester 863116-67-0 C31H31N3O5
2-(3-amino-3-{4-[2-(4-methoxy-phenyl)-quinolin-4-ylmethoxy]-phenyl}-2-oxo-pyrrolidin-l-yl)-propionic acid methyl ester
—— N,N'-bis(2-phosphonoethyl)-3,4;9,10-perylenediimide 869371-15-3 C28H20N2O10P2
N,N'-bis(2-phosphonoethyl)-3,4;9,10-perylenediimide
—— tert-butyl [2-(1-hydroxy-1-methylethyl)-3-methylimidazo[1,2-a]pyridin-6-yl]carbamate 869109-46-6 C16H23N3O3
tert-butyl [2-(1-hydroxy-1-methylethyl)-3-methylimidazo[1,2-a]pyridin-6-yl]carbamate