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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-(2-(6-((2-(dimethylamino)ethyl)(ethyl)amino)-2-phenylpyrimidine-4-carboxamido)phenyl)-1,3,4-thiadiazole-2-carboxamide 1148120-99-3 C26H28N8O2S
5-(2-(6-((2-(dimethylamino)ethyl)(ethyl)amino)-2-phenylpyrimidine-4-carboxamido)phenyl)-1,3,4-thiadiazole-2-carboxamide
—— methyl 3,3-bis(3,5-di-t-butyl-4-hydroxyphenylthio)butanoate 1029421-72-4 C33H50O4S2
methyl 3,3-bis(3,5-di-t-butyl-4-hydroxyphenylthio)butanoate
—— 7-chloro-1-(2,4-difluorobenzyl)-3-[3-(trifluoromethoxy)phenyl]cinnolin-4(1H)-one 1204653-00-8 C22H12ClF5N2O2
7-chloro-1-(2,4-difluorobenzyl)-3-[3-(trifluoromethoxy)phenyl]cinnolin-4(1H)-one
—— 1-(tetrahydro-pyran-4-yl)-azetidine-2-carboxylic acid methyl ester 1450977-82-8 C10H17NO3
1-(tetrahydro-pyran-4-yl)-azetidine-2-carboxylic acid methyl ester
—— (S)-5-bromo-1-sec-butyl-6-methyl-4-oxo-1,4-dihydro-pyridine-3-carboxylic acid (5-methyl-[1,3,4]oxadiazol-2-ylmethyl)-amide 1569651-74-6 C15H19BrN4O3
(S)-5-bromo-1-sec-butyl-6-methyl-4-oxo-1,4-dihydro-pyridine-3-carboxylic acid (5-methyl-[1,3,4]oxadiazol-2-ylmethyl)-amide
—— (5-bromopyrazin-2-yl)[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazin-1-yl]methanone 1346124-39-7 C18H20BrN5O
(5-bromopyrazin-2-yl)[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazin-1-yl]methanone
—— 2-chloro-N-cyano-4-pyrimidinecarboximidamide 1150111-26-4 C6H4ClN5
2-chloro-N-cyano-4-pyrimidinecarboximidamide
—— 4-(but-1-en-3-ylamino)-2,5-dichloro-6-methoxycarbonyl-pyrimidine 1292286-77-1 C10H11Cl2N3O2
4-(but-1-en-3-ylamino)-2,5-dichloro-6-methoxycarbonyl-pyrimidine
—— N-(4-{2-[4-(chloromethyl)-2-fluorophenyl]ethyl}-1,3-thiazol-2-yl)acetamide 1174633-16-9 C14H14ClFN2OS
N-(4-{2-[4-(chloromethyl)-2-fluorophenyl]ethyl}-1,3-thiazol-2-yl)acetamide
—— (3R,5S)-7-chloro-5-(2,4-dimethoxyphenyl)-1-isobutyl-2-oxo-1,2,3,5-tetrahydro-4,1-benzothiazepine-3-acetic acid 179124-77-7 C23H26ClNO5S
(3R,5S)-7-chloro-5-(2,4-dimethoxyphenyl)-1-isobutyl-2-oxo-1,2,3,5-tetrahydro-4,1-benzothiazepine-3-acetic acid
—— 1-[({2-[2,3-bis(nitrooxy)propoxy]ethoxy}carbonyl)oxy]-1-methylethyl 2-ethoxy-1-{[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-1H-benzimidazole-7-carboxylate 1034453-34-3 C33H34N8O13
1-[({2-[2,3-bis(nitrooxy)propoxy]ethoxy}carbonyl)oxy]-1-methylethyl 2-ethoxy-1-{[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-1H-benzimidazole-7-carboxylate
—— N-[4-(4-methoxybenzyl)-1,3-thiazol-2-yl]-2-(3-methoxy-9H-xanthen-9-yl)-2-methylpropanamide 1008113-70-9 C29H28N2O4S
N-[4-(4-methoxybenzyl)-1,3-thiazol-2-yl]-2-(3-methoxy-9H-xanthen-9-yl)-2-methylpropanamide
—— cis-3-[1-(6-chloro-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]carbonyl}pyridin-2-yl)piperidin-4-yl]-1,3,4,5-tetrahydro-2H-1,3-benzodiazepin-2-one 1028319-42-7 C26H32ClN5O3
cis-3-[1-(6-chloro-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]carbonyl}pyridin-2-yl)piperidin-4-yl]-1,3,4,5-tetrahydro-2H-1,3-benzodiazepin-2-one
—— (3R,4S)-N-cyclopropyl-4-{4-(2-(2,6-dichloro-4-methyl-phenoxy)ethoxy)-phenyl}-N-[3-{[(1R,2R)-2-(hydroxymethyl)-cyclopropyl]methoxy}-5-(3-methoxy-propyl)benzyl]-piperidine-3-carboxamide 1026787-29-0 C40H50Cl2N2O6
(3R,4S)-N-cyclopropyl-4-{4-(2-(2,6-dichloro-4-methyl-phenoxy)ethoxy)-phenyl}-N-[3-{[(1R,2R)-2-(hydroxymethyl)-cyclopropyl]methoxy}-5-(3-methoxy-propyl)benzyl]-piperidine-3-carboxamide
—— N-[(3S)-1-({6-chloro-3-[1-(4-chlorobenzyl)-4-phenyl-1H-imidazol-5-yl]-1H-indol-2-yl}carbonyl)pyrrolidin-3-yl]-N,N',N'-trimethylpropane-1,3-diamine 1067654-70-9 C35H38Cl2N6O
N-[(3S)-1-({6-chloro-3-[1-(4-chlorobenzyl)-4-phenyl-1H-imidazol-5-yl]-1H-indol-2-yl}carbonyl)pyrrolidin-3-yl]-N,N',N'-trimethylpropane-1,3-diamine
—— 7-chloro-3,6-bis(6-fluoropyridin-3-yl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinoline 1021911-53-4 C26H23ClF2N4O
7-chloro-3,6-bis(6-fluoropyridin-3-yl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinoline
—— N-[(1S,2S,4R)-4-((S)-1-benzylcarbamoyl-2-methyl-propylcarbamoyl)-1-(3,5-difluorobenzyloxymethyl)-2-hydroxy-4-methoxy-butyl]-5-(methanesulfonyl(methyl)amino)-N'-((R)-1-phenyl-ethyl)-isophthalamide 1067651-18-6 C44H53F2N5O9S
N-[(1S,2S,4R)-4-((S)-1-benzylcarbamoyl-2-methyl-propylcarbamoyl)-1-(3,5-difluorobenzyloxymethyl)-2-hydroxy-4-methoxy-butyl]-5-(methanesulfonyl(methyl)amino)-N'-((R)-1-phenyl-ethyl)-isophthalamide
—— 2-(4-[5-bromo-2-(2-chloro-6-fluorophenyl)-1H-imidazol-4-yl]phenyl)-1,6-dimethyl-1H-benzoimidazole 1038842-25-9 C24H17BrClFN4
2-(4-[5-bromo-2-(2-chloro-6-fluorophenyl)-1H-imidazol-4-yl]phenyl)-1,6-dimethyl-1H-benzoimidazole
—— N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenyl-propan-2-yl]butanesulfonamide 1028458-79-8 C26H28FN3O3S
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenyl-propan-2-yl]butanesulfonamide
—— 7-fluoromethyl-2-(4-hydroxy-phenyl)-3-phenyl-1H-inden-5-ol 1019985-19-3 C22H17FO2
7-fluoromethyl-2-(4-hydroxy-phenyl)-3-phenyl-1H-inden-5-ol
—— 1-adamantan-2-yl-3-cyclopropyl-4-isobutyl-1,3-dihydro-imidazol-2-one 1021390-08-8 C20H30N2O
1-adamantan-2-yl-3-cyclopropyl-4-isobutyl-1,3-dihydro-imidazol-2-one
—— 1-(5-isopropyl-[1,2,4]oxadiazol-3-yl)-4-((R)-3-(4-methanesulfonylphenoxy)-1-methylpropyl)piperidine 1037779-21-7 C21H31N3O4S
1-(5-isopropyl-[1,2,4]oxadiazol-3-yl)-4-((R)-3-(4-methanesulfonylphenoxy)-1-methylpropyl)piperidine
—— —— 1609529-74-9 C29H29FN6O4
—— 4-hydroxy-3-[(3,5-difluoro-6-(3-dimethylaminocarbonylphenoxy)-4-(4-carboxymethyl-piperazin-1-yl)pyridin-2-yl)oxy]benzamidine, trifluoroacetic acid salt 183304-53-2 C2HF3O2*C27H28F2N6O6
4-hydroxy-3-[(3,5-difluoro-6-(3-dimethylaminocarbonylphenoxy)-4-(4-carboxymethyl-piperazin-1-yl)pyridin-2-yl)oxy]benzamidine, trifluoroacetic acid salt
—— —— 1186105-18-9 C32H37N5O3
—— N-[4-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)-3-fluorophenyl]-1-(3,4-difluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide 1195779-66-8 C30H22F3N5O4
N-[4-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-a]pyridin-6-yl}oxy)-3-fluorophenyl]-1-(3,4-difluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
—— N-[4-(2-oxo-4-phenylpyrrolidin-1-yl)pyridin-2-yl]cyclohexanecarboxamide 1019649-47-8 C22H25N3O2
N-[4-(2-oxo-4-phenylpyrrolidin-1-yl)pyridin-2-yl]cyclohexanecarboxamide
—— N-[(2-chloro-4-fluorophenyl)methyl]-2-[1-(2,6-dimethyl-3-pyridinyl)-3,5-dimethyl-1H-pyrazol-4-yl]acetamide 1082826-88-7 C21H22ClFN4O
N-[(2-chloro-4-fluorophenyl)methyl]-2-[1-(2,6-dimethyl-3-pyridinyl)-3,5-dimethyl-1H-pyrazol-4-yl]acetamide
—— 9-[1-(2-aminoethyl)piperidin-4-yl]-8-(2-chloro-6-fluorophenyl)-N-[(2-fluorophenyl)methyl]purin-2-amine 1021694-67-6 C25H26ClF2N7
9-[1-(2-aminoethyl)piperidin-4-yl]-8-(2-chloro-6-fluorophenyl)-N-[(2-fluorophenyl)methyl]purin-2-amine
—— —— 1245516-86-2 C27H28N2O2S
—— 2-(dipropylamino)methyl-4-({4-[4-(2-(pyrrolidin-1-yl)pyridin-4-ylamino)phenyl]pyrimidin-2-ylamino}methyl)phenol 1609657-65-9 C33H41N7O
2-(dipropylamino)methyl-4-({4-[4-(2-(pyrrolidin-1-yl)pyridin-4-ylamino)phenyl]pyrimidin-2-ylamino}methyl)phenol
—— —— 1179323-23-9 C22H29N3O4S2
—— —— 1008518-43-1 C22H21NO4
—— —— 1092932-20-1 C20H19N3O3
—— 5-[(1R)-5-(2-methylpyridin-4-yl)oxy-2,3-dihydro-1H-inden-1-yl]-1,3-thiazolidine-2,4-dione 1021935-17-0 C18H16N2O3S
5-[(1R)-5-(2-methylpyridin-4-yl)oxy-2,3-dihydro-1H-inden-1-yl]-1,3-thiazolidine-2,4-dione
—— N-(3,5-bis(trifluoromethyl)benzyl)-4-(cyclopropylmethyl)-1-(2-methyl-2-morpholinopropyl)piperidine-4-carboxamide 1018991-59-7 C27H37F6N3O2
N-(3,5-bis(trifluoromethyl)benzyl)-4-(cyclopropylmethyl)-1-(2-methyl-2-morpholinopropyl)piperidine-4-carboxamide
—— [3-[4-(4-cyclopentyl-piperazin-1-ylmethyl)-phenyl]-3-(4-trifluoromethyl-phenoxy)-propyl]-dimethyl-amine 1029648-56-3 C28H38F3N3O
[3-[4-(4-cyclopentyl-piperazin-1-ylmethyl)-phenyl]-3-(4-trifluoromethyl-phenoxy)-propyl]-dimethyl-amine
—— 2-(3,5-dichloro-pyridin-4-yl)-1-{2-[2-(2-fluoro-phenyl)-ethoxy]-3,4-dimethoxy-phenyl}-ethanone 1035571-58-4 C23H20Cl2FNO4
2-(3,5-dichloro-pyridin-4-yl)-1-{2-[2-(2-fluoro-phenyl)-ethoxy]-3,4-dimethoxy-phenyl}-ethanone
—— (5S,7a'S)-N-(1-(cyclopropylamino)-1,2-dioxohexan-3-yl)-1-((S)-2-(3-cyclopropylureido)-3,3-dimethylbutanoyl)-1'-oxohexahydrospiro[pyrrolidine-3,3'-pyrrolo[1,2-c]imidazole]-5-carboxamide 1024615-82-4 C29H45N7O6
(5S,7a'S)-N-(1-(cyclopropylamino)-1,2-dioxohexan-3-yl)-1-((S)-2-(3-cyclopropylureido)-3,3-dimethylbutanoyl)-1'-oxohexahydrospiro[pyrrolidine-3,3'-pyrrolo[1,2-c]imidazole]-5-carboxamide
—— 2-{4-[2-(dimethylamino)ethoxy]-9H-xanthen-9-yl}-N-[4-(4-methoxybenzyl)-1,3-thiazol-2-yl]-2-methylpropanamide 1008114-10-0 C32H35N3O4S
2-{4-[2-(dimethylamino)ethoxy]-9H-xanthen-9-yl}-N-[4-(4-methoxybenzyl)-1,3-thiazol-2-yl]-2-methylpropanamide
—— (E)-N-(4-{[3-(4-bromophenyl)-2-propen-1-yl]amino}butyl)-5-isoquinolinesulfonamide 1415682-29-9 C22H24BrN3O2S
(E)-N-(4-{[3-(4-bromophenyl)-2-propen-1-yl]amino}butyl)-5-isoquinolinesulfonamide
—— 1H-Indole-3-methanamine, 2,3-dihydro-, hydrochloride (1:2) 1408058-15-0 C9H13ClN2
1H-Indole-3-methanamine, 2,3-dihydro-, hydrochloride (1:2)
—— N-(3-(5-(2-Aminopyrimidin-4-yl)-2-cyclopropyl-1H-imidazol-4-yl)-5-chloro-2-fluorophenyl)methanesulfonamide 1269231-67-5 C17H16ClFN6O2S
N-(3-(5-(2-Aminopyrimidin-4-yl)-2-cyclopropyl-1H-imidazol-4-yl)-5-chloro-2-fluorophenyl)methanesulfonamide
—— N-[(2-chloro-4-fluorophenyl)methyl]-2-[3,5-dimethyl-1-(2-phenylcyclohexyl)-1H-pyrazol-4-yl]acetamide 1082826-09-2 C26H29ClFN3O
N-[(2-chloro-4-fluorophenyl)methyl]-2-[3,5-dimethyl-1-(2-phenylcyclohexyl)-1H-pyrazol-4-yl]acetamide
—— Bouvardin, 5-(N-methyl-L-tyrosine)-6-(O-beta-D-glucopyranosyl-3-hydroxy-N-methyl-L-tyrosine)- 143343-98-0 C46H58N6O14
Bouvardin, 5-(N-methyl-L-tyrosine)-6-(O-beta-D-glucopyranosyl-3-hydroxy-N-methyl-L-tyrosine)-
—— —— 1116105-85-1 C18H16FN3O3*ClH
—— N-(3,5-dimethylisooxazol-4-yl)sulfonyl-3-amino-4-oxo-5-(5-(2,6-dichlorophenylmethyl)tetrazol-2-yl)pentanoic acid 192504-93-1 C18H18Cl2N6O6S
N-(3,5-dimethylisooxazol-4-yl)sulfonyl-3-amino-4-oxo-5-(5-(2,6-dichlorophenylmethyl)tetrazol-2-yl)pentanoic acid
—— N-(3-(2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)phenyl)-2-hydroxyacetamide 1231714-64-9 C18H17ClN4O3S
N-(3-(2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)phenyl)-2-hydroxyacetamide
—— 2,4,5,6-tetrahydro-1H-oxepino[4,5-b]indole 1279723-15-7 C12H13NO
2,4,5,6-tetrahydro-1H-oxepino[4,5-b]indole
—— 6'-methoxy-3,4,5,6-tetrahydro-2H-[1,3']bipyridinyl-4-carboxylic acid 1268692-84-7 C12H16N2O3
6'-methoxy-3,4,5,6-tetrahydro-2H-[1,3']bipyridinyl-4-carboxylic acid