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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-fluoro-4-[1-methyl-5-(trifluoromethyl)-1H-benzimidazol-2-yl]isoquinoline 1356480-62-0 C18H11F4N3
6-fluoro-4-[1-methyl-5-(trifluoromethyl)-1H-benzimidazol-2-yl]isoquinoline
—— (cis)-4-(4-(4-chloro-3-cyclopropylphenyl)-2-(2,6-dimethylmorpholine-4-carbonyl)thiazol-5-yl)benzenesulfonamide 1454649-51-4 C25H26ClN3O4S2
(cis)-4-(4-(4-chloro-3-cyclopropylphenyl)-2-(2,6-dimethylmorpholine-4-carbonyl)thiazol-5-yl)benzenesulfonamide
—— 1-(3-methoxybenzyl)-1-methyl-3-(2-(2-morpholinoethoxy)-4-(1H-pyrazol-4-yl)phenyl)urea 1219726-80-3 C25H31N5O4
1-(3-methoxybenzyl)-1-methyl-3-(2-(2-morpholinoethoxy)-4-(1H-pyrazol-4-yl)phenyl)urea
—— ethyl 3-[(1-naphthylsulfonyl)amino]-2-(4-nitrobenzyl)-3-oxopropionate 1094201-58-7 C22H20N2O7S
ethyl 3-[(1-naphthylsulfonyl)amino]-2-(4-nitrobenzyl)-3-oxopropionate
—— 2-chloro-N-[(S)-1-(3,4-difluoro-phenyl)-ethyl]-4-pyridin-4-yl-benzamide 1127309-82-3 C20H15ClF2N2O
2-chloro-N-[(S)-1-(3,4-difluoro-phenyl)-ethyl]-4-pyridin-4-yl-benzamide
—— 2-methyl-5-(2-(2-(((R)-1-(naphthalen-1-yl)ethyl)amino)ethyl)morpholino)benzoic acid 1398393-69-5 C26H30N2O3
2-methyl-5-(2-(2-(((R)-1-(naphthalen-1-yl)ethyl)amino)ethyl)morpholino)benzoic acid
—— ethyl 3-{3-(2-phenylethyl)-1-[4-(2-pyridin-2-ylethoxy)phenyl]-1H-indol-5-yl}propanoate 1069044-68-3 C34H34N2O3
ethyl 3-{3-(2-phenylethyl)-1-[4-(2-pyridin-2-ylethoxy)phenyl]-1H-indol-5-yl}propanoate
—— N-phenyl-N-(piperidin-4-yl)-3-(piperidin-1-yl)propionamide 1186213-15-9 C19H29N3O
N-phenyl-N-(piperidin-4-yl)-3-(piperidin-1-yl)propionamide
—— 3-fluoro-N-((1R,2S)-2-hydroxy-indan-1-yl)-4-pyridin-4-yl-benzamide 1127309-94-7 C21H17FN2O2
3-fluoro-N-((1R,2S)-2-hydroxy-indan-1-yl)-4-pyridin-4-yl-benzamide
—— 4-[cyclohexyl(5-cyclohexyl-2-ethylthiophen-3-yl)methoxy]benzoic acid 1150223-15-6 C26H34O3S
4-[cyclohexyl(5-cyclohexyl-2-ethylthiophen-3-yl)methoxy]benzoic acid
—— 2-{4-[(2-chlorobenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide 1094194-90-7 C31H30ClN3O5S
2-{4-[(2-chlorobenzoyl)amino]benzyl}-N, N-diethyl-N'-(2-naphthylsulfonyl)malonamide
—— 4-[2-(4-fluorophenyl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxaazin-3-yl]-N-(1-methylethyl)-2-aminopyrimidine 1161076-09-0 C19H20FN5O
4-[2-(4-fluorophenyl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxaazin-3-yl]-N-(1-methylethyl)-2-aminopyrimidine
—— N-[1-(2,4-dimethylphenyl)-2-hydroxyethyl]-4-pyridin-4-ylbenzamide 1127308-04-6 C22H22N2O2
N-[1-(2,4-dimethylphenyl)-2-hydroxyethyl]-4-pyridin-4-ylbenzamide
