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苯并噁庚英

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-((4aR,11bR)-2-amino-3,3,11b-trimethyl-4,4-dioxido-4a,5,6,11b-tetrahydro-3H-benzo[6,7]oxepino[4,5-b][1,4]thiazin-10-yl)-5-((R)-pent-3-yn-2-yloxy)picolinamide —— C26H30N4O5S
N-((4aR,11bR)-2-amino-3,3,11b-trimethyl-4,4-dioxido-4a,5,6,11b-tetrahydro-3H-benzo[6,7]oxepino[4,5-b][1,4]thiazin-10-yl)-5-((R)-pent-3-yn-2-yloxy)picolinamide
—— tert-butyl N-[(4aS,6S,11bS)-10-amino-11b-(fluoromethyl)-3,3,6-trimethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-2-yl]-N-tert-butoxycarbonylcarbamate 1620981-06-7 C26H38FN3O7S
tert-butyl N-[(4aS,6S,11bS)-10-amino-11b-(fluoromethyl)-3,3,6-trimethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-2-yl]-N-tert-butoxycarbonylcarbamate
—— (4aR,11bR)-2,3,3,6,6,11b-hexamethyl-4,4-dioxo-4a,5-dihydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine —— C18H26N2O3S
(4aR,11bR)-2,3,3,6,6,11b-hexamethyl-4,4-dioxo-4a,5-dihydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine
—— (11bR)-2,3,3,4a,11b-pentamethyl-10-nitro-5,6-dihydro-[1]benzoxepino[4,5-b][1,4]thiazine 4,4-dioxide —— C17H22N2O5S
(11bR)-2,3,3,4a,11b-pentamethyl-10-nitro-5,6-dihydro-[1]benzoxepino[4,5-b][1,4]thiazine 4,4-dioxide
—— (4aR,11bR)-2,3,3,11b-tetramethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine —— C16H22N2O3S
(4aR,11bR)-2,3,3,11b-tetramethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine
—— (4aR,11bS)-11b-(fluoromethyl)-2,3,3-trimethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine —— C16H21FN2O3S
(4aR,11bS)-11b-(fluoromethyl)-2,3,3-trimethyl-4,4-dioxo-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine
—— (11bR)-2,3,3,4a,11b-pentamethyl-4,4-dioxo-5,6-dihydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine —— C17H24N2O3S
(11bR)-2,3,3,4a,11b-pentamethyl-4,4-dioxo-5,6-dihydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine
—— 5-(4a-methyl-3,5,6,11b-tetrahydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl)-2-(dimethylamino)-4,4-dihydroxy-6,8-dimethyl-1H-1,7-naphthyridine-3-carbonitrile —— C26H29N5O3S
5-(4a-methyl-3,5,6,11b-tetrahydro-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl)-2-(dimethylamino)-4,4-dihydroxy-6,8-dimethyl-1H-1,7-naphthyridine-3-carbonitrile
—— 1-amino-3-(4,4-dioxo-4a,5,6,11b-tetrahydro-3H-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl)-3,5,7,8-tetramethyl-4H-pyrido[3,4-b]pyrazin-2-one —— C23H27N5O4S
1-amino-3-(4,4-dioxo-4a,5,6,11b-tetrahydro-3H-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl)-3,5,7,8-tetramethyl-4H-pyrido[3,4-b]pyrazin-2-one
—— 2-(Fluoromethyl)-4,4-dihydroxy-3,3,6-trimethyl-4a,5,6,11b-tetrahydro-[1]benzoxepino[4,5-b][1,4]thiazine —— C16H22FNO3S
2-(Fluoromethyl)-4,4-dihydroxy-3,3,6-trimethyl-4a,5,6,11b-tetrahydro-[1]benzoxepino[4,5-b][1,4]thiazine
—— 2,3,3,4a-tetramethyl-4,4-dioxo-N-[3-(trifluoromethyl)-1,7-naphthyridin-8-yl]-6,11b-dihydro-5H-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine —— C25H25F3N4O3S
2,3,3,4a-tetramethyl-4,4-dioxo-N-[3-(trifluoromethyl)-1,7-naphthyridin-8-yl]-6,11b-dihydro-5H-[1]benzoxepino[4,5-b][1,4]thiazin-10-amine
—— 3H-[1]benzoxepino[4,5-b][1,4]thiazine —— C12H9NOS
3H-[1]benzoxepino[4,5-b][1,4]thiazine
—— N-[(4aS,11bS)-2-amino-4,4-dihydroxy-3,3,11b-trimethyl-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl]-5-chloro-3-methylpyridine-2-carboxamide —— C22H27ClN4O4S
N-[(4aS,11bS)-2-amino-4,4-dihydroxy-3,3,11b-trimethyl-5,6-dihydro-4aH-[1]benzoxepino[4,5-b][1,4]thiazin-10-yl]-5-chloro-3-methylpyridine-2-carboxamide
—— 7-nitro-N-pyridin-3-yl-2,3,4,5-tetrahydro-1-benzoxepine-8-carboxamide —— C16H15N3O4
7-nitro-N-pyridin-3-yl-2,3,4,5-tetrahydro-1-benzoxepine-8-carboxamide
—— 3-[(3E)-3-chloroiminospiro[1H-indene-2,4'-3,5-dihydro-2H-1-benzoxepine]-5-yl]benzonitrile —— C25H19ClN2O
3-[(3E)-3-chloroiminospiro[1H-indene-2,4'-3,5-dihydro-2H-1-benzoxepine]-5-yl]benzonitrile
—— (9-Methyl-6,7-dihydro-[1]benzofuro[3,2-d][1]benzoxepin-3-yl) trifluoromethanesulfonate —— C18H13F3O5S
(9-Methyl-6,7-dihydro-[1]benzofuro[3,2-d][1]benzoxepin-3-yl) trifluoromethanesulfonate
—— 3-[(1Z)-1-[8-[(7-ethynyl-2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C29H21FN4O3
3-[(1Z)-1-[8-[(7-ethynyl-2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— 3-[(1Z)-1-[3-fluoro-8-[[8-methoxy-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C29H25FN4O5
3-[(1Z)-1-[3-fluoro-8-[[8-methoxy-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (E)-2-{3-fluoro-8-[(8-methyl-2-propylimidazo[1,2-a]pyrazin-3-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}propanenitrile 1421787-45-2 C28H25FN4O
(E)-2-{3-fluoro-8-[(8-methyl-2-propylimidazo[1,2-a]pyrazin-3-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}propanenitrile
—— 3-[(1Z)-1-[8-[[7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C28H22ClFN4O4
3-[(1Z)-1-[8-[[7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (E)-2-(8-{[4-(difluoromethoxy)-2-(methoxymethyl)-1H-benzo[d]imidazol-1-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile 1421785-22-9 C28H22F3N3O3
(E)-2-(8-{[4-(difluoromethoxy)-2-(methoxymethyl)-1H-benzo[d]imidazol-1-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile
—— (E)-3-(1-{3-fluoro-8-[(2-isopropyl-1H-benzo[d]imidazol-1-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one 1421783-68-7 C29H25FN4O3
(E)-3-(1-{3-fluoro-8-[(2-isopropyl-1H-benzo[d]imidazol-1-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one
—— (2Z)-2-[3-fluoro-8-[(5-fluoro-2-propylimidazo[4,5-b]pyridin-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C27H22F2N4O
(2Z)-2-[3-fluoro-8-[(5-fluoro-2-propylimidazo[4,5-b]pyridin-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile
—— (E)-3-[1-(3-fluoro-8-{[2-(methoxymethyl)-4-(methylthio)-1H-benzo[d]imidazol-1-yl]methyl}dibenzo[b,e]oxepin-11(6H)-ylidene)ethyl]-1,2,4-oxadiazol-5(4H)-one 1421783-91-6 C29H25FN4O4S
(E)-3-[1-(3-fluoro-8-{[2-(methoxymethyl)-4-(methylthio)-1H-benzo[d]imidazol-1-yl]methyl}dibenzo[b,e]oxepin-11(6H)-ylidene)ethyl]-1,2,4-oxadiazol-5(4H)-one
—— 8-bromo-1,3-difluorospiro[6H-benzo[c][1]benzoxepine-11,2'-cyclopropane]-1'-carbonitrile —— C17H10BrF2NO
8-bromo-1,3-difluorospiro[6H-benzo[c][1]benzoxepine-11,2'-cyclopropane]-1'-carbonitrile
—— (11R)-8-bromo-1,3-difluorospiro[6H-benzo[c][1]benzoxepine-11,2'-cyclopropane]-1'-carbonitrile —— C17H10BrF2NO
(11R)-8-bromo-1,3-difluorospiro[6H-benzo[c][1]benzoxepine-11,2'-cyclopropane]-1'-carbonitrile
—— 3-[(1Z)-1-[8-[[8-(difluoromethoxy)-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C29H23F3N4O5
3-[(1Z)-1-[8-[[8-(difluoromethoxy)-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— 3-[(1Z)-1-[3-fluoro-8-[[2-(methoxymethyl)thieno[3,4-d]imidazol-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C26H21FN4O4S
3-[(1Z)-1-[3-fluoro-8-[[2-(methoxymethyl)thieno[3,4-d]imidazol-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— methyl 1-[[(11E)-11-(2-cyanoethylidene)-3-fluoro-6H-benzo[c][1]benzoxepin-8-yl]methyl]-2-propylbenzimidazole-4-carboxylate —— C30H26FN3O3
methyl 1-[[(11E)-11-(2-cyanoethylidene)-3-fluoro-6H-benzo[c][1]benzoxepin-8-yl]methyl]-2-propylbenzimidazole-4-carboxylate
—— (2Z)-2-[3,4-difluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C28H23F2N3O
(2Z)-2-[3,4-difluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile
—— 2-(8-bromo-3,4-difluoro-6H-benzo[c][1]benzoxepin-11-ylidene)propanenitrile —— C17H10BrF2NO
2-(8-bromo-3,4-difluoro-6H-benzo[c][1]benzoxepin-11-ylidene)propanenitrile
—— (E)-3-(1-{8-[(8-chloro-2-cyclobutylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one 1421784-27-1 C30H24ClFN4O3
(E)-3-(1-{8-[(8-chloro-2-cyclobutylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one
—— 3-[(1Z)-1-[8-[[2-(dimethylamino)benzimidazol-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C28H24FN5O3
3-[(1Z)-1-[8-[[2-(dimethylamino)benzimidazol-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— 3-[(1Z)-1-[3-fluoro-8-[[2-methyl-8-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C28H20F4N4O3
3-[(1Z)-1-[3-fluoro-8-[[2-methyl-8-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (E)-2-(8-{[8-(difluoromethoxy)-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile 1421786-42-6 C28H22F3N3O3
(E)-2-(8-{[8-(difluoromethoxy)-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile
—— (E)-3-(1-{3-fluoro-8-[(2-isopropyl-8-methoxyimidazo[1,2-a]pyridin-3-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one 1421784-35-1 C30H27FN4O4
(E)-3-(1-{3-fluoro-8-[(2-isopropyl-8-methoxyimidazo[1,2-a]pyridin-3-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one
—— (2E)-2-[3-fluoro-8-(hydroxymethyl)-6H-benzo[c][1]benzoxepin-11-ylidene]butanenitrile —— C19H16FNO2
(2E)-2-[3-fluoro-8-(hydroxymethyl)-6H-benzo[c][1]benzoxepin-11-ylidene]butanenitrile
—— 1-[[(11E)-11-(2-cyanoethylidene)-3-fluoro-6H-benzo[c][1]benzoxepin-8-yl]methyl]-5-methyl-2-propylbenzimidazole-4-carboxylic acid —— C30H26FN3O3
1-[[(11E)-11-(2-cyanoethylidene)-3-fluoro-6H-benzo[c][1]benzoxepin-8-yl]methyl]-5-methyl-2-propylbenzimidazole-4-carboxylic acid
—— (E)-2-cyclopropyl-2-(8-{[2-(3,3-difluorocyclobutyl)-1H-benzo[d]imidazol-1-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)acetonitrile 1421785-70-7 C31H24F3N3O
(E)-2-cyclopropyl-2-(8-{[2-(3,3-difluorocyclobutyl)-1H-benzo[d]imidazol-1-yl]methyl}-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)acetonitrile
—— (2Z)-2-[8-[[8-(difluoromethoxy)-2-propan-2-ylimidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C29H24F3N3O2
(2Z)-2-[8-[[8-(difluoromethoxy)-2-propan-2-ylimidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile
—— 3-[(1Z)-1-[8-[(2-ethylbenzimidazol-1-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C28H23FN4O3
3-[(1Z)-1-[8-[(2-ethylbenzimidazol-1-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (E)-3-(1-{3-fluoro-8-[(2-propyl-1H-imidazo[4,5-c]pyridin-1-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one 1421783-94-9 C28H24FN5O3
(E)-3-(1-{3-fluoro-8-[(2-propyl-1H-imidazo[4,5-c]pyridin-1-yl)methyl]dibenzo[b,e]oxepin-11(6H)-ylidene}ethyl)-1,2,4-oxadiazol-5(4H)-one
—— 3-[(1Z)-1-[8-[(2-cyclopropyl-8-methylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C30H25FN4O3
3-[(1Z)-1-[8-[(2-cyclopropyl-8-methylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (2Z)-2-[3-fluoro-8-[(8-methoxy-2-propan-2-ylimidazo[1,2-a]pyridin-3-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C29H26FN3O2
(2Z)-2-[3-fluoro-8-[(8-methoxy-2-propan-2-ylimidazo[1,2-a]pyridin-3-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile
—— 3-[(1Z)-1-[8-[[2-(cyclobutadienyl)-5-fluoroimidazo[4,5-b]pyridin-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C29H19F2N5O3
3-[(1Z)-1-[8-[[2-(cyclobutadienyl)-5-fluoroimidazo[4,5-b]pyridin-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (E)-2-{8-[(7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl)methyl]-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene}-2-cyclopropylacetonitrile 1421787-12-3 C29H23ClFN3O2
(E)-2-{8-[(7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl)methyl]-3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene}-2-cyclopropylacetonitrile
—— 3-[(1Z)-1-[3-fluoro-8-[[2-methoxy-7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C28H20F4N4O4
3-[(1Z)-1-[3-fluoro-8-[[2-methoxy-7-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (2Z)-2-[8-[[8-chloro-2-(cyclobutadienyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C29H19ClFN3O
(2Z)-2-[8-[[8-chloro-2-(cyclobutadienyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile
—— 3-[(1Z)-1-[8-[[4-(difluoromethoxy)-2-(methoxymethyl)benzimidazol-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one —— C29H23F3N4O5
3-[(1Z)-1-[8-[[4-(difluoromethoxy)-2-(methoxymethyl)benzimidazol-1-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
—— (2Z)-2-[3-fluoro-8-[[2-(methoxymethyl)-4-methylsulfanylbenzimidazol-1-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile —— C28H24FN3O2S
(2Z)-2-[3-fluoro-8-[[2-(methoxymethyl)-4-methylsulfanylbenzimidazol-1-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]propanenitrile