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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-2-[2,4-dioxo-1-(1,4,6-trimethyl-1H-indol-3-ylmethyl)-1,4-dihydro-2H-quinazolin-3-yl]-pentanoic acid 1115352-99-2 C25H27N3O4
(R)-2-[2,4-dioxo-1-(1,4,6-trimethyl-1H-indol-3-ylmethyl)-1,4-dihydro-2H-quinazolin-3-yl]-pentanoic acid
—— 4-[6-({[3-(2,6-dichlorophenyl)-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1-benzothien-2-yl]benzoic acid 1097776-63-0 C28H21Cl2NO4S
4-[6-({[3-(2,6-dichlorophenyl)-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1-benzothien-2-yl]benzoic acid
—— 4-[[4-(2,4-Dichlorophenyl)-3-phenylpiperazin-1-yl]methyl]benzonitrile 1097636-39-9 C24H21Cl2N3
4-[[4-(2,4-Dichlorophenyl)-3-phenylpiperazin-1-yl]methyl]benzonitrile
—— 1-(2,3-dimethoxybenzyl)-2-(4-sulfamoylphenylamino)-1H-benzo[d]imidazole-5-carboxamide 1092829-80-5 C23H23N5O5S
1-(2,3-dimethoxybenzyl)-2-(4-sulfamoylphenylamino)-1H-benzo[d]imidazole-5-carboxamide
—— 3-fluoro-8-methyl-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine 1097265-39-8 C25H25FN4OS
3-fluoro-8-methyl-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine
—— (4S)-4-(2-amino-4-oxo-6-phenoxyquinazolin-3-yl)-N,4-dicyclohexyl-N-methylbutanamide 1100393-40-5 C31H40N4O3
(4S)-4-(2-amino-4-oxo-6-phenoxyquinazolin-3-yl)-N,4-dicyclohexyl-N-methylbutanamide
—— 2-[3-[1-[2-[4-[4-[4-[(2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxybutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine 1005839-57-5 C38H62N18O6
2-[3-[1-[2-[4-[4-[4-[(2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxybutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine
—— 3-{[5-({[3-{[(2,6-dichlorophenyl)amino]methyl}-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1H-indol-1-yl]methyl}benzoic acid 1097776-40-3 C30H27Cl2N3O4
3-{[5-({[3-{[(2,6-dichlorophenyl)amino]methyl}-5-(1-methylethyl)-4-isoxazolyl]methyl}oxy)-1H-indol-1-yl]methyl}benzoic acid
—— (2R,3R)-2-(benzenesulfonyl)-2-benzyl-3-(2-oxopropyl)cyclohexan-1-one 1134193-15-9 C22H24O4S
(2R,3R)-2-(benzenesulfonyl)-2-benzyl-3-(2-oxopropyl)cyclohexan-1-one
—— 2-[[4-Amino-5-(2-furanyl)-4H-1,2,4-triazol-3-yl]thio]-N-(2-methylcyclohexyl)propanamide 1186646-12-7 C16H23N5O2S
2-[[4-Amino-5-(2-furanyl)-4H-1,2,4-triazol-3-yl]thio]-N-(2-methylcyclohexyl)propanamide
—— 4-(acetylamino)-1-[(6-bromo-1,3-benzodioxol-5-yl)methyl]-5-methyl-1H-pyrazole-3-carboxamide 1102467-12-8 C15H15BrN4O4
4-(acetylamino)-1-[(6-bromo-1,3-benzodioxol-5-yl)methyl]-5-methyl-1H-pyrazole-3-carboxamide
—— (2S)-6-amino-1-[4-[4-[4-[(2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxybutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-(4-butyltriazol-1-yl)hexan-1-one 1005839-54-2 C42H70N16O6
(2S)-6-amino-1-[4-[4-[4-[(2S,3R)-2-[4-(4-aminobutyl)triazol-1-yl]-3-hydroxybutanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-(4-butyltriazol-1-yl)hexan-1-one
—— (2S)-2-(3-{[6-methoxy-3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridine-1-yl]methyl}phenoxy)propanoic acid 1071811-78-3 C27H26N2O6
(2S)-2-(3-{[6-methoxy-3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridine-1-yl]methyl}phenoxy)propanoic acid
