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—— Ethyl 3-[(4-cyano-3-methylsulfanyl-1,2-thiazol-5-yl)hydrazinylidene]-4,4-difluorobutanoate —— C11H12F2N4O2S2
Ethyl 3-[(4-cyano-3-methylsulfanyl-1,2-thiazol-5-yl)hydrazinylidene]-4,4-difluorobutanoate
—— ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C21H27ClN6O3S2
ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 5-(diethylcarbamoyl)-4-methyl-2-({[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}amino)thiophene-3-carboxylate —— C19H23F3N4O4S
ethyl 5-(diethylcarbamoyl)-4-methyl-2-({[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}amino)thiophene-3-carboxylate
—— ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C25H28N6O3S2
ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 2-{[(4-bromo-1-methyl-1H-pyrazol-5-yl)carbonyl]amino}-4,5-dimethylthiophene-3-carboxylate —— C14H16BrN3O3S
ethyl 2-{[(4-bromo-1-methyl-1H-pyrazol-5-yl)carbonyl]amino}-4,5-dimethylthiophene-3-carboxylate
—— ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H28ClFN6O3S2
ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[2-[1-[2-[4-[(2R)-butan-2-yl]phenoxy]ethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C30H33N3O2
(E)-N-[2-[1-[2-[4-[(2R)-butan-2-yl]phenoxy]ethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— Ethyl 4-{3-[(4-chlorophenoxy)methyl]-2,4,6-trimethylphenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate —— C31H36ClNO4
Ethyl 4-{3-[(4-chlorophenoxy)methyl]-2,4,6-trimethylphenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
—— (E)-N-[2-[1-[2-[4-[(2S)-butan-2-yl]phenoxy]ethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C30H33N3O2
(E)-N-[2-[1-[2-[4-[(2S)-butan-2-yl]phenoxy]ethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— Ethyl 4-{5-bromo-2-[(3-fluorobenzyl)oxy]phenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate —— C28H29BrFNO4
Ethyl 4-{5-bromo-2-[(3-fluorobenzyl)oxy]phenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
—— Ethyl 5-methyl-7-(1,1,2,2,2-pentafluoroethyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate —— C12H10F5N3O2
Ethyl 5-methyl-7-(1,1,2,2,2-pentafluoroethyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
—— (E)-N-[2-[1-[2-[bis[(2S)-butan-2-yl]amino]-2-oxoethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C28H36N4O2
(E)-N-[2-[1-[2-[bis[(2S)-butan-2-yl]amino]-2-oxoethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— ethyl 2-[({[5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C24H24ClFN6O3S2
ethyl 2-[({[5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C25H28N6O3S2
ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-N-[2-[1-[(2R)-2-methylbutyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C23H27N3O
(E)-N-[2-[1-[(2R)-2-methylbutyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— Ethyl 7-[chloro(difluoro)methyl]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxylate —— C11H10ClF2N3O2
Ethyl 7-[chloro(difluoro)methyl]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxylate
—— Ethyl 4-{5-bromo-2-[(4-chlorobenzyl)oxy]phenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate —— C28H29BrClNO4
Ethyl 4-{5-bromo-2-[(4-chlorobenzyl)oxy]phenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
—— ethyl 6-ethyl-2-[({[5-(1-methyl-1H-pyrazol-3-yl)-4-(tetrahydrofuran-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H34N6O4S2
ethyl 6-ethyl-2-[({[5-(1-methyl-1H-pyrazol-3-yl)-4-(tetrahydrofuran-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 1-methyl-3-{[3-(morpholinosulfonyl)anilino]carbonyl}-1H-pyrazole-5-carboxylate —— C18H22N4O6S
ethyl 1-methyl-3-{[3-(morpholinosulfonyl)anilino]carbonyl}-1H-pyrazole-5-carboxylate
—— ethyl 3-[(2,3-dichloroanilino)carbonyl]-1-methyl-1H-pyrazole-5-carboxylate —— C14H13Cl2N3O3
ethyl 3-[(2,3-dichloroanilino)carbonyl]-1-methyl-1H-pyrazole-5-carboxylate
—— ethyl 2-[({[4-butyl-5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C21H27ClN6O3S2
ethyl 2-[({[4-butyl-5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— Ethyl 2-[3-[3-[(4-bromophenoxy)methyl]-4-methoxyphenyl]prop-2-enoylamino]-4,5-dimethylthiophene-3-carboxylate —— C26H26BrNO5S
Ethyl 2-[3-[3-[(4-bromophenoxy)methyl]-4-methoxyphenyl]prop-2-enoylamino]-4,5-dimethylthiophene-3-carboxylate
—— Ethyl 2-[(2-{[4-butyl-5-(4-chloro-1-methyl-1H-pyrazol-3-YL)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H33ClN6O3S2
Ethyl 2-[(2-{[4-butyl-5-(4-chloro-1-methyl-1H-pyrazol-3-YL)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[({[5-(4-bromo-1,5-dimethyl-1H-pyrazol-3-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H30BrFN6O3S2
ethyl 2-[({[5-(4-bromo-1,5-dimethyl-1H-pyrazol-3-yl)-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 7-(difluoromethyl)-5-(naphthalen-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate —— C20H15F2N3O2
Ethyl 7-(difluoromethyl)-5-(naphthalen-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
—— ethyl 4-carbamoyl-5-({[5-cyclopropyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]acetyl}amino)-3-methylthiophene-2-carboxylate —— C18H19F3N4O4S
ethyl 4-carbamoyl-5-({[5-cyclopropyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]acetyl}amino)-3-methylthiophene-2-carboxylate
—— ethyl 7-(difluoromethyl)-5-(4-ethylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 678190-43-7 C18H17F2N3O2
ethyl 7-(difluoromethyl)-5-(4-ethylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
—— Ethyl 3-({4-[(1-adamantylamino)sulfonyl]anilino}carbonyl)-1-methyl-1H-pyrazole-5-carboxylate —— C24H30N4O5S
Ethyl 3-({4-[(1-adamantylamino)sulfonyl]anilino}carbonyl)-1-methyl-1H-pyrazole-5-carboxylate
—— Ethyl 4-carbamoyl-3-methyl-5-{[(2,3,5,6-tetrafluorophenoxy)acetyl]amino}thiophene-2-carboxylate —— C17H14F4N2O5S
Ethyl 4-carbamoyl-3-methyl-5-{[(2,3,5,6-tetrafluorophenoxy)acetyl]amino}thiophene-2-carboxylate
—— Ethyl 2-[(2-{[5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-YL)-4-(2-furylmethyl)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H31ClN6O4S2
Ethyl 2-[(2-{[5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-YL)-4-(2-furylmethyl)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[(2-{[4-benzyl-5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-YL)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-4,5-dimethyl-3-thiophenecarboxylate —— C25H27ClN6O3S2
Ethyl 2-[(2-{[4-benzyl-5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-YL)-4H-1,2,4-triazol-3-YL]sulfanyl}acetyl)amino]-4,5-dimethyl-3-thiophenecarboxylate
—— ethyl 1-methyl-3-{[2-(propan-2-yl)phenyl]carbamoyl}-1H-pyrazole-5-carboxylate —— C17H21N3O3
ethyl 1-methyl-3-{[2-(propan-2-yl)phenyl]carbamoyl}-1H-pyrazole-5-carboxylate
—— ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H34N6O3S2
ethyl 2-[({[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 5-(diethylcarbamoyl)-2-{[(2,5-difluorophenyl)carbonyl]amino}-4-methylthiophene-3-carboxylate —— C20H22F2N2O4S
Ethyl 5-(diethylcarbamoyl)-2-{[(2,5-difluorophenyl)carbonyl]amino}-4-methylthiophene-3-carboxylate
—— ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(furan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H29ClN6O4S2
ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(furan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]acetate —— C8H9F3N2O3
ethyl 2-[3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]acetate
—— Ethyl 4-{5-bromo-2-[(4-chlorobenzyl)oxy]phenyl}-2-methyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate —— C26H25BrClNO4
Ethyl 4-{5-bromo-2-[(4-chlorobenzyl)oxy]phenyl}-2-methyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
—— Ethyl 13-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C27H21ClN2O5S
Ethyl 13-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— (E)-N-[2-[1-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C26H30N4O2
(E)-N-[2-[1-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— ethyl 2-[({[5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C20H25ClN6O3S2
ethyl 2-[({[5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-N-[2-[1-[3-[4-[(2R)-butan-2-yl]phenoxy]propyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C31H35N3O2
(E)-N-[2-[1-[3-[4-[(2R)-butan-2-yl]phenoxy]propyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— (E)-N-[2-[1-[[4-[(2R)-butan-2-yl]phenyl]methyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide —— C29H31N3O
(E)-N-[2-[1-[[4-[(2R)-butan-2-yl]phenyl]methyl]benzimidazol-2-yl]ethyl]-3-phenylprop-2-enamide
—— Ethyl 1-methyl-3-{[(5-nitro-2-pyridyl)amino]carbonyl}-1H-pyrazole-5-carboxylate —— C13H13N5O5
Ethyl 1-methyl-3-{[(5-nitro-2-pyridyl)amino]carbonyl}-1H-pyrazole-5-carboxylate
—— Ethyl 4-{3-[(4-chloro-2-methylphenoxy)methyl]-2,5-dimethylphenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate —— C31H36ClNO4
Ethyl 4-{3-[(4-chloro-2-methylphenoxy)methyl]-2,5-dimethylphenyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
—— ethyl 2-[2-[2-[[(2R)-oxolane-2-carbonyl]amino]ethyl]benzimidazol-1-yl]acetate —— C18H23N3O4
ethyl 2-[2-[2-[[(2R)-oxolane-2-carbonyl]amino]ethyl]benzimidazol-1-yl]acetate
—— ethyl 2-[2-[2-[[(2S)-oxolane-2-carbonyl]amino]ethyl]benzimidazol-1-yl]acetate —— C18H23N3O4
ethyl 2-[2-[2-[[(2S)-oxolane-2-carbonyl]amino]ethyl]benzimidazol-1-yl]acetate
—— ethyl 4,5-dimethyl-2-({[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}amino)thiophene-3-carboxylate —— C15H16F3N3O3S
ethyl 4,5-dimethyl-2-({[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl}amino)thiophene-3-carboxylate
—— Ethyl 4-carbamoyl-5-{[(4-fluorophenoxy)acetyl]amino}-3-methylthiophene-2-carboxylate —— C17H17FN2O5S
Ethyl 4-carbamoyl-5-{[(4-fluorophenoxy)acetyl]amino}-3-methylthiophene-2-carboxylate
—— ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-5-yl)-4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C24H25ClN6O3S2
ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-5-yl)-4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(furan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate —— C22H23ClN6O4S2
ethyl 2-[({[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-(furan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]-4,5-dimethylthiophene-3-carboxylate