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—— ethyl 6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H23F2N5O3S
ethyl 6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 5-amino-3-[[3-(4-butan-2-ylphenyl)-4-oxoquinazolin-2-yl]sulfanylmethyl]-4-cyanothiophene-2-carboxylate —— C27H26N4O3S2
Ethyl 5-amino-3-[[3-(4-butan-2-ylphenyl)-4-oxoquinazolin-2-yl]sulfanylmethyl]-4-cyanothiophene-2-carboxylate
—— Ethyl 4-[2-(4-chloro-3-morpholin-4-ylsulfonylanilino)-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C23H25ClN4O6S3
Ethyl 4-[2-(4-chloro-3-morpholin-4-ylsulfonylanilino)-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 1-[5-amino-6-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-4-carboxylate —— C18H29N5O2
ethyl 1-[5-amino-6-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 5-[2-[2,4-dichloro-5-[(4-ethoxyphenyl)sulfamoyl]benzoyl]oxypropanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C27H28Cl2N2O8S
ethyl 5-[2-[2,4-dichloro-5-[(4-ethoxyphenyl)sulfamoyl]benzoyl]oxypropanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[[5-amino-6-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]amino]benzoate —— C19H25N5O2
ethyl 4-[[5-amino-6-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]amino]benzoate
—— ethyl (3R)-1-[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate —— C18H29N5O2
ethyl (3R)-1-[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate —— C18H29N5O2
ethyl (3S)-1-[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl 4-[[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]amino]benzoate —— C19H25N5O2
ethyl 4-[[5-amino-6-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]amino]benzoate
—— ethyl (3R)-1-[5-amino-6-(4-benzylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C23H32N6O2
ethyl (3R)-1-[5-amino-6-(4-benzylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-benzhydrylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C29H36N6O2
ethyl (3R)-1-[5-amino-6-(4-benzhydrylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(4-benzylpiperidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C24H33N5O2
ethyl (3S)-1-[5-amino-6-(4-benzylpiperidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C17H28N6O2
ethyl (3S)-1-[5-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate —— C23H32N6O3
ethyl (3R)-1-[5-amino-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C22H30N6O2
ethyl (3S)-1-[5-amino-6-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-benzylpiperidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C24H33N5O2
ethyl (3R)-1-[5-amino-6-(4-benzylpiperidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C17H28N6O2
ethyl (3R)-1-[5-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(2-phenylethylamino)pyrimidin-4-yl]piperidine-3-carboxylate —— C20H27N5O2
ethyl (3R)-1-[5-amino-6-(2-phenylethylamino)pyrimidin-4-yl]piperidine-3-carboxylate
—— Ethyl 2-[5-[(3,5-dimethoxyphenyl)methylidene]-4-oxo-3-[2-oxo-2-(thiophen-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C23H24N2O6S2
Ethyl 2-[5-[(3,5-dimethoxyphenyl)methylidene]-4-oxo-3-[2-oxo-2-(thiophen-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (3S)-1-[5-amino-6-(4-ethylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C18H30N6O2
ethyl (3S)-1-[5-amino-6-(4-ethylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(azepan-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C18H29N5O2
ethyl (3R)-1-[5-amino-6-(azepan-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-(5-amino-6-piperidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate —— C17H27N5O2
ethyl (3R)-1-(5-amino-6-piperidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(diethylamino)pyrimidin-4-yl]piperidine-3-carboxylate —— C16H27N5O2
ethyl (3S)-1-[5-amino-6-(diethylamino)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C22H30N6O2
ethyl (3R)-1-[5-amino-6-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-propan-2-ylphenoxy)pyrimidin-4-yl]piperidine-3-carboxylate —— C21H28N4O3
ethyl (3R)-1-[5-amino-6-(4-propan-2-ylphenoxy)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate —— C23H32N6O3
ethyl (3S)-1-[5-amino-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-(5-amino-6-piperidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate —— C17H27N5O2
ethyl (3S)-1-(5-amino-6-piperidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(2-phenylethylamino)pyrimidin-4-yl]piperidine-3-carboxylate —— C20H27N5O2
ethyl (3S)-1-[5-amino-6-(2-phenylethylamino)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-(5-amino-6-morpholin-4-ylpyrimidin-4-yl)piperidine-3-carboxylate —— C16H25N5O3
ethyl (3R)-1-(5-amino-6-morpholin-4-ylpyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(diethylamino)pyrimidin-4-yl]piperidine-3-carboxylate —— C16H27N5O2
ethyl (3R)-1-[5-amino-6-(diethylamino)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(4-propan-2-ylphenoxy)pyrimidin-4-yl]piperidine-3-carboxylate —— C21H28N4O3
ethyl (3S)-1-[5-amino-6-(4-propan-2-ylphenoxy)pyrimidin-4-yl]piperidine-3-carboxylate
—— Ethyl 6-methyl-2-[2-[methyl-[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]propanoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H28F3N3O4S
Ethyl 6-methyl-2-[2-[methyl-[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]propanoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (3S)-1-(5,6-diaminopyrimidin-4-yl)piperidine-3-carboxylate —— C12H19N5O2
ethyl (3S)-1-(5,6-diaminopyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3R)-1-(5-amino-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate —— C16H25N5O2
ethyl (3R)-1-(5-amino-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(dimethylamino)pyrimidin-4-yl]piperidine-3-carboxylate —— C14H23N5O2
ethyl (3S)-1-[5-amino-6-(dimethylamino)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-amino-6-(4-chlorophenyl)sulfanylpyrimidin-4-yl]piperidine-3-carboxylate —— C18H21ClN4O2S
ethyl (3S)-1-[5-amino-6-(4-chlorophenyl)sulfanylpyrimidin-4-yl]piperidine-3-carboxylate
—— Ethyl 2-[2-[3-[(4-butylphenyl)sulfamoyl]benzoyl]oxypropanoylamino]-4-phenylthiophene-3-carboxylate —— C33H34N2O7S2
Ethyl 2-[2-[3-[(4-butylphenyl)sulfamoyl]benzoyl]oxypropanoylamino]-4-phenylthiophene-3-carboxylate
—— ethyl (3S)-1-(5-amino-6-morpholin-4-ylpyrimidin-4-yl)piperidine-3-carboxylate —— C16H25N5O3
ethyl (3S)-1-(5-amino-6-morpholin-4-ylpyrimidin-4-yl)piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-ethylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate —— C18H30N6O2
ethyl (3R)-1-[5-amino-6-(4-ethylpiperazin-1-yl)pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-amino-6-(4-chlorophenyl)sulfanylpyrimidin-4-yl]piperidine-3-carboxylate —— C18H21ClN4O2S
ethyl (3R)-1-[5-amino-6-(4-chlorophenyl)sulfanylpyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl 6-[[2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]phenyl]acetyl]oxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H27N3O7S
ethyl 6-[[2-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]phenyl]acetyl]oxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-4-[(3R)-3-methylpyrrolidin-1-yl]-4-oxobut-2-enoic acid —— C9H13NO3
(E)-4-[(3R)-3-methylpyrrolidin-1-yl]-4-oxobut-2-enoic acid
—— (E)-4-[(3S)-3-methylpyrrolidin-1-yl]-4-oxobut-2-enoic acid —— C9H13NO3
(E)-4-[(3S)-3-methylpyrrolidin-1-yl]-4-oxobut-2-enoic acid
—— ethyl 6-[3-[(4-chlorophenyl)sulfonylamino]propanoyloxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H22ClN3O7S2
ethyl 6-[3-[(4-chlorophenyl)sulfonylamino]propanoyloxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-oxo-4-thiophen-2-yl-6-[[5-[3-(trifluoromethyl)phenyl]furan-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H19F3N2O6S
ethyl 2-oxo-4-thiophen-2-yl-6-[[5-[3-(trifluoromethyl)phenyl]furan-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[2-(3,4-dihydro-2H-quinolin-1-yl)propanoylamino]-5-phenylthiophene-3-carboxylate —— C25H26N2O3S
ethyl 2-[2-(3,4-dihydro-2H-quinolin-1-yl)propanoylamino]-5-phenylthiophene-3-carboxylate
—— Ethyl 3-(4-chlorophenyl)-6-[4-[(4-methoxycarbonylphenyl)methoxy]phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C29H27ClN2O6
Ethyl 3-(4-chlorophenyl)-6-[4-[(4-methoxycarbonylphenyl)methoxy]phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 2,4-dimethyl-5-[2-[2-[2-(4-methylphenyl)ethenylsulfonylamino]acetyl]oxypropanoyl]-1H-pyrrole-3-carboxylate —— C23H28N2O7S
ethyl 2,4-dimethyl-5-[2-[2-[2-(4-methylphenyl)ethenylsulfonylamino]acetyl]oxypropanoyl]-1H-pyrrole-3-carboxylate
—— ethyl 6-[[4-methyl-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H16F3N5O3S2
ethyl 6-[[4-methyl-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2,4-dimethyl-5-[2-[3-[[3-(trifluoromethyl)phenyl]sulfonylamino]propanoyloxy]propanoyl]-1H-pyrrole-3-carboxylate —— C22H25F3N2O7S
ethyl 2,4-dimethyl-5-[2-[3-[[3-(trifluoromethyl)phenyl]sulfonylamino]propanoyloxy]propanoyl]-1H-pyrrole-3-carboxylate