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中文名称 英文名称 CAS号 化学式 结构式图片
—— [5-(2,2,2-trifluoro-acetyl)-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-yl]-carbamic acid tert-butyl ester 1454648-79-3 C13H16F3N3O3S
[5-(2,2,2-trifluoro-acetyl)-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-yl]-carbamic acid tert-butyl ester
—— (9H-fluoren-9-yl)methyl (S)-1-((benzo[b]thiophen-3-ylmethyl)((S)-1,1-diethoxypropan-2-yl)amino)-3-(4-tert-butoxyphenyl)-1-oxopropan-2-ylcarbamate 1198778-32-3 C44H50N2O6S
(9H-fluoren-9-yl)methyl (S)-1-((benzo[b]thiophen-3-ylmethyl)((S)-1,1-diethoxypropan-2-yl)amino)-3-(4-tert-butoxyphenyl)-1-oxopropan-2-ylcarbamate
—— (2,2-difluoro-ethyl)-(4-iodo-pyridin-3-yl)-amine 1395416-10-0 C7H7F2IN2
(2,2-difluoro-ethyl)-(4-iodo-pyridin-3-yl)-amine
—— N-{4-[4-(cyclobutylmethoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl}-2-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidin-5-yl)acetamide 1246275-32-0 C24H23F2N5O4S
N-{4-[4-(cyclobutylmethoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl}-2-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidin-5-yl)acetamide
—— (2S,4R)-N-(1-cyanocyclopropyl)-4-(2-methoxyphenylthio)pyrrolidine-2-carboxamide 1450977-55-5 C16H19N3O2S
(2S,4R)-N-(1-cyanocyclopropyl)-4-(2-methoxyphenylthio)pyrrolidine-2-carboxamide
—— (R)-ethyl 2-(1-allyl-2-(1-phenylethylcarbamoyl)hydrazinyl)acetate 1198777-78-4 C16H23N3O3
(R)-ethyl 2-(1-allyl-2-(1-phenylethylcarbamoyl)hydrazinyl)acetate
—— N-(3-{4-[(6-chloro-3-nitropyridin-2-yl)amino]phenyl}oxetan-3-yl)-2-methylpropane-2-sulfinamide 1313883-49-6 C18H21ClN4O4S
N-(3-{4-[(6-chloro-3-nitropyridin-2-yl)amino]phenyl}oxetan-3-yl)-2-methylpropane-2-sulfinamide
—— (R)-7-((3-fluoro-4-((6-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1,2-dimethyl-2,3-dihydroimidazo[1,2-c]pyrimidin-5(1H)-one 1620578-66-6 C21H18F4N4O3
(R)-7-((3-fluoro-4-((6-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1,2-dimethyl-2,3-dihydroimidazo[1,2-c]pyrimidin-5(1H)-one
—— N-(4-chlorobenzyl)-2-((2R,6S,11R,E)-11-methyl-5,12-dioxo-2-phenyl-1-oxa-4-azacyclododec-8-en-6-yl)acetamide 1589555-46-3 C26H29ClN2O4
N-(4-chlorobenzyl)-2-((2R,6S,11R,E)-11-methyl-5,12-dioxo-2-phenyl-1-oxa-4-azacyclododec-8-en-6-yl)acetamide
—— 5-[3-(Difluoromethyl)-1,2,4-triazol-1-yl]-2-methylbenzenesulfonyl chloride 1267995-30-1 C10H8ClF2N3O2S
5-[3-(Difluoromethyl)-1,2,4-triazol-1-yl]-2-methylbenzenesulfonyl chloride
—— N-ethyl-6-fluoro-8-methyl-3,4-dihydro-2H-1-benzopyran-4-amine 1554168-99-8 C12H16FNO
N-ethyl-6-fluoro-8-methyl-3,4-dihydro-2H-1-benzopyran-4-amine
—— 3-(7-isopropyl-4(R)-methyl-3-oxo-2,3,4,10-tetrahydro-9-oxa-1,2,4a-triazaphenanthren-6-yloxy)azetidine-1-carboxylic acid tert-butyl ester 1613722-20-5 C22H30N4O5
3-(7-isopropyl-4(R)-methyl-3-oxo-2,3,4,10-tetrahydro-9-oxa-1,2,4a-triazaphenanthren-6-yloxy)azetidine-1-carboxylic acid tert-butyl ester
—— ethyl (3-{[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]methyl}oxetan-3-yl)methyl(4-{[4-{[6-bromo-2-(methylcarbamoyl)pyridin-3-yl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-2-chloro-3-methoxybenzyl)phosphonate 1380308-10-0 C36H43BBrClF3N8O8P
ethyl (3-{[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]methyl}oxetan-3-yl)methyl(4-{[4-{[6-bromo-2-(methylcarbamoyl)pyridin-3-yl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-2-chloro-3-methoxybenzyl)phosphonate
—— 4-{[3,5-bis(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-2,6-dibromoaniline 1207089-08-4 C11H6Br2F6N4
4-{[3,5-bis(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-2,6-dibromoaniline
—— tert-butyl 4-(4-(7-cyano-4-(2,6-dichlorobenzyl)-1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazo[4,5-c]pyridin-6-ylamino)-3-(trifluoromethyl)phenyl)piperazine-1-carboxylate 1386949-86-5 C36H42Cl2F3N7O3Si
tert-butyl 4-(4-(7-cyano-4-(2,6-dichlorobenzyl)-1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazo[4,5-c]pyridin-6-ylamino)-3-(trifluoromethyl)phenyl)piperazine-1-carboxylate
—— (4-benzylamino-1-hydroxy-cyclohexyl)-acetic acid benzyl ester 1613269-43-4 C22H27NO3
(4-benzylamino-1-hydroxy-cyclohexyl)-acetic acid benzyl ester
—— 2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[2-(tetrahydro-2H-pyran-4-yl)ethyl]-1,3-thiazole-4-carboxamide 1421847-16-6 C24H29FN4O2S
2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[2-(tetrahydro-2H-pyran-4-yl)ethyl]-1,3-thiazole-4-carboxamide
—— methyl 4-(3-(2-(((4S,5R)-5-(3,5-bis(trifluoromethyl)phenyl)-4-methyl-2-oxooxazolidin-3-yl)methyl)-4,4-dimethylcyclohex-1-enyl)-4-methoxyphenyl)cyclohex-3-enecarboxylate 1402799-15-8 C36H39F6NO5
methyl 4-(3-(2-(((4S,5R)-5-(3,5-bis(trifluoromethyl)phenyl)-4-methyl-2-oxooxazolidin-3-yl)methyl)-4,4-dimethylcyclohex-1-enyl)-4-methoxyphenyl)cyclohex-3-enecarboxylate
—— tert-butyl {1-[4-(6-amino-3-phenylimidazo[1,2-b]pyridazin-2-yl)phenyl]cyclobutyl}carbamate 1402608-85-8 C27H29N5O2
tert-butyl {1-[4-(6-amino-3-phenylimidazo[1,2-b]pyridazin-2-yl)phenyl]cyclobutyl}carbamate
—— 2-(3-chloro-4-fluorophenoxy)-5-formylbenzonitrile 1420365-41-8 C14H7ClFNO2
2-(3-chloro-4-fluorophenoxy)-5-formylbenzonitrile
—— 3,5,8-trimethyl-1-adamantane carboxylic acid 1430847-62-3 C14H22O2
3,5,8-trimethyl-1-adamantane carboxylic acid
—— N-(3-{1-[7-cyano-1-(2-methoxy-ethyl)-1H-indole-3-carbonyl]-piperidin-4-yl}-4-fluoro-benzyl)-2,2,2-trifluoro-acetamide 1313042-08-8 C27H26F4N4O3
N-(3-{1-[7-cyano-1-(2-methoxy-ethyl)-1H-indole-3-carbonyl]-piperidin-4-yl}-4-fluoro-benzyl)-2,2,2-trifluoro-acetamide
—— (S)-O-methyl (3-(4-(4-(6-amino-nicotinoyl)-piperazin-1-yl)-3-fluorophenyl)-2-oxo-oxazoIidin-5-yl)-methyl-carbamothioate 1094617-88-5 C22H25FN6O4S
(S)-O-methyl (3-(4-(4-(6-amino-nicotinoyl)-piperazin-1-yl)-3-fluorophenyl)-2-oxo-oxazoIidin-5-yl)-methyl-carbamothioate
—— 4-methyl-2-{[(3R,6R)-6-methyl-1-{[4-(2H-1,2,3-triazol-2-yl)pyridin-3-yl]carbonyl}piperidin-3-yl]oxy}pyridin-3-carbonitrile 1616373-41-1 C21H21N7O2
4-methyl-2-{[(3R,6R)-6-methyl-1-{[4-(2H-1,2,3-triazol-2-yl)pyridin-3-yl]carbonyl}piperidin-3-yl]oxy}pyridin-3-carbonitrile
—— β-[[2-[[[3-[(aminoiminomethyl)amino]phenyl]carbonyl]amino]acetyl]amino]-3,5-bis(1-methylethoxy)benzenepropanoic acid 188809-39-4 C25H33N5O6
β-[[2-[[[3-[(aminoiminomethyl)amino]phenyl]carbonyl]amino]acetyl]amino]-3,5-bis(1-methylethoxy)benzenepropanoic acid
—— 2-((2-chloropyridin-4-yl)oxy)-5-(((1-methyl-5-oxo-1,2,3,5-tetrahydroimidazo[1,2-c]pyrimidin-7-yl)oxy)methyl)benzonitrile 1421433-29-5 C20H16ClN5O3
2-((2-chloropyridin-4-yl)oxy)-5-(((1-methyl-5-oxo-1,2,3,5-tetrahydroimidazo[1,2-c]pyrimidin-7-yl)oxy)methyl)benzonitrile
—— 4-(1-(3-(difluoromethyl)phenyl)-3-methyl-2,5-dioxo-1,2,3,4,5,6,7,8-octahydroquinazolin-4-yl)-3-(methylsulfonyl)benzonitrile 1625669-86-4 C24H21F2N3O4S
4-(1-(3-(difluoromethyl)phenyl)-3-methyl-2,5-dioxo-1,2,3,4,5,6,7,8-octahydroquinazolin-4-yl)-3-(methylsulfonyl)benzonitrile
—— N-((2S)-1-((2-(5-(benzyloxy)pyridin-2-yl)-7-fluoro[1,3]oxazolo[4,5-c]pyridin-6-yl)oxy)propan-2-yl)acetamide 1431535-26-0 C23H21FN4O4
N-((2S)-1-((2-(5-(benzyloxy)pyridin-2-yl)-7-fluoro[1,3]oxazolo[4,5-c]pyridin-6-yl)oxy)propan-2-yl)acetamide
—— ((S)-6-{(R)-4-[2-cyano-4-(morpholin-4-ylmethyl)phenoxy]-7-fluoroindan-1-yloxy}-2,3-dihydrobenzofuran-3-yl)acetic acid methyl ester 1613301-92-0 C32H31FN2O6
((S)-6-{(R)-4-[2-cyano-4-(morpholin-4-ylmethyl)phenoxy]-7-fluoroindan-1-yloxy}-2,3-dihydrobenzofuran-3-yl)acetic acid methyl ester
—— (S)-2-(2-amino-6-fluorobenzamido)propanoic acid 1585988-33-5 C10H11FN2O3
(S)-2-(2-amino-6-fluorobenzamido)propanoic acid
—— 6-(2-fluoro-4-iodophenylamino)-N-(2-methoxyethoxy)-5-methyl-4-oxo-4,5-dihydrofuro[3,2-c]pyridine-7-carboxamide 1289571-40-9 C18H17FIN3O5
6-(2-fluoro-4-iodophenylamino)-N-(2-methoxyethoxy)-5-methyl-4-oxo-4,5-dihydrofuro[3,2-c]pyridine-7-carboxamide
—— 6-chloro-7-ethyl-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]-7,9-dihydro-8H-purin-8-one 1361570-00-4 C20H15ClFN7O
6-chloro-7-ethyl-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]-7,9-dihydro-8H-purin-8-one
—— 8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[(3S)-pyrrolidin-3-yl]imidazo[1,2-a]pyridine-3-carboxamide 1609340-71-7 C20H20F2N4O2
8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[(3S)-pyrrolidin-3-yl]imidazo[1,2-a]pyridine-3-carboxamide
—— 6-(2,4-dichloro-benzylcarbamoyl)-1,6-diaza-spiro[3.3]heptane-1-carboxylic acid tert-butyl ester 1431868-77-7 C18H23Cl2N3O3
6-(2,4-dichloro-benzylcarbamoyl)-1,6-diaza-spiro[3.3]heptane-1-carboxylic acid tert-butyl ester
—— N-(4b-hydroxy-7-isopropyl-1-nitro-10-oxo-9b,10-dihydro-4bH-benzo[d]indeno[1,2-b]furan-9b-yl)-1H-indazole-3-carboxamide 1416238-45-3 C26H20N4O6
N-(4b-hydroxy-7-isopropyl-1-nitro-10-oxo-9b,10-dihydro-4bH-benzo[d]indeno[1,2-b]furan-9b-yl)-1H-indazole-3-carboxamide
—— 2-chloro-N-(3-cyclopropyl-2-(6-(trifluoromethyl)pyridin-3-yl)propyl)-3-fluorobenzamide 1600496-95-4 C19H17ClF4N2O
2-chloro-N-(3-cyclopropyl-2-(6-(trifluoromethyl)pyridin-3-yl)propyl)-3-fluorobenzamide
—— N-{4-[4-(difluoromethoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl}-2-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidin-5-yl)acetamide 1246275-24-0 C20H15F4N5O4S
N-{4-[4-(difluoromethoxy)-3,5-difluorophenyl]-1,3-thiazol-2-yl}-2-(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidin-5-yl)acetamide
—— 4-(3-methylsulfanyl-6-(piperazin-1-ylmethyl)indazol-1-yl)phenylamine 1345405-43-7 C19H23N5S
4-(3-methylsulfanyl-6-(piperazin-1-ylmethyl)indazol-1-yl)phenylamine
—— 9-benzyloxy-2-cyclobutyl-6-(1-pyrrolo[2,3-b]pyridin-1-ylcyclopentylmethyl)-3,4-dihydro-2H-pyrazino[1,2-c]pyrimidine-1,8-dione 1616925-54-2 C31H33N5O3
9-benzyloxy-2-cyclobutyl-6-(1-pyrrolo[2,3-b]pyridin-1-ylcyclopentylmethyl)-3,4-dihydro-2H-pyrazino[1,2-c]pyrimidine-1,8-dione
—— (E)-2-(3-fluoro-{8-[2-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl]methyl}dibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile 1421785-02-5 C26H17F4N3O
(E)-2-(3-fluoro-{8-[2-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl]methyl}dibenzo[b,e]oxepin-11(6H)-ylidene)propanenitrile
—— (R)-tert-butyl 2-(2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)propylcarbamate 1338543-85-3 C20H31BFNO4
(R)-tert-butyl 2-(2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)propylcarbamate
—— 2-chloro-N-(2-(pyridin-4-yl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)benzamide 1600496-05-6 C19H14ClF3N4O
2-chloro-N-(2-(pyridin-4-yl)-2-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)benzamide
—— 2-(6-cyclopropyl-pyridin-3-yl)-2-morpholin-4-yl-ethylamine 1601471-96-8 C14H21N3O
2-(6-cyclopropyl-pyridin-3-yl)-2-morpholin-4-yl-ethylamine
—— 6-[8-(2,5-difluorophenyl)-3-methoxy-6,7-dihydro-5H-benzo[7]annulen-9-yl]hex-5-yn-1-ol 1353008-29-3 C24H24F2O2
6-[8-(2,5-difluorophenyl)-3-methoxy-6,7-dihydro-5H-benzo[7]annulen-9-yl]hex-5-yn-1-ol
—— N-(6-chloro-[2,4']bipyridinyl-3'-yl)-N-methyl-3,5-bis-trifluoromethylbenzamide 1395412-72-2 C20H12ClF6N3O
N-(6-chloro-[2,4']bipyridinyl-3'-yl)-N-methyl-3,5-bis-trifluoromethylbenzamide
—— 3-(5-amino-2-fluorophenyl)-5-tert-butoxycarbonylamino-3-difluoromethyl-3,6-dihydro-2H-pyrazine-1-carboxylic acid 2,2,2-trichloroethyl ester 1313526-25-8 C19H22Cl3F3N4O4
3-(5-amino-2-fluorophenyl)-5-tert-butoxycarbonylamino-3-difluoromethyl-3,6-dihydro-2H-pyrazine-1-carboxylic acid 2,2,2-trichloroethyl ester
—— 3-[3-(1-methyl-1H-indazol-4-yl)thioureido]-4-trifluoromethoxy-benzamide 1378079-31-2 C17H14F3N5O2S
3-[3-(1-methyl-1H-indazol-4-yl)thioureido]-4-trifluoromethoxy-benzamide
—— 4-Chlor-5-hydroxy-2-oxo-2,5-dihydro-1H-1-benzazepin 16511-41-4 C10H8ClNO2
4-Chlor-5-hydroxy-2-oxo-2,5-dihydro-1H-1-benzazepin
—— 4-methoxy-6-methylfuro[2,3-b]pyridin-3(2H)-one O-methyl oxime 1421621-23-9 C10H12N2O3
4-methoxy-6-methylfuro[2,3-b]pyridin-3(2H)-one O-methyl oxime
—— 3-(methoxymethoxy)-1-(methoxymethyl)-5-{[(3-methylpyridin-2-yl)methyl]sulfanyl}pyridin-2(1H)-one 1417710-48-5 C16H20N2O4S
3-(methoxymethoxy)-1-(methoxymethyl)-5-{[(3-methylpyridin-2-yl)methyl]sulfanyl}pyridin-2(1H)-one