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—— Piperidine-3-carboxylic acid {2-[5-(1-{2-hydroxy-3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-phenylsulfanyl]-ethyl}-amide 1049095-32-0 C34H48F3N7O5S2
Piperidine-3-carboxylic acid {2-[5-(1-{2-hydroxy-3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-phenylsulfanyl]-ethyl}-amide
—— (2R)-2-({4-[(2,3-dihydro[1,4]oxathiino [2,3-c]pyridin-7-ylmethyl)amino]-1-piperidinyl}methyl)-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione 1075235-07-2 C23H26N6O3S
(2R)-2-({4-[(2,3-dihydro[1,4]oxathiino [2,3-c]pyridin-7-ylmethyl)amino]-1-piperidinyl}methyl)-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione
—— 6-(5-bromo-2-hydroxyphenyl)-2-(2-chlorophenyl)pyrimidin-4(3H)-one 1076188-12-9 C16H10BrClN2O2
6-(5-bromo-2-hydroxyphenyl)-2-(2-chlorophenyl)pyrimidin-4(3H)-one
—— 3-(3,5-difluorophenyl)-1-ethylpyrrolidin-3-ol 1092572-17-2 C12H15F2NO
3-(3,5-difluorophenyl)-1-ethylpyrrolidin-3-ol
—— (E)-3-amino-1-(3-(2,6-dichlorostyryl)phenyl)propan-1-ol 1075174-91-2 C17H17Cl2NO
(E)-3-amino-1-(3-(2,6-dichlorostyryl)phenyl)propan-1-ol
—— (2S)-6-amino-1-[4-[4-[4-[2-[4-(2-hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-[4-(2-hydroxypropyl)triazol-1-yl]hexan-1-one 1005839-24-6 C37H59N15O7
(2S)-6-amino-1-[4-[4-[4-[2-[4-(2-hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-[4-(2-hydroxypropyl)triazol-1-yl]hexan-1-one
—— 3-[1-[(2S)-6-amino-1-[4-[4-[4-[(2S,3S)-2-[4-(2-carboxyethyl)triazol-1-yl]-3-methylpentanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-1-oxohexan-2-yl]triazol-4-yl]propanoic acid 1005839-16-6 C42H65N15O9
3-[1-[(2S)-6-amino-1-[4-[4-[4-[(2S,3S)-2-[4-(2-carboxyethyl)triazol-1-yl]-3-methylpentanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-1-oxohexan-2-yl]triazol-4-yl]propanoic acid
—— N-carbamimidoyl-2-(4-chlorophenyl)-5-methyl-1,3-oxazole-4-carboxamide 1144520-81-9 C12H11ClN4O2
N-carbamimidoyl-2-(4-chlorophenyl)-5-methyl-1,3-oxazole-4-carboxamide
—— N-carbamimidoyl-5-methyl-2-(3-methylphenyl)-1,3-oxazole-4-carboxamide 1144520-68-2 C13H14N4O2
N-carbamimidoyl-5-methyl-2-(3-methylphenyl)-1,3-oxazole-4-carboxamide
—— 3-[1-[(2S,3S)-1-[4-[4-[4-[(2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-methylbutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methyl-1-oxopentan-2-yl]triazol-4-yl]propanoic acid 1005839-11-1 C40H62N14O8
3-[1-[(2S,3S)-1-[4-[4-[4-[(2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-methylbutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methyl-1-oxopentan-2-yl]triazol-4-yl]propanoic acid
—— 2-[3-[1-[2-[4-[4-[4-[2-[4-(2-Hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine 1005839-29-1 C34H53N17O6
2-[3-[1-[2-[4-[4-[4-[2-[4-(2-Hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine
—— (3S,5S)-5-(methoxymethoxymethyl)-3-phenylmethoxyoxolan-2-one 1056441-24-7 C14H18O5
(3S,5S)-5-(methoxymethoxymethyl)-3-phenylmethoxyoxolan-2-one
—— (2S)-1-[4-[4-[4-[2-[4-(4-aminobutyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-(4-hydroxyphenyl)propan-1-one 1005839-06-4 C41H59N15O7
(2S)-1-[4-[4-[4-[2-[4-(4-aminobutyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-(4-hydroxyphenyl)propan-1-one
—— 3-[1-[(2S,3S)-1-[4-[4-[4-[(2S)-6-amino-2-[4-(2-hydroxypropyl)triazol-1-yl]hexanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methyl-1-oxopentan-2-yl]triazol-4-yl]propanoic acid 1005839-13-3 C42H67N15O8
3-[1-[(2S,3S)-1-[4-[4-[4-[(2S)-6-amino-2-[4-(2-hydroxypropyl)triazol-1-yl]hexanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methyl-1-oxopentan-2-yl]triazol-4-yl]propanoic acid
—— 2-[[5-[3-(Carboxymethylcarbamoyl)-4-hydroxyphenyl]seleninyloxyseleninyl-2-hydroxybenzoyl]amino]acetic acid 1071918-62-1 C18H16N2O11Se2
2-[[5-[3-(Carboxymethylcarbamoyl)-4-hydroxyphenyl]seleninyloxyseleninyl-2-hydroxybenzoyl]amino]acetic acid
—— (E)-6-(t-butyldimethylsilyl)oxy-2-hexen-4-ynal 1056417-36-7 C12H20O2Si
(E)-6-(t-butyldimethylsilyl)oxy-2-hexen-4-ynal
—— N-carbamimidoyl-2-(3-fluorophenyl)-5-methyl-1,3-oxazole-4-carboxamide 1144520-74-0 C12H11FN4O2
N-carbamimidoyl-2-(3-fluorophenyl)-5-methyl-1,3-oxazole-4-carboxamide
—— (2S,3S)-2-[4-(4-aminobutyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylpentan-1-one 1005838-83-4 C39H63N15O6
(2S,3S)-2-[4-(4-aminobutyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylpentan-1-one
—— 2-(cyclobutylamino)-4-(3-ethyl-6,6-dimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)-6-fluorobenzamide 1073969-30-8 C22H27FN4O2
2-(cyclobutylamino)-4-(3-ethyl-6,6-dimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)-6-fluorobenzamide
—— 2-[4-(2-Hydroxyethyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]ethanone 1005839-22-4 C33H50N14O7
2-[4-(2-Hydroxyethyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]ethanone
—— 2-(1-(2-(isobutylamino)ethyl)-1H-pyrazol-4-ylamino)-4-(3,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzamide 1073969-16-0 C26H35N7O2
2-(1-(2-(isobutylamino)ethyl)-1H-pyrazol-4-ylamino)-4-(3,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzamide
—— 4-Acetamido-2-[3-(trifluoromethyl)anilino]benzoic acid 1019854-44-4 C16H13F3N2O3
4-Acetamido-2-[3-(trifluoromethyl)anilino]benzoic acid
—— 5-Methanesulfonyl-1-(3-morpholin-4-yl-propyl)-3-[3-(2-piperidin-1-yl-ethylsulfanyl)-4-trifluoromethyl-phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine 1049094-68-9 C28H40F3N5O3S2
5-Methanesulfonyl-1-(3-morpholin-4-yl-propyl)-3-[3-(2-piperidin-1-yl-ethylsulfanyl)-4-trifluoromethyl-phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine
—— (3S,4aS,8aS)-2-[(2R)-3-[(4-aminophenyl)sulfonyl-(1,3-benzodioxol-5-ylmethyl)amino]-2-hydroxypropyl]-N-tert-butyl-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-3-carboxamide 1083099-03-9 C31H44N4O6S
(3S,4aS,8aS)-2-[(2R)-3-[(4-aminophenyl)sulfonyl-(1,3-benzodioxol-5-ylmethyl)amino]-2-hydroxypropyl]-N-tert-butyl-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-3-carboxamide
—— 4-Thiazolemethanamine, 2-methyl-N-(tetrahydro-4,4-dimethyl-2H-thiopyran-3-yl)- 1534482-04-6 C12H20N2S2
4-Thiazolemethanamine, 2-methyl-N-(tetrahydro-4,4-dimethyl-2H-thiopyran-3-yl)-
—— 1-((6-chloro-5-(trifluoromethyl)pyridin-2-yl)amino)-3-((3,3-dimethylbutoxy)methyl)-4-methyl-1H-pyrrole-2,5-dione 1076235-04-5 C18H21ClF3N3O3
1-((6-chloro-5-(trifluoromethyl)pyridin-2-yl)amino)-3-((3,3-dimethylbutoxy)methyl)-4-methyl-1H-pyrrole-2,5-dione
—— tert-butyl N-(2-methyl-3-oxopropyl)-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 1075218-31-3 C14H25NO5
tert-butyl N-(2-methyl-3-oxopropyl)-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— 5-chloro-2-(pyrazol-3-yl)benzoxazole 1073468-74-2 C10H6ClN3O
5-chloro-2-(pyrazol-3-yl)benzoxazole
—— 2-(1-(4-chlorophenyl)cyclopropyl)-3-hydroxy-8-methyl-6-(trifluoromethyl)quinoline-4-carboxylic acid 1067187-16-9 C21H15ClF3NO3
2-(1-(4-chlorophenyl)cyclopropyl)-3-hydroxy-8-methyl-6-(trifluoromethyl)quinoline-4-carboxylic acid
—— (3S,4aS,8aS)-2-[(2R)-3-[(3-aminophenyl)methyl-(4-methoxyphenyl)sulfonylamino]-2-hydroxypropyl]-N-tert-butyl-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-3-carboxamide 1083098-97-8 C31H46N4O5S
(3S,4aS,8aS)-2-[(2R)-3-[(3-aminophenyl)methyl-(4-methoxyphenyl)sulfonylamino]-2-hydroxypropyl]-N-tert-butyl-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline-3-carboxamide
—— 3-(5-{6-[2-(N-acetyl-N-methylamino)ethoxy]-2,3-difluorobenzyloxy}-2-fluorophenyl)-5-carboxythieno[3,4-d]pyrimidine-2,4(1H,3H)-dione 1075700-58-1 C25H20F3N3O7S
3-(5-{6-[2-(N-acetyl-N-methylamino)ethoxy]-2,3-difluorobenzyloxy}-2-fluorophenyl)-5-carboxythieno[3,4-d]pyrimidine-2,4(1H,3H)-dione
—— 5-carboxy-3-(2-fluoro-5-{2,3-difluoro-6-[2-(oxazolidin-2-one-3-yl)ethoxy]benzyloxy}phenyl)thieno[3,4-d]pyrimidine-2,4(1H,3H)-dione 1075700-73-0 C25H18F3N3O8S
5-carboxy-3-(2-fluoro-5-{2,3-difluoro-6-[2-(oxazolidin-2-one-3-yl)ethoxy]benzyloxy}phenyl)thieno[3,4-d]pyrimidine-2,4(1H,3H)-dione
—— (2R,3R,4R)-2-benzyloxycarbonylamino-2-benzyloxymethyl-6-(tertbutyldimethylsilanyloxy)-3,4-dihydroxyhexanoic acid 8-phenylmenthyl ester 1059067-72-9 C44H63NO8Si
(2R,3R,4R)-2-benzyloxycarbonylamino-2-benzyloxymethyl-6-(tertbutyldimethylsilanyloxy)-3,4-dihydroxyhexanoic acid 8-phenylmenthyl ester
—— 3-[4-(4-hydroxyphenyl)-2-thienyl]phenol 1078733-89-7 C16H12O2S
3-[4-(4-hydroxyphenyl)-2-thienyl]phenol
—— (2S,3S)-1-[(2S,6R)-6-allyl-3,6-dihydro-2H-pyran-2-yl]-4-(benzyloxy)-methylbutan-2-ol 1088779-94-5 C20H28O3
(2S,3S)-1-[(2S,6R)-6-allyl-3,6-dihydro-2H-pyran-2-yl]-4-(benzyloxy)-methylbutan-2-ol
—— 2-(cyclopent-3-enylamino)-6-fluoro-4-(3,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzamide 1073969-27-3 C22H25FN4O2
2-(cyclopent-3-enylamino)-6-fluoro-4-(3,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzamide
—— (2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxy-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]butan-1-one 1005839-33-7 C37H59N15O7
(2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxy-1-[4-[4-[4-[2-[4-(2-hydroxypropyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]butan-1-one
—— 3-(2-methylphenyl)-1-(3-(1-naphthyloxy)propyl)-1H-indole-2-carboxylic acid 1072899-65-0 C29H25NO3
