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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4-[2-oxo-2-(4-pyridin-2-ylpiperazin-1-yl)ethyl]-1,4-benzoxazin-3-one —— C26H33N5O5S
6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4-[2-oxo-2-(4-pyridin-2-ylpiperazin-1-yl)ethyl]-1,4-benzoxazin-3-one
—— N-[(1R,2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide —— C24H28N4O2S
N-[(1R,2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide
—— 3-methyl-6-[(3S)-3-[(3S)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-1,3-benzoxazol-2-one —— C26H32N4O5S
3-methyl-6-[(3S)-3-[(3S)-3-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-1,3-benzoxazol-2-one
—— N-[(1S,2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-2-thiophen-2-ylacetamide —— C24H29N3O2S2
N-[(1S,2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-2-thiophen-2-ylacetamide
—— N'-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(2-morpholin-4-ylethyl)oxamide —— C25H34FN5O3S
N'-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(2-morpholin-4-ylethyl)oxamide
—— 3-(4-chlorophenyl)-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine —— C23H22ClN5O
3-(4-chlorophenyl)-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine
—— N-[(1R,2S)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide —— C23H27N3O3S
N-[(1R,2S)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide
—— N-[(1R,2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide —— C24H28N4O2S
N-[(1R,2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide
—— 3-methyl-6-[(3R)-3-(4-pyrimidin-2-ylpiperazine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3-benzoxazol-2-one —— C22H26N6O5S
3-methyl-6-[(3R)-3-(4-pyrimidin-2-ylpiperazine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3-benzoxazol-2-one
—— N-[(2-methoxyphenyl)methyl]-N'-[(1R,2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide —— C28H34N4O4S
N-[(2-methoxyphenyl)methyl]-N'-[(1R,2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide
—— N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-2-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-2-ylmethyl)oxamide
—— N-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide —— C23H25FN4OS
N-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide
—— N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide
—— N'-[(1R,2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1R,2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide
—— N-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide —— C22H25N3O2S
N-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide
—— 2-fluoro-N-[(1S,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]benzamide —— C24H26FN3OS
2-fluoro-N-[(1S,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]benzamide
—— N-[(1R,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide —— C21H29N3OS
N-[(1R,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide
—— 3-fluoro-N-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]benzamide —— C24H25F2N3OS
3-fluoro-N-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]benzamide
—— N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide
—— N-[2-(dimethylamino)ethyl]-N'-[(1R,2R)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide —— C24H35N5O3S
N-[2-(dimethylamino)ethyl]-N'-[(1R,2R)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide
—— N'-[(1S,2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1S,2R)-1-[4-(4-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide
—— [(3R)-1-(1H-imidazol-5-ylsulfonyl)piperidin-3-yl]-[4-(2-methoxyphenyl)piperazin-1-yl]methanone —— C20H27N5O4S
[(3R)-1-(1H-imidazol-5-ylsulfonyl)piperidin-3-yl]-[4-(2-methoxyphenyl)piperazin-1-yl]methanone
—— N-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide —— C23H25FN4OS
N-[(1R,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]pyridine-3-carboxamide
—— N-[2-(diethylamino)ethyl]-N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide —— C25H36FN5O2S
N-[2-(diethylamino)ethyl]-N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide
—— N-[(1R,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide —— C22H25N3O2S
N-[(1R,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]furan-2-carboxamide
—— ethyl (4R)-4-(2,3-dimethoxyphenyl)-6-[[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H36N4O5
ethyl (4R)-4-(2,3-dimethoxyphenyl)-6-[[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(1R,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide —— C21H29N3OS
N-[(1R,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide
—— ethyl (4S)-4-(2,3-dimethoxyphenyl)-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H31N5O7
ethyl (4S)-4-(2,3-dimethoxyphenyl)-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(4-methoxyphenyl)methyl]-N'-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide —— C27H32N4O3S
N-[(4-methoxyphenyl)methyl]-N'-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide
—— 1-[5-[(1R)-1-hydroxy-2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]-2,3-dihydroindol-1-yl]ethanone —— C23H29N3O3
1-[5-[(1R)-1-hydroxy-2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]-2,3-dihydroindol-1-yl]ethanone
—— (1S)-1-(2,3-dihydro-1H-indol-5-yl)-2-[4-(4-nitrophenyl)piperazin-1-yl]ethanol —— C20H24N4O3
(1S)-1-(2,3-dihydro-1H-indol-5-yl)-2-[4-(4-nitrophenyl)piperazin-1-yl]ethanol
—— N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-2-ylmethyl)oxamide —— C25H28FN5O2S
N'-[(1S,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-2-ylmethyl)oxamide
—— ethyl (4R)-6-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-4-(2,3-dimethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H31ClN4O5
ethyl (4R)-6-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-4-(2,3-dimethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(4-methoxyphenyl)methyl]-N'-[(1R,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide —— C27H32N4O3S
N-[(4-methoxyphenyl)methyl]-N'-[(1R,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide
—— 1-[5-[(1S)-1-hydroxy-2-[4-(4-nitrophenyl)piperazin-1-yl]ethyl]-2,3-dihydroindol-1-yl]ethanone —— C22H26N4O4
1-[5-[(1S)-1-hydroxy-2-[4-(4-nitrophenyl)piperazin-1-yl]ethyl]-2,3-dihydroindol-1-yl]ethanone
—— (E)-3-[4-(difluoromethoxy)phenyl]-1-(4-pyrimidin-2-ylpiperazin-1-yl)prop-2-en-1-one —— C18H18F2N4O2
(E)-3-[4-(difluoromethoxy)phenyl]-1-(4-pyrimidin-2-ylpiperazin-1-yl)prop-2-en-1-one
—— N-[(4-fluorophenyl)methyl]-N'-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide —— C26H29FN4O2S
N-[(4-fluorophenyl)methyl]-N'-[(1S,2S)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]oxamide
—— ethyl (4R)-4-(2,3-dimethoxyphenyl)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H36N4O5
ethyl (4R)-4-(2,3-dimethoxyphenyl)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-oxo-N-[(2S)-1-oxo-3-phenyl-1-(4-phenylpiperazin-1-yl)propan-2-yl]-3,4-dihydro-1H-quinoline-6-sulfonamide —— C28H30N4O4S
2-oxo-N-[(2S)-1-oxo-3-phenyl-1-(4-phenylpiperazin-1-yl)propan-2-yl]-3,4-dihydro-1H-quinoline-6-sulfonamide
—— 2-oxo-N-[(2R)-1-oxo-3-phenyl-1-(4-phenylpiperazin-1-yl)propan-2-yl]-3,4-dihydro-1H-quinoline-6-sulfonamide —— C28H30N4O4S
2-oxo-N-[(2R)-1-oxo-3-phenyl-1-(4-phenylpiperazin-1-yl)propan-2-yl]-3,4-dihydro-1H-quinoline-6-sulfonamide
—— (E)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-3-thiophen-2-ylprop-2-en-1-one —— C18H20N2O2S
(E)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-3-thiophen-2-ylprop-2-en-1-one
—— (E)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-(3-fluorophenyl)prop-2-en-1-one —— C19H18ClFN2O
(E)-1-[4-(3-chlorophenyl)piperazin-1-yl]-3-(3-fluorophenyl)prop-2-en-1-one
—— ethyl (4S)-6-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-4-(2,3-dimethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H31ClN4O5
ethyl (4S)-6-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-4-(2,3-dimethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(2,3-dimethoxyphenyl)-6-[[4-(3-methoxyphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H34N4O6
ethyl (4S)-4-(2,3-dimethoxyphenyl)-6-[[4-(3-methoxyphenyl)piperazin-1-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(2S)-1-(2,1,3-benzothiadiazol-4-ylsulfonyl)pyrrolidin-2-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone —— C20H22N6O3S2
[(2S)-1-(2,1,3-benzothiadiazol-4-ylsulfonyl)pyrrolidin-2-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone
—— N'-[(1S,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(2-morpholin-4-ylethyl)oxamide —— C25H34FN5O3S
N'-[(1S,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(2-morpholin-4-ylethyl)oxamide
—— 3-methyl-2-oxo-N-[(2R)-1-oxo-3-phenyl-1-(4-pyridin-2-ylpiperazin-1-yl)propan-2-yl]-1,3-benzoxazole-6-sulfonamide —— C26H27N5O5S
3-methyl-2-oxo-N-[(2R)-1-oxo-3-phenyl-1-(4-pyridin-2-ylpiperazin-1-yl)propan-2-yl]-1,3-benzoxazole-6-sulfonamide
—— N-[(1S,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide —— C21H29N3OS
N-[(1S,2R)-1-(4-phenylpiperazin-1-yl)-1-thiophen-2-ylpropan-2-yl]butanamide
—— N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-[(2-methoxyphenyl)methyl]oxamide —— C27H31FN4O3S
N'-[(1R,2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-[(2-methoxyphenyl)methyl]oxamide
—— N-[2-(dimethylamino)ethyl]-N'-[(1S,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide —— C23H32FN5O2S
N-[2-(dimethylamino)ethyl]-N'-[(1S,2S)-1-[4-(2-fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide