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中文名称 英文名称 CAS号 化学式 结构式图片
—— benzyl-(3-bromo-quinolin-2-ylmethyl)-carbamic acid tert-butyl ester 1219696-53-3 C22H23BrN2O2
benzyl-(3-bromo-quinolin-2-ylmethyl)-carbamic acid tert-butyl ester
—— 7-[4-(2-phenylethyl)piperazine-1-carbonyl]-1-propyl-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one 1243157-57-4 C25H28N6O2
7-[4-(2-phenylethyl)piperazine-1-carbonyl]-1-propyl-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one
—— 5-propyl-2,3-dihydro-1H-phenothiazin-4-one 106513-71-7 C15H17NOS
5-propyl-2,3-dihydro-1H-phenothiazin-4-one
—— (2R,5S)-5-(5,5-dimethyl-2-oxo-oxazolidin-3-ylmethyl)-4-{2-[6-(4-fluoro-benzyl)-3,3-dimethyl-2,3-dihydro-pyrrolo[3,2-b]pyridin-1-yl]-2-oxo-ethyl}-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1605312-05-7 C34H46FN5O5
(2R,5S)-5-(5,5-dimethyl-2-oxo-oxazolidin-3-ylmethyl)-4-{2-[6-(4-fluoro-benzyl)-3,3-dimethyl-2,3-dihydro-pyrrolo[3,2-b]pyridin-1-yl]-2-oxo-ethyl}-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— 1-((1R,8S,8aS)-8-Hydroxy-1,2,3,5,6,7,8,8a-octahydro-naphthalen-1-yl)-ethanone 126397-39-5 C12H18O2
1-((1R,8S,8aS)-8-Hydroxy-1,2,3,5,6,7,8,8a-octahydro-naphthalen-1-yl)-ethanone
—— prop-2-enyl N-(4-bromophenyl)-4-methoxybenzenecarboximidate 1337937-60-6 C17H16BrNO2
prop-2-enyl N-(4-bromophenyl)-4-methoxybenzenecarboximidate
—— 3,7,7-trimethyl-4-(4-(trifluoromethyl)phenyl)-6,7,8,9-tetrahydro-2H-pyrazolo[3,4-b]quinolin-5(4H)-one 1597439-13-8 C20H20F3N3O
3,7,7-trimethyl-4-(4-(trifluoromethyl)phenyl)-6,7,8,9-tetrahydro-2H-pyrazolo[3,4-b]quinolin-5(4H)-one
—— 2-Methyl-2-[[4-[5-[4-(2-methylphenyl)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]methylamino]propanoic acid 1355157-97-9 C27H24F3N3O3
2-Methyl-2-[[4-[5-[4-(2-methylphenyl)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenyl]methylamino]propanoic acid
—— 2-((3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)methyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one 1354198-66-5 C21H18F3N5O2
2-((3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)methyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— {4-chloro-2-[(5-isobutylsulfonyl-2-methylphenyl)ethynyl]phenoxy}acetic acid 1240285-60-2 C21H21ClO5S
{4-chloro-2-[(5-isobutylsulfonyl-2-methylphenyl)ethynyl]phenoxy}acetic acid
—— 1-[2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carbonyl]-piperidine-4-carboxylic acid methyl ester 1333399-64-6 C27H28N4O4
1-[2'-aminomethyl-5'-(pyridin-4-ylcarbamoyl)-biphenyl-3-carbonyl]-piperidine-4-carboxylic acid methyl ester
—— 12-[2-(3-ethylbenzylamino)-1-hydroxyethyl]-16-fluoro-9-isopropyl-2-oxa-8,11-diazabicyclo[12.3.1]octadeca-1(17),14(18),15-triene-7,10-dione 1175396-84-5 C29H40FN3O4
12-[2-(3-ethylbenzylamino)-1-hydroxyethyl]-16-fluoro-9-isopropyl-2-oxa-8,11-diazabicyclo[12.3.1]octadeca-1(17),14(18),15-triene-7,10-dione
