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—— (6Z)-6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H15ClF3N5O2S
(6Z)-6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(3,4-Dimethoxyphenyl)methyl]-9-methoxyindolo[3,2-b]quinoxaline —— C24H21N3O3
6-[(3,4-Dimethoxyphenyl)methyl]-9-methoxyindolo[3,2-b]quinoxaline
—— (6S)-2-bromo-5-(5-chloro-1-methyl-6-oxopyridin-3-yl)-6-(4-chlorophenyl)-1-[(2R)-1-methoxypropan-2-yl]-6H-pyrrolo[3,4-b]pyrrol-4-one —— C22H20BrCl2N3O3
(6S)-2-bromo-5-(5-chloro-1-methyl-6-oxopyridin-3-yl)-6-(4-chlorophenyl)-1-[(2R)-1-methoxypropan-2-yl]-6H-pyrrolo[3,4-b]pyrrol-4-one
—— (6Z)-6-({1-[2-(2,6-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-methyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C26H24N4O2S
(6Z)-6-({1-[2-(2,6-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-methyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 6-(1,4-dioxa-8-azaspiro[4.5]dec-8-ylsulfonyl)-1,3-benzoxazol-2(3H)-one —— C14H16N2O6S
6-(1,4-dioxa-8-azaspiro[4.5]dec-8-ylsulfonyl)-1,3-benzoxazol-2(3H)-one
—— (6Z)-6-[[1-(2-ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(4-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22FN5O2S
(6Z)-6-[[1-(2-ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(4-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Amino-5-(4-bromophenyl)sulfonyl-11-methyl-7-propyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C21H20BrN4O3S+
6-Amino-5-(4-bromophenyl)sulfonyl-11-methyl-7-propyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— (6Z)-6-{[1-(3,4-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C25H18Cl2N4OS
(6Z)-6-{[1-(3,4-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7-(furan-2-ylmethyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C25H23N4O4S+
6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7-(furan-2-ylmethyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— (6Z)-6-[[1-(3,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(3-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5OS
(6Z)-6-[[1-(3,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(3-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(4-fluorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22FN5O2S
(6E)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(4-fluorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-chloro-phenyl)-5-(1,3-dimethyl-1H-pyrazol-4-yl)-1-isopropyl-2-(5-methoxy-1-methyl-2-oxo-1,2-dihydro-pyridin-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C27H28ClN5O3
6-(4-chloro-phenyl)-5-(1,3-dimethyl-1H-pyrazol-4-yl)-1-isopropyl-2-(5-methoxy-1-methyl-2-oxo-1,2-dihydro-pyridin-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7-prop-2-enyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C22H21N4O3S+
6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7-prop-2-enyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— 6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7,11-dimethyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C21H21N4O3S+
6-Amino-5-(3,4-dimethylphenyl)sulfonyl-7,11-dimethyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— 6-(4-chloro-2-methylphenyl)-2-(2,4-dimethoxypyrimidin-5-yl)-5-(4-hydroxycyclohexyl)-1-propan-2-yl-6H-pyrrolo[3,4-b]pyrrol-4-one —— C28H33ClN4O4
6-(4-chloro-2-methylphenyl)-2-(2,4-dimethoxypyrimidin-5-yl)-5-(4-hydroxycyclohexyl)-1-propan-2-yl-6H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-amino-3-chloro-5-methyl-4-sulfanylidene-N-(1-trimethylsilylpropan-2-yl)cyclohexa-1,5-diene-1-carboxamide —— C14H23ClN2OSSi
6-amino-3-chloro-5-methyl-4-sulfanylidene-N-(1-trimethylsilylpropan-2-yl)cyclohexa-1,5-diene-1-carboxamide
—— 6-chloro-9-[(2-chlorophenyl)methyl]-3,4-dimethyl-9,10-dihydro-8H-pyrano[2,3-f][1,3]benzoxazin-9-ium-2-one —— C20H18Cl2NO3+
6-chloro-9-[(2-chlorophenyl)methyl]-3,4-dimethyl-9,10-dihydro-8H-pyrano[2,3-f][1,3]benzoxazin-9-ium-2-one
—— 6-[(2,4-dichlorobenzyl)oxy]-2-[(Z,2E)-3-(2-methoxyphenyl)-2-propenylidene]-1-benzofuran-3-one —— C25H18Cl2O4
6-[(2,4-dichlorobenzyl)oxy]-2-[(Z,2E)-3-(2-methoxyphenyl)-2-propenylidene]-1-benzofuran-3-one
—— (6E)-6-({1-[3-(2,3-dimethylphenoxy)propyl]-1H-indol-3-yl}methylidene)-5-imino-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H26N6O2S
(6E)-6-({1-[3-(2,3-dimethylphenoxy)propyl]-1H-indol-3-yl}methylidene)-5-imino-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Amino-5-(4-bromophenyl)sulfonyl-7-(2-methoxyethyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one —— C21H20BrN4O4S+
6-Amino-5-(4-bromophenyl)sulfonyl-7-(2-methoxyethyl)-11-methyl-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaen-2-one
—— 6,6-dimethyl-4-(4-methylpiperidin-1-yl)-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine —— C18H25N3OS2
6,6-dimethyl-4-(4-methylpiperidin-1-yl)-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine
—— 6-(4-Chlorophenyl)-1-propan-2-yl-5,6-dihydropyrrolo[3,4-b]pyrrol-4-one —— C15H15ClN2O
6-(4-Chlorophenyl)-1-propan-2-yl-5,6-dihydropyrrolo[3,4-b]pyrrol-4-one
—— 6-amino-N-[(4-methoxyphenyl)methyl]-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C26H28N5O4+
6-amino-N-[(4-methoxyphenyl)methyl]-11-methyl-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-(4-chloro-phenyl)-1-isopropyl-5-(tetrahydro-pyran-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C20H23ClN2O2
6-(4-chloro-phenyl)-1-isopropyl-5-(tetrahydro-pyran-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-Hydroxy-5-methyl-3-pyridinsulfonsaeure —— C6H7NO4S
6-Hydroxy-5-methyl-3-pyridinsulfonsaeure
—— (6Z)-6-[[1-[2-(2-chlorophenoxy)ethyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H19ClN6O2S
(6Z)-6-[[1-[2-(2-chlorophenoxy)ethyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[1-[3-(2,3-dimethylphenoxy)propyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H26N6O2S
(6Z)-6-[[1-[3-(2,3-dimethylphenoxy)propyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-chloro-phenyl)-1-isopropyl-5-(1-methyl-6-oxo-piperidin-3-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C21H24ClN3O2
6-(4-chloro-phenyl)-1-isopropyl-5-(1-methyl-6-oxo-piperidin-3-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-chloro-9-(2-chlorobenzyl)-3,4-dimethyl-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one —— C20H17Cl2NO3
6-chloro-9-(2-chlorobenzyl)-3,4-dimethyl-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one
—— 6-amino-N-butyl-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-9-aza-1,7-diazoniatricyclo[8.4.0.03,8]tetradeca-1(14),3,5,7,10,12-hexaene-5-carboxamide —— C23H32N6O3+2
6-amino-N-butyl-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-9-aza-1,7-diazoniatricyclo[8.4.0.03,8]tetradeca-1(14),3,5,7,10,12-hexaene-5-carboxamide
—— 6-amino-N-butyl-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C23H31N6O3+
6-amino-N-butyl-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-[4-[(4-Chlorophenyl)methyl]piperazine-1-carbonyl]-2-phenyl-1,4-dihydropyridazin-3-one —— C22H23ClN4O2
6-[4-[(4-Chlorophenyl)methyl]piperazine-1-carbonyl]-2-phenyl-1,4-dihydropyridazin-3-one
—— 6-({(7RS)-7-[(9aRS)-octahydro-2H-pyrido[1,2-a]pyrazin-2-ylcarbonyl]-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl}amino)-1,3-benzothiazol-2(3H)-one —— C26H28N6O2S2
6-({(7RS)-7-[(9aRS)-octahydro-2H-pyrido[1,2-a]pyrazin-2-ylcarbonyl]-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl}amino)-1,3-benzothiazol-2(3H)-one
—— 6-[4-[(4-Chlorophenyl)methyl]piperazin-4-ium-1-carbonyl]-2-phenyl-1,4-dihydropyridazin-3-one —— C22H24ClN4O2+
6-[4-[(4-Chlorophenyl)methyl]piperazin-4-ium-1-carbonyl]-2-phenyl-1,4-dihydropyridazin-3-one