—— 2-[3-[1-[2-[4-[4-[4-[(2S)-6-amino-2-(4-butyltriazol-1-yl)hexanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine 1005839-78-0 C40H66N18O5
2-[3-[1-[2-[4-[4-[4-[(2S)-6-amino-2-(4-butyltriazol-1-yl)hexanoyl]piperazin-1-yl]-6-[2-[2-(2-prop-2-ynoxyethoxy)ethoxy]ethylamino]-1,3,5-triazin-2-yl]piperazin-1-yl]-2-oxoethyl]triazol-4-yl]propyl]guanidine
—— (Z)-3-(4-{2-[4-(acetyl-methyl-amino)-phenyl]-ethoxy}-3-butoxy-phenyl)-2-ethoxy-acrylic acid 1092167-45-7 C26H33NO6
(Z)-3-(4-{2-[4-(acetyl-methyl-amino)-phenyl]-ethoxy}-3-butoxy-phenyl)-2-ethoxy-acrylic acid
—— ethyl 6-{4-[(benzylsulfonyl)carbamoyl]piperidin-1-yl}-5-cyano-2-(2-methoxyethyl)nicotinate 1039068-10-4 C25H30N4O6S
ethyl 6-{4-[(benzylsulfonyl)carbamoyl]piperidin-1-yl}-5-cyano-2-(2-methoxyethyl)nicotinate
—— (Z)-3-(3-butoxy-4-{2-[4-(methanesulfonyl-methyl-amino)-phenyl]-ethoxy}-phenyl)-2-ethoxy-acrylic acid 1092167-33-3 C25H33NO7S
(Z)-3-(3-butoxy-4-{2-[4-(methanesulfonyl-methyl-amino)-phenyl]-ethoxy}-phenyl)-2-ethoxy-acrylic acid
—— ethyl 2-[(benzyloxy)methyl]-6-{4-[(benzylsulfonyl)carbamoyl]piperidin-1-yl}-5-cyanonicotinate 1039068-00-2 C30H32N4O6S
ethyl 2-[(benzyloxy)methyl]-6-{4-[(benzylsulfonyl)carbamoyl]piperidin-1-yl}-5-cyanonicotinate
—— 2-[(2R)-2-(4-chlorophenyl)piperazin-1-yl]-5-(2-methoxyethoxy)benzonitrile 1097206-36-4 C20H22ClN3O2
2-[(2R)-2-(4-chlorophenyl)piperazin-1-yl]-5-(2-methoxyethoxy)benzonitrile
—— 5-[(2R)-1-[(3R)-4-(2-chloro-4-cyanophenyl)-3-(4-chlorophenyl)piperazin-1-yl]-2-hydroxypropan-2-yl]-N-cyclopropylpyrazine-2-carboxamide 1097078-32-4 C28H28Cl2N6O2
5-[(2R)-1-[(3R)-4-(2-chloro-4-cyanophenyl)-3-(4-chlorophenyl)piperazin-1-yl]-2-hydroxypropan-2-yl]-N-cyclopropylpyrazine-2-carboxamide
—— 5-amino-1-(3-isopropylamino-propyl)-2-(naphthalen-2-ylsulfanyl)-1H-imidazole-4-carboxamide 1102466-77-2 C20H25N5OS
5-amino-1-(3-isopropylamino-propyl)-2-(naphthalen-2-ylsulfanyl)-1H-imidazole-4-carboxamide
—— N-hydroxy-2-isobutyl-N'-(2-{pentanoyl[2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethyl]amino}ethyl)malonamide 1043607-90-4 C28H37N7O4
N-hydroxy-2-isobutyl-N'-(2-{pentanoyl[2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethyl]amino}ethyl)malonamide
—— N,N'-bis(2,3-dihydroxybenzoyl)-N''-hexanoyltren 1120366-33-7 C26H36N4O7
N,N'-bis(2,3-dihydroxybenzoyl)-N''-hexanoyltren
—— 2-fluoro-4-[(5,6,6a,7,8,9-hexahydro-4H-2-phenalenyl)carboxamido]benzoic acid 1117680-81-5 C21H20FNO3
2-fluoro-4-[(5,6,6a,7,8,9-hexahydro-4H-2-phenalenyl)carboxamido]benzoic acid
—— methyl (2S)-1-[(2S)-2-(1,3-dioxoisoindol-2-yl)-3-phenylpropanoyl]-2,3-dihydropyrrole-2-carboxylate 114486-37-2 C23H20N2O5
methyl (2S)-1-[(2S)-2-(1,3-dioxoisoindol-2-yl)-3-phenylpropanoyl]-2,3-dihydropyrrole-2-carboxylate
—— 1-(3-((2,6-dimethyl-4-(((2S)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-2-yl)methoxy)benzoyl)amino)-4-(trifluoromethyl)phenyl)cyclopropanecarboxylic acid 1116623-84-7 C30H29F3N2O5
1-(3-((2,6-dimethyl-4-(((2S)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-2-yl)methoxy)benzoyl)amino)-4-(trifluoromethyl)phenyl)cyclopropanecarboxylic acid