—— 12-{2-[(5-ethylpyridin-3-ylmethyl)amino]-1-hydroxyethyl}-16-fluoro-2-oxa-8,11-diazabicyclo[12.2.2]octadeca-1(17),14(18),15-triene-7,10-dione 1175397-74-6 C25H33FN4O4
12-{2-[(5-ethylpyridin-3-ylmethyl)amino]-1-hydroxyethyl}-16-fluoro-2-oxa-8,11-diazabicyclo[12.2.2]octadeca-1(17),14(18),15-triene-7,10-dione
—— t-butyl 4-[N-(t-butoxycarbonyl)-N-(methyl)amino-methyl]-3-nitrobenzoate 165529-27-1 C18H26N2O6
t-butyl 4-[N-(t-butoxycarbonyl)-N-(methyl)amino-methyl]-3-nitrobenzoate
—— (2R,5S)-4-{2-[6-(4-fluoro-benzyl)-3,3-dimethyl-2,3-dihydro-pyrrolo[3,2-b]pyridin-1-yl]-2-oxo-ethyl}-2-methyl-5-(5-oxo-5,7-dihydro-pyrrolo[3,4-b]pyridin-6-ylmethyl)-piperazine-1-carboxylic acid tert-butyl ester 1605315-03-4 C36H43FN6O4
(2R,5S)-4-{2-[6-(4-fluoro-benzyl)-3,3-dimethyl-2,3-dihydro-pyrrolo[3,2-b]pyridin-1-yl]-2-oxo-ethyl}-2-methyl-5-(5-oxo-5,7-dihydro-pyrrolo[3,4-b]pyridin-6-ylmethyl)-piperazine-1-carboxylic acid tert-butyl ester
—— ethyl 7-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxylate 1391938-58-1 C11H13NO3
ethyl 7-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxylate
—— 2-(3-(2-((4-(4-ethylpiperazin-1-yl)-3-fluorophenyl)amino)-5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)acetonitrile 1239875-91-2 C27H28FN7
2-(3-(2-((4-(4-ethylpiperazin-1-yl)-3-fluorophenyl)amino)-5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)acetonitrile
—— N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-2-(5-phenyl-1H-imidazol-2-yl)pyridine-3-carboxamide 1241025-06-8 C25H21N5O3
N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-2-(5-phenyl-1H-imidazol-2-yl)pyridine-3-carboxamide
—— N-(4-chloro-3-(trifluoromethyl)benzyl)-2-methyl-1,8-naphthyridine-3-carboxamide 1241909-52-3 C18H13ClF3N3O
N-(4-chloro-3-(trifluoromethyl)benzyl)-2-methyl-1,8-naphthyridine-3-carboxamide
—— 1-(4-{3-phenyl-5-[2-(tetrahydro-2H-pyran-4-yl)ethoxy]-1,6-naphthyridin-2-yl}phenyl)methanamine 1238318-98-3 C28H29N3O2
1-(4-{3-phenyl-5-[2-(tetrahydro-2H-pyran-4-yl)ethoxy]-1,6-naphthyridin-2-yl}phenyl)methanamine
—— 8-cyclobutyl-2-(pyrimidin-2-yl)-1,2,3,6,7,8,9,10-octahydro-[1,4]diazepino[1',7':1,2]imidazo[4,5-f]isoindole 1239878-60-4 C21H24N6
8-cyclobutyl-2-(pyrimidin-2-yl)-1,2,3,6,7,8,9,10-octahydro-[1,4]diazepino[1',7':1,2]imidazo[4,5-f]isoindole
—— (6-bromo-3-chloro-8-trifluoromethyl-imidazo[1,2-a]pyridin-2-yl)-(3-fluoro-3',6'-dihydro-2'H-[2,4']bipyridinyl-1'-yl)-methanone 1239205-28-7 C19H12BrClF4N4O
(6-bromo-3-chloro-8-trifluoromethyl-imidazo[1,2-a]pyridin-2-yl)-(3-fluoro-3',6'-dihydro-2'H-[2,4']bipyridinyl-1'-yl)-methanone
—— 3-methylbut-2-enyl (2S)-2-[[4-(2-cyanophenyl)phenyl]methyl-pentanoylamino]-3-methylbutanoate 1298055-63-6 C29H36N2O3
3-methylbut-2-enyl (2S)-2-[[4-(2-cyanophenyl)phenyl]methyl-pentanoylamino]-3-methylbutanoate
—— 8-methyl-9-phenyl-N-(2-prop-2-enoxyphenyl)-5,6-dihydropyrazolo[3,4-h]quinazolin-2-amine 1356588-88-9 C25H23N5O
8-methyl-9-phenyl-N-(2-prop-2-enoxyphenyl)-5,6-dihydropyrazolo[3,4-h]quinazolin-2-amine
—— 2-methoxy-N-(3-(3-(trifluoromethyl)benzamido)phenyl)benzamide 1202038-25-2 C22H17F3N2O3
2-methoxy-N-(3-(3-(trifluoromethyl)benzamido)phenyl)benzamide
—— 1-[4-(2-pyrrolidin-1-ylethoxy)benzoyl]-2-phenylnaphthalene, citrate salt 170847-24-2 C6H8O7*C29H27NO2
1-[4-(2-pyrrolidin-1-ylethoxy)benzoyl]-2-phenylnaphthalene, citrate salt
—— N-[3-[(4S)-2-amino-4-methyl-1,3-thiazin-4-yl]-4-fluorophenyl]-5-(2-methoxyethoxy)pyridine-2-carboxamide 1200494-10-5 C20H21FN4O3S
N-[3-[(4S)-2-amino-4-methyl-1,3-thiazin-4-yl]-4-fluorophenyl]-5-(2-methoxyethoxy)pyridine-2-carboxamide
—— 4-(1-(4-methyl-3-(5-(methylsulfonyl)-4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)benzoyl)piperidin-4-yl)benzonitrile 1399175-90-6 C27H29N5O3S
4-(1-(4-methyl-3-(5-(methylsulfonyl)-4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)benzoyl)piperidin-4-yl)benzonitrile
—— {4-[cyclobutyl(difluoro)methyl]phenyl}methanol 1400701-90-7 C12H14F2O
{4-[cyclobutyl(difluoro)methyl]phenyl}methanol
—— 7-(2-fluoro-4-methanesulfonylphenyl)-4-[1-(5-cyclopropylpyrimidin-2-yl)piperidin-4-yloxy]thieno[3,2-d]pyrimidine 1384951-27-2 C25H24FN5O3S2
7-(2-fluoro-4-methanesulfonylphenyl)-4-[1-(5-cyclopropylpyrimidin-2-yl)piperidin-4-yloxy]thieno[3,2-d]pyrimidine
—— 1-[(1S,3R,4R,7S)-7-hydroxy-1-(hydroxymethyl)-2,5-dioxabicyclo[2.2.1]heptan-3-yl]-5-(1,3-thiazol-2-yl)pyrimidine-2,4-dione 1314716-24-9 C13H13N3O6S
1-[(1S,3R,4R,7S)-7-hydroxy-1-(hydroxymethyl)-2,5-dioxabicyclo[2.2.1]heptan-3-yl]-5-(1,3-thiazol-2-yl)pyrimidine-2,4-dione
—— 7-[3-(butylsulfamoyl)anilino]-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214931-73-3 C24H27N5O4S
7-[3-(butylsulfamoyl)anilino]-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— N-tert-butyl-5-(8-fluoro-2-(3-(2-oxo-2-(pyrrolidin-1-yl)ethyl)ureido)-[1,2,4]triazolo[1,5-a]pyridin-6-yl)pyridine-3-sulfonamide 1240282-45-4 C22H27FN8O4S
N-tert-butyl-5-(8-fluoro-2-(3-(2-oxo-2-(pyrrolidin-1-yl)ethyl)ureido)-[1,2,4]triazolo[1,5-a]pyridin-6-yl)pyridine-3-sulfonamide
—— 2-[(2-Chlorophenyl)methylamino]-1-[[3-(trifluoromethoxy)phenyl]methyl]imidazo[4,5-b]pyridine-5-carboxamide 1202159-43-0 C22H17ClF3N5O2
2-[(2-Chlorophenyl)methylamino]-1-[[3-(trifluoromethoxy)phenyl]methyl]imidazo[4,5-b]pyridine-5-carboxamide
—— (S)-3-{4-propyl-6-[3-(pyridin-2-ylmethylamino)pyrrolidin-1-yl]pyrimidin-2-ylamino}benzonitrile 1394314-94-3 C24H27N7
(S)-3-{4-propyl-6-[3-(pyridin-2-ylmethylamino)pyrrolidin-1-yl]pyrimidin-2-ylamino}benzonitrile
—— 2-(4-(3-(1-(quinolin-6-yl)cyclopropyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)-1H-pyrazol-1-yl)ethanol 1313724-18-3 C22H19N7O
2-(4-(3-(1-(quinolin-6-yl)cyclopropyl)-3H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)-1H-pyrazol-1-yl)ethanol
—— (5R,8S)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-vinylcyclopropyl}-7-{(2S)-2-[({(1S)-2,2-dimethyl-1-[(4-methylpiperazin-1-yl)methyl]propyl}carbamoyl)amino]-3,3-dimethylbutanoyl}-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide 1247707-90-9 C39H65N7O6S
(5R,8S)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-vinylcyclopropyl}-7-{(2S)-2-[({(1S)-2,2-dimethyl-1-[(4-methylpiperazin-1-yl)methyl]propyl}carbamoyl)amino]-3,3-dimethylbutanoyl}-10,10-dimethyl-7-azadispiro[3.0.4.1]decane-8-carboxamide
—— 1-{5-({1-[(3,5-difluoro-4-pyridinyl)methyl]-1H-pyrazol-3-yl}amino)-1,3,4-thiadiazol-2-yl}-1-(4-methyl-1,3-thiazol-2-yl)ethanol 1372891-26-3 C17H15F2N7OS2
1-{5-({1-[(3,5-difluoro-4-pyridinyl)methyl]-1H-pyrazol-3-yl}amino)-1,3,4-thiadiazol-2-yl}-1-(4-methyl-1,3-thiazol-2-yl)ethanol
—— 2-{1-[2-(1H-indol-6-ylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol 1394803-87-2 C22H29N5O
2-{1-[2-(1H-indol-6-ylamino)-6-propylpyrimidin-4-yl]piperidin-2-yl}ethanol
—— 4-nitro-3-(3,4,5-trimethoxyphenoxy)phenol 1393831-68-9 C15H15NO7
4-nitro-3-(3,4,5-trimethoxyphenoxy)phenol
—— 4-(2-methyl-3-propionyl-5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1H-pyrrol-1-yl)benzenesulfonamide 1392286-11-1 C24H26N2O3S
4-(2-methyl-3-propionyl-5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1H-pyrrol-1-yl)benzenesulfonamide
—— 1-(4-(benzyloxy)-3-chlorobenzyl)azetidine-3-carboxylic acid 1240307-27-0 C18H18ClNO3
1-(4-(benzyloxy)-3-chlorobenzyl)azetidine-3-carboxylic acid
—— N-(2-methyl-6-(methylsulfonyl)pyridin-3-yl)-3-(1-(pyrimidin-2-yl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyrazin-8-amine 1236354-57-6 C22H22N8O2S
N-(2-methyl-6-(methylsulfonyl)pyridin-3-yl)-3-(1-(pyrimidin-2-yl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyrazin-8-amine
—— 3-ethoxycarbonyl-6-(5-fluoro-2H-spiro[benzofuran-3,4'-piperidine]-1'-ylcarbonyl)-7-(2-methylphenylamino)pyrazolo[1,5-a]pyrimidine 1138521-66-0 C29H28FN5O4
3-ethoxycarbonyl-6-(5-fluoro-2H-spiro[benzofuran-3,4'-piperidine]-1'-ylcarbonyl)-7-(2-methylphenylamino)pyrazolo[1,5-a]pyrimidine
—— (2S)-1-{4-[(5-fluoro-1-methyl-1H-benzimidazol-2-yl)oxy]piperidin-1-yl}-3-methyl-1-oxobutan-2-amine hydrochloride 1189550-65-9 C18H25FN4O2*ClH
(2S)-1-{4-[(5-fluoro-1-methyl-1H-benzimidazol-2-yl)oxy]piperidin-1-yl}-3-methyl-1-oxobutan-2-amine hydrochloride
—— 6,7-dichloro-4-(1-methylcyclopropyl)-4H-1,2,4-benzothiadiazine 1,1-dioxide 1204574-36-6 C11H10Cl2N2O2S
6,7-dichloro-4-(1-methylcyclopropyl)-4H-1,2,4-benzothiadiazine 1,1-dioxide
—— 2-bromothieno[2,3-c]furan-6(4H)-one 1374574-30-7 C6H3BrO2S
2-bromothieno[2,3-c]furan-6(4H)-one
—— (3S,5S)-5-(3-cyclopentyloxy-4-methoxyphenyl)-3-(pyridin-3-ylmethyl)piperidin-2-one 1058223-06-5 C23H28N2O3
(3S,5S)-5-(3-cyclopentyloxy-4-methoxyphenyl)-3-(pyridin-3-ylmethyl)piperidin-2-one
—— 2-(benzylamino)-1-(4,5-dimethoxy-2-nitrophenyl)-2-oxoethyl 4-methoxybenzoate 1622384-53-5 C25H24N2O8
2-(benzylamino)-1-(4,5-dimethoxy-2-nitrophenyl)-2-oxoethyl 4-methoxybenzoate
—— 2-chloro-N-(2,6-diisopropylphenyl)-5-methylaniline 1227188-09-1 C19H24ClN
2-chloro-N-(2,6-diisopropylphenyl)-5-methylaniline