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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-methyl-N-[[(2R)-oxolan-2-yl]methyl]-4-(4-phenylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide —— C23H27N5O2S
5-methyl-N-[[(2R)-oxolan-2-yl]methyl]-4-(4-phenylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
—— N-[(2R)-butan-2-yl]-4-[4-(2-fluorophenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide —— C22H26FN5OS
N-[(2R)-butan-2-yl]-4-[4-(2-fluorophenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
—— [(3S,5S)-3,5-dimethylpiperidin-1-yl]-[5-methyl-4-(4-phenylpiperazin-1-yl)thieno[2,3-d]pyrimidin-6-yl]methanone —— C25H31N5OS
[(3S,5S)-3,5-dimethylpiperidin-1-yl]-[5-methyl-4-(4-phenylpiperazin-1-yl)thieno[2,3-d]pyrimidin-6-yl]methanone
—— [4-[4-(2-methoxyphenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidin-6-yl]-[(2R)-2-methylpiperidin-1-yl]methanone —— C25H31N5O2S
[4-[4-(2-methoxyphenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidin-6-yl]-[(2R)-2-methylpiperidin-1-yl]methanone
—— [4-[4-(2-fluorophenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidin-6-yl]-[(2R)-2-methylpiperidin-1-yl]methanone —— C24H28FN5OS
[4-[4-(2-fluorophenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidin-6-yl]-[(2R)-2-methylpiperidin-1-yl]methanone
—— 6-[(3S)-3-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C25H29ClN4O5S
6-[(3S)-3-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— N-[(2S)-butan-2-yl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide —— C23H29N5O2S
N-[(2S)-butan-2-yl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
—— [4-(4-fluorophenyl)piperazin-1-yl]-[(3S)-1-quinolin-8-ylsulfonylpiperidin-3-yl]methanone —— C25H27FN4O3S
[4-(4-fluorophenyl)piperazin-1-yl]-[(3S)-1-quinolin-8-ylsulfonylpiperidin-3-yl]methanone
—— (1R,2R,6S,7S)-4-[3-[4-(3-chlorophenyl)piperazin-1-yl]-3-oxopropyl]-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione —— C22H24ClN3O3
(1R,2R,6S,7S)-4-[3-[4-(3-chlorophenyl)piperazin-1-yl]-3-oxopropyl]-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
—— 6-[(3S)-3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C25H30N4O6S
6-[(3S)-3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one —— C26H32N6O3S
3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C27H32FN5O3S
3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one —— C27H33N5O3S
3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one
—— (2R)-1-acetyl-5-bromo-N-[4-(4-chlorophenyl)piperazin-1-yl]-2-methyl-2,3-dihydroindole-7-sulfonamide —— C21H24BrClN4O3S
(2R)-1-acetyl-5-bromo-N-[4-(4-chlorophenyl)piperazin-1-yl]-2-methyl-2,3-dihydroindole-7-sulfonamide
—— 3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one —— C27H33N5O3S
3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one —— C26H32N6O3S
3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C27H32FN5O3S
3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C27H32FN5O3S
3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— ethyl 5-methoxy-3-{[3-(4-phenylpiperazin-1-yl)propanoyl]amino}-1H-indole-2-carboxylate —— C25H30N4O4
ethyl 5-methoxy-3-{[3-(4-phenylpiperazin-1-yl)propanoyl]amino}-1H-indole-2-carboxylate
—— 4-(5-cyanopyridin-2-yl)-N-(2-thiophen-2-ylethyl)piperazine-1-carboxamide —— C17H19N5OS
4-(5-cyanopyridin-2-yl)-N-(2-thiophen-2-ylethyl)piperazine-1-carboxamide
—— 2-[5-methyl-2-(propan-2-yl)phenoxy]-N-{4-[4-(thiophen-2-ylcarbonyl)piperazin-1-yl]phenyl}acetamide —— C27H31N3O3S
2-[5-methyl-2-(propan-2-yl)phenoxy]-N-{4-[4-(thiophen-2-ylcarbonyl)piperazin-1-yl]phenyl}acetamide
—— 1-(4-Chlorophenoxy)-3-[4-[2-(trifluoromethyl)quinolin-4-yl]piperazin-1-yl]propan-2-ol —— C23H23ClF3N3O2
1-(4-Chlorophenoxy)-3-[4-[2-(trifluoromethyl)quinolin-4-yl]piperazin-1-yl]propan-2-ol
—— 3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one —— C26H32N6O3S
3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-6-(4-pyridin-2-ylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-one
—— N-(4-butyl-2-methylphenyl)-4-(4-methoxyphenyl)-3-methylpiperazine-1-carbothioamide —— C24H33N3OS
N-(4-butyl-2-methylphenyl)-4-(4-methoxyphenyl)-3-methylpiperazine-1-carbothioamide
—— N-(4-bromo-3-methylphenyl)-4-(2-cyanophenyl)piperazine-1-carbothioamide —— C19H19BrN4S
N-(4-bromo-3-methylphenyl)-4-(2-cyanophenyl)piperazine-1-carbothioamide
—— 1-(2-Fluorophenyl)sulfonyl-4-(3-methoxyphenyl)piperazine —— C17H19FN2O3S
1-(2-Fluorophenyl)sulfonyl-4-(3-methoxyphenyl)piperazine
—— [4-(3-chlorophenyl)piperazin-1-yl]-[5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone —— C24H28ClN5OS
[4-(3-chlorophenyl)piperazin-1-yl]-[5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone
—— 3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C27H32FN5O3S
3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 4-(2-Cyanophenyl)piperazine-1-carboxylic acid (3,5-bis-trifluoromethyl-phenyl)-amide —— C20H16F6N4O
4-(2-Cyanophenyl)piperazine-1-carboxylic acid (3,5-bis-trifluoromethyl-phenyl)-amide
—— 3-(4-Chlorophenyl)-1-[4-[4-nitro-2-(trifluoromethyl)phenyl]piperazin-1-yl]prop-2-en-1-one —— C20H17ClF3N3O3
3-(4-Chlorophenyl)-1-[4-[4-nitro-2-(trifluoromethyl)phenyl]piperazin-1-yl]prop-2-en-1-one
—— 6-methyl-5-[(3R)-3-methyl-4-(4-methylphenyl)piperazin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione —— C17H22N4O4S
6-methyl-5-[(3R)-3-methyl-4-(4-methylphenyl)piperazin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione
—— 3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C27H32FN5O3S
3-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-6-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— (2-Prop-2-enylsulfanylpyridin-3-yl)-[4-[4-[4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl]-1,3-thiazol-2-yl]piperidin-1-yl]methanone —— C29H30F3N5O2S2
(2-Prop-2-enylsulfanylpyridin-3-yl)-[4-[4-[4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl]-1,3-thiazol-2-yl]piperidin-1-yl]methanone
—— [2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone —— C26H33N5O2S
[2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone
—— [5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone —— C24H29N5OS
[5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone
—— [2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone —— C25H31N5OS
[2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone
—— [2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone —— C25H31N5OS
[2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone
—— [2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone —— C26H33N5O2S
[2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone
—— [2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone —— C25H30FN5OS
[2,5-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone
—— [2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone —— C25H30FN5OS
[2,5-dimethyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone
—— [5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone —— C24H29N5OS
[5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]-(4-phenylpiperazin-1-yl)methanone
—— [4-(2-fluorophenyl)piperazin-1-yl]-[5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone —— C24H28FN5OS
[4-(2-fluorophenyl)piperazin-1-yl]-[5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone
—— [4-(2-fluorophenyl)piperazin-1-yl]-[5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone —— C24H28FN5OS
[4-(2-fluorophenyl)piperazin-1-yl]-[5-methyl-4-[(2S)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone
—— 1-(2,3-dimethylphenyl)-3-[(E)-[2-oxo-1-[(4-phenylpiperazin-1-yl)methyl]indol-3-ylidene]amino]thiourea —— C28H30N6OS
1-(2,3-dimethylphenyl)-3-[(E)-[2-oxo-1-[(4-phenylpiperazin-1-yl)methyl]indol-3-ylidene]amino]thiourea
—— 1-(4,5-Dibromothiophen-2-yl)sulfonyl-4-(3-methoxyphenyl)piperazine —— C15H16Br2N2O3S2
1-(4,5-Dibromothiophen-2-yl)sulfonyl-4-(3-methoxyphenyl)piperazine
—— 1-(2,3-dimethylphenyl)-3-[(E)-[1-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-2-oxoindol-3-ylidene]amino]thiourea —— C28H29FN6OS
1-(2,3-dimethylphenyl)-3-[(E)-[1-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-2-oxoindol-3-ylidene]amino]thiourea
—— [4-(3-chlorophenyl)piperazin-1-yl]-[5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone —— C24H28ClN5OS
[4-(3-chlorophenyl)piperazin-1-yl]-[5-methyl-4-[(2R)-2-methylpiperidin-1-yl]thieno[2,3-d]pyrimidin-6-yl]methanone
—— 1-[1-(Bicyclo[2.2.1]hept-5-en-2-ylmethyl)piperidin-4-yl]-4-methylpiperazine —— C18H31N3
1-[1-(Bicyclo[2.2.1]hept-5-en-2-ylmethyl)piperidin-4-yl]-4-methylpiperazine
—— 1-[(E)-[1-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-2-oxoindol-3-ylidene]amino]-3-(3-methoxyphenyl)thiourea —— C27H27FN6O2S
1-[(E)-[1-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-2-oxoindol-3-ylidene]amino]-3-(3-methoxyphenyl)thiourea
—— ethyl 3-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propanoyl)amino]-1H-indole-2-carboxylate —— C25H27F3N4O3
ethyl 3-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propanoyl)amino]-1H-indole-2-carboxylate