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中文名称 英文名称 CAS号 化学式 结构式图片
—— US9434719, 279 as TFA salt —— C16H16BrF2N5O3
US9434719, 279 as TFA salt
—— US9434719, 241 as TFA salt —— C20H22ClN7O3
US9434719, 241 as TFA salt
—— US9434719, 218 as TFA salt —— C20H19ClFN5O4
US9434719, 218 as TFA salt
—— US9434719, 434 as TFA salt —— C20H18F4N6O2
US9434719, 434 as TFA salt
—— US9434719, 325 as TFA salt —— C23H20F5N5O3
US9434719, 325 as TFA salt
—— US9434719, 264 as TFA salt —— C20H20F2N6O3
US9434719, 264 as TFA salt
—— US9434719, 245 as TFA salt —— C20H21F5N4O4
US9434719, 245 as TFA salt
—— US9434719, 442 as TFA salt —— C22H19F4N5O2
US9434719, 442 as TFA salt
—— US9434719, 209 as TFA salt —— C21H22ClFN6O3
US9434719, 209 as TFA salt
—— US9434719, 234 as TFA salt —— C19H19ClN6O3S
US9434719, 234 as TFA salt
—— US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile —— C29H31FN8O2S
US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile
—— US9670204, 162 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile —— C30H33FN8O2S
US9670204, 162 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile
—— US9670204, 67 N-(6-(1-(chloromethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C25H25ClFN5O2S2
US9670204, 67 N-(6-(1-(chloromethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine
—— US9670204, 182 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-thiomorpholine1,1-dioxide —— C23H24FN5O2S2
US9670204, 182 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-thiomorpholine1,1-dioxide
—— US9670204, 75 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-ylsulfonyl)propan-1-ol —— C27H30FN5O3S2
US9670204, 75 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-ylsulfonyl)propan-1-ol
—— US9670204, 151 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(pyrrolidin-1-yl)ethanone —— C31H37FN6O2S
US9670204, 151 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(pyrrolidin-1-yl)ethanone
—— US9670204, 49 (4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)(1-(methylsulfonyl)pyrrolidin-3-yl)methanone —— C29H34FN7O3S2
US9670204, 49 (4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)(1-(methylsulfonyl)pyrrolidin-3-yl)methanone
—— US9670204, 108 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-yl)acetate —— C28H30FN5O2S
US9670204, 108 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-yl)acetate
—— US9670204, 130 3-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one —— C29H35FN6OS
US9670204, 130 3-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one
—— US9670204, 203 (S)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-hydroxypropan-1-one —— C26H29FN6O2S
US9670204, 203 (S)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-hydroxypropan-1-one
—— US9670204, 159 1-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl)-2,2,2-trifluoroethanone —— C31H32F4N6O3S
US9670204, 159 1-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl)-2,2,2-trifluoroethanone
—— US9670204, 189 N-(2-ethyl-6-(1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyridin-3-yl)-3-(4-fluorophenyl)-N-methyl-1,2,4-oxadiazol-5-amine —— C24H25FN6O3S
US9670204, 189 N-(2-ethyl-6-(1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyridin-3-yl)-3-(4-fluorophenyl)-N-methyl-