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中文名称 英文名称 CAS号 化学式 结构式图片
—— —— 137648-22-7 C26H38O3
—— —— 1609529-42-1 C19H18FN5O3S
—— N-[(2-chlorophenyl)methyl]-8-(4-fluorophenyl)-9-(2-piperidin-4-ylethyl)purin-2-amine 1021696-53-6 C25H26ClFN6
N-[(2-chlorophenyl)methyl]-8-(4-fluorophenyl)-9-(2-piperidin-4-ylethyl)purin-2-amine
—— 4-butyl-5-[(2'-carboxybiphenyl-4-yl)methyl]-6-[(3-carboxythien-2-yl) methoxy]-2-methylpyrimidine 148564-19-6 C29H28N2O5S
4-butyl-5-[(2'-carboxybiphenyl-4-yl)methyl]-6-[(3-carboxythien-2-yl) methoxy]-2-methylpyrimidine
—— 1-{2-[(3R,4S)-4-amino-3-hydroxy-1-piperidinyl]ethyl}-1,5-naphthyridin-2(1H)-one 1173897-81-8 C15H20N4O2
1-{2-[(3R,4S)-4-amino-3-hydroxy-1-piperidinyl]ethyl}-1,5-naphthyridin-2(1H)-one
—— 1-fluoro-4-((3-methylenepentan-2-yl)oxy)benzene 1352740-20-5 C12H15FO
1-fluoro-4-((3-methylenepentan-2-yl)oxy)benzene
—— 1-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-phenylpiperidin-3-yl}methaneamine 1178882-08-0 C16H22N4O2S
1-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-phenylpiperidin-3-yl}methaneamine
—— 7-((4-fluorophenyl)ethynyl)-3-propylquinazolin-4(3H)-one 1312448-40-0 C19H15FN2O
7-((4-fluorophenyl)ethynyl)-3-propylquinazolin-4(3H)-one
—— [4-[(2S)-3-[[(3S,6S,10aS)-3-[[(2S)-5-amino-1-(benzylamino)-1,5-dioxopentan-2-yl]carbamoyl]-5-oxo-2,3,6,7,8,9,10,10a-octahydro-1H-pyrrolo[1,2-a]azocin-6-yl]amino]-2-amino-3-oxopropyl]phenyl]methylphosphonic acid 1233085-38-5 C33H45N6O8P
[4-[(2S)-3-[[(3S,6S,10aS)-3-[[(2S)-5-amino-1-(benzylamino)-1,5-dioxopentan-2-yl]carbamoyl]-5-oxo-2,3,6,7,8,9,10,10a-octahydro-1H-pyrrolo[1,2-a]azocin-6-yl]amino]-2-amino-3-oxopropyl]phenyl]methylphosphonic acid
—— 4-((3R,4R)-3-(6-imidazo[1,5-a]pyrrolo[2,3-e]pyrazin-1-yl)-4-methylpiperidin-1-yl)-4-oxobutanenitrile 1310724-07-2 C18H20N6O
4-((3R,4R)-3-(6-imidazo[1,5-a]pyrrolo[2,3-e]pyrazin-1-yl)-4-methylpiperidin-1-yl)-4-oxobutanenitrile
—— ethyl 3-[2-[1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]ethyl]-3,4-difluorophenyl]propanoate 1232405-74-1 C29H39F2NO4
ethyl 3-[2-[1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]ethyl]-3,4-difluorophenyl]propanoate
—— (S)-2-(5-((5-chloro-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)-2,3-dihydro-1H-inden-1-yl)acetic acid 1234843-70-9 C22H23ClO4
(S)-2-(5-((5-chloro-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)-2,3-dihydro-1H-inden-1-yl)acetic acid
—— 3-[4-(2,4-Dichlorophenyl)piperazin-1-yl]-1-[4-[4-nitro-3-(trifluoromethyl)phenoxy]piperidin-1-yl]propan-1-one 1247031-31-7 C25H27Cl2F3N4O4
3-[4-(2,4-Dichlorophenyl)piperazin-1-yl]-1-[4-[4-nitro-3-(trifluoromethyl)phenoxy]piperidin-1-yl]propan-1-one
—— methyl N[(2S)-1-({4[1-(propan-2-yl)-3-(2,4,5-trifluoro-3-methanesulfonamidophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)propan-2-yl]carbamate 1269440-30-3 C22H26F3N7O4S
