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—— ethyl 2-[[5-amino-4-[(2R)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C22H26N6O4S2
ethyl 2-[[5-amino-4-[(2R)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 4-acetyl-2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-5-methylfuran-3-carboxylate —— C19H25N5O7S
ethyl 4-acetyl-2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C24H25N5O4S
ethyl 2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[[5-amino-4-[(2S)-1-[4-(dimethylsulfamoyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H26N6O5S2
ethyl 2-[[5-amino-4-[(2S)-1-[4-(dimethylsulfamoyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— Ethyl 4-[3-(4-carbamoylpiperidin-1-ium-1-yl)-2,5-dioxopyrrolidin-1-yl]benzoate —— C19H24N3O5+
Ethyl 4-[3-(4-carbamoylpiperidin-1-ium-1-yl)-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C24H25N5O4S
ethyl 2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[[5-amino-4-[(2S)-1-[(3-cyano-4,5-diphenylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C26H24N6O4S
ethyl 2-[[5-amino-4-[(2S)-1-[(3-cyano-4,5-diphenylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-benzothiazole-6-carboxylate —— C27H25N5O4S
ethyl 2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-benzothiazole-6-carboxylate
—— ethyl 2-[[5-amino-4-[(2S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C15H22N6O3S2
ethyl 2-[[5-amino-4-[(2S)-1-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[4-[(2S)-1-(4-acetylanilino)-1-oxopropan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H21N5O4S
ethyl 2-[[4-[(2S)-1-(4-acetylanilino)-1-oxopropan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[(6-methyl-1,3-benzothiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H22N6O3S2
ethyl 2-[[5-amino-4-[(2R)-1-[(6-methyl-1,3-benzothiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C19H22N6O3S2
ethyl 2-[[5-amino-4-[(2R)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C22H26N6O4S2
ethyl 2-[[5-amino-4-[(2S)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-oxo-1-[2-(trifluoromethyl)anilino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H20F3N5O3S
ethyl 2-[[5-amino-4-[(2S)-1-oxo-1-[2-(trifluoromethyl)anilino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-benzothiazole-6-carboxylate —— C27H25N5O4S
ethyl 2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-benzothiazole-6-carboxylate
—— ethyl 4-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]benzoate —— C26H26N4O4
ethyl 4-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]benzoate
—— ethyl 2-[2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-thiazol-4-yl]acetate —— C24H25N5O4S
ethyl 2-[2-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 5-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate —— C18H24N6O7S
ethyl 5-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate
—— ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H22N6O4S
ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-phenylthiophene-3-carboxylate —— C23H27N5O5S2
ethyl 2-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl 2-[[5-amino-4-[(2R)-1-(2-ethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H25N5O3S
ethyl 2-[[5-amino-4-[(2R)-1-(2-ethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[[3-cyano-4-(4-methoxyphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C22H24N6O4S2
ethyl 2-[[5-amino-4-[(2R)-1-[[3-cyano-4-(4-methoxyphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H22N6O4S
ethyl 2-[[5-amino-4-[(2S)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 5-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate —— C18H24N6O7S
ethyl 5-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate
—— Ethyl 7-(4-methoxyphenyl)-2-methylidene-5-oxo-4-(4-phenylmethoxyphenyl)-1,3,4,6,7,8-hexahydroquinoline-3-carboxylate —— C33H33NO5
Ethyl 7-(4-methoxyphenyl)-2-methylidene-5-oxo-4-(4-phenylmethoxyphenyl)-1,3,4,6,7,8-hexahydroquinoline-3-carboxylate
—— ethyl 2-[2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-thiazol-4-yl]acetate —— C24H25N5O4S
ethyl 2-[2-[[(2S)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 5-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate —— C19H26N6O7S
ethyl 5-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate
—— ethyl 2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H27N5O5S2
ethyl 2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[4-[(2R)-1-(4-acetylanilino)-1-oxobutan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H23N5O4S
ethyl 2-[[4-[(2R)-1-(4-acetylanilino)-1-oxobutan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-(2,4-dimethoxyanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H25N5O5S
ethyl 2-[[5-amino-4-[(2S)-1-(2,4-dimethoxyanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H27N5O5S2
ethyl 2-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[5-amino-4-[(2R)-1-[4-(dimethylsulfamoyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H26N6O5S2
ethyl 2-[[5-amino-4-[(2R)-1-[4-(dimethylsulfamoyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[4-[(2S)-1-(4-acetamidoanilino)-1-oxobutan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H24N6O4S
ethyl 2-[[4-[(2S)-1-(4-acetamidoanilino)-1-oxobutan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-(4-methoxyanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H23N5O4S
ethyl 2-[[5-amino-4-[(2S)-1-(4-methoxyanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[4-(azepan-1-ylsulfonyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C22H32N6O5S2
ethyl 2-[[5-amino-4-[(2R)-1-[4-(azepan-1-ylsulfonyl)anilino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C16H20N6O4S
ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-dimethylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-[[3-cyano-4-(4-methoxyphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C22H24N6O4S2
ethyl 2-[[5-amino-4-[(2S)-1-[[3-cyano-4-(4-methoxyphenyl)thiophen-2-yl]amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-(2-chloroanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C16H20ClN5O3S
ethyl 2-[[5-amino-4-[(2S)-1-(2-chloroanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-[(4-methyl-1,3-thiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C14H20N6O3S2
ethyl 2-[[5-amino-4-[(2S)-1-[(4-methyl-1,3-thiazol-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-phenylthiophene-3-carboxylate —— C23H27N5O5S2
ethyl 2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl 4-acetyl-2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-5-methylfuran-3-carboxylate —— C20H27N5O7S
ethyl 4-acetyl-2-[[(2R)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 2-[[4-[(2R)-1-(4-acetamidophenyl)-1-oxopropan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H21N5O4S
ethyl 2-[[4-[(2R)-1-(4-acetamidophenyl)-1-oxopropan-2-yl]-5-amino-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-diphenylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C26H24N6O4S
ethyl 2-[[5-amino-4-[(2R)-1-[(3-cyano-4,5-diphenylfuran-2-yl)amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-(2,4-dimethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H25N5O3S
ethyl 2-[[5-amino-4-[(2S)-1-(2,4-dimethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C21H24N6O4S2
ethyl 2-[[5-amino-4-[(2R)-1-[[3-carbamoyl-4-(4-methylphenyl)thiophen-2-yl]amino]-1-oxopropan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 4-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]benzoate —— C26H26N4O4
ethyl 4-[[(2R)-2-(3,4-dimethyl-6-oxo-1-phenylpyrazolo[3,4-b]pyridin-7-yl)propanoyl]amino]benzoate
—— ethyl 2-[[5-amino-4-[(2R)-1-(2,3-dimethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H25N5O3S
ethyl 2-[[5-amino-4-[(2R)-1-(2,3-dimethylanilino)-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2R)-1-[(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C19H26N6O4S2
ethyl 2-[[5-amino-4-[(2R)-1-[(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-1-oxobutan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 2-[[5-amino-4-[(2S)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C19H22N6O3S2
ethyl 2-[[5-amino-4-[(2S)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]butan-2-yl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl 5-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate —— C19H26N6O7S
ethyl 5-[[(2S)-2-[3-amino-5-(2-ethoxy-2-oxoethyl)sulfanyl-1,2,4-triazol-4-yl]butanoyl]amino]-4-carbamoyl-2-methylfuran-3-carboxylate