—— 4-[(2R)-4-benzyl-2-phenylpiperazin-1-yl]-3-chlorobenzonitrile 1097636-06-0 C24H22ClN3
4-[(2R)-4-benzyl-2-phenylpiperazin-1-yl]-3-chlorobenzonitrile
—— 5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyran-4-ylmethyl)piperazin-1-yl]carbonyl}-N-[5-fluoro-2-(methoxymethyl)pyrimidin-4-yl]-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine 1046789-95-0 C26H39FN8O3
5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyran-4-ylmethyl)piperazin-1-yl]carbonyl}-N-[5-fluoro-2-(methoxymethyl)pyrimidin-4-yl]-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine
—— (S)-2-hydroxy-3-methyl-N-[(S)-1-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-azepin-3-ylcarbamoyl)-ethyl]-butyramide 1116395-10-8 C21H27N3O4
(S)-2-hydroxy-3-methyl-N-[(S)-1-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-azepin-3-ylcarbamoyl)-ethyl]-butyramide
—— 3-chloro-7-(methyloxy)-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl} methyl)imidazo[1,2-a]pyridine 1097265-45-6 C25H25ClN4O2S
3-chloro-7-(methyloxy)-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl} methyl)imidazo[1,2-a]pyridine
—— 4-(4-chlorophenyl)-3-[4-[4-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione 156525-77-8 C22H14Cl2N6S2
4-(4-chlorophenyl)-3-[4-[4-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]phenyl]-1H-1,2,4-triazole-5-thione
—— (1S,5S,8R,10S)-10-bromo-5-([tert-butyldimethylsilyl]oxymethyl)-2-oxa-4-azatricyclo[6.2.1.0(4,8)]undecan-3-one 1107601-94-4 C16H28BrNO3Si
(1S,5S,8R,10S)-10-bromo-5-([tert-butyldimethylsilyl]oxymethyl)-2-oxa-4-azatricyclo[6.2.1.0(4,8)]undecan-3-one
—— 3-(6-fluoro-1H-benzimidazol-2-yl)-5-[4-(2-pyrazol-1-ylethoxy)phenyl]pyrazin-2-amine 1100094-66-3 C22H18FN7O
3-(6-fluoro-1H-benzimidazol-2-yl)-5-[4-(2-pyrazol-1-ylethoxy)phenyl]pyrazin-2-amine
—— 3-chloro-6-fluoro-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine 1097265-41-2 C24H22ClFN4OS
3-chloro-6-fluoro-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine
—— N,N'-bis(2-((2-(7-chloro-6-oxo-6H-dibenzo[cd,g]indazol-2-yl)ethyl)methylamino)ethyl)malonamide 1096533-22-0 C41H38Cl2N8O4
N,N'-bis(2-((2-(7-chloro-6-oxo-6H-dibenzo[cd,g]indazol-2-yl)ethyl)methylamino)ethyl)malonamide
—— 8-fluoro-2-[((2S)-1-{[5-(4-fluorophenyl)-2-methyl-1,3-thiazol-4-yl]carbonyl}-2-piperidinyl)methyl]imidazo[1,2-a]pyridine 1097265-57-0 C24H22F2N4OS
8-fluoro-2-[((2S)-1-{[5-(4-fluorophenyl)-2-methyl-1,3-thiazol-4-yl]carbonyl}-2-piperidinyl)methyl]imidazo[1,2-a]pyridine
—— Bis[2-[2-(6-chloro-8-oxo-14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-14-yl)ethyl-methylamino]ethyl] propanedioate 1033203-79-0 C41H36Cl2N6O6
Bis[2-[2-(6-chloro-8-oxo-14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-14-yl)ethyl-methylamino]ethyl] propanedioate
—— ethyl 6-(3-{[(4-chloro-2-fluorobenzyl)sulfonyl]carbamoyl}azetidin-1-yl)-5-cyano-2-methoxynicotinate 1039067-95-2 C21H20ClFN4O6S
ethyl 6-(3-{[(4-chloro-2-fluorobenzyl)sulfonyl]carbamoyl}azetidin-1-yl)-5-cyano-2-methoxynicotinate
—— 6-[2-(4-cyclobutylpiperazin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydropyrazolo[1,5-a]pyrido[3,4-d]pyrimidine 1094706-11-2 C19H26N6O
6-[2-(4-cyclobutylpiperazin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydropyrazolo[1,5-a]pyrido[3,4-d]pyrimidine
—— allyl (2,3,4,6-tetra-O-benzyl-α-D-glucopyranosyl)-(1→3)-4-O-benzyl-2-O-levulinoyl-α-L-rhamnopyranoside 1091625-34-1 C55H62O12
allyl (2,3,4,6-tetra-O-benzyl-α-D-glucopyranosyl)-(1→3)-4-O-benzyl-2-O-levulinoyl-α-L-rhamnopyranoside
—— (Z)-2-ethoxy-3-{4-[2-(4-methanesulfonyloxy-phenyl)-ethoxy]-3-methoxy-phenyl}-acrylic acid 1092167-21-9 C21H24O8S
(Z)-2-ethoxy-3-{4-[2-(4-methanesulfonyloxy-phenyl)-ethoxy]-3-methoxy-phenyl}-acrylic acid
—— 3-(1H-benzimidazol-2-yl)-5-[3-[3-(piperidin-1-yl)propoxy]phenyl]pyrazin-2-amine 1100094-65-2 C25H28N6O
3-(1H-benzimidazol-2-yl)-5-[3-[3-(piperidin-1-yl)propoxy]phenyl]pyrazin-2-amine
—— 5-amino-2-(7-chloro-benzothiazol-2-ylsulfanyl)-1-(3-isopropylamino-propyl)-1H-imidazole-4-carboxamide 1102466-71-6 C17H21ClN6OS2
5-amino-2-(7-chloro-benzothiazol-2-ylsulfanyl)-1-(3-isopropylamino-propyl)-1H-imidazole-4-carboxamide
—— (R)-1-(3,4-difluorobenzyl)-2-(6-(3,3-difluoropiperidine-1-carbonyl)pyridin-3-yl)-5-ethyl-7-isopropyl-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one 1314080-44-8 C30H31F4N7O2
(R)-1-(3,4-difluorobenzyl)-2-(6-(3,3-difluoropiperidine-1-carbonyl)pyridin-3-yl)-5-ethyl-7-isopropyl-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one
—— (Z)-3-{3-butoxy-4-[2-(4-methanesulfonylamino-phenyl)-ethoxy]-phenyl}-2-ethoxy-acrylic acid 1092167-36-6 C24H31NO7S
(Z)-3-{3-butoxy-4-[2-(4-methanesulfonylamino-phenyl)-ethoxy]-phenyl}-2-ethoxy-acrylic acid
—— (R)-dibenzyl 2-(6-(2-ethoxy-2-oxoethoxy)naphthalene-2-sulfonamido)pentanedioate 1092117-64-0 C33H33NO9S
(R)-dibenzyl 2-(6-(2-ethoxy-2-oxoethoxy)naphthalene-2-sulfonamido)pentanedioate
—— (3E)-5-hydroxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one 1087343-95-0 C22H17N3O2S
(3E)-5-hydroxy-3-[[2-methyl-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylidene]-1H-indol-2-one
—— propyl α-D-glucopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-rhamnopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→3)-2-acetamido-2-deoxy-β-D-glucopyranoside 1091625-90-9 C35H61NO23
propyl α-D-glucopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-rhamnopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→3)-2-acetamido-2-deoxy-β-D-glucopyranoside
—— 8-ethenyl-6-fluoro-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine 1097265-49-0 C26H25FN4OS
8-ethenyl-6-fluoro-2-({(2S)-1-[(2-methyl-5-phenyl-1,3-thiazol-4-yl)carbonyl]-2-piperidinyl}methyl)imidazo[1,2-a]pyridine
—— methyl (13S,15R)-13-[(1R,9R,10S,11R,12R,19R)-11-acetyloxy-10-[(cyclobutanecarbonylamino)methyl]-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2,4,6,13-tetraen-4-yl]-17-ethyl-1,11-diazatetracyclo[13.3.1.04,12.05,10]nonadeca-4(12),5,7,9,16-pentaene-13-carboxylate 1043910-80-0 C50H63N5O7
methyl (13S,15R)-13-[(1R,9R,10S,11R,12R,19R)-11-acetyloxy-10-[(cyclobutanecarbonylamino)methyl]-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2,4,6,13-tetraen-4-yl]-17-ethyl-1,11-diazatetracyclo[13.3.1.04,12.05,10]nonadeca-4(12),5,7,9,16-pentaene-13-carboxylate