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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-4-[4-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)phenyl]piperazine-1-carbonyl]-1-(4-methylphenyl)pyrrolidin-2-one —— C26H29N5O3
(4S)-4-[4-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)phenyl]piperazine-1-carbonyl]-1-(4-methylphenyl)pyrrolidin-2-one
—— 5-(methanesulfonamido)-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]benzoic acid —— C20H25N3O4S
5-(methanesulfonamido)-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]benzoic acid
—— (4S)-4-[4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one —— C24H25N5O3
(4S)-4-[4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one
—— 5-(methanesulfonamido)-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C19H24N4O4S
5-(methanesulfonamido)-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— 5-[(3,5-dimethylphenyl)sulfonylamino]-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C26H30N4O4S
5-[(3,5-dimethylphenyl)sulfonylamino]-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— (7R)-2-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H32N4O2S
(7R)-2-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 5-(benzenesulfonamido)-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C24H26N4O4S
5-(benzenesulfonamido)-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— N-[(2R)-1-[4-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)phenyl]piperazin-1-yl]-1-oxopropan-2-yl]-4-methylbenzenesulfonamide —— C24H29N5O4S
N-[(2R)-1-[4-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)phenyl]piperazin-1-yl]-1-oxopropan-2-yl]-4-methylbenzenesulfonamide
—— (7R)-2-[3-[4-(3-methoxyphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H30N4O3S
(7R)-2-[3-[4-(3-methoxyphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 5-(methanesulfonamido)-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C19H24N4O4S
5-(methanesulfonamido)-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— 5-(benzenesulfonamido)-6-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C24H26N4O4S
5-(benzenesulfonamido)-6-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— 5-[(3-fluorophenyl)sulfonylamino]-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C24H25FN4O4S
5-[(3-fluorophenyl)sulfonylamino]-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— (7S)-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H27FN4O2S
(7S)-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-(4-methylpiperidin-1-yl)sulfonylquinoline —— C27H34N4O2S
2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-6-(4-methylpiperidin-1-yl)sulfonylquinoline
—— (7R)-2-[3-[4-(4-methoxyphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H30N4O3S
(7R)-2-[3-[4-(4-methoxyphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 5-[(4-fluorophenyl)sulfonylamino]-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid —— C24H25FN4O4S
5-[(4-fluorophenyl)sulfonylamino]-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]pyridine-3-carboxylic acid
—— (7R)-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H27FN4O2S
(7R)-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-tert-butyl-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H33FN4O2S
(7R)-7-tert-butyl-2-[3-[4-(2-fluorophenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H32N4O2S
(7S)-2-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H29ClN4O2S
(7R)-2-[3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-[(3-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid —— C25H28N4O4S
2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-[(3-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid
—— (6S)-N-cyclopentyl-5-ethyl-2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O4
(6S)-N-cyclopentyl-5-ethyl-2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-butyl-N-cyclopentyl-6-methyl-4-oxo-2-(4-pyridin-2-ylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H37N7O3
(6S)-5-butyl-N-cyclopentyl-6-methyl-4-oxo-2-(4-pyridin-2-ylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclopentyl-6-methyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O3
(6R)-N-cyclopentyl-6-methyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-butyl-N-cyclopentyl-2-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H40N6O4
(6S)-5-butyl-N-cyclopentyl-2-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H33FN6O3
(6S)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— N-[(Z)-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylideneamino]pyridine-3-carboxamide —— C18H20N6O3
N-[(Z)-[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylideneamino]pyridine-3-carboxamide
—— (6S)-N-cycloheptyl-5,6-dimethyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O3
(6S)-N-cycloheptyl-5,6-dimethyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (E)-ethyl 4-(5-(2-(benzo[d]thiazol-2-yl)-2-cyanovinyl)furan-2-yl)piperazine-1-carboxylate —— C21H20N4O3S
(E)-ethyl 4-(5-(2-(benzo[d]thiazol-2-yl)-2-cyanovinyl)furan-2-yl)piperazine-1-carboxylate
—— (6R)-N-cyclopentyl-5,6-dimethyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H32N6O3
(6R)-N-cyclopentyl-5,6-dimethyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclopentyl-2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O3
(6S)-N-cyclopentyl-2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (5Z)-5-(2,4-diethoxybenzylidene)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione —— C26H29N3O5S
(5Z)-5-(2,4-diethoxybenzylidene)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,3-thiazolidine-2,4-dione
—— (6S)-N-cyclopentyl-2-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H31FN6O3
(6S)-N-cyclopentyl-2-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (3S)-3-[(1-acetyl-2,3-dihydroindol-5-yl)sulfonyl]-1-[4-(3-chlorophenyl)piperazin-1-yl]butan-1-one —— C24H28ClN3O4S
(3S)-3-[(1-acetyl-2,3-dihydroindol-5-yl)sulfonyl]-1-[4-(3-chlorophenyl)piperazin-1-yl]butan-1-one
—— 1-[[4-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]phenyl]methyl]pyrido[2,3-b][1,4]thiazin-2-one —— C27H28N4O2S
1-[[4-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]phenyl]methyl]pyrido[2,3-b][1,4]thiazin-2-one
—— (3S)-3-[(1-acetyl-2,3-dihydroindol-5-yl)sulfonyl]-1-[4-(2,4-dimethylphenyl)piperazin-1-yl]butan-1-one —— C26H33N3O4S
(3S)-3-[(1-acetyl-2,3-dihydroindol-5-yl)sulfonyl]-1-[4-(2,4-dimethylphenyl)piperazin-1-yl]butan-1-one
—— (2R)-N-cyclohexyl-1-(3,5-dimethoxyphenyl)-4-ethylsulfonyl-2-methyl-6-oxopiperazine-2-carboxamide —— C22H33N3O6S
(2R)-N-cyclohexyl-1-(3,5-dimethoxyphenyl)-4-ethylsulfonyl-2-methyl-6-oxopiperazine-2-carboxamide
—— (2R)-1-(5-chloro-2-methoxyphenyl)-N-cyclohexyl-4-ethylsulfonyl-2-methyl-6-oxopiperazine-2-carboxamide —— C21H30ClN3O5S
(2R)-1-(5-chloro-2-methoxyphenyl)-N-cyclohexyl-4-ethylsulfonyl-2-methyl-6-oxopiperazine-2-carboxamide
—— (2S)-4-(benzenesulfonyl)-N-cyclopentyl-1-(4-ethylphenyl)-2-methyl-6-oxopiperazine-2-carboxamide —— C25H31N3O4S
(2S)-4-(benzenesulfonyl)-N-cyclopentyl-1-(4-ethylphenyl)-2-methyl-6-oxopiperazine-2-carboxamide
—— (2S)-N-cyclohexyl-1-(2,4-dimethoxyphenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C21H31N3O6S
(2S)-N-cyclohexyl-1-(2,4-dimethoxyphenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide
—— cyclobutyl-[(2S)-5-[4-(2,4-dimethylphenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]methanone —— C26H33N3O3S
cyclobutyl-[(2S)-5-[4-(2,4-dimethylphenyl)piperazin-1-yl]sulfonyl-2-methyl-2,3-dihydroindol-1-yl]methanone
—— (2R)-1-(5-chloro-2,4-dimethoxyphenyl)-N-cyclopentyl-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C20H28ClN3O6S
(2R)-1-(5-chloro-2,4-dimethoxyphenyl)-N-cyclopentyl-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide
—— (2S)-N-cyclohexyl-1-(2,3-dimethylphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide —— C23H35N3O4S
(2S)-N-cyclohexyl-1-(2,3-dimethylphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide
—— (2R)-N-cyclopentyl-1-(3,5-dimethylphenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C20H29N3O4S
(2R)-N-cyclopentyl-1-(3,5-dimethylphenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide
—— (2S)-4-(benzenesulfonyl)-2-methyl-1-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-6-oxopiperazine-2-carboxamide —— C27H29N3O4S
(2S)-4-(benzenesulfonyl)-2-methyl-1-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-6-oxopiperazine-2-carboxamide
—— (2S)-N-cyclohexyl-1-(2,4-dimethoxyphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide —— C23H35N3O6S
(2S)-N-cyclohexyl-1-(2,4-dimethoxyphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide
—— (2R)-N-cyclohexyl-1-(2,4-difluorophenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C19H25F2N3O4S
(2R)-N-cyclohexyl-1-(2,4-difluorophenyl)-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide
—— (2R)-1-(4-chloro-2-methylphenyl)-N-cyclohexyl-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C20H28ClN3O4S
(2R)-1-(4-chloro-2-methylphenyl)-N-cyclohexyl-2-methyl-4-methylsulfonyl-6-oxopiperazine-2-carboxamide
—— (2R)-N-cyclohexyl-1-(3,5-dimethoxyphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide —— C23H35N3O6S
(2R)-N-cyclohexyl-1-(3,5-dimethoxyphenyl)-2-methyl-6-oxo-4-propylsulfonylpiperazine-2-carboxamide
—— (2R)-N-cyclopentyl-2-methyl-1-(4-methylphenyl)-4-methylsulfonyl-6-oxopiperazine-2-carboxamide —— C19H27N3O4S
(2R)-N-cyclopentyl-2-methyl-1-(4-methylphenyl)-4-methylsulfonyl-6-oxopiperazine-2-carboxamide