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二嗪烷类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4-(2-fluorophenyl)piperazin-1-yl]-2-[[(1R)-1-(2-methoxyphenyl)ethyl]-methylamino]ethanone —— C22H28FN3O2
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-[[(1R)-1-(2-methoxyphenyl)ethyl]-methylamino]ethanone
—— (2S)-2-[4-[[5-(3-fluorophenyl)thiophen-2-yl]methyl]piperazin-1-yl]-1-morpholin-4-ylpropan-1-one —— C22H28FN3O2S
(2S)-2-[4-[[5-(3-fluorophenyl)thiophen-2-yl]methyl]piperazin-1-yl]-1-morpholin-4-ylpropan-1-one
—— N-[(2R)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propyl]-4-pyrimidin-2-ylpiperazine-1-carboxamide —— C18H30N6O2
N-[(2R)-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propyl]-4-pyrimidin-2-ylpiperazine-1-carboxamide
—— (2R)-2-[4-[[5-(3-fluorophenyl)thiophen-2-yl]methyl]piperazin-1-yl]-1-morpholin-4-ylpropan-1-one —— C22H28FN3O2S
(2R)-2-[4-[[5-(3-fluorophenyl)thiophen-2-yl]methyl]piperazin-1-yl]-1-morpholin-4-ylpropan-1-one
—— N-cyclohexyl-4-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide —— C21H34N4O3S2
N-cyclohexyl-4-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide
—— 1-[4-[5-[3-[2-(3,4-Dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-oxopropyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]-2-methylguanidine —— C35H41Cl2N7O2
1-[4-[5-[3-[2-(3,4-Dichlorophenyl)-4-(3,5-dimethylbenzoyl)piperazin-1-yl]-3-oxopropyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]-2-methylguanidine
—— N-cyclohexyl-4-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide —— C21H34N4O3S2
N-cyclohexyl-4-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide
—— 1-Oxido-7-[12-(1-oxido-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ium-7-yl)-3,12-diaza-6,9-diazoniadispiro[5.2.59.26]hexadecan-3-yl]-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ium;dichloride —— C20H26Cl2N12O4
1-Oxido-7-[12-(1-oxido-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ium-7-yl)-3,12-diaza-6,9-diazoniadispiro[5.2.59.26]hexadecan-3-yl]-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ium;dichloride
—— N-[(2R)-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propyl]-4-pyrimidin-2-ylpiperazine-1-carboxamide —— C18H30N6O2
N-[(2R)-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propyl]-4-pyrimidin-2-ylpiperazine-1-carboxamide
—— 1-[4-(2-fluorophenyl)piperazin-1-yl]-2-[[(1S)-1-(2-methoxyphenyl)ethyl]-methylamino]ethanone —— C22H28FN3O2
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-[[(1S)-1-(2-methoxyphenyl)ethyl]-methylamino]ethanone
—— (2S)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C24H26F3N3O2
(2S)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— (2S)-2-phenyl-1-piperidin-1-yl-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]ethanone —— C25H28F3N3O2
(2S)-2-phenyl-1-piperidin-1-yl-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]ethanone
—— 1-(5-methyl-1,2-oxazol-3-yl)-3-[2-[(2R)-4-methyl-2-phenylpiperazin-1-yl]ethyl]urea —— C18H25N5O2
1-(5-methyl-1,2-oxazol-3-yl)-3-[2-[(2R)-4-methyl-2-phenylpiperazin-1-yl]ethyl]urea
—— 4-[3,6-bis(diethylamino)pyridin-2-yl]-N-[4-(2,3-dihydroxyphenyl)-1,3-thiazol-2-yl]piperazine-1-carboxamide —— C27H37N7O3S
4-[3,6-bis(diethylamino)pyridin-2-yl]-N-[4-(2,3-dihydroxyphenyl)-1,3-thiazol-2-yl]piperazine-1-carboxamide
—— (2S)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C24H26F3N3O2
(2S)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— N-(cyclohexanecarbonyl)-N-[1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-phenylpropan-2-yl]cyclohexanecarboxamide —— C34H47N3O3
N-(cyclohexanecarbonyl)-N-[1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-phenylpropan-2-yl]cyclohexanecarboxamide
—— (2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C22H24F3N3O2S
(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— (2R)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C24H26F3N3O2
(2R)-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— tert-butyl 4-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate —— C23H35N3O4
tert-butyl 4-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate
—— 3-(4-methylphenyl)-5-[(1R)-1-[4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C27H26N6OS
3-(4-methylphenyl)-5-[(1R)-1-[4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— (2R)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C24H26F3N3O2
(2R)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— 3-(4-methylphenyl)-5-[(1S)-1-[4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C27H26N6OS
3-(4-methylphenyl)-5-[(1S)-1-[4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— (2S)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-2-methyl-3-[3-thieno[2,3-d]isoxazol-3-yl-phenoxy]propan-2-ol —— C26H29N3O4S
(2S)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-2-methyl-3-[3-thieno[2,3-d]isoxazol-3-yl-phenoxy]propan-2-ol
—— N-{(S)-2-Hydroxy-3-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-propyl}-2-p-tolyloxy-nicotinamide —— C29H36N4O4
N-{(S)-2-Hydroxy-3-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-propyl}-2-p-tolyloxy-nicotinamide
—— (2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one —— C22H24F3N3O2S
(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]propan-1-one
—— 3,5-dimethyl-4-[(2R)-4-methyl-2-phenylpiperazin-1-yl]sulfonyl-1,2-oxazole —— C16H21N3O3S
3,5-dimethyl-4-[(2R)-4-methyl-2-phenylpiperazin-1-yl]sulfonyl-1,2-oxazole
—— 5-[(1R)-1-[4-(6-tert-butylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperazin-1-yl]ethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole —— C23H29N7OS
5-[(1R)-1-[4-(6-tert-butylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperazin-1-yl]ethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole
—— (2R)-2-phenyl-1-piperidin-1-yl-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]ethanone —— C25H28F3N3O2
(2R)-2-phenyl-1-piperidin-1-yl-2-[4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl]ethanone
—— tert-butyl 4-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate —— C23H35N3O4
tert-butyl 4-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate
—— 2-[2-propoxy-5-(4-pyridin-2-ylpiperazin-1-yl)sulfonylphenyl]-7-propyl-1H-purin-6-one —— C26H31N7O4S
2-[2-propoxy-5-(4-pyridin-2-ylpiperazin-1-yl)sulfonylphenyl]-7-propyl-1H-purin-6-one
—— N-cyclohexyl-4-[(1R)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl]-N-methylpiperazine-1-sulfonamide —— C21H31F2N5O2S
N-cyclohexyl-4-[(1R)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl]-N-methylpiperazine-1-sulfonamide
—— 3-[[1-[3-[4-(2-ethoxyphenyl)piperazin-1-yl]propyl]piperidin-4-yl]methyl]-5-fluoro-1H-indole —— C29H39FN4O
3-[[1-[3-[4-(2-ethoxyphenyl)piperazin-1-yl]propyl]piperidin-4-yl]methyl]-5-fluoro-1H-indole
—— 5-[(1S)-1-[4-(6-tert-butylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperazin-1-yl]ethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole —— C23H29N7OS
5-[(1S)-1-[4-(6-tert-butylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperazin-1-yl]ethyl]-3-(4-methylphenyl)-1,2,4-oxadiazole
—— N-cyclohexyl-4-[(1S)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl]-N-methylpiperazine-1-sulfonamide —— C21H31F2N5O2S
N-cyclohexyl-4-[(1S)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl]-N-methylpiperazine-1-sulfonamide
—— 2-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone —— C21H30N4O4S
2-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone
—— tert-butyl 4-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate —— C23H35N3O4
tert-butyl 4-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoyl]piperazine-1-carboxylate
—— N-cyclohexyl-4-[(1R)-1-(4-fluorophenyl)ethyl]-N-methylpiperazine-1-sulfonamide —— C19H30FN3O2S
N-cyclohexyl-4-[(1R)-1-(4-fluorophenyl)ethyl]-N-methylpiperazine-1-sulfonamide
—— (2R)-4-methyl-1-(1-methylpyrazol-4-yl)sulfonyl-2-phenylpiperazine —— C15H20N4O2S
(2R)-4-methyl-1-(1-methylpyrazol-4-yl)sulfonyl-2-phenylpiperazine
—— 2-[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone —— C21H30N4O4S
2-[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone
—— N-cyclohexyl-4-[(2R)-1-(1H-indol-3-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide —— C22H32N4O3S
N-cyclohexyl-4-[(2R)-1-(1H-indol-3-yl)-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide
—— N-cyclohexyl-4-[(2R)-1-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide —— C21H40N4O3S
N-cyclohexyl-4-[(2R)-1-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide
—— ethyl 6-[4-[(2R)-1-[N-(2-cyanoethyl)anilino]-1-oxopropan-2-yl]piperazin-1-yl]pyridine-3-carboxylate —— C24H29N5O3
ethyl 6-[4-[(2R)-1-[N-(2-cyanoethyl)anilino]-1-oxopropan-2-yl]piperazin-1-yl]pyridine-3-carboxylate
—— 2-[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone —— C21H30N4O4S
2-[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylpiperazin-1-yl]-1-(2-methyl-1H-indol-3-yl)ethanone
—— N-cyclohexyl-4-[(1S)-1-(4-fluorophenyl)ethyl]-N-methylpiperazine-1-sulfonamide —— C19H30FN3O2S
N-cyclohexyl-4-[(1S)-1-(4-fluorophenyl)ethyl]-N-methylpiperazine-1-sulfonamide
—— 1-[4-[[(3R,5R)-5-(2,4-difluorophenyl)-5-(1,2,4-triazol-1-ylmethyl)oxolan-3-yl]methoxy]phenyl]-4-propan-2-ylpiperazine —— C27H33F2N5O2
1-[4-[[(3R,5R)-5-(2,4-difluorophenyl)-5-(1,2,4-triazol-1-ylmethyl)oxolan-3-yl]methoxy]phenyl]-4-propan-2-ylpiperazine
—— ethyl (4S)-6-[[4-[cyclohexyl(methyl)sulfamoyl]piperazin-1-yl]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H35N5O5S
ethyl (4S)-6-[[4-[cyclohexyl(methyl)sulfamoyl]piperazin-1-yl]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-[(4-chlorophenyl)amino]-2-[4-[(2E)-2-hydroxyiminopropanoyl]piperazin-1-yl]-6-propan-2-yl-5H-pyrrolo[4,3-e]pyrimidin-7-one —— C22H26ClN7O3
4-[(4-chlorophenyl)amino]-2-[4-[(2E)-2-hydroxyiminopropanoyl]piperazin-1-yl]-6-propan-2-yl-5H-pyrrolo[4,3-e]pyrimidin-7-one
—— (2S,6S)-4-[4-[2-(4-chlorophenyl)sulfanylethyl]piperazin-1-yl]sulfonyl-2,6-dimethylmorpholine —— C18H28ClN3O3S2
(2S,6S)-4-[4-[2-(4-chlorophenyl)sulfanylethyl]piperazin-1-yl]sulfonyl-2,6-dimethylmorpholine
—— 2-[4-[2-(3,4-Difluorophenyl)ethyl]piperazin-1-yl]-6,7-dimethoxyquinazolin-4-amine;dihydrochloride —— C22H27Cl2F2N5O2
2-[4-[2-(3,4-Difluorophenyl)ethyl]piperazin-1-yl]-6,7-dimethoxyquinazolin-4-amine;dihydrochloride
—— N-cyclohexyl-4-[(2R)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide —— C21H40N4O3S
N-cyclohexyl-4-[(2R)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1-oxopropan-2-yl]-N-methylpiperazine-1-sulfonamide