3-(2-methylphenyl)-1-(3-(1-naphthyloxy)propyl)-1H-indole-2-carboxylic acid
—— (3S,5Z,7E)-3-(methoxy-methoxy)-9-(tetrahydro-2H-pyran-2-yloxy)-5,7-nonadienal 1071075-98-3 C16H26O5
(3S,5Z,7E)-3-(methoxy-methoxy)-9-(tetrahydro-2H-pyran-2-yloxy)-5,7-nonadienal
—— (2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-1-[4-[4-[4-[(2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-(4-hydroxyphenyl)propanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylbutan-1-one 1005839-49-5 C42H60N14O8
(2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-1-[4-[4-[4-[(2S)-2-[4-(2-hydroxyethyl)triazol-1-yl]-3-(4-hydroxyphenyl)propanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylbutan-1-one
—— 5-(4-chloro-phenyl)-2-trifluoromethyl-furan-3-carboxylic acid [5-chloro-2-(1H-tetrazol-5-ylmethoxy)-phenyl]-amide 1083418-41-0 C20H12Cl2F3N5O3
5-(4-chloro-phenyl)-2-trifluoromethyl-furan-3-carboxylic acid [5-chloro-2-(1H-tetrazol-5-ylmethoxy)-phenyl]-amide
—— 2-methylspiro[oxaol-4(5H),2'-tricyclo[3.3.1.1.(3,7)]decane] 1059192-56-1 C13H19NO
2-methylspiro[oxaol-4(5H),2'-tricyclo[3.3.1.1.(3,7)]decane]
—— 2,3-dimethoxy-N-[2-[6-(oxiran-2-yl)-1,3-benzodioxol-5-yl]ethyl]benzamide 1075231-78-5 C20H21NO6
2,3-dimethoxy-N-[2-[6-(oxiran-2-yl)-1,3-benzodioxol-5-yl]ethyl]benzamide
—— (2S,3S)-2-[4-(4-aminobutyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylpentan-1-one 1005838-82-3 C38H61N15O6
(2S,3S)-2-[4-(4-aminobutyl)triazol-1-yl]-1-[4-[4-[4-[2-[4-(2-hydroxyethyl)triazol-1-yl]acetyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-3-methylpentan-1-one
—— 3-[4-(1,3,3-trimethyl-6-aza-bicyclo[3.2.1]octane-6-carbonyl)-indol-1-yl]-propionic acid 1057653-91-4 C22H28N2O3
3-[4-(1,3,3-trimethyl-6-aza-bicyclo[3.2.1]octane-6-carbonyl)-indol-1-yl]-propionic acid
—— (4-[6-(2-ethoxy-phenyl)-pyrimidin-4-ylamino]-phenyl)-methanesulfonamide 1073589-70-4 C19H20N4O3S
(4-[6-(2-ethoxy-phenyl)-pyrimidin-4-ylamino]-phenyl)-methanesulfonamide
—— 3-[3-(5-methyl-1H-imidazol-1-yl)propyl]-2-thioxo-2,3,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-4(1H)-one 1072441-38-3 C17H20N4OS2
3-[3-(5-methyl-1H-imidazol-1-yl)propyl]-2-thioxo-2,3,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-4(1H)-one
—— (2R)-2-[(4-{[(8-fluoro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}-1-piperidinyl)methyl]-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione 1075236-91-7 C24H26FN5O4
(2R)-2-[(4-{[(8-fluoro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}-1-piperidinyl)methyl]-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione
—— Ethyl 4-[[2-methoxy-6-(4-methoxyphenyl)pyridin-3-yl]methyl]piperazine-1-carboxylate 1061733-45-6 C21H27N3O4
Ethyl 4-[[2-methoxy-6-(4-methoxyphenyl)pyridin-3-yl]methyl]piperazine-1-carboxylate
—— 6-benzyl-2,3-dihydro-3-(3-(5-methyl-1H-imidazol-1-yl)propyl)-2-thioxothieno[2,3-d]pyrimidin-4(1H)-one 1072441-48-5 C20H20N4OS2
6-benzyl-2,3-dihydro-3-(3-(5-methyl-1H-imidazol-1-yl)propyl)-2-thioxothieno[2,3-d]pyrimidin-4(1H)-one