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苯并噁庚英

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4,5-dihydro-[1]benzoxepino[4,5-d][1,3]thiazol-2-yl N-(2-chlorophenyl)-N-methylcarbamate —— C19H15ClN2O3S
4,5-dihydro-[1]benzoxepino[4,5-d][1,3]thiazol-2-yl N-(2-chlorophenyl)-N-methylcarbamate
—— (3R)-2-[4-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde —— C27H25F2N5O2S
(3R)-2-[4-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde
—— 5-[2-propan-2-yl-4-(1H-1,2,4-triazol-5-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl]pyridin-2-amine —— C21H20N6OS
5-[2-propan-2-yl-4-(1H-1,2,4-triazol-5-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl]pyridin-2-amine
—— 2-[2-[2-(2-Hydroxy-2-methylpropyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C24H29N5O3S
2-[2-[2-(2-Hydroxy-2-methylpropyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— 2-[4-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C26H23F2N5O2S
2-[4-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— 2-[5-(1,1,1-trifluoropropan-2-yl)-1H-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide —— C17H14F3N5O2S
2-[5-(1,1,1-trifluoropropan-2-yl)-1H-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide
—— [2-[5-(2,4-Difluorophenyl)-1,2,4-triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl] carbamate —— C20H13F2N5O3S
[2-[5-(2,4-Difluorophenyl)-1,2,4-triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl] carbamate
—— 2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide —— C17H17N5O2S
2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxamide
—— 2-[4-[2-(2-Hydroxy-2-methylpropyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C24H29N5O3S
2-[4-[2-(2-Hydroxy-2-methylpropyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— 4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-yl N-[2-chloro-4-(methylcarbamoyl)phenyl]-N-methylcarbamate —— C21H18ClN3O4S
4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-yl N-[2-chloro-4-(methylcarbamoyl)phenyl]-N-methylcarbamate
—— 8-(1H-imidazol-2-yl)-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole —— C19H18N6OS
8-(1H-imidazol-2-yl)-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole
—— 8-(1H-pyrazol-4-yl)-2-[5-(1,1,1-trifluoropropan-2-yl)-1H-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole —— C19H15F3N6OS
8-(1H-pyrazol-4-yl)-2-[5-(1,1,1-trifluoropropan-2-yl)-1H-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole
—— (8-cyano-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-yl) N-[2-chloro-4-(methylcarbamoyl)phenyl]-N-methylcarbamate —— C22H17ClN4O4S
(8-cyano-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-yl) N-[2-chloro-4-(methylcarbamoyl)phenyl]-N-methylcarbamate
—— (3S)-2-[4-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde —— C27H25F2N5O2S
(3S)-2-[4-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde
—— 2-methylsulfonyl-N-[2-(4-propan-2-yl-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl]acetamide —— C19H21N5O4S2
2-methylsulfonyl-N-[2-(4-propan-2-yl-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl]acetamide
—— 2-[4-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C26H23F2N5O2S
2-[4-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— [2-[5-(2,4-Difluorophenyl)triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl] carbamate —— C20H13F2N5O3S
[2-[5-(2,4-Difluorophenyl)triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl] carbamate
—— (2R)-2-[2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde —— C27H25F2N5O2S
(2R)-2-[2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde
—— 9-bromo-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole —— C16H15BrN4OS
9-bromo-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole
—— 2-[2-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C26H23F2N5O2S
2-[2-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— 2-[2-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]piperazine-1-carbaldehyde —— C25H21F2N5O2S
2-[2-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]piperazine-1-carbaldehyde
—— 2-[2-[2-(2-Chlorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde —— C26H24ClN5O2S
2-[2-[2-(2-Chlorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-4-methylpiperazine-1-carbaldehyde
—— (2S)-2-[2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde —— C27H25F2N5O2S
(2S)-2-[2-[2-(2,4-difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]-3-(dimethylamino)pyrrolidine-1-carbaldehyde
—— 2-[4-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]piperazine-1-carbaldehyde —— C25H21F2N5O2S
2-[4-[2-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-9-yl]piperazine-1-carbaldehyde
—— [2-[4-(2-Chlorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl]-methylcarbamic acid —— C22H17ClN4O3S
[2-[4-(2-Chlorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl]-methylcarbamic acid
—— 8-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole —— C21H22N6OS
8-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole
—— [2-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl] carbamate —— C20H13F2N5O3S
[2-[4-(2,4-Difluorophenyl)-1,2,4-triazol-3-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl] carbamate
—— 2-[5-(2,4-Difluorophenyl)-1,2,4-triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxylic acid —— C20H12F2N4O3S
2-[5-(2,4-Difluorophenyl)-1,2,4-triazol-1-yl]-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-8-carboxylic acid
