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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-­5-bromo-­3-chloro-3-((S)-2-nitro-1-phenylethyl)indolin-2-one 1398566-73-8 C14H10BrClN2O3S
(R)-­5-bromo-­3-chloro-3-((S)-2-nitro-1-phenylethyl)indolin-2-one
—— —— 1173722-14-9 C32H23FN2O5S
—— 6-methoxy-pyridine-3-sulfonic acid [5-(1-methyl-2-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-pyridin-3-ylmethyl]-amide 1427586-18-2 C22H22N4O4S
6-methoxy-pyridine-3-sulfonic acid [5-(1-methyl-2-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-pyridin-3-ylmethyl]-amide
—— (3S,3aR,6R,6aR)-6-[(1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl)oxymethoxy]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol 1418018-47-9 C17H28O5
(3S,3aR,6R,6aR)-6-[(1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl)oxymethoxy]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol
—— 5-(2-hydroxyphenyl)-N-[2-(phenylsulfanyl)pyridin-3-yl]3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide 1035233-63-6 C26H21N5O2S
5-(2-hydroxyphenyl)-N-[2-(phenylsulfanyl)pyridin-3-yl]3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide
—— N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-(2-hydroxyphenyl)-3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide 1035234-14-0 C27H28N4O3
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-(2-hydroxyphenyl)-3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide
—— N-[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)phenyl]-5-(2-hydroxyphenyl)-3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide 1035234-25-3 C29H21N5O4
N-[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)phenyl]-5-(2-hydroxyphenyl)-3-pyridin-3-yl-4,5-dihydro-1H-pyrazole-1-carboxamide
—— 1-(2-methoxy-pyridin-4-yl)-3-(4-methyl-pyridin-3-yl)-imidazolidin-2-one 1260006-42-5 C15H16N4O2
1-(2-methoxy-pyridin-4-yl)-3-(4-methyl-pyridin-3-yl)-imidazolidin-2-one
—— 4-{(S)-2-[(S)-2-(methoxycarbonylamino)-3-phenylpropanamido]-2-[2-(6-methylpyridin-3-yl)thiazol-4-yl]ethyl}phenylsulfamic acid 1008510-45-9 C28H29N5O6S2
4-{(S)-2-[(S)-2-(methoxycarbonylamino)-3-phenylpropanamido]-2-[2-(6-methylpyridin-3-yl)thiazol-4-yl]ethyl}phenylsulfamic acid
—— N-(5-tert-butyl-2-methylphenyl)-6,7-dimethoxy-2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]quinazolin-4-amine 1048388-93-7 C34H43N5O3
N-(5-tert-butyl-2-methylphenyl)-6,7-dimethoxy-2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]quinazolin-4-amine
—— 2-(4-fluorophenoxy)-5-(((1,2,2-trimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile 1620679-92-6 C24H23FN4O3
2-(4-fluorophenoxy)-5-(((1,2,2-trimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile
—— [D-Leu<sup>7</sup>]-ternatin 1005766-32-4 C37H67N7O7
[D-Leu<sup>7</sup>]-ternatin
—— N-cyclopropyl-4-[(3-{5-methoxy-4-[(pyridin-4-yl)amino]pyrimidin-2-yl}-1H-indazol-1-yl)methyl]benzenesulfonamide 1429745-46-9 C27H25N7O3S
N-cyclopropyl-4-[(3-{5-methoxy-4-[(pyridin-4-yl)amino]pyrimidin-2-yl}-1H-indazol-1-yl)methyl]benzenesulfonamide
—— (tetraphenylporphyrin)(germanium(IV))(ethylhydroperoxide)2 126327-28-4 C48H38GeN4O4
(tetraphenylporphyrin)(germanium(IV))(ethylhydroperoxide)2
—— [4-(4-Ethoxy-2-fluorobenzoyl)oxyphenyl] 4-ethoxy-2-fluorobenzoate 1189397-87-2 C24H20F2O6
[4-(4-Ethoxy-2-fluorobenzoyl)oxyphenyl] 4-ethoxy-2-fluorobenzoate
—— (η(5)-C9H7)IrH2(PiPr3) 163317-88-2 C18H30IrP
(η(5)-C9H7)IrH2(PiPr3)
—— 4',4'''-divinyl-2,2':6',2'':6'',2''':6''',2''''-quinquepyridine 126257-34-9 C29H21N5
4',4'''-divinyl-2,2':6',2'':6'',2''':6''',2''''-quinquepyridine
—— 1-t-butyl-3,3-dichloro-2-methoxy-1,2-epoxycyclohexane 116625-43-5 C11H18Cl2O2
1-t-butyl-3,3-dichloro-2-methoxy-1,2-epoxycyclohexane
—— [(1S,2S,4R)-5,8,8-trimethyl-2-bicyclo[2.2.2]oct-5-enyl] 2-chloroacetate 137330-35-9 C13H19ClO2
[(1S,2S,4R)-5,8,8-trimethyl-2-bicyclo[2.2.2]oct-5-enyl] 2-chloroacetate
—— N-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-morpholin-4-ylethanimine 110718-35-9 C15H18N4OS
N-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-morpholin-4-ylethanimine
—— 3-(2-amino-6-(3-chlorophenyl)-pyrimidin-4-yl)-6-bromo-2H-chromen-2-one 1309189-49-8 C19H11BrClN3O2
3-(2-amino-6-(3-chlorophenyl)-pyrimidin-4-yl)-6-bromo-2H-chromen-2-one
—— 6-(difluoromethyl)-2,4-difluorophenanthridine 1610500-99-6 C14H7F4N
6-(difluoromethyl)-2,4-difluorophenanthridine
—— (R)-5-[(methysulfonyl)oxy]-3-phenylpentyl acetate 1312363-61-3 C14H20O5S
(R)-5-[(methysulfonyl)oxy]-3-phenylpentyl acetate
—— 1,4-bis-(1-phenoxy-ethoxy)-benzene 125667-46-1 C22H22O4
1,4-bis-(1-phenoxy-ethoxy)-benzene
—— (4S,1'R,2'S)-N(3)-[1'-(m-chlorobenzoyl)-2'-hydroxy-propan-1'-yl]-4-phenyl-5,5-dimethyloxazolidin-2-one 1067232-34-1 C21H22ClNO5
(4S,1'R,2'S)-N(3)-[1'-(m-chlorobenzoyl)-2'-hydroxy-propan-1'-yl]-4-phenyl-5,5-dimethyloxazolidin-2-one
—— N-(2,4-difluorophenyl)-4-{[(3,5-dimethyl-4-isoxazolyl)methyl]oxy}-N-(2-methylpropyl)benzenesulfonamide 1429345-97-0 C22H24F2N2O4S
N-(2,4-difluorophenyl)-4-{[(3,5-dimethyl-4-isoxazolyl)methyl]oxy}-N-(2-methylpropyl)benzenesulfonamide
—— 1,3-dihydroisoindole-2-carboxylic acid adamantan-1-ylamide 1422444-13-0 C19H24N2O
1,3-dihydroisoindole-2-carboxylic acid adamantan-1-ylamide
—— 2-acetonyl-5-allyl-4,6-dimethoxy-5-nitro-2,5-dihydroryrimidine 177851-25-1 C12H17N3O5
2-acetonyl-5-allyl-4,6-dimethoxy-5-nitro-2,5-dihydroryrimidine
—— methyl (E)-4-[hydroxy-[[1-[[4-(naphthalen-1-ylcarbamoyloxymethyl)phenyl]methyl]piperidin-4-yl]methyl]amino]-4-oxobut-2-enoate 1439845-17-6 C30H33N3O6
methyl (E)-4-[hydroxy-[[1-[[4-(naphthalen-1-ylcarbamoyloxymethyl)phenyl]methyl]piperidin-4-yl]methyl]amino]-4-oxobut-2-enoate
—— (2S)-5-(diaminomethylideneamino)-2-[[2-[(1S,2S)-1-[[4-(dimethylamino)benzoyl]amino]-2-methylbutyl]-1,3-oxazole-4-carbonyl]amino]pentanoic acid 1434871-89-2 C24H35N7O5
(2S)-5-(diaminomethylideneamino)-2-[[2-[(1S,2S)-1-[[4-(dimethylamino)benzoyl]amino]-2-methylbutyl]-1,3-oxazole-4-carbonyl]amino]pentanoic acid
—— US9598416, Example 50 1443617-09-1 C22H26N6OS
US9598416, Example 50
—— 7-amino-2-(2,4-difluorophenyl)phthalazin-1(2H)-one 1436504-01-6 C14H9F2N3O
7-amino-2-(2,4-difluorophenyl)phthalazin-1(2H)-one
—— 5-tert-butyl-2-(2-methanesulfonyl-benzyl)-7-(2-oxa-6-aza-spiro[3.3]hept-6-yl)-2H-[1,2,3]triazolo[4,5-d]pyrimidine 1438466-64-8 C21H26N6O3S
5-tert-butyl-2-(2-methanesulfonyl-benzyl)-7-(2-oxa-6-aza-spiro[3.3]hept-6-yl)-2H-[1,2,3]triazolo[4,5-d]pyrimidine
—— [5-chloro-2-methoxy-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-phenyl]-(3,3-difluoro-pyrrolidin-1-yl)-methanone 1441200-99-2 C18H17ClF5N5O2
[5-chloro-2-methoxy-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-phenyl]-(3,3-difluoro-pyrrolidin-1-yl)-methanone
—— (8S,11S,14S,17S)-10-[(2S)-2-[[(2S)-2-(methylamino)propanoyl]amino]-3-phenylpropanoyl]-12,15-dioxo-14-(2-phenylethyl)-2-oxa-5,6,7,10,13,16-hexazatetracyclo[17.2.2.14,7.18,11]pentacosa-1(22),4(25),5,19(23),20-pentaene-17-carboxylic acid 1432734-38-7 C40H46N8O7
(8S,11S,14S,17S)-10-[(2S)-2-[[(2S)-2-(methylamino)propanoyl]amino]-3-phenylpropanoyl]-12,15-dioxo-14-(2-phenylethyl)-2-oxa-5,6,7,10,13,16-hexazatetracyclo[17.2.2.14,7.18,11]pentacosa-1(22),4(25),5,19(23),20-pentaene-17-carboxylic acid
—— Bis(trifluoromethylsulfonyl)azanide;3,5-dimethyl-1-propylpyridin-1-ium 1456878-04-8 C2F6NO4S2*C10H16N
Bis(trifluoromethylsulfonyl)azanide;3,5-dimethyl-1-propylpyridin-1-ium
—— N-benzyl-3-(2-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)benzamide 1246083-12-4 C23H20N2O3
N-benzyl-3-(2-methyl-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)benzamide
—— 6-[3-cyano-1-cyclohexyl-6-(difluoromethoxy)-1H-indol-2-yl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide 1248577-12-9 C24H23F5N4O3S
6-[3-cyano-1-cyclohexyl-6-(difluoromethoxy)-1H-indol-2-yl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide
—— 1-[(7-amino-5-ethyl[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)ethynyl]cyclopentanol 1075216-94-2 C14H17N5O
1-[(7-amino-5-ethyl[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)ethynyl]cyclopentanol
—— N-(1-butylpiperidin-4-yl)-1-ethyl-5-(1-oxa-2-azaspiro[4.4]noN-2-en-3-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine 1057635-54-7 C24H36N6O
N-(1-butylpiperidin-4-yl)-1-ethyl-5-(1-oxa-2-azaspiro[4.4]noN-2-en-3-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine
—— methyl (1R,9R,10S,11R,12R,19R)-11-acetyloxy-4-[(13S,15R,17S)-17-(butylcarbamoylamino)-17-ethyl-13-methoxycarbonyl-1,11-diazatetracyclo[13.3.1.04,12.05,10]nonadeca-4(12),5,7,9-tetraen-13-yl]-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2,4,6,13-tetraene-10-carboxylate 1416208-90-6 C51H68N6O9
methyl (1R,9R,10S,11R,12R,19R)-11-acetyloxy-4-[(13S,15R,17S)-17-(butylcarbamoylamino)-17-ethyl-13-methoxycarbonyl-1,11-diazatetracyclo[13.3.1.04,12.05,10]nonadeca-4(12),5,7,9-tetraen-13-yl]-12-ethyl-10-hydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2,4,6,13-tetraene-10-carboxylate
—— 4-(4-chloro-2-(imidazolo[1,2-a]pyridin-5-yl)phenoxy)-N-(3-chloropyrazin-2-yl)-2,5-difluorobenzenesulfonamide 1432913-22-8 C23H13Cl2F2N5O3S
4-(4-chloro-2-(imidazolo[1,2-a]pyridin-5-yl)phenoxy)-N-(3-chloropyrazin-2-yl)-2,5-difluorobenzenesulfonamide
—— 1-N-(4,4'-Dimethoxytrityl)-biotinyl-6-amino-1-tert-butyldimethylsilylhexan-1-ol 135137-85-8 C43H61N3O5SSi
1-N-(4,4'-Dimethoxytrityl)-biotinyl-6-amino-1-tert-butyldimethylsilylhexan-1-ol
—— tert-butyl (R)-(4-((2-(2-((tert-butoxycarbonyl)amino)-N-ethylpropanamido)ethyl)(ethyl)carbamoyl)-1H-imidazole-5-carbonyl)glycinate 1393747-76-6 C25H42N6O7
tert-butyl (R)-(4-((2-(2-((tert-butoxycarbonyl)amino)-N-ethylpropanamido)ethyl)(ethyl)carbamoyl)-1H-imidazole-5-carbonyl)glycinate
—— tert-butyl (S,E)-5-(N-(benzoyloxy)-5-((tert-butyldiphenylsilyl)oxy)-3-methylpent-2-enamido)-2-((tert-butoxycarbonyl)amino)pentanoate 1224926-52-6 C43H58N2O8Si
tert-butyl (S,E)-5-(N-(benzoyloxy)-5-((tert-butyldiphenylsilyl)oxy)-3-methylpent-2-enamido)-2-((tert-butoxycarbonyl)amino)pentanoate
—— 2-(selenocyanatomethyl)prop-2-en-1-ol 1407967-77-4 C5H7NOSe
2-(selenocyanatomethyl)prop-2-en-1-ol
—— 4-{3-Benzyloxy-5-[3-(3,5-bis-benzyloxy-benzyloxy)-5-bromomethyl-phenoxymethyl]-phenoxymethyl}-benzonitrile 134868-81-8 C50H42BrNO6
4-{3-Benzyloxy-5-[3-(3,5-bis-benzyloxy-benzyloxy)-5-bromomethyl-phenoxymethyl]-phenoxymethyl}-benzonitrile
—— 4,8-bis(hexyloxy)-2,6-di(thiophen-2-yl)benzo[1,2-d:4,5-d']bis([1,3]thiaphosphole) 1618089-37-4 C28H32O2P2S4
4,8-bis(hexyloxy)-2,6-di(thiophen-2-yl)benzo[1,2-d:4,5-d']bis([1,3]thiaphosphole)
—— 5-(2-amino-4-methyl-pyrimidin-5-yl)-2,n,N-trimethyl-benzenesulfonamide 1106312-61-1 C14H18N4O2S
5-(2-amino-4-methyl-pyrimidin-5-yl)-2,n,N-trimethyl-benzenesulfonamide
—— 1-(3-isopropyl-1-(4-(2-morpholinoethoxy)phenyl)-1H-pyrazol-5-yl)-3-(4-((2-((2-oxoindolin-6-yl)amino)pyrimidin-4-yl)oxy)naphthalen-1-yl)urea 1574358-28-3 C41H41N9O5
1-(3-isopropyl-1-(4-(2-morpholinoethoxy)phenyl)-1H-pyrazol-5-yl)-3-(4-((2-((2-oxoindolin-6-yl)amino)pyrimidin-4-yl)oxy)naphthalen-1-yl)urea