中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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US9434719, 279 as TFA salt |
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C16H16BrF2N5O3 |
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—— |
US9434719, 241 as TFA salt |
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C20H22ClN7O3 |
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—— |
US9434719, 218 as TFA salt |
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C20H19ClFN5O4 |
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—— |
US9434719, 434 as TFA salt |
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C20H18F4N6O2 |
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—— |
US9434719, 325 as TFA salt |
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C23H20F5N5O3 |
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—— |
US9434719, 264 as TFA salt |
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C20H20F2N6O3 |
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—— |
US9434719, 245 as TFA salt |
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C20H21F5N4O4 |
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—— |
US9434719, 442 as TFA salt |
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C22H19F4N5O2 |
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—— |
US9434719, 209 as TFA salt |
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C21H22ClFN6O3 |
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—— |
US9434719, 234 as TFA salt |
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C19H19ClN6O3S |
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—— |
US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile |
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C29H31FN8O2S |
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—— |
US9670204, 162 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile |
—— |
C30H33FN8O2S |
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—— |
US9670204, 67 N-(6-(1-(chloromethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine |
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C25H25ClFN5O2S2 |
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—— |
US9670204, 182 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-thiomorpholine1,1-dioxide |
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C23H24FN5O2S2 |
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—— |
US9670204, 75 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-ylsulfonyl)propan-1-ol |
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C27H30FN5O3S2 |
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—— |
US9670204, 151 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(pyrrolidin-1-yl)ethanone |
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C31H37FN6O2S |
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US9670204, 49 (4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)(1-(methylsulfonyl)pyrrolidin-3-yl)methanone |
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C29H34FN7O3S2 |
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US9670204, 108 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-yl)acetate |
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C28H30FN5O2S |
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—— |
US9670204, 130 3-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one |
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C29H35FN6OS |
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—— |
US9670204, 203 (S)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-hydroxypropan-1-one |
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C26H29FN6O2S |
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—— |
US9670204, 159 1-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl)-2,2,2-trifluoroethanone |
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C31H32F4N6O3S |
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—— |
US9670204, 189 N-(2-ethyl-6-(1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyridin-3-yl)-3-(4-fluorophenyl)-N-methyl-1,2,4-oxadiazol-5-amine |
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C24H25FN6O3S |
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—— |
US9670204, 149 (2-((6-(1-(3-(dimethylamino)propyl-sulfonyl)piperidin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl) |
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C30H39FN6O3S2 |
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—— |
US9670204, 207 2-(2-ethyl-4-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-1-[1,2]thiazinane-1,1-dioxide |
—— |
C23H24ClN5O2S2 |
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—— |
US9670204, 97 2-(2-((2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile |
—— |
C27H29FN6O2S2 |
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—— |
US9670204, 57 N-(2-ethyl-6-(4-(3-(pyrrolidin-1-yl)propylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine |
—— |
C30H38FN7O2S2 |
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—— |
US9670204, 208 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-N-(thiophen-2-yl)-5,6-dihydropyridine-1(2H)-carboxamide |
—— |
C29H27FN6OS2 |
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—— |
Unk-N(Tfa)4Abz-hTyr-OH |
—— |
C26H22F3N7O6 |
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—— |
Unk-N(Tfa)4Abz-Tyr-OBn |
—— |
C32H26F3N7O6 |
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—— |
Unk-N(Tfa)4Abz-N(Me)Tyr-OH |
—— |
C26H22F3N7O6 |
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—— |
US9611261, Example 276 |
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C18H15Cl2FN4O2 |
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—— |
US9611261, Example 341 |
—— |
C20H15ClF3N5O |
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—— |
Undecane-1,8,10-triol |
—— |
C11H24O3 |
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—— |
US9624241, Example 103 |
—— |
C24H25N5O2 |
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—— |
US9624241, Example 89 |
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C21H20N4O4 |
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—— |
undecan-6-yl (10R,15S)-12-[4-(4-fluorophenyl)-4-oxobutyl]-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-triene-4-carboxylate |
—— |
C35H48FN3O3 |
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—— |
US9617282, Example 219 |
—— |
C23H27N7O4S |
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—— |
US9617282, Example 192 |
—— |
C21H22N6O3S |
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—— |
US9617282, Example 222 |
—— |
C19H21N7O3S |
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—— |
US9617282, Example 207 |
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C19H19N5O4S |
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—— |
US9617282, Example 45 |
—— |
C18H19N7O3S |
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—— |
US9617282, Example 59 |
—— |
C19H24N4O3 |
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—— |
US9617282, Example 217 |
—— |
C20H22N6O3S |
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—— |
US9617282, Example 170 |
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C25H29N7O4S |
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—— |
US9617282, Example 202 |
—— |
C18H19N7O4 |
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—— |
US9617282, Example 50 |
—— |
C20H23N5O3 |
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—— |
US9617282, Example 20 |
—— |
C23H25N5O3S |
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—— |
US9617282, Example 215 |
—— |
C20H22N6O3S |
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—— |
US9617282, Example 203 |
—— |
C20H20N6O4 |
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—— |
US9617282, Example 169 |
—— |
C24H29N7O3S |
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