—— 2-methylsulfonyl-N-[2-(4-propan-2-yl-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl]acetamide —— C19H21N5O4S2
2-methylsulfonyl-N-[2-(4-propan-2-yl-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-9-yl]acetamide
—— 5-[2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl]pyridin-2-amine —— C21H20N6OS
5-[2-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-8-yl]pyridin-2-amine
—— N-(9-fluoro-5,6-dihydrobenzo[b][1]benzoxepin-3-yl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C24H19FN4O2S
N-(9-fluoro-5,6-dihydrobenzo[b][1]benzoxepin-3-yl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— Methyl 5-[(3-fluoro-7-oxo-7lambda6-thia-8-azabicyclo[4.2.0]octa-1(6),2,4,7-tetraen-7-yl)-methoxycarbonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate —— C20H17FN2O6S
Methyl 5-[(3-fluoro-7-oxo-7lambda6-thia-8-azabicyclo[4.2.0]octa-1(6),2,4,7-tetraen-7-yl)-methoxycarbonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— tert-butyl 3-[(Z)-2-[5-fluoro-2-[(4-methoxycarbonyl-1,1a,2,7b-tetrahydrocyclopropa[c]chromen-5-yl)sulfamoyl]phenyl]ethenyl]azetidine-1-carboxylate —— C28H31FN2O7S
tert-butyl 3-[(Z)-2-[5-fluoro-2-[(4-methoxycarbonyl-1,1a,2,7b-tetrahydrocyclopropa[c]chromen-5-yl)sulfamoyl]phenyl]ethenyl]azetidine-1-carboxylate
—— Methyl 5-[[2-[[acetyl(methyl)amino]methyl]-4-fluorophenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate —— C22H23FN2O6S
Methyl 5-[[2-[[acetyl(methyl)amino]methyl]-4-fluorophenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— methyl (1aR,7bS)-5-[2-((R)-1-ethylpyrrolidin-3-yloxymethyl)-4-fluorobenzene-sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate 1412979-29-3 C25H29FN2O6S
methyl (1aR,7bS)-5-[2-((R)-1-ethylpyrrolidin-3-yloxymethyl)-4-fluorobenzene-sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— Tert-butyl 5-acetamido-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate —— C17H21NO4
Tert-butyl 5-acetamido-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— 5-Acetamido-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid —— C13H13NO4
5-Acetamido-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— (1aRS,7bSR)-5-[2-((Z)-3-diethylaminoprop-1-enyl)-4-fluorobenzene-sulfonylamino]-1,1-difluoro-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid 1412974-09-4 C24H25F3N2O5S
(1aRS,7bSR)-5-[2-((Z)-3-diethylaminoprop-1-enyl)-4-fluorobenzene-sulfonylamino]-1,1-difluoro-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— (1aRS,7bSR)-5-{2[(Z)-3-(pyrrolidin-1-yl)prop-1-enyl]-4-fluorobenzene-sulfonylamino}-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid 1412974-21-0 C24H25FN2O5S
(1aRS,7bSR)-5-{2[(Z)-3-(pyrrolidin-1-yl)prop-1-enyl]-4-fluorobenzene-sulfonylamino}-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— Methyl 5-[[2-(1-acetylazetidin-3-yl)-4-fluorophenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate —— C23H23FN2O6S
Methyl 5-[[2-(1-acetylazetidin-3-yl)-4-fluorophenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— methyl 5-[[4-fluoro-2-[(Z)-3-[(3S)-3-hydroxypyrrolidin-1-yl]prop-1-enyl]phenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate —— C25H27FN2O6S
methyl 5-[[4-fluoro-2-[(Z)-3-[(3S)-3-hydroxypyrrolidin-1-yl]prop-1-enyl]phenyl]sulfonylamino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylate
—— (1aRS,7bSR)-5-{2[(Z)-3-(azetidin-1-yl)prop-1-enyl]-4-fluorobenzenesulfonyl-amino}-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid 1412974-55-0 C23H23FN2O5S
(1aRS,7bSR)-5-{2[(Z)-3-(azetidin-1-yl)prop-1-enyl]-4-fluorobenzenesulfonyl-amino}-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— 5-[2-[5-(dimethylamino)pentylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid —— C24H31N3O5S
5-[2-[5-(dimethylamino)pentylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— 4-carboxy-5-[4-fluoro-2-(2-methoxy-2-oxoethyl)-N-sulfinatoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene —— C20H17FNO7S-
4-carboxy-5-[4-fluoro-2-(2-methoxy-2-oxoethyl)-N-sulfinatoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene
—— 5-[2-[[(3R)-1-ethylpyrrolidin-3-yl]methylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid —— C24H29N3O5S
5-[2-[[(3R)-1-ethylpyrrolidin-3-yl]methylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— (1aR,7bS)-5-[2((Z)-4-diethylaminobut-1-enyl)-4-fluorobenzenesulfonyl-amino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid 1412974-49-2 C25H29FN2O5S
(1aR,7bS)-5-[2((Z)-4-diethylaminobut-1-enyl)-4-fluorobenzenesulfonyl-amino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— 5-[2-[4-(dimethylamino)butylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid —— C23H29N3O5S
5-[2-[4-(dimethylamino)butylamino]-N-sulfinoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene-4-carboxylic acid
—— (3R)-3-[[2-[(4-carboxy-1,1a,2,7b-tetrahydrocyclopropa[c]chromen-5-yl)-sulfinatoamino]anilino]methyl]-1-ethylpyrrolidine —— C24H28N3O5S-
(3R)-3-[[2-[(4-carboxy-1,1a,2,7b-tetrahydrocyclopropa[c]chromen-5-yl)-sulfinatoamino]anilino]methyl]-1-ethylpyrrolidine
—— 4-carboxy-5-[2-[5-(dimethylamino)pentylamino]-N-sulfinatoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene —— C24H30N3O5S-
4-carboxy-5-[2-[5-(dimethylamino)pentylamino]-N-sulfinatoanilino]-1,1a,2,7b-tetrahydrocyclopropa[c]chromene
—— (2R)-7'-methyl-3-[(4-methylphenyl)methyl]spiro[1H-quinazoline-2,5'-3,4-dihydro-2H-1-benzoxepine]-4-one —— C26H26N2O2
(2R)-7'-methyl-3-[(4-methylphenyl)methyl]spiro[1H-quinazoline-2,5'-3,4-dihydro-2H-1-benzoxepine]-4-one