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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S,4R)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-(4-phenylpiperazine-1-carbonyl)-3,4-dihydroisoquinolin-1-one —— C30H33N3O4S
(3S,4R)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-(4-phenylpiperazine-1-carbonyl)-3,4-dihydroisoquinolin-1-one
—— 5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32FN5O4S2
5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— (3R,4R)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one —— C30H32N4O6S
(3R,4R)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one
—— (3R,4R)-6,7-dimethoxy-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one —— C31H35N3O5S
(3R,4R)-6,7-dimethoxy-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one
—— (3R,4S)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one —— C30H32N4O6S
(3R,4S)-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one
—— (3R,4R)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one —— C30H32ClN3O4S
(3R,4R)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one
—— (3R)-N-[[(3aR,4S,7R,7aR)-2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-4,7-epoxyisoindol-4-yl]methyl]-3-methyl-4-(3-methylphenyl)piperazine-1-carbothioamide —— C29H32N4O3S
(3R)-N-[[(3aR,4S,7R,7aR)-2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-4,7-epoxyisoindol-4-yl]methyl]-3-methyl-4-(3-methylphenyl)piperazine-1-carbothioamide
—— 6-bromo-3-[4-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-quinazoline-2,4-dione —— C24H27BrN4O3
6-bromo-3-[4-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-quinazoline-2,4-dione
—— 5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32FN5O4S2
5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— 2-[(3S)-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]piperidin-1-yl]thieno[3,2-d][1,3]thiazin-4-one —— C22H23N5O4S2
2-[(3S)-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]piperidin-1-yl]thieno[3,2-d][1,3]thiazin-4-one
—— 3-[(4-methoxyphenyl)methyl]-7-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-quinazoline-2,4-dione —— C29H30N4O4
3-[(4-methoxyphenyl)methyl]-7-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-quinazoline-2,4-dione
—— (3S,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one —— C30H32ClN3O4S
(3S,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one
—— 5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C27H35N5O5S2
5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-one —— C26H33N5O4S2
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-one
—— (5R,6S)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H37N3O6
(5R,6S)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-one —— C26H33N5O4S2
5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-one
—— (5S,6S)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H37N3O6
(5S,6S)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— (5R,6R)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H36ClN3O6
(5R,6R)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32FN5O4S2
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— (5R,6S)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C33H39N3O7
(5R,6S)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C27H35N5O5S2
5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— 5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-[4-(4-nitrophenyl)piperazin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C26H32N6O6S2
5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-[4-(4-nitrophenyl)piperazin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— N-[3-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-3-oxopropyl]-2-(1-oxoisoquinolin-2-yl)acetamide —— C26H30N4O3
N-[3-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-3-oxopropyl]-2-(1-oxoisoquinolin-2-yl)acetamide
—— (5R,6R)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C33H39N3O7
(5R,6R)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C27H35N5O5S2
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— (5R,6S)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H36ClN3O6
(5R,6S)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— N-[(2S)-1-[4-(2,5-dimethylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C25H29N3O3S2
N-[(2S)-1-[4-(2,5-dimethylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— 5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32FN5O4S2
5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— (5R,6R)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H36FN3O6
(5R,6R)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 3-[4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione —— C22H26N4O3S
3-[4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
—— 3-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]-5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32ClN5O4S2
3-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]-5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methylthieno[2,3-d]pyrimidin-4-one
—— 3-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]-5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32ClN5O4S2
3-[2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl]-5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methylthieno[2,3-d]pyrimidin-4-one
—— 3-[6-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-oxohexyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione —— C24H30N4O3S
3-[6-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-oxohexyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
—— (5S,6S)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C33H39N3O7
(5S,6S)-6-(4-methoxyphenyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H37N3O6
(5R,6R)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-[4-(4-nitrophenyl)piperazin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C26H32N6O6S2
5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-6-methyl-3-[2-[4-(4-nitrophenyl)piperazin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— (5S,6R)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H37N3O6
(5S,6R)-6-(4-methoxyphenyl)-5-(4-phenylpiperazine-1-carbonyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— (5S,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H36FN3O6
(5S,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— (5S,6S)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one —— C32H36ClN3O6
(5S,6S)-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-(3,4,5-trimethoxyphenyl)piperidin-2-one
—— 3-[6-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-oxohexyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione —— C24H30N4O3S
3-[6-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-oxohexyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
—— 3-[(5-bromo-1-propanoyl-2,3-dihydroindol-7-yl)sulfonyl]-1-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]propan-1-one —— C26H32BrN3O4S
3-[(5-bromo-1-propanoyl-2,3-dihydroindol-7-yl)sulfonyl]-1-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]propan-1-one
—— 6,7-dimethoxy-4-[(3S)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one —— C28H35N3O4
6,7-dimethoxy-4-[(3S)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one
—— N'-methyl-2-[1-(4-pyridin-2-ylpiperazine-1-carbonyl)piperidin-4-yl]-N'-quinoxalin-2-yl-1,3-thiazole-4-carbohydrazide —— C28H31N9O2S
N'-methyl-2-[1-(4-pyridin-2-ylpiperazine-1-carbonyl)piperidin-4-yl]-N'-quinoxalin-2-yl-1,3-thiazole-4-carbohydrazide
—— N-[(2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C23H24FN3O3S2
N-[(2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C31H33ClFN5O2S
N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— 4-[5-Nitro-6-(4-pyridin-2-ylpiperazin-1-yl)pyrimidin-4-yl]oxybenzene-1,2-dicarbonitrile —— C21H16N8O3
4-[5-Nitro-6-(4-pyridin-2-ylpiperazin-1-yl)pyrimidin-4-yl]oxybenzene-1,2-dicarbonitrile
—— 3-[4-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione —— C22H26N4O3S
3-[4-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-4-oxobutyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
—— [4-(2-fluorophenyl)piperazin-1-yl]-[(2R)-1-(2,4,6-trimethylphenyl)sulfonylpiperidin-2-yl]methanone —— C25H32FN3O3S
[4-(2-fluorophenyl)piperazin-1-yl]-[(2R)-1-(2,4,6-trimethylphenyl)sulfonylpiperidin-2-yl]methanone
—— N-(4-chlorophenyl)-2-[(4S)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methoxyphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C31H33ClFN5O3S
N-(4-chlorophenyl)-2-[(4S)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methoxyphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— 2-ethyl-6,7-dimethoxy-4-[(3R)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]isoquinolin-1-one —— C26H31N3O4
2-ethyl-6,7-dimethoxy-4-[(3R)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]isoquinolin-1-one