—— 6-(4-chloro-phenyl)-2-(2-dimethylamino-4-methoxy-pyrimidin-5-yl)-5-(1,3-dimethyl-2-oxo-hexahydro-pyrimidin-5-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C28H34ClN7O3
6-(4-chloro-phenyl)-2-(2-dimethylamino-4-methoxy-pyrimidin-5-yl)-5-(1,3-dimethyl-2-oxo-hexahydro-pyrimidin-5-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— (6S)-2-bromo-5-(3-chloro-4-fluorophenyl)-6-(4-chlorophenyl)-1-[(2R)-1-methoxypropan-2-yl]-6H-pyrrolo[3,4-b]pyrrol-4-one —— C22H18BrCl2FN2O2
(6S)-2-bromo-5-(3-chloro-4-fluorophenyl)-6-(4-chlorophenyl)-1-[(2R)-1-methoxypropan-2-yl]-6H-pyrrolo[3,4-b]pyrrol-4-one
—— (6Z)-2-(2-chlorophenyl)-6-{[1-(2,6-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22ClN5OS
(6Z)-2-(2-chlorophenyl)-6-{[1-(2,6-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-benzhydrylpiperazine-1-carbonyl)pyridazin-3(2H)-one —— C22H22N4O2
6-(4-benzhydrylpiperazine-1-carbonyl)pyridazin-3(2H)-one
—— 6,6-difluoro-N-[2-methoxy-5-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b]indol-4-amine —— C18H15F5N4O
6,6-difluoro-N-[2-methoxy-5-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b]indol-4-amine
—— 6-amino-N-[(4-methoxyphenyl)methyl]-11-methyl-2-oxo-7-[[(2R)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C26H28N5O4+
6-amino-N-[(4-methoxyphenyl)methyl]-11-methyl-2-oxo-7-[[(2R)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6,8-Difluoro-1-(2-fluoroethyl)-7-(4-methylpiperazin-1-yl)-4-oxoquinoline-3-carboxylic acid;1-ethyl-6-fluoro-7-(4-methylpiperazin-1-yl)-4-oxoquinoline-3-carboxylic acid —— C34H38F4N6O6
6,8-Difluoro-1-(2-fluoroethyl)-7-(4-methylpiperazin-1-yl)-4-oxoquinoline-3-carboxylic acid;1-ethyl-6-fluoro-7-(4-methylpiperazin-1-yl)-4-oxoquinoline-3-carboxylic acid
—— (6E)-6-{[1-(3,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H15Cl2N5O2S
(6E)-6-{[1-(3,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-chloro-phenyl)-2-(2-dimethylamino-4-methoxy-pyrimidin-5-yl)-5-(2,5-dimethyl-2H-pyrazol-3-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C27H30ClN7O2
6-(4-chloro-phenyl)-2-(2-dimethylamino-4-methoxy-pyrimidin-5-yl)-5-(2,5-dimethyl-2H-pyrazol-3-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-[2-(1,4-dioxaspiro[4.5]dec-8-ylidene)hydrazino]pyrimidin-4-ol —— C12H16N4O3
6-[2-(1,4-dioxaspiro[4.5]dec-8-ylidene)hydrazino]pyrimidin-4-ol
—— 6-(4-chloro-phenyl)-5-(4-fluoro-2,5-dimethyl-2H-pyrazol-3-yl)-1-isopropyl-2-(5-methoxy-1-methyl-2-oxo-1,2-dihydro-pyridin-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C27H27ClFN5O3
6-(4-chloro-phenyl)-5-(4-fluoro-2,5-dimethyl-2H-pyrazol-3-yl)-1-isopropyl-2-(5-methoxy-1-methyl-2-oxo-1,2-dihydro-pyridin-4-yl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-chloro-4-[1-(oxetan-3-yl)piperidin-4-yl]-N-pyridin-2-ylpyridin-2-amine —— C18H21ClN4O
6-chloro-4-[1-(oxetan-3-yl)piperidin-4-yl]-N-pyridin-2-ylpyridin-2-amine
—— 6-(4-chlorophenyl)-2-(2,4-dimethoxypyrimidin-5-yl)-5-(4-methoxycyclohexyl)-1-propan-2-yl-6H-pyrrolo[3,4-b]pyrrol-4-one —— C28H33ClN4O4
6-(4-chlorophenyl)-2-(2,4-dimethoxypyrimidin-5-yl)-5-(4-methoxycyclohexyl)-1-propan-2-yl-6H-pyrrolo[3,4-b]pyrrol-4-one
—— 6-amino-7-[(4-fluorophenyl)methyl]-11-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C25H25FN5O3+
6-amino-7-[(4-fluorophenyl)methyl]-11-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— (6Z)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C25H19ClN4OS
(6Z)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 6-{[(7RS)-7-{[(3RS)-3-fluoropiperidin-1-yl]carbonyl}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]amino}-1,3-benzothiazol-2(3H)-one —— C23H22FN5O2S2
6-{[(7RS)-7-{[(3RS)-3-fluoropiperidin-1-yl]carbonyl}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]amino}-1,3-benzothiazol-2(3H)-one