methyl N[(2S)-1-({4[1-(propan-2-yl)-3-(2,4,5-trifluoro-3-methanesulfonamidophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)propan-2-yl]carbamate
—— 2-((1-phenylprop-2-yn-1-yl)oxy)isoindoline-1,3-dione 1226968-93-9 C17H11NO3
2-((1-phenylprop-2-yn-1-yl)oxy)isoindoline-1,3-dione
—— (2S,4S,5S)-5-Amino-6-cyclohexyl-4-hydroxy-2-isopropyl-hexanoic acid {(1S,2S)-2-methyl-1-[(pyridin-2-ylmethyl)-carbamoyl]-butyl}-amide; hydrochloride 136520-80-4 C27H46N4O3*2ClH
(2S,4S,5S)-5-Amino-6-cyclohexyl-4-hydroxy-2-isopropyl-hexanoic acid {(1S,2S)-2-methyl-1-[(pyridin-2-ylmethyl)-carbamoyl]-butyl}-amide; hydrochloride
—— N-(3-propan-2-yl-3,4,10,11-tetrazatricyclo[8.3.0.02,6]trideca-1(13),2(6),4,11-tetraen-12-yl)acetamide 1221884-35-0 C14H19N5O
N-(3-propan-2-yl-3,4,10,11-tetrazatricyclo[8.3.0.02,6]trideca-1(13),2(6),4,11-tetraen-12-yl)acetamide
—— 1-[(4-Chlorophenyl)methyl]-3-(2-hydroxyethyl)-6-(4-phenoxyanilino)-1,3,5-triazine-2,4-dione 1239688-66-4 C24H21ClN4O4
1-[(4-Chlorophenyl)methyl]-3-(2-hydroxyethyl)-6-(4-phenoxyanilino)-1,3,5-triazine-2,4-dione
—— ethyl 3-(3-fluoro-4-hydroxy-2-propylphenyl)propanoate 1234845-91-0 C14H19FO3
ethyl 3-(3-fluoro-4-hydroxy-2-propylphenyl)propanoate
—— N-[4-bromo-2-methyl-6-(methylcarbamoyl)phenyl]-5-(2-chlorophenyl)-2-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]-1,3-oxazole-4-carboxamide 1352315-38-8 C22H16BrClF3N7O3
N-[4-bromo-2-methyl-6-(methylcarbamoyl)phenyl]-5-(2-chlorophenyl)-2-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]-1,3-oxazole-4-carboxamide
—— 5-fluoro-6-(4-morpholinyl)-3-pyridinamine 1244642-62-3 C9H12FN3O
5-fluoro-6-(4-morpholinyl)-3-pyridinamine
—— 2-[5-[2-(5-Propoxyspiro[3,4-dihydrochromene-2,4'-piperidine]-1'-yl)-1,3-thiazol-5-yl]tetrazol-2-yl]acetic acid 1241952-79-3 C22H26N6O4S
2-[5-[2-(5-Propoxyspiro[3,4-dihydrochromene-2,4'-piperidine]-1'-yl)-1,3-thiazol-5-yl]tetrazol-2-yl]acetic acid
—— (R)-8-cyclohexyl-6-(4-(2-(2-methoxyphenyl)acetyl)-3-methylpiperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-82-7 C29H36N4O3
(R)-8-cyclohexyl-6-(4-(2-(2-methoxyphenyl)acetyl)-3-methylpiperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— 2-(((3-chloropyridin-2-yl)methyl)thio)-N-((1,3-dimethyl-1H-pyrazol-4-yl)methyl)-1-(4-fluorophenyl)-N-methyl-1H-imidazole-5-carboxamide 1416264-24-8 C23H22ClFN6OS
2-(((3-chloropyridin-2-yl)methyl)thio)-N-((1,3-dimethyl-1H-pyrazol-4-yl)methyl)-1-(4-fluorophenyl)-N-methyl-1H-imidazole-5-carboxamide
—— 2-(2-(pyrazin-2-yl)ethyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one 1354199-62-4 C19H14F3N5O2
2-(2-(pyrazin-2-yl)ethyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— 1-methyl-5-phenyl-3-(thiophen-3-yl)-4,5-dihydro-1H-pyrazole 1334222-46-6 C14H14N2S
1-methyl-5-phenyl-3-(thiophen-3-yl)-4,5-dihydro-1H-pyrazole
—— 4-(4-methylpyridin-3-yl)-1-o-tolyl-1H-pyrazolo[3,4-b]pyridine 1356054-02-8 C19H16N4
4-(4-methylpyridin-3-yl)-1-o-tolyl-1H-pyrazolo[3,4-b]pyridine
—— 4-(4-{[4-(4-chlorophenyl)-6,6-dimethyl-5,6-dihydro-2H-pyran-3-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-N-({4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]-3-[(trifluoromethyl)sulfonyl]phenyl}sulfonyl)benzamide 1257044-85-1 C45H48ClF3N6O8S2
4-(4-{[4-(4-chlorophenyl)-6,6-dimethyl-5,6-dihydro-2H-pyran-3-yl]methyl}piperazin-1-yl)-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-N-({4-[(tetrahydro-2H-pyran-4-ylmethyl)amino]-3-[(trifluoromethyl)sulfonyl]phenyl}sulfonyl)benzamide
—— ethyl (3-{2-[(1R)-1-({(5R)-3-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-oxo-1,3-oxazolidin-5-yl}methoxy)ethyl]phenyl}propoxy)acetate 1232407-17-8 C32H43NO6
ethyl (3-{2-[(1R)-1-({(5R)-3-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-oxo-1,3-oxazolidin-5-yl}methoxy)ethyl]phenyl}propoxy)acetate
—— 4-(4-((5-chloro-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)phenyl)butanoic acid 1234843-58-3 C21H23ClO4
4-(4-((5-chloro-2,2-dimethyl-2,3-dihydrobenzofuran-7-yl)methoxy)phenyl)butanoic acid
—— 6-amino-N'-hydroxy-2-(trifluoromethyl)pyridine-3-carboximidamide 1233243-97-4 C7H7F3N4O
6-amino-N'-hydroxy-2-(trifluoromethyl)pyridine-3-carboximidamide
—— ethyl 1-ethyl-6,6-dimethyl-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole-3-carboxylate 1233244-07-9 C13H20N2O3
ethyl 1-ethyl-6,6-dimethyl-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole-3-carboxylate
—— (2R)-2-[[(8R,11S,14R,17S)-8-benzyl-3,6,9,12,15-pentaoxo-14-(2-phenylethyl)-11-[(4-phenylphenyl)methyl]-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carbonyl]amino]propanoic acid 1211443-35-4 C50H52N6O8
(2R)-2-[[(8R,11S,14R,17S)-8-benzyl-3,6,9,12,15-pentaoxo-14-(2-phenylethyl)-11-[(4-phenylphenyl)methyl]-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carbonyl]amino]propanoic acid
—— N<sup>b</sup>-Ethyl-N<sup>b</sup>-(4-hydroxy-butyl)-tryptamin 1029-41-0 C16H24N2O
N<sup>b</sup>-Ethyl-N<sup>b</sup>-(4-hydroxy-butyl)-tryptamin
—— 4-(2-dimethylamino-1-[3-(3-fluoro-4-methoxy-benzoylamino)phenyl]ethylamino)quinazoline-8-carboxylic acid amide 1240474-49-0 C27H27FN6O3
4-(2-dimethylamino-1-[3-(3-fluoro-4-methoxy-benzoylamino)phenyl]ethylamino)quinazoline-8-carboxylic acid amide
—— N-[2-[[(4S,5R,6Z,9S,10S,12E)-9,10,18-trihydroxy-4,5-dimethyl-2,8-dioxo-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaen-16-yl]oxy]ethyl]acetamide 1228924-62-6 C23H29NO8
N-[2-[[(4S,5R,6Z,9S,10S,12E)-9,10,18-trihydroxy-4,5-dimethyl-2,8-dioxo-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaen-16-yl]oxy]ethyl]acetamide
—— 4-{[(S)-2-tert-butoxycarbonyl-7-dimethylamino-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]amino}-2,3,6-trimethylphenyl acetate 1370262-47-7 C28H37N3O5
4-{[(S)-2-tert-butoxycarbonyl-7-dimethylamino-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]amino}-2,3,6-trimethylphenyl acetate
—— 2-(2-Hydroxyphenyl)-2-(2-methylanilino)acetonitrile 1235590-64-3 C15H14N2O
2-(2-Hydroxyphenyl)-2-(2-methylanilino)acetonitrile
—— (S)-1-((R)-3-(6H-imidazo[1,5-a]pyrrolo[2,3-e]pyrazin-1-yl)piperidine-1-carbonyl)pyrrolidine-3-carbonitrile 1310725-05-3 C19H21N7O
(S)-1-((R)-3-(6H-imidazo[1,5-a]pyrrolo[2,3-e]pyrazin-1-yl)piperidine-1-carbonyl)pyrrolidine-3-carbonitrile
—— 3-(7-chlorospiro[benzo[b]pyrrolo[1,2-d][1,4]oxazine-4,4'-piperidine]-1'-ylcarbonyl)-1-ethylpyridin-2(1H)-one 1346615-52-8 C23H22ClN3O3
3-(7-chlorospiro[benzo[b]pyrrolo[1,2-d][1,4]oxazine-4,4'-piperidine]-1'-ylcarbonyl)-1-ethylpyridin-2(1H)-one
—— 1-(5-(4-(2-ethylphenylcarbamoyl)-3,4.dihydro-2H-benzo[b][1,4]oxazin-7-yl)pyrimidin-2-yl)pyrrolidine-3-carboxylic acid 1246211-36-8 C26H27N5O4
1-(5-(4-(2-ethylphenylcarbamoyl)-3,4.dihydro-2H-benzo[b][1,4]oxazin-7-yl)pyrimidin-2-yl)pyrrolidine-3-carboxylic acid
—— N-[(1-cyclohexylpiperidin-4-yl)methyl]-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide 1247035-48-8 C25H36F3N5O3
N-[(1-cyclohexylpiperidin-4-yl)methyl]-4-[4-nitro-3-(trifluoromethyl)anilino]piperidine-1-carboxamide
—— ethyl (2E)-3-(3-fluoro-6-{(1R)-1-[(2R)-oxiran-2-yl methoxy]ethyl}phenyl)prop-2-enoate 1232829-11-6 C16H19FO4
ethyl (2E)-3-(3-fluoro-6-{(1R)-1-[(2R)-oxiran-2-yl methoxy]ethyl}phenyl)prop-2-enoate
—— 8-[1-(4-Fluorophenyl)-5-(4-methoxyphenyl)pyrazol-3-yl]-1,4-dioxaspiro[4.5]decan-8-ol 1224949-76-1 C24H25FN2O4
8-[1-(4-Fluorophenyl)-5-(4-methoxyphenyl)pyrazol-3-yl]-1,4-dioxaspiro[4.5]decan-8-ol
—— 3-(Imidazo[1,2-a]pyridin-6-ylmethyl)-5-pyridin-4-yltriazolo[4,5-b]pyrazine 1313723-24-8 C17H12N8
3-(Imidazo[1,2-a]pyridin-6-ylmethyl)-5-pyridin-4-yltriazolo[4,5-b]pyrazine
—— N-cyclopropyl-N-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-oxazol-5-ylbenzamide 1400707-33-6 C24H27N5O2
N-cyclopropyl-N-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-oxazol-5-ylbenzamide
—— N-(7-(5-fluoro-2-methylphenyl)-5-(piperazin-1-yl)-2,6-naphthyridin-3-yl)cyclopropanecarboxamide 1382846-02-7 C23H24FN5O
N-(7-(5-fluoro-2-methylphenyl)-5-(piperazin-1-yl)-2,6-naphthyridin-3-yl)cyclopropanecarboxamide
—— 1-(4-fluorophenyl)-2-(2-methyl-1-(2,3,6-trifluorophenyl)propan-2-yl)-1H-imidazole-5-carboxylic acid 1416266-62-0 C20H16F4N2O2
1-(4-fluorophenyl)-2-(2-methyl-1-(2,3,6-trifluorophenyl)propan-2-yl)-1H-imidazole-5-carboxylic acid
—— N'-(3-fluoro-4-{[6-methoxy-7-({1-[(methylamino)-2-oxoethyl]piperidin-4-yl}methoxy)quinolin-4-yl]oxy}phenyl)-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide 1416320-92-7 C36H37F2N5O6
N'-(3-fluoro-4-{[6-methoxy-7-({1-[(methylamino)-2-oxoethyl]piperidin-4-yl}methoxy)quinolin-4-yl]oxy}phenyl)-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— ethyl 3-[2-[(1R)-1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]ethyl]-4-fluoro-5-methylphenyl]propanoate 1232405-31-0 C30H42FNO4
ethyl 3-[2-[(1R)-1-[(2R)-3-[[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino]-2-hydroxypropoxy]ethyl]-4-fluoro-5-methylphenyl]propanoate