—— methyl 3-{1-[4-(diethylamino)phenyl]-3-(2-phenylethyl)-1H-indol-5-yl}propanoate 1069043-08-8 C30H34N2O2
methyl 3-{1-[4-(diethylamino)phenyl]-3-(2-phenylethyl)-1H-indol-5-yl}propanoate
—— 4-[[3-butoxy-4-(difluoromethoxy)phenyl](pyridin-3-ylmethyl)amino]benzoic acid tert-butyl ester 1203597-17-4 C28H32F2N2O4
4-[[3-butoxy-4-(difluoromethoxy)phenyl](pyridin-3-ylmethyl)amino]benzoic acid tert-butyl ester
—— [3-(3,3'-dichloro-2'-fluorobiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1035927-06-0 C20H18Cl2FN3OS
[3-(3,3'-dichloro-2'-fluorobiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— 1-(3-hydroxy-1-(3-methoxyphenyl)propyl)-3-(2-(2-hydroxyethoxy)-4-(1H-pyrazol-4-yl)phenyl)urea 1219723-55-3 C22H26N4O5
1-(3-hydroxy-1-(3-methoxyphenyl)propyl)-3-(2-(2-hydroxyethoxy)-4-(1H-pyrazol-4-yl)phenyl)urea
—— 1,2,4-trifluoro-3-[1-(4-nitrophenoxy)ethyl]benzene 1146853-98-6 C14H10F3NO3
1,2,4-trifluoro-3-[1-(4-nitrophenoxy)ethyl]benzene
—— 6-{4-fluoro-3-[(4-oxooctahydro-2H-pyrido[1,2-a]pyrazin-2-yl)carbonyl]benzyl}-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate 1154869-32-5 C2HF3O2*C22H25FN4O3
6-{4-fluoro-3-[(4-oxooctahydro-2H-pyrido[1,2-a]pyrazin-2-yl)carbonyl]benzyl}-4,5-dimethyl-3-oxo-2,3-dihydropyridazin-1-ium trifluoroacetate
—— 6-(3-{[4-(3,5-dimethylbenzyl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one trifluoroacetate 1154869-06-3 C2HF3O2*C27H29FN4O3
6-(3-{[4-(3,5-dimethylbenzyl)-3-oxopiperazin-1-yl]carbonyl}-4-fluorobenzyl)-4,5-dimethylpyridazin-3(2H)-one trifluoroacetate
—— ethyl 4-[3-(4-bromo-2-tert-butylphenoxy)azetidin-1-yl]-4-oxobutanoate 1146957-00-7 C19H26BrNO4
ethyl 4-[3-(4-bromo-2-tert-butylphenoxy)azetidin-1-yl]-4-oxobutanoate
—— rac-3-{2,6-dimethyl-4-[5-(6-methyl-2-propoxy-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenoxy}-propane-1,2-diol 1150645-56-9 C21H26N4O5
rac-3-{2,6-dimethyl-4-[5-(6-methyl-2-propoxy-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-phenoxy}-propane-1,2-diol
—— 2-[(4-benzoylamino)benzyl]-3-(4-methylpiperazino)-N-(2-naphthylsulfonyl)-3-oxopropanamide 1094197-04-2 C32H32N4O5S
2-[(4-benzoylamino)benzyl]-3-(4-methylpiperazino)-N-(2-naphthylsulfonyl)-3-oxopropanamide
—— (3S,5S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3,5-dimethyl-N-[2-methyl-4-(trifluoromethoxy)phenyl]piperazine-1-carboxamide 1616415-24-7 C21H25F3N8O2
(3S,5S)-4-(6-amino-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)-3,5-dimethyl-N-[2-methyl-4-(trifluoromethoxy)phenyl]piperazine-1-carboxamide
—— {2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}(phenyl)methanol 1150221-38-7 C20H17F3O2
{2-ethyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}(phenyl)methanol
—— 4-fluoro-N-{[2-oxo-7-(1H-pyrazol-4-yl)-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide 1141878-20-7 C20H14F4N4O3
4-fluoro-N-{[2-oxo-7-(1H-pyrazol-4-yl)-4-(trifluoromethyl)-1,4-dihydro-2H-3,1-benzoxazin-4-yl]methyl}benzamide
—— 4-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-ylsulfamoyl]benzoic acid 1150342-40-7 C35H32F3N5O7S
4-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-ylsulfamoyl]benzoic acid
—— N-[(S)-1-(4-chloro-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide 1127308-91-1 C21H19ClN2O2
N-[(S)-1-(4-chloro-phenyl)-ethyl]-2-methoxy-4-pyridin-4-yl-benzamide
—— cyclohexyl[5-(6-fluoropyridin-3-yl)-2-methylfuran-3-yl]methanol 1150225-60-7 C17H20FNO2
cyclohexyl[5-(6-fluoropyridin-3-yl)-2-methylfuran-3-yl]methanol
—— 6-[5-(3,4-dichlorobenzenesulfonylamino)-4-methylpyridin-2-yloxy]-1-methyl-1H-indole-2-carboxylic acid 1150744-93-6 C22H17Cl2N3O5S
6-[5-(3,4-dichlorobenzenesulfonylamino)-4-methylpyridin-2-yloxy]-1-methyl-1H-indole-2-carboxylic acid
—— 3-methoxy-N-(1-{2-[7-(methoxymethyl)naphthalen-2-yl]ethyl}piperidin-4-yl)benzamide 1018072-99-5 C27H32N2O3
3-methoxy-N-(1-{2-[7-(methoxymethyl)naphthalen-2-yl]ethyl}piperidin-4-yl)benzamide
—— 5-bromo-2-(3-chloropyridin-4-yl)-1-cyclopropyl-1H-benzimidazole 1356480-52-8 C15H11BrClN3
5-bromo-2-(3-chloropyridin-4-yl)-1-cyclopropyl-1H-benzimidazole
—— 5-fluoro-2-(5-fluoropyridin-3-yl)-1-methyl-1H-benzimidazole 1356482-25-1 C13H9F2N3
5-fluoro-2-(5-fluoropyridin-3-yl)-1-methyl-1H-benzimidazole
—— methyl 2-(4-(3-(2-(methylsulfonyl)-1,2,3,4-tetrahydroisoquinolin-6-yloxy)propyl)piperidin-1-yl)pyrimidine-5-carboxylate 1046816-62-9 C24H32N4O5S
methyl 2-(4-(3-(2-(methylsulfonyl)-1,2,3,4-tetrahydroisoquinolin-6-yloxy)propyl)piperidin-1-yl)pyrimidine-5-carboxylate
—— 2-[4-chloro-2-(trifluoromethoxy)phenyl]-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079362-06-3 C20H21ClF3N3O2
2-[4-chloro-2-(trifluoromethoxy)phenyl]-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 6-(cyclopropylamino)-9-[1-(2-(4-methoxyphenyl)ethyl)]-2-(trifluoromethyl)purine 1082247-79-7 C18H18F3N5O
6-(cyclopropylamino)-9-[1-(2-(4-methoxyphenyl)ethyl)]-2-(trifluoromethyl)purine
—— 5-(2,4-dimethylphenyl)isoxazole-4-carboxylic acid 1173711-05-1 C12H11NO3
5-(2,4-dimethylphenyl)isoxazole-4-carboxylic acid
—— 5-(1-ethylpropyl)-2-(2-methoxy-6-methylphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079352-90-1 C21H27N3O2
5-(1-ethylpropyl)-2-(2-methoxy-6-methylphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— ethyl 3-{3-(2-phenylethyl)-1-[4-(tetrahydro-2H-pyran-4-yloxy)phenyl]-1H-indol-5-yl}propanoate 1069044-37-6 C32H35NO4
ethyl 3-{3-(2-phenylethyl)-1-[4-(tetrahydro-2H-pyran-4-yloxy)phenyl]-1H-indol-5-yl}propanoate
—— N-{[6-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-3-({[(2-fluorobenzyl)-carbamoyl]amino}methyl)pyrid-2-yl]methyl}-2-methoxyacetamide 1173144-24-5 C30H26Cl3FN4O3
N-{[6-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-3-({[(2-fluorobenzyl)-carbamoyl]amino}methyl)pyrid-2-yl]methyl}-2-methoxyacetamide
—— 5-[bis(4-fluorophenyl)methyl]-1-[2-(tetrahydro-2H-pyran-2-yloxy)ethyl]pyridin-2(1H)-one 1034019-87-8 C25H25F2NO3
5-[bis(4-fluorophenyl)methyl]-1-[2-(tetrahydro-2H-pyran-2-yloxy)ethyl]pyridin-2(1H)-one
—— 5-isopropyl-2-[4-methoxy-2-(trifluoromethyl)phenyl]-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079361-09-3 C19H20F3N3O2
5-isopropyl-2-[4-methoxy-2-(trifluoromethyl)phenyl]-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— N-[2-(2,4-dichlorobenzoyl)phenyl]-4-[4-(3-piperidin-1-ylpropyl)piperazine-1-carbonyl]benzenesulfonamide 1021363-09-6 C32H36Cl2N4O4S
N-[2-(2,4-dichlorobenzoyl)phenyl]-4-[4-(3-piperidin-1-ylpropyl)piperazine-1-carbonyl]benzenesulfonamide
—— 5-chloro-3-methyl-1-benzothiophene-2-carboxylic acid hydrazide 1035928-09-6 C10H9ClN2OS
5-chloro-3-methyl-1-benzothiophene-2-carboxylic acid hydrazide
—— 3-(4-(1H-pyrazol-4-yl)phenyl)-1-(3-ethoxybenzyl)-1-methylurea 1219726-63-2 C20H22N4O2
3-(4-(1H-pyrazol-4-yl)phenyl)-1-(3-ethoxybenzyl)-1-methylurea
—— 2-(3-chloropyridin-4-yl)-1-cyclopropyl-4,6-difluoro-1H-benzimidazole 1356482-36-4 C15H10ClF2N3
2-(3-chloropyridin-4-yl)-1-cyclopropyl-4,6-difluoro-1H-benzimidazole
—— 8-({[t-butyl(dimethyl)silyl]oxy}methyl)-3-(3-chloro-3'-methoxybiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1035928-46-1 C27H36ClN3O2SSi
8-({[t-butyl(dimethyl)silyl]oxy}methyl)-3-(3-chloro-3'-methoxybiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 1-methyl-2-(pyridin-3-yl)-5-(trifluoromethyl)-1H-benzimidazole 1356480-55-1 C14H10F3N3
1-methyl-2-(pyridin-3-yl)-5-(trifluoromethyl)-1H-benzimidazole
—— ethyl 2-amino-5-methyl-4-(n-pentyl)-thiophene-3-carboxylate 1186474-60-1 C13H21NO2S
ethyl 2-amino-5-methyl-4-(n-pentyl)-thiophene-3-carboxylate
—— tert-butyl 4-(2-{3,5-dichloro-6-[(E)-2-(3-nitrophenyl)vinyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoate 1091598-80-9 C26H24Cl2N2O5
tert-butyl 4-(2-{3,5-dichloro-6-[(E)-2-(3-nitrophenyl)vinyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoate