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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone —— C21H28F3N3O2
1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone
—— 2-[4-[2-(4-bromo-2-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C20H27BrFN3O3
2-[4-[2-(4-bromo-2-fluorophenoxy)acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 3-(4-methylphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one —— C22H33N3O2
3-(4-methylphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one
—— 1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone —— C21H28F3N3O2
1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone
—— 2-[4-(1-benzylpyrrole-2-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C24H32N4O2
2-[4-(1-benzylpyrrole-2-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C23H32ClN3O4
2-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 3-(4-methylphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one —— C22H33N3O2
3-(4-methylphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one
—— 2-[4-(1-benzylpyrrole-2-carbonyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C24H32N4O2
2-[4-(1-benzylpyrrole-2-carbonyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— [(5S,7R)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone —— C26H37N3O4S
[(5S,7R)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone
—— 1-[(2S)-2-methylpiperidin-1-yl]-2-[4-[2-[2-(methylsulfanylmethyl)benzimidazol-1-yl]acetyl]piperazin-1-yl]ethanone —— C23H33N5O2S
1-[(2S)-2-methylpiperidin-1-yl]-2-[4-[2-[2-(methylsulfanylmethyl)benzimidazol-1-yl]acetyl]piperazin-1-yl]ethanone
—— 2-[4-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C23H35N3O2S
2-[4-(4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-2-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-[1-(4-bromophenyl)cyclobutanecarbonyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C23H32BrN3O2
2-[4-[1-(4-bromophenyl)cyclobutanecarbonyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-(4-methylphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C21H31N3O2
2-(4-methylphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 3-(3-bromo-4-methoxyphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one —— C22H32BrN3O3
3-(3-bromo-4-methoxyphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one
—— 3-(3-bromo-4-methoxyphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one —— C22H32BrN3O3
3-(3-bromo-4-methoxyphenyl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]propan-1-one
—— 2-(1,2-benzoxazol-3-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C21H28N4O3
2-(1,2-benzoxazol-3-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 2-(4-methylphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C21H31N3O2
2-(4-methylphenyl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 5-(1,3-benzothiazol-2-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pentan-1-one —— C24H34N4O2S
5-(1,3-benzothiazol-2-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pentan-1-one
—— 2-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C23H32ClN3O4
2-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 2-(1,2-benzoxazol-3-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C21H28N4O3
2-(1,2-benzoxazol-3-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 5-(1,3-benzothiazol-2-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pentan-1-one —— C24H34N4O2S
5-(1,3-benzothiazol-2-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pentan-1-one
—— [(5S,7S)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone —— C26H37N3O4S
[(5S,7S)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone
—— [(5R,7R)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone —— C26H37N3O4S
[(5R,7R)-3-(4-methylphenyl)-1-adamantyl]-(4-morpholin-4-ylsulfonylpiperazin-1-yl)methanone
—— 2-[4-[2-[4-(1,3-dithian-2-yl)phenoxy]acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C24H35N3O3S2
2-[4-[2-[4-(1,3-dithian-2-yl)phenoxy]acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-[2-[4-(1,3-dithian-2-yl)phenoxy]acetyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C24H35N3O3S2
2-[4-[2-[4-(1,3-dithian-2-yl)phenoxy]acetyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-[2-[(4-methylphenyl)methylsulfanyl]acetyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C22H33N3O2S
2-[4-[2-[(4-methylphenyl)methylsulfanyl]acetyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-[2-[(4-methylphenyl)methylsulfanyl]acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C22H33N3O2S
2-[4-[2-[(4-methylphenyl)methylsulfanyl]acetyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 2-(6,7-dimethyl-1-benzofuran-3-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C24H33N3O3
2-(6,7-dimethyl-1-benzofuran-3-yl)-1-[4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— 1-[4-[4-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-nitrophenyl]piperazin-1-yl]ethanone —— C23H25FN4O5
1-[4-[4-[(2S)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-nitrophenyl]piperazin-1-yl]ethanone
—— 2-[4-(3,4-dipropoxybenzoyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C25H39N3O4
2-[4-(3,4-dipropoxybenzoyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-(3,4-dipropoxybenzoyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C25H39N3O4
2-[4-(3,4-dipropoxybenzoyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 1-[4-[4-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-nitrophenyl]piperazin-1-yl]ethanone —— C23H25FN4O5
1-[4-[4-[(2R)-2-(4-fluorophenyl)morpholine-4-carbonyl]-2-nitrophenyl]piperazin-1-yl]ethanone
—— 2-[4-(2-ethoxypyridine-3-carbonyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C20H30N4O3
2-[4-(2-ethoxypyridine-3-carbonyl)piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 2-[4-(2-ethoxypyridine-3-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C20H30N4O3
2-[4-(2-ethoxypyridine-3-carbonyl)piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-(6,7-dimethyl-1-benzofuran-3-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone —— C24H33N3O3
2-(6,7-dimethyl-1-benzofuran-3-yl)-1-[4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]piperazin-1-yl]ethanone
—— [1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone —— C28H33N5O4S
[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone
—— [4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C31H38N4O4S
[4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [4-(3-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C30H36N4O5S
[4-(3-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C30H36N4O5S
[4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-phenylpiperazin-1-yl)methanone —— C29H34N4O4S
[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-phenylpiperazin-1-yl)methanone
—— [4-(5-chloro-2-methylphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C30H35ClN4O4S
[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone —— C28H30F2N4O4S
[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone
—— [1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone —— C28H30F2N4O4S
[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(2-fluorophenyl)piperazin-1-yl]methanone
—— [4-(2-fluorophenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C29H33FN4O4S
[4-(2-fluorophenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(4-methylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C30H35FN4O4S
[4-(2,5-dimethylphenyl)piperazin-1-yl]-[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(3-methoxyphenyl)piperazin-1-yl]methanone —— C29H33FN4O5S
[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-[4-(3-methoxyphenyl)piperazin-1-yl]methanone
—— [4-(3-chlorophenyl)piperazin-1-yl]-[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C28H30ClFN4O4S
[4-(3-chlorophenyl)piperazin-1-yl]-[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-phenylpiperazin-1-yl)methanone —— C28H31FN4O4S
[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-phenylpiperazin-1-yl)methanone
—— [4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(2,4,6-trimethylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone —— C32H40N4O5S
[4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[3-methyl-5-[(Z)-2-(2,4,6-trimethylphenyl)ethenyl]-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]methanone
—— [1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone —— C27H30FN5O4S
[1-[[5-[(Z)-2-(2-fluorophenyl)ethenyl]-3-methyl-1,2-oxazol-4-yl]sulfonyl]piperidin-4-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone