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—— Methyl 2-[2-(4-chlorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19ClN4O5S
Methyl 2-[2-(4-chlorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-prop-2-enoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H24N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-prop-2-enoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H26N4O7S
Methyl 2-[2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-[3-(3-methylbutoxy)phenyl]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H30N4O6S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-[3-(3-methylbutoxy)phenyl]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(3-ethoxy-4-prop-2-enoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H28N4O7S
Methyl 2-[2-(3-ethoxy-4-prop-2-enoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-bromophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19BrN4O5S
Methyl 2-[2-(4-bromophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-hydroxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H20N4O6S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-hydroxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H30N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H26N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxy-4-pentoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N4O7S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxy-4-pentoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(3-ethoxy-4-pentoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H34N4O7S
Methyl 2-[2-(3-ethoxy-4-pentoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxy-4-phenylmethoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H28N4O7S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxy-4-phenylmethoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl N-[4-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylcarbamoylamino]phenyl]-N-methylcarbamate —— C19H21N3O5
methyl N-[4-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylcarbamoylamino]phenyl]-N-methylcarbamate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H19N5O5S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 3-[[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]amino]-4-methylbenzoate —— C20H21ClN2O4
methyl 3-[[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]amino]-4-methylbenzoate
—— morpholin-4-yl-[(3R)-1-[3-(4-nitrophenoxy)propyl]piperidin-3-yl]methanone —— C19H27N3O5
morpholin-4-yl-[(3R)-1-[3-(4-nitrophenoxy)propyl]piperidin-3-yl]methanone
—— methyl 2-ethyl-4-methyl-5-[[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate —— C22H27N3O4
methyl 2-ethyl-4-methyl-5-[[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate
—— Methyl 2,5-dihydroxy-3-(4-methylphenyl)sulfonylbenzoate —— C15H14O6S
Methyl 2,5-dihydroxy-3-(4-methylphenyl)sulfonylbenzoate
—— methyl 4-[1-[2-(diethylamino)ethyl]-4-hydroxy-3-(5-methyl-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-2-yl]benzoate —— C28H30N2O6
methyl 4-[1-[2-(diethylamino)ethyl]-4-hydroxy-3-(5-methyl-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-2-yl]benzoate
—— Methyl 4-[(3,6,6-trimethyl-4-oxo-5,7-dihydro-1-benzofuran-2-carbonyl)amino]benzoate —— C20H21NO5
Methyl 4-[(3,6,6-trimethyl-4-oxo-5,7-dihydro-1-benzofuran-2-carbonyl)amino]benzoate
—— methyl 4-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]carbamoyl-methylamino]methyl]benzoate —— C18H23N3O3S
methyl 4-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]carbamoyl-methylamino]methyl]benzoate
—— Methyl 2-[(3,6,6-trimethyl-4-oxo-5,6,7-trihydrobenzo[2,1-d]furan-2-yl)carbonyl amino]benzoate —— C20H21NO5
Methyl 2-[(3,6,6-trimethyl-4-oxo-5,6,7-trihydrobenzo[2,1-d]furan-2-yl)carbonyl amino]benzoate
—— methyl 4-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]carbamoyl-methylamino]methyl]benzoate —— C18H23N3O3S
methyl 4-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]carbamoyl-methylamino]methyl]benzoate
—— Methyl 4-[(7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl)methylsulfonylamino]benzoate —— C18H23NO5S
Methyl 4-[(7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl)methylsulfonylamino]benzoate
—— methyl 2-ethyl-4-methyl-5-[[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate —— C22H27N3O4
methyl 2-ethyl-4-methyl-5-[[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate
—— methyl 2,4-dimethyl-5-[[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate —— C21H25N3O4
methyl 2,4-dimethyl-5-[[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]carbamoyl]-1H-pyrrole-3-carboxylate
—— Methyl 2-[(3,6,6-trimethyl-4-oxo-5,7-dihydro-1-benzofuran-2-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H25NO5S
