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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-1-(4-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-ethoxyphenyl)acetamide —— C32H36ClN5O3S
2-[(4R)-1-(4-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-ethoxyphenyl)acetamide
—— N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methylsulfanylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C31H33ClFN5O2S2
N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methylsulfanylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— N-[(2R)-1-[4-(2-chlorophenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C23H24ClN3O3S2
N-[(2R)-1-[4-(2-chlorophenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— N-(4-ethoxyphenyl)-2-[(4R)-1-(4-methylphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide —— C33H39N5O3S
N-(4-ethoxyphenyl)-2-[(4R)-1-(4-methylphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide
—— N-[(2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C24H27N3O4S2
N-[(2S)-1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— 3-(2-methoxyethyl)-7-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-quinazoline-2,4-dione —— C24H28N4O4
3-(2-methoxyethyl)-7-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-quinazoline-2,4-dione
—— N-[(2S)-1-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C24H26ClN3O3S2
N-[(2S)-1-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— 2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide —— C34H40FN5O3S
2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide
—— (4S,5R)-1,5-bis(4-methoxyphenyl)-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one —— C30H33N3O5
(4S,5R)-1,5-bis(4-methoxyphenyl)-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
—— 2-[(4R)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-methoxyphenyl)acetamide —— C31H34ClN5O3S
2-[(4R)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-methoxyphenyl)acetamide
—— 2-[(4S)-1-(4-ethoxyphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide —— C35H43N5O4S
2-[(4S)-1-(4-ethoxyphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide
—— N-(4-chlorophenyl)-2-[(4R)-1-(4-chlorophenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C30H30Cl2FN5O2S
N-(4-chlorophenyl)-2-[(4R)-1-(4-chlorophenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— N-(4-ethoxyphenyl)-2-[(4S)-1-(4-methylphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide —— C33H39N5O3S
N-(4-ethoxyphenyl)-2-[(4S)-1-(4-methylphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide
—— (2S)-1-acetyl-5-bromo-N-[3-[4-(2-fluorophenyl)piperazin-1-yl]propyl]-2-methyl-2,3-dihydroindole-7-sulfonamide —— C24H30BrFN4O3S
(2S)-1-acetyl-5-bromo-N-[3-[4-(2-fluorophenyl)piperazin-1-yl]propyl]-2-methyl-2,3-dihydroindole-7-sulfonamide
—— (3R,4R)-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one —— C29H29FN4O6
(3R,4R)-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-4-[4-(4-nitrophenyl)piperazine-1-carbonyl]-3,4-dihydroisoquinolin-1-one
—— N-(4-methoxyphenyl)-2-[(4R)-1-(3-methoxyphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide —— C32H37N5O4S
N-(4-methoxyphenyl)-2-[(4R)-1-(3-methoxyphenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]acetamide
—— 5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one —— C26H32FN5O4S2
5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-3-[2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-6-methylthieno[2,3-d]pyrimidin-4-one
—— N-(4-chlorophenyl)-2-[(4S)-1-(3-chlorophenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C30H30Cl2FN5O2S
N-(4-chlorophenyl)-2-[(4S)-1-(3-chlorophenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— (4S,5R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,5-bis(4-methoxyphenyl)pyrrolidin-2-one —— C29H30FN3O4
(4S,5R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,5-bis(4-methoxyphenyl)pyrrolidin-2-one
—— 2-[(4S)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide —— C33H38ClN5O3S
2-[(4S)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-propoxyphenyl)acetamide
—— (4S,5R)-1,5-bis(4-methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one —— C30H33N3O5
(4S,5R)-1,5-bis(4-methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
—— (3S,4R)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one —— C30H32FN3O4S
(3S,4R)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one
—— N-(4-chlorophenyl)-2-[(4S)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methylsulfanylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C31H33ClFN5O2S2
N-(4-chlorophenyl)-2-[(4S)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(3-methylsulfanylphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— 2-[(4R)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-ethoxyphenyl)acetamide —— C32H36ClN5O3S
2-[(4R)-1-(3-chlorophenyl)-5-oxo-3-[3-(4-phenylpiperazin-1-yl)propyl]-2-sulfanylideneimidazolidin-4-yl]-N-(4-ethoxyphenyl)acetamide
—— 2-[(4R)-1-(4-ethoxyphenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]-N-(4-methoxyphenyl)acetamide —— C33H38FN5O4S
2-[(4R)-1-(4-ethoxyphenyl)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-5-oxo-2-sulfanylideneimidazolidin-4-yl]-N-(4-methoxyphenyl)acetamide
—— N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methoxyphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide —— C31H33ClFN5O3S
N-(4-chlorophenyl)-2-[(4R)-3-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-1-(4-methoxyphenyl)-5-oxo-2-sulfanylideneimidazolidin-4-yl]acetamide
—— (4R,5R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,5-bis(4-methoxyphenyl)pyrrolidin-2-one —— C29H30FN3O4
(4R,5R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,5-bis(4-methoxyphenyl)pyrrolidin-2-one
—— N-[(2R)-1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide —— C25H29N3O3S2
N-[(2R)-1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-1-oxo-3-phenylpropan-2-yl]thiophene-2-sulfonamide
—— (3S,4S)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one —— C31H35N3O5S
(3S,4S)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-(4-methylsulfanylphenyl)-3,4-dihydroisoquinolin-1-one
—— [(2R)-1-(4-tert-butylphenyl)sulfonylpiperidin-2-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone —— C26H34FN3O3S
[(2R)-1-(4-tert-butylphenyl)sulfonylpiperidin-2-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone
—— (3R,4R)-3-(2-fluorophenyl)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3,4-dihydroisoquinolin-1-one —— C30H32FN3O5
(3R,4R)-3-(2-fluorophenyl)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3,4-dihydroisoquinolin-1-one
—— (3R,4R)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one —— C27H28FN3O4S
(3R,4R)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one
—— (5S,6R)-1-(1,3-benzodioxol-5-yl)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)piperidin-2-one —— C30H30FN3O5
(5S,6R)-1-(1,3-benzodioxol-5-yl)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)piperidin-2-one
—— (3R,4R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one —— C27H28FN3O4S
(3R,4R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one
—— (3R,4R)-N-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-1-oxo-3,4-dihydroisoquinoline-4-carboxamide —— C32H36ClFN4O4
(3R,4R)-N-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-1-oxo-3,4-dihydroisoquinoline-4-carboxamide
—— (3R,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-3,4-dihydroisoquinolin-1-one —— C29H29ClFN3O4
(3R,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-3-(2-fluorophenyl)-6,7-dimethoxy-2-methyl-3,4-dihydroisoquinolin-1-one
—— (3R,4S)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one —— C27H28FN3O4S
(3R,4S)-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one
—— (3R,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one —— C27H28ClN3O4S
(3R,4S)-4-[4-(3-chlorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-thiophen-2-yl-3,4-dihydroisoquinolin-1-one
—— 1-[(2R)-5-bromo-7-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone —— C21H23BrClN3O3S
1-[(2R)-5-bromo-7-[4-(3-chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone
—— 2-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-{(Z)-[3-(2-methylpropyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one —— C28H29N5O4S2
2-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-{(Z)-[3-(2-methylpropyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
—— (3S,4R)-6,7-dimethoxy-2-methyl-3-pyridin-3-yl-4-(4-pyridin-2-ylpiperazine-1-carbonyl)-3,4-dihydroisoquinolin-1-one —— C27H29N5O4
(3S,4R)-6,7-dimethoxy-2-methyl-3-pyridin-3-yl-4-(4-pyridin-2-ylpiperazine-1-carbonyl)-3,4-dihydroisoquinolin-1-one
—— 3-[(1-acetyl-5-bromo-2,3-dihydroindol-7-yl)sulfonyl]-1-[(3R)-3-methyl-4-(4-methylphenyl)piperazin-1-yl]propan-1-one —— C25H30BrN3O4S
3-[(1-acetyl-5-bromo-2,3-dihydroindol-7-yl)sulfonyl]-1-[(3R)-3-methyl-4-(4-methylphenyl)piperazin-1-yl]propan-1-one
—— (3S,4R)-6,7-dimethoxy-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one —— C29H32N4O5
(3S,4R)-6,7-dimethoxy-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one
—— (E)-N-[4-[4-(2-methylpropanoyl)piperazin-1-yl]phenyl]-3-(3-nitrophenyl)prop-2-enamide —— C23H26N4O4
(E)-N-[4-[4-(2-methylpropanoyl)piperazin-1-yl]phenyl]-3-(3-nitrophenyl)prop-2-enamide
—— (3S,4S)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one —— C29H32N4O5
(3S,4S)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one
—— (5R,6R)-1-(1,3-benzodioxol-5-yl)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)piperidin-2-one —— C30H30FN3O5
(5R,6R)-1-(1,3-benzodioxol-5-yl)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)piperidin-2-one
—— 1-[(2R)-5-bromo-7-[4-(2-chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone —— C21H23BrClN3O3S
1-[(2R)-5-bromo-7-[4-(2-chlorophenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone
—— (3S,4R)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one —— C29H32N4O5
(3S,4R)-6,7-dimethoxy-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one
—— 1-[(2S)-5-bromo-7-[4-(2,5-dimethylphenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone —— C23H28BrN3O3S
1-[(2S)-5-bromo-7-[4-(2,5-dimethylphenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]ethanone
—— (3S,4R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one —— C28H29FN4O4
(3S,4R)-4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6,7-dimethoxy-2-methyl-3-pyridin-3-yl-3,4-dihydroisoquinolin-1-one