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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-((S)-4-carboxy-2-{[2-phenyl-6-(piperidin-4-yloxy)-pyrimidine-4-carbonyl]-amino}-butyryl)-piperazine-1-carboxylic acid ethyl ester 1021702-91-9 C28H36N6O7
4-((S)-4-carboxy-2-{[2-phenyl-6-(piperidin-4-yloxy)-pyrimidine-4-carbonyl]-amino}-butyryl)-piperazine-1-carboxylic acid ethyl ester
—— (S)-N-[methyl(oxo)phenyl-λ<sup>6</sup>-sulfanylidene]-5-({3-[(2-thienylcarbonyl)amino]phenyl}ethynyl)nicotinamide 1027726-11-9 C26H19N3O3S2
(S)-N-[methyl(oxo)phenyl-λ<sup>6</sup>-sulfanylidene]-5-({3-[(2-thienylcarbonyl)amino]phenyl}ethynyl)nicotinamide
—— 2-ethyl-N-(5-ethyl-4-(morpholinomethyl)pyridin-2-yl)-2-methylbutanamide 1029126-91-7 C19H31N3O2
2-ethyl-N-(5-ethyl-4-(morpholinomethyl)pyridin-2-yl)-2-methylbutanamide
—— [5-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-1-ethyl-1H-pyrazol-3-yl]-(4-fluorobenzyl)amine 1029051-56-6 C20H19ClFN5
[5-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-1-ethyl-1H-pyrazol-3-yl]-(4-fluorobenzyl)amine
—— (4-{4-[1-methylethoxy]-9-[(1-methylpropyl)oxy]-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid 1028542-55-3 C27H27NO6
(4-{4-[1-methylethoxy]-9-[(1-methylpropyl)oxy]-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid
—— 3,5-dimethyl-4-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrazole-1-carboxylic acid 3-fluorobenzylamide 1029046-85-2 C21H20FN5O
3,5-dimethyl-4-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrazole-1-carboxylic acid 3-fluorobenzylamide
—— 2-(2-chloro-4-hydroxy-phenyl)-7-methyl-3-phenyl-1H-inden-5-ol 1019984-56-5 C22H17ClO2
2-(2-chloro-4-hydroxy-phenyl)-7-methyl-3-phenyl-1H-inden-5-ol
—— 2-(2-chloro-6-(2-((4aS,5R)-1-(4-fluorophenyl)-5-hydroxy-4a-methyl-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl)ethyl)phenyl)acetamide 1021539-19-4 C27H27ClFN3O2
2-(2-chloro-6-(2-((4aS,5R)-1-(4-fluorophenyl)-5-hydroxy-4a-methyl-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl)ethyl)phenyl)acetamide
—— (4aR,6R,8aS)-6-(4-chlorophenyl)-8a-(2,4-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-amine 1622328-05-5 C19H17ClF2N2OS
(4aR,6R,8aS)-6-(4-chlorophenyl)-8a-(2,4-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-amine
—— 4-(2-cyclopentyl-acetyl)-[1,4]diazepane-1-carboxylic acid (4-bromo-phenyl)-amide 1028852-26-7 C19H26BrN3O2
4-(2-cyclopentyl-acetyl)-[1,4]diazepane-1-carboxylic acid (4-bromo-phenyl)-amide
—— (4,6-dimethyl-pyrimidin-5-yl)-{5-[3-phenyl-3-(1-phenylmethanesulfonyl-piperidin-4-yl)-propyl]-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl}-methanone 1014701-96-2 C34H43N5O3S
(4,6-dimethyl-pyrimidin-5-yl)-{5-[3-phenyl-3-(1-phenylmethanesulfonyl-piperidin-4-yl)-propyl]-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl}-methanone
—— 5-fluoro-2-(4-(2-methoxyethyl)phenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)benzamide 1620847-08-6 C21H19FN2O4
5-fluoro-2-(4-(2-methoxyethyl)phenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)benzamide
—— 4-(2-(2,4-dimethoxyphenoxy)quinoline-3-carboxamido)benzoic acid 1621108-36-8 C25H20N2O6
4-(2-(2,4-dimethoxyphenoxy)quinoline-3-carboxamido)benzoic acid
—— N-(3-fluorophenyl)-3-[5-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-3-yl]propanamide 1353542-78-5 C25H21F2N3O2
N-(3-fluorophenyl)-3-[5-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-3-yl]propanamide
—— N-[(3-chloro-2-methylphenyl)methyl]-2-[1-(2-hydroxy-2-methylpropyl)-3,5-dimethyl-1H-pyrazol-4-yl]acetamide 1082827-07-3 C19H26ClN3O2
N-[(3-chloro-2-methylphenyl)methyl]-2-[1-(2-hydroxy-2-methylpropyl)-3,5-dimethyl-1H-pyrazol-4-yl]acetamide
—— N',4-diethyl-N-(3-hydroxyphenyl)sulfonyl-3,4-dihydropyrazole-2-carboximidamide 1187966-00-2 C14H20N4O3S
N',4-diethyl-N-(3-hydroxyphenyl)sulfonyl-3,4-dihydropyrazole-2-carboximidamide
—— 1-{[4-(trifluoromethyl)phenyl]ethynyl}benzo[c]-1,8-naphthyridin-6(5H)-one 1186376-83-9 C21H11F3N2O
1-{[4-(trifluoromethyl)phenyl]ethynyl}benzo[c]-1,8-naphthyridin-6(5H)-one
—— N,N-diphenyl-4-[6,7,16,17-tetramethyl-15-[4-(N-phenylanilino)phenyl]-8,15-diazapentacyclo[11.7.0.02,10.05,9.014,18]icosa-1(13),2(10),3,5(9),6,11,14(18),16,19-nonaen-8-yl]aniline 1268697-08-0 C58H46N4
N,N-diphenyl-4-[6,7,16,17-tetramethyl-15-[4-(N-phenylanilino)phenyl]-8,15-diazapentacyclo[11.7.0.02,10.05,9.014,18]icosa-1(13),2(10),3,5(9),6,11,14(18),16,19-nonaen-8-yl]aniline
—— 5-Bromo-4-(chloromethyl)-1,3-thiazole 1936260-42-2 C4H3BrClNS
5-Bromo-4-(chloromethyl)-1,3-thiazole
—— N-{2-[6-(biphenyl-2-yloxy)-hexahydro-pyrrolo[3,2-b]pyrrol-1-yl]-1-cyclohexyl-2-oxo-ethyl}-2-methylamino-propionamide 1257233-23-0 C30H40N4O3
N-{2-[6-(biphenyl-2-yloxy)-hexahydro-pyrrolo[3,2-b]pyrrol-1-yl]-1-cyclohexyl-2-oxo-ethyl}-2-methylamino-propionamide
—— 1-(tert-butoxycarbonyl)-4-methylazetidine-2-carboxylic acid 1822530-58-4 C10H17NO4
1-(tert-butoxycarbonyl)-4-methylazetidine-2-carboxylic acid
—— 11-ethyl-2-methoxy-6,11-dihydro-5H-dibenz[b,e]azepine 1228434-98-7 C17H19NO
11-ethyl-2-methoxy-6,11-dihydro-5H-dibenz[b,e]azepine
—— 4-methylpentanesulfonic acid 1048111-02-9 C6H14O3S
4-methylpentanesulfonic acid
—— N-hydroxy-2-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide 1259297-14-7 C18H20N2O3
N-hydroxy-2-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide
—— 8-({4-[4-(4-ethylpiperazin-1-yl)cyclohexyl]phenyl}amino)-6-(pyrimidin-5-yl)-1,2-dihydro-2,7-naphthyridin-1-one 1263390-06-2 C30H35N7O
8-({4-[4-(4-ethylpiperazin-1-yl)cyclohexyl]phenyl}amino)-6-(pyrimidin-5-yl)-1,2-dihydro-2,7-naphthyridin-1-one
—— 2-(2,1,3-benzoxadiazol-5-ylmethyl)-N-hydroxy-1,2,3,4-tetrahydroisoquinoline-6-carboxamide 1259297-16-9 C17H16N4O3
2-(2,1,3-benzoxadiazol-5-ylmethyl)-N-hydroxy-1,2,3,4-tetrahydroisoquinoline-6-carboxamide
—— N-(3-chloro-4-hydroxyphenyl)sulfonyl-N'-ethyl-2,3-diazaspiro[4.4]non-3-ene-2-carboximidamide 1187965-93-0 C16H21ClN4O3S
N-(3-chloro-4-hydroxyphenyl)sulfonyl-N'-ethyl-2,3-diazaspiro[4.4]non-3-ene-2-carboximidamide
—— 11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-1,5,7,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-2(27),3,5,8(26),9,11,16-heptaene 1083089-70-6 C27H37N5O3
11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-1,5,7,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-2(27),3,5,8(26),9,11,16-heptaene
—— N-[4-[2-(methoxymethyl)phenyl]but-3-ynyl]thieno[3,2-d]pyrimidin-4-amine 1262024-75-8 C18H17N3OS
N-[4-[2-(methoxymethyl)phenyl]but-3-ynyl]thieno[3,2-d]pyrimidin-4-amine
—— 2-((2-furfurylidenehydrazono)(4-methoxyphenyl)methyl)-4'-methoxybenzophenone 1390649-53-2 C27H22N2O4
2-((2-furfurylidenehydrazono)(4-methoxyphenyl)methyl)-4'-methoxybenzophenone
—— Yxa2JN5ftq 1217800-23-1 C23H30N2O2
Yxa2JN5ftq
—— N-{[4-({[5-phenylsulfonyl-2-trifluoromethyl-phenyl]thio}methyl)piperidin-1-yl]carbonyl}glycine 1027094-61-6 C22H23F3N2O5S2
N-{[4-({[5-phenylsulfonyl-2-trifluoromethyl-phenyl]thio}methyl)piperidin-1-yl]carbonyl}glycine
—— 2-(4-(difluoromethoxy)phenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)-5-(trifluoromethyl)benzamide 1620846-79-8 C20H13F5N2O4
2-(4-(difluoromethoxy)phenoxy)-N-(2-oxo-1,2-dihydropyridin-4-yl)-5-(trifluoromethyl)benzamide
—— 3-(4-chlorophenyl)-7-(3-fluorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one 1621967-23-4 C18H10ClFN2OS
3-(4-chlorophenyl)-7-(3-fluorophenyl)thieno[3,2-d]pyrimidin-4(3H)-one
—— N-(2,2-dimethylpropyl)-2-fluoro-6-(2-((4aS,5R)-1-(4-fluorophenyl)-5-hydroxy-4a-methyl-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl)ethyl)benzamide 1021537-77-8 C31H35F2N3O2
N-(2,2-dimethylpropyl)-2-fluoro-6-(2-((4aS,5R)-1-(4-fluorophenyl)-5-hydroxy-4a-methyl-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl)ethyl)benzamide
—— N-(1-(1-(3-fluorobenzyl)-1H-benzo[d]imidazol-2-yl)piperidin-4-yl)tetrahydrothiophene-3-sulfonamide 1,1-dioxide 1568976-89-5 C23H27FN4O4S2
N-(1-(1-(3-fluorobenzyl)-1H-benzo[d]imidazol-2-yl)piperidin-4-yl)tetrahydrothiophene-3-sulfonamide 1,1-dioxide
—— 8-(tert-butylamino)-2-(2-hydroxyethyl)-6-[(6-{[1-(2-hydroxyethyl)piperidin-4-yl]oxy}pyrimidin-4-yl)amino]-1,2-dihydro-2,7-naphthyridin-1-one 1263395-43-2 C25H35N7O4
8-(tert-butylamino)-2-(2-hydroxyethyl)-6-[(6-{[1-(2-hydroxyethyl)piperidin-4-yl]oxy}pyrimidin-4-yl)amino]-1,2-dihydro-2,7-naphthyridin-1-one
—— 6-{[1-({4-[2-(4-ethylpiperazin-1-yl)ethyl]phenyl}amino)-8-oxo-7,8-dihydro-2,7-naphthyridin-3-yl]amino}pyridine-3-carboxylic acid 1263394-78-0 C28H31N7O3
6-{[1-({4-[2-(4-ethylpiperazin-1-yl)ethyl]phenyl}amino)-8-oxo-7,8-dihydro-2,7-naphthyridin-3-yl]amino}pyridine-3-carboxylic acid
—— 6-(2-(2-(2-fluoroethoxy)ethoxy)ethoxy)-9-(methoxymethyl)-N,N-dimethyl-9H-carbazol-3-amine 1181376-36-2 C22H29FN2O4
6-(2-(2-(2-fluoroethoxy)ethoxy)ethoxy)-9-(methoxymethyl)-N,N-dimethyl-9H-carbazol-3-amine
—— N-[(2-chloro-4-fluorophenyl)methyl]-2-[3,5-dimethyl-1-(6-methyl-3-pyridinyl)-1H-pyrazol-4-yl]acetamide 1082826-87-6 C20H20ClFN4O
N-[(2-chloro-4-fluorophenyl)methyl]-2-[3,5-dimethyl-1-(6-methyl-3-pyridinyl)-1H-pyrazol-4-yl]acetamide
—— butyl-[2-(3,4-dimethoxy-phenyl)-benzofuran-5-yl]-amine 1018948-84-9 C20H23NO3
butyl-[2-(3,4-dimethoxy-phenyl)-benzofuran-5-yl]-amine
—— 4-chloro-1-(phenylsulfonyl)-N-(2-pyridin-3-ylethyl)-1H-indole-3-sulfonamide 1027068-81-0 C21H18ClN3O4S2
4-chloro-1-(phenylsulfonyl)-N-(2-pyridin-3-ylethyl)-1H-indole-3-sulfonamide
—— (4-chlorobenzyl)-[5-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrimidin-2-yl]amine 1029047-73-1 C19H16ClN5
(4-chlorobenzyl)-[5-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrimidin-2-yl]amine
—— 2-(3-(2-fluorophenethyl)-4-oxo-5-(trifluoromethyl)-3,4-dihydroquinazolin-2-yl)benzonitrile 1018678-24-4 C24H15F4N3O
2-(3-(2-fluorophenethyl)-4-oxo-5-(trifluoromethyl)-3,4-dihydroquinazolin-2-yl)benzonitrile
—— 4-(3-cyclopentyl-propionyl)-[1,4]diazepane-1-carboxylic acid (4-ethyl-phenyl)-amide 1028851-43-5 C22H33N3O2
4-(3-cyclopentyl-propionyl)-[1,4]diazepane-1-carboxylic acid (4-ethyl-phenyl)-amide
—— 2-formyl-4-methoxy-butyric acid methyl ester 1058159-85-5 C7H12O4
2-formyl-4-methoxy-butyric acid methyl ester
—— ((4S,5S)-5-((1S,2S)-3-benzamido-2-(benzo[d][1,3]dioxol-5-yl)-1-(methoxymethoxy)propyl)-2,2-dimethyl-1,3-dioxolan-4-yl)methyl 4-methylbenzenesulfonate 1226976-45-9 C32H37NO10S
((4S,5S)-5-((1S,2S)-3-benzamido-2-(benzo[d][1,3]dioxol-5-yl)-1-(methoxymethoxy)propyl)-2,2-dimethyl-1,3-dioxolan-4-yl)methyl 4-methylbenzenesulfonate
—— 2-(4-(((2-(2,4-Dimethylphenylamino)-2-oxoethyl)(4-methoxybenzyl)amino)methyl)phenoxy)-2-methylpropanoic acid 1235514-82-5 C29H34N2O5
2-(4-(((2-(2,4-Dimethylphenylamino)-2-oxoethyl)(4-methoxybenzyl)amino)methyl)phenoxy)-2-methylpropanoic acid
—— 3-(Ethanesulfonyl)-2-ethyl-4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)benzoic acid 1355555-11-1 C14H13F7O4S
3-(Ethanesulfonyl)-2-ethyl-4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)benzoic acid
—— N-acetyl-N-tert-butylmorpholine-4-carboxamide 1542248-05-4 C11H20N2O3
N-acetyl-N-tert-butylmorpholine-4-carboxamide