Methyl 2-[(3,6,6-trimethyl-4-oxo-5,7-dihydro-1-benzofuran-2-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 4-[4-hydroxy-3-(5-methyl-1-benzofuran-2-carbonyl)-1-(2-morpholin-4-ylethyl)-5-oxo-2H-pyrrol-2-yl]benzoate —— C28H28N2O7
methyl 4-[4-hydroxy-3-(5-methyl-1-benzofuran-2-carbonyl)-1-(2-morpholin-4-ylethyl)-5-oxo-2H-pyrrol-2-yl]benzoate
—— Methyl 4-[[5-(dibenzylsulfamoyl)pyridin-2-yl]amino]benzoate —— C27H25N3O4S
Methyl 4-[[5-(dibenzylsulfamoyl)pyridin-2-yl]amino]benzoate
—— methyl 4-[1-[3-(diethylamino)propyl]-4-hydroxy-3-(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)-5-oxo-2H-pyrrol-2-yl]benzoate —— C30H33N3O5S
methyl 4-[1-[3-(diethylamino)propyl]-4-hydroxy-3-(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)-5-oxo-2H-pyrrol-2-yl]benzoate
—— methyl 4-[4-hydroxy-3-(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)-1-(3-morpholin-4-ylpropyl)-5-oxo-2H-pyrrol-2-yl]benzoate —— C30H31N3O6S
methyl 4-[4-hydroxy-3-(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)-1-(3-morpholin-4-ylpropyl)-5-oxo-2H-pyrrol-2-yl]benzoate
—— Methyl 2-[[5-(dibenzylsulfamoyl)pyridin-2-yl]amino]benzoate —— C27H25N3O4S
Methyl 2-[[5-(dibenzylsulfamoyl)pyridin-2-yl]amino]benzoate
—— Methyl 4-[[5-[ethyl(phenyl)sulfamoyl]pyridin-2-yl]amino]benzoate —— C21H21N3O4S
Methyl 4-[[5-[ethyl(phenyl)sulfamoyl]pyridin-2-yl]amino]benzoate
—— methyl 3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidine-1-carbonyl]benzoate —— C20H24N4O3
methyl 3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidine-1-carbonyl]benzoate
—— Methyl 4-[[5-(4-methylpiperazin-1-yl)sulfonylpyridin-2-yl]amino]benzoate —— C18H22N4O4S
Methyl 4-[[5-(4-methylpiperazin-1-yl)sulfonylpyridin-2-yl]amino]benzoate
—— methyl 4-[[1-[2-(diethylamino)ethyl]-2-(4-ethoxy-3-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O7
methyl 4-[[1-[2-(diethylamino)ethyl]-2-(4-ethoxy-3-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[2-(3-ethoxyphenyl)-1-(2-morpholin-4-ylethyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H33N3O7
methyl 4-[[2-(3-ethoxyphenyl)-1-(2-morpholin-4-ylethyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-(3-propoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O6
methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-(3-propoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(diethylamino)ethyl]-4,5-dioxo-2-(4-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H35N3O6
methyl 4-[[1-[2-(diethylamino)ethyl]-4,5-dioxo-2-(4-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-pyridin-2-ylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C22H26N4O5
methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-pyridin-2-ylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[2-(2,4-dimethoxyphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H31N3O7
methyl 4-[[2-(2,4-dimethoxyphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-(3-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H31N3O6
methyl 4-[[1-[2-(dimethylamino)ethyl]-4,5-dioxo-2-(3-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(diethylamino)ethyl]-4,5-dioxo-2-(4-propoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O6
methyl 4-[[1-[2-(diethylamino)ethyl]-4,5-dioxo-2-(4-propoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[hydroxy-[1-(2-morpholin-4-ylethyl)-4,5-dioxo-2-(3-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H33N3O7
methyl 4-[hydroxy-[1-(2-morpholin-4-ylethyl)-4,5-dioxo-2-(3-prop-2-enoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[2-(2,4-dimethoxyphenyl)-1-(2-morpholin-4-ylethyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H33N3O8
methyl 4-[[2-(2,4-dimethoxyphenyl)-1-(2-morpholin-4-ylethyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[2-(2,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O7
methyl 4-[[2-(2,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(3-propoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H37N3O7
methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(3-propoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[3-(diethylamino)propyl]-2-(3-ethoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O6
methyl 4-[[1-[3-(diethylamino)propyl]-2-(3-ethoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[[1-[2-(diethylamino)ethyl]-2-(3-ethoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H35N3O6
methyl 4-[[1-[2-(diethylamino)ethyl]-2-(3-ethoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(4-propoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H37N3O7
methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(4-propoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate