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—— Methyl 4-[1-[5-[(2,4-dichlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H21Cl2N5O5S2
Methyl 4-[1-[5-[(2,4-dichlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-methyl-5-[[(4-phenoxypiperidine-1-carbonyl)amino]methyl]furan-3-carboxylate —— C20H24N2O5
methyl 2-methyl-5-[[(4-phenoxypiperidine-1-carbonyl)amino]methyl]furan-3-carboxylate
—— methyl N-[[(Z)-2-phenylethenyl]sulfonylamino]carbamate —— C10H12N2O4S
methyl N-[[(Z)-2-phenylethenyl]sulfonylamino]carbamate
—— Methyl 4-[1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H22ClN5O5S2
Methyl 4-[1-[5-[(2-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 5-[[2-[[(E)-3-(furan-2-yl)prop-2-enoyl]amino]acetyl]amino]-1H-indazole-3-carboxylate —— C18H16N4O5
methyl 5-[[2-[[(E)-3-(furan-2-yl)prop-2-enoyl]amino]acetyl]amino]-1H-indazole-3-carboxylate
—— Methyl 4-[1-[5-[(4-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H22ClN5O5S2
Methyl 4-[1-[5-[(4-chlorophenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 4-[[(1S)-5-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoylamino]benzoate —— C18H17FN2O3
methyl 4-[[(1S)-5-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoylamino]benzoate
—— methyl 5-[[(2R)-2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-1H-indazole-3-carboxylate —— C15H16N6O3S
methyl 5-[[(2R)-2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[(2S)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1H-indazole-3-carboxylate —— C18H16FN3O5S
methyl 5-[[(2S)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[2-[(2S)-oxolan-2-yl]acetyl]amino]-1H-indazole-3-carboxylate —— C15H17N3O4
methyl 5-[[2-[(2S)-oxolan-2-yl]acetyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[1-(3-chlorophenyl)-5-methyltriazole-4-carbonyl]amino]-1H-indazole-3-carboxylate —— C19H15ClN6O3
methyl 5-[[1-(3-chlorophenyl)-5-methyltriazole-4-carbonyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[(2S)-3-methyl-2-(3-methylbutanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate —— C19H26N4O4
methyl 5-[[(2S)-3-methyl-2-(3-methylbutanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate
—— Methyl 4-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-1-[5-[(4-methylphenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-4,5-dioxopyrrolidin-2-yl]benzoate —— C31H25N5O5S2
Methyl 4-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-1-[5-[(4-methylphenyl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 4-[[(1R)-5-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoylamino]benzoate —— C18H17FN2O3
methyl 4-[[(1R)-5-fluoro-2,3-dihydro-1H-inden-1-yl]carbamoylamino]benzoate
—— methyl 5-[[2-[(4-cyanophenyl)methylsulfanyl]acetyl]amino]-1H-indazole-3-carboxylate —— C19H16N4O3S
methyl 5-[[2-[(4-cyanophenyl)methylsulfanyl]acetyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[(2R)-4-methylsulfanyl-2-(propanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate —— C17H22N4O4S
methyl 5-[[(2R)-4-methylsulfanyl-2-(propanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[5-[(2-cyanophenoxy)methyl]furan-2-carbonyl]amino]-1H-indazole-3-carboxylate —— C22H16N4O5
methyl 5-[[5-[(2-cyanophenoxy)methyl]furan-2-carbonyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[2-[[(Z)-3-(furan-2-yl)prop-2-enoyl]amino]acetyl]amino]-1H-indazole-3-carboxylate —— C18H16N4O5
methyl 5-[[2-[[(Z)-3-(furan-2-yl)prop-2-enoyl]amino]acetyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[(2R)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1H-indazole-3-carboxylate —— C18H16FN3O5S
methyl 5-[[(2R)-2-(4-fluorophenyl)sulfonylpropanoyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[(5-chloro-2-pyrrolidin-1-ylpyrimidine-4-carbonyl)amino]-1H-indazole-3-carboxylate —— C18H17ClN6O3
methyl 5-[(5-chloro-2-pyrrolidin-1-ylpyrimidine-4-carbonyl)amino]-1H-indazole-3-carboxylate
—— methyl 5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]butanoylamino]-1H-indazole-3-carboxylate —— C18H24N4O5
methyl 5-[4-[(2-methylpropan-2-yl)oxycarbonylamino]butanoylamino]-1H-indazole-3-carboxylate
—— methyl 5-[[(2R)-3-methyl-2-(3-methylbutanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate —— C19H26N4O4
methyl 5-[[(2R)-3-methyl-2-(3-methylbutanoylamino)butanoyl]amino]-1H-indazole-3-carboxylate
—— methyl 5-[[1-(diethylcarbamoyl)piperidine-4-carbonyl]amino]-1H-indazole-3-carboxylate —— C20H27N5O4
methyl 5-[[1-(diethylcarbamoyl)piperidine-4-carbonyl]amino]-1H-indazole-3-carboxylate
—— methyl 3-[(E)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]furan-2-carboxylate —— C10H7NO4S2
methyl 3-[(E)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]furan-2-carboxylate
—— methyl N-[3-[[(2R)-2-(3-fluorophenyl)pyrrolidine-1-carbonyl]amino]phenyl]carbamate —— C19H20FN3O3
methyl N-[3-[[(2R)-2-(3-fluorophenyl)pyrrolidine-1-carbonyl]amino]phenyl]carbamate
—— Methyl 2-[2-(2-fluorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19FN4O5S
Methyl 2-[2-(2-fluorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 4-[1-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C27H22N4O6S
Methyl 4-[1-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— Methyl 4-[1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H23N5O5S2
Methyl 4-[1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H26N4O8S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-chloro-5-[4-(3-propyl-1,2,4-oxadiazol-5-yl)butanoylamino]benzoate —— C17H20ClN3O4
methyl 2-chloro-5-[4-(3-propyl-1,2,4-oxadiazol-5-yl)butanoylamino]benzoate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-propoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H26N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-propoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H22N4O7S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-hydroxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H20N4O6S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-hydroxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-ethoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H24N4O6S
Methyl 2-[2-(4-ethoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-propoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H26N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-propoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H22N4O6S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(3-chlorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19ClN4O5S
Methyl 2-[2-(3-chlorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-fluorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19FN4O5S
Methyl 2-[2-(4-fluorophenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 4-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxo-1-(1,3-thiazol-2-yl)pyrrolidin-2-yl]benzoate —— C24H18N4O5S
Methyl 4-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxo-1-(1,3-thiazol-2-yl)pyrrolidin-2-yl]benzoate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19N5O7S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-hexoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N4O6S
Methyl 2-[2-(4-hexoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H24N4O7S
Methyl 2-[2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H26N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-tert-butylphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H28N4O5S
Methyl 2-[2-(4-tert-butylphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H20N4O5S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(4-butoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H28N4O6S
Methyl 2-[2-(4-butoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H30N4O6S
Methyl 2-[4-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2,3-dioxo-5-(4-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H22N4O6S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H19N5O7S
Methyl 2-[3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-2-(3-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-(3-bromo-4-hydroxy-5-methoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H21BrN4O7S
Methyl 2-[2-(3-bromo-4-hydroxy-5-methoxyphenyl)-3-[hydroxy-(2-methylimidazo[1,2-a]pyridin-3-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate