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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-[3-[(2-methoxyphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-(pyridin-3-ylmethyl)butanamide —— C26H26N4O3S
(2R)-2-[3-[(2-methoxyphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-(pyridin-3-ylmethyl)butanamide
—— 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazoline-7-carboxamide —— C25H29N5O6S
2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazoline-7-carboxamide
—— 4-oxo-N,3-bis[[(2S)-oxolan-2-yl]methyl]-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazoline-7-carboxamide —— C25H32N4O5S
4-oxo-N,3-bis[[(2S)-oxolan-2-yl]methyl]-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazoline-7-carboxamide
—— 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N,3-bis[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxamide —— C25H29N5O6S
2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N,3-bis[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxamide
—— N-[(2-chlorophenyl)methyl]-2-[3-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide —— C27H33ClN4O2S
N-[(2-chlorophenyl)methyl]-2-[3-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-[4-oxo-3-(3-piperidin-1-ylpropyl)quinazolin-2-yl]sulfanylacetamide —— C23H32N4O3S
N-[[(2S)-oxolan-2-yl]methyl]-2-[4-oxo-3-(3-piperidin-1-ylpropyl)quinazolin-2-yl]sulfanylacetamide
—— ethyl (3S)-1-[2-[3-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate —— C27H29N3O6S
ethyl (3S)-1-[2-[3-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate
—— 4-[2-[(2-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C24H26FN3O3S
4-[2-[(2-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[2-(4-ethylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C27H32N4O4S
4-[2-[2-(4-ethylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 3-[(2-chlorophenyl)methyl]-2-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanylquinazolin-4-one —— C23H24ClN3O2S
3-[(2-chlorophenyl)methyl]-2-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]sulfanylquinazolin-4-one
—— (2R)-2-[[2-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]sulfanyl]-N-(pyridin-3-ylmethyl)butanamide —— C26H28N8OS
(2R)-2-[[2-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]sulfanyl]-N-(pyridin-3-ylmethyl)butanamide
—— 4-[2-[2-(2-chloroanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C25H27ClN4O4S
4-[2-[2-(2-chloroanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C27H32N4O4S
4-[2-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[2-(3-methoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C26H30N4O5S
4-[2-[2-(3-methoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[(3-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C24H26FN3O3S
4-[2-[(3-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— methyl 2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxo-3-[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxylate —— C24H24ClN3O5S
methyl 2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxo-3-[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxylate
—— N-(furan-2-ylmethyl)-4-[4-oxo-2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]butanamide —— C24H28N4O5S
N-(furan-2-ylmethyl)-4-[4-oxo-2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]butanamide
—— 6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]hexanamide —— C30H39N3O3S
6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]hexanamide
—— 3-benzyl-6-morpholin-4-yl-2-[(2R)-1-morpholin-4-yl-1-oxobutan-2-yl]sulfanylquinazolin-4-one —— C27H32N4O4S
3-benzyl-6-morpholin-4-yl-2-[(2R)-1-morpholin-4-yl-1-oxobutan-2-yl]sulfanylquinazolin-4-one
—— 4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-3-[[(2R)-oxolan-2-yl]methyl]-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazoline-7-carboxamide —— C25H32N4O5S
4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-3-[[(2R)-oxolan-2-yl]methyl]-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazoline-7-carboxamide
—— ethyl (3S)-1-[2-[3-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate —— C27H29N3O6S
ethyl (3S)-1-[2-[3-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate
—— 4-[2-[2-(3-methoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C26H30N4O5S
4-[2-[2-(3-methoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[(2-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C24H26FN3O3S
4-[2-[(2-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— (2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-(3-methoxypropyl)butanamide —— C22H23BrN4O2S
(2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-(3-methoxypropyl)butanamide
—— 2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-[(2S)-butan-2-yl]acetamide —— C20H19BrN4OS
2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-[(2S)-butan-2-yl]acetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-[4-oxo-3-(3-piperidin-1-ylpropyl)quinazolin-2-yl]sulfanylacetamide —— C23H32N4O3S
N-[[(2R)-oxolan-2-yl]methyl]-2-[4-oxo-3-(3-piperidin-1-ylpropyl)quinazolin-2-yl]sulfanylacetamide
—— 6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]hexanamide —— C30H39N3O3S
6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]hexanamide
—— ethyl (3R)-1-[2-[3-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate —— C27H29N3O6S
ethyl (3R)-1-[2-[3-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-3-carboxylate
—— 4-[2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C26H29ClN4O4S
4-[2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— N-[(2S)-butan-2-yl]-2-[3-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide —— C24H36N4O2S
N-[(2S)-butan-2-yl]-2-[3-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-4-[4-oxo-2-[2-oxo-2-(2-phenylethylamino)ethyl]sulfanylquinazolin-3-yl]butanamide —— C27H32N4O4S
N-[[(2R)-oxolan-2-yl]methyl]-4-[4-oxo-2-[2-oxo-2-(2-phenylethylamino)ethyl]sulfanylquinazolin-3-yl]butanamide
—— 4-[2-[(2-methylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C25H29N3O3S
4-[2-[(2-methylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— N-cyclohexyl-3-[(2R)-5-[2-(2-methoxyethylamino)-2-oxoethyl]sulfanyl-3-oxo-2H-imidazo[1,2-c]quinazolin-2-yl]propanamide —— C24H31N5O4S
N-cyclohexyl-3-[(2R)-5-[2-(2-methoxyethylamino)-2-oxoethyl]sulfanyl-3-oxo-2H-imidazo[1,2-c]quinazolin-2-yl]propanamide
—— 4-[4-oxo-2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]-N-(2-phenylethyl)butanamide —— C27H32N4O4S
4-[4-oxo-2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]-N-(2-phenylethyl)butanamide
—— N-[(2S)-butan-2-yl]-2-[3-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide —— C24H36N4O2S
N-[(2S)-butan-2-yl]-2-[3-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinazolin-2-yl]sulfanylacetamide
—— 4-[2-[(2-methylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C25H29N3O3S
4-[2-[(2-methylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[2-(benzylamino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C26H30N4O4S
4-[2-[2-(benzylamino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 3-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanylquinazolin-4-one —— C26H29N3O4S
3-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanylquinazolin-4-one
—— [(2R)-1-(4-cyanoanilino)-1-oxopropan-2-yl] 3-hexyl-4-oxophthalazine-1-carboxylate —— C25H26N4O4
[(2R)-1-(4-cyanoanilino)-1-oxopropan-2-yl] 3-hexyl-4-oxophthalazine-1-carboxylate
—— 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-3-[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxamide —— C25H29N5O6S
2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanyl-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-3-[[(2R)-oxolan-2-yl]methyl]quinazoline-7-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-4-[4-oxo-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazolin-3-yl]butanamide —— C23H30N4O4S
N-[[(2S)-oxolan-2-yl]methyl]-4-[4-oxo-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylquinazolin-3-yl]butanamide
—— 4-[2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C26H29ClN4O4S
4-[2-[2-(3-chloro-4-methylanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— ethyl 4-[2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]piperidine-1-carboxylate —— C25H34N4O4S
ethyl 4-[2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]piperidine-1-carboxylate
—— (2R)-N-cyclohexyl-2-[[2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]sulfanyl]butanamide —— C26H33N7OS
(2R)-N-cyclohexyl-2-[[2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]sulfanyl]butanamide
—— (2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-1-morpholin-4-ylbutan-1-one —— C22H21BrN4O2S
(2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-1-morpholin-4-ylbutan-1-one
—— (2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C23H23BrN4O2S
(2S)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— N-(furan-2-ylmethyl)-4-[4-oxo-2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]butanamide —— C24H28N4O5S
N-(furan-2-ylmethyl)-4-[4-oxo-2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]sulfanylquinazolin-3-yl]butanamide
—— 4-[2-[(3-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C24H26FN3O3S
4-[2-[(3-fluorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 4-[2-[2-(4-ethoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide —— C27H32N4O5S
4-[2-[2-(4-ethoxyanilino)-2-oxoethyl]sulfanyl-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]butanamide
—— (2R)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-(3-methoxypropyl)butanamide —— C22H23BrN4O2S
(2R)-2-(2-bromobenzimidazolo[1,2-c]quinazolin-6-yl)sulfanyl-N-(3-methoxypropyl)butanamide