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—— Ethyl 1-[3-[4-[(3-benzyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazol-3-yl]phenyl]sulfonylpiperidine-4-carboxylate —— C34H32N4O5S3
Ethyl 1-[3-[4-[(3-benzyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazol-3-yl]phenyl]sulfonylpiperidine-4-carboxylate
—— Ethyl 1-[3-[4-[2-cyano-3-(furan-2-ylmethylamino)-3-oxoprop-1-enyl]-1-phenylpyrazol-3-yl]phenyl]sulfonylpiperidine-4-carboxylate —— C32H31N5O6S
Ethyl 1-[3-[4-[2-cyano-3-(furan-2-ylmethylamino)-3-oxoprop-1-enyl]-1-phenylpyrazol-3-yl]phenyl]sulfonylpiperidine-4-carboxylate
—— Ethyl 4-[[3-[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate —— C39H37N5O8S
Ethyl 4-[[3-[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate
—— (E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[(2S)-2-methyl-2H-chromen-3-yl]prop-2-enamide —— C17H19NO4S
(E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[(2S)-2-methyl-2H-chromen-3-yl]prop-2-enamide
—— Ethyl 1-[4-oxo-5-[[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C31H33N5O5S2
Ethyl 1-[4-oxo-5-[[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— Ethyl 1-[5-[[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C33H37N5O5S2
Ethyl 1-[5-[[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]benzoate —— C43H43N5O8S
Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]benzoate
—— Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoyl]amino]benzoate —— C41H39N5O8S
Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoyl]amino]benzoate
—— Ethyl 2-cyano-3-[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enoate —— C27H28N4O4S
Ethyl 2-cyano-3-[3-[3-(4-methylpiperidin-1-yl)sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enoate
—— ethyl (4S)-2-amino-6-(hydroxymethyl)-4-(4-methoxyphenyl)-8-oxo-4H-pyrano[3,2-b]pyran-3-carboxylate —— C19H19NO7
ethyl (4S)-2-amino-6-(hydroxymethyl)-4-(4-methoxyphenyl)-8-oxo-4H-pyrano[3,2-b]pyran-3-carboxylate
—— Ethyl 2-cyano-3-[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoate —— C25H24N4O4S
Ethyl 2-cyano-3-[1-phenyl-3-(3-pyrrolidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoate
—— Ethyl 1-[5-[[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C29H31N5O5S2
Ethyl 1-[5-[[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— Ethyl 1-[5-[[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C31H35N5O5S2
Ethyl 1-[5-[[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— ethyl (7S)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C18H23N5O4
ethyl (7S)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— Ethyl 4-[[3-[3-(3-chloro-4-ethoxyphenyl)-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate —— C39H35ClN4O7
Ethyl 4-[[3-[3-(3-chloro-4-ethoxyphenyl)-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate
—— Ethyl 3-[3-(3-chloro-4-propoxyphenyl)-1-phenylpyrazol-4-yl]-2-cyanoprop-2-enoate —— C24H22ClN3O3
Ethyl 3-[3-(3-chloro-4-propoxyphenyl)-1-phenylpyrazol-4-yl]-2-cyanoprop-2-enoate
—— ethyl (7S)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H24N4O4
ethyl (7S)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 6-[2-[(1R)-4,4-dimethyl-1-oxo-2,3-dihydrothiochromen-6-yl]ethynyl]pyridine-3-carboxylate —— C21H21NO3S
ethyl 6-[2-[(1R)-4,4-dimethyl-1-oxo-2,3-dihydrothiochromen-6-yl]ethynyl]pyridine-3-carboxylate
—— (E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[(2R)-2-methyl-2H-chromen-3-yl]prop-2-enamide —— C17H19NO4S
(E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[(2R)-2-methyl-2H-chromen-3-yl]prop-2-enamide
—— Ethyl 1-[4-oxo-5-[[1-phenyl-3-(3-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C32H35N5O5S2
Ethyl 1-[4-oxo-5-[[1-phenyl-3-(3-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[1-phenyl-3-(3-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoyl]amino]benzoate —— C42H41N5O8S
Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[1-phenyl-3-(3-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]prop-2-enoyl]amino]benzoate
—— ethyl (7R)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H24N4O4
ethyl (7R)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C17H21N5O4
ethyl (7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-1-[(3S,3aR,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one —— C27H24N2O2
(E)-1-[(3S,3aR,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one
—— ethyl (1S)-7-fluoro-4-oxo-2,3-dihydro-1H-naphthalene-1-carboxylate —— C13H13FO3
ethyl (1S)-7-fluoro-4-oxo-2,3-dihydro-1H-naphthalene-1-carboxylate
—— ethyl (2S)-2-(4-tert-butylphenyl)-2-cyanoacetate —— C15H19NO2
ethyl (2S)-2-(4-tert-butylphenyl)-2-cyanoacetate
—— (E)-N-[(2S)-2-(3,4-dimethoxyphenyl)-2-hydroxyethyl]-3-phenylprop-2-enamide —— C19H21NO4
(E)-N-[(2S)-2-(3,4-dimethoxyphenyl)-2-hydroxyethyl]-3-phenylprop-2-enamide
—— (E)-4-[(3S)-5-(4-bromophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]-4-oxobut-2-enoic acid —— C19H15BrN2O4
(E)-4-[(3S)-5-(4-bromophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]-4-oxobut-2-enoic acid
—— ethyl (7R)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C18H21BrN4O4
ethyl (7R)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-4-(3,4-dichlorobenzylidene)-5-methyl-2-phenyl-2,4-dihydro-3H-pyrazol-3-one —— C17H12Cl2N2O
(E)-4-(3,4-dichlorobenzylidene)-5-methyl-2-phenyl-2,4-dihydro-3H-pyrazol-3-one
—— ethyl (2R)-2-(4-tert-butylphenyl)-2-cyanoacetate —— C15H19NO2
ethyl (2R)-2-(4-tert-butylphenyl)-2-cyanoacetate
—— ethyl (7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C18H21BrN4O4
ethyl (7S)-7-(3-bromo-5-ethoxy-4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— [(E)-[(2S)-2-(2,4-dinitrophenyl)cyclohexylidene]amino] 4-tert-butylbenzoate —— C23H25N3O6
[(E)-[(2S)-2-(2,4-dinitrophenyl)cyclohexylidene]amino] 4-tert-butylbenzoate
—— ethyl (7R)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C18H23N5O4
ethyl (7R)-7-(3,4-diethoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— Ethyl 1-[5-[[3-(3-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C31H33N5O6S2
Ethyl 1-[5-[[3-(3-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— (E)-4-[2-[(1R,2R)-2-methyl-2-phenylcyclopropanecarbonyl]hydrazinyl]-4-oxobut-2-enoic acid —— C15H16N2O4
(E)-4-[2-[(1R,2R)-2-methyl-2-phenylcyclopropanecarbonyl]hydrazinyl]-4-oxobut-2-enoic acid
—— (E)-1-[(3R,3aR,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one —— C27H24N2O2
(E)-1-[(3R,3aR,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one
—— [(E)-1-[(1R,2S)-2-(4-methoxyphenyl)cyclopropyl]ethylideneamino] cyclopropanecarboxylate —— C16H19NO3
[(E)-1-[(1R,2S)-2-(4-methoxyphenyl)cyclopropyl]ethylideneamino] cyclopropanecarboxylate
—— Ethyl 5-hydroxy-2-(1-methylbenzotriazol-1-ium-2-yl)-5-phenylpenta-2,4-dienoate —— C20H20N3O3+
Ethyl 5-hydroxy-2-(1-methylbenzotriazol-1-ium-2-yl)-5-phenylpenta-2,4-dienoate
—— Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[3-(3-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]benzoate —— C41H39N5O9S
Ethyl 4-[[2-[(4-ethoxycarbonylphenyl)carbamoyl]-3-[3-(3-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]benzoate
—— Ethyl 1-[5-[[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate —— C31H33ClN4O4S
Ethyl 1-[5-[[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-4-oxo-1,3-thiazol-2-yl]piperidine-4-carboxylate
—— [(E)-[[(1S,2S)-2-(1,3-benzodioxol-5-yl)cyclopropyl]-(4-methoxyphenyl)methylidene]amino] 4-methoxybenzoate —— C26H23NO6
[(E)-[[(1S,2S)-2-(1,3-benzodioxol-5-yl)cyclopropyl]-(4-methoxyphenyl)methylidene]amino] 4-methoxybenzoate
—— Ethyl 3-[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]-2-cyanoprop-2-enoate —— C25H24ClN3O3
Ethyl 3-[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]-2-cyanoprop-2-enoate
—— ethyl (2Z,5R)-7-methyl-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H30N2O4S
ethyl (2Z,5R)-7-methyl-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E,4E)-4-[cyano-[(2S,3S,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethylidene]hex-2-enedioic acid —— C14H17NO10
(E,4E)-4-[cyano-[(2S,3S,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethylidene]hex-2-enedioic acid
—— ethyl (2Z,5S)-7-methyl-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H30N2O4S
ethyl (2Z,5S)-7-methyl-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-7-methyl-2-[[(2S)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H30N2O4S
ethyl (2Z,5S)-7-methyl-2-[[(2S)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H28N4O4
ethyl (7S)-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-1-[(3R,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one —— C27H24N2O2
(E)-1-[(3R,3aS,7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-3-(furan-2-yl)prop-2-en-1-one
—— Ethyl 4-[[3-[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate —— C41H39ClN4O7
Ethyl 4-[[3-[3-(4-butoxy-3-chlorophenyl)-1-phenylpyrazol-4-yl]-2-[(4-ethoxycarbonylphenyl)carbamoyl]prop-2-enoyl]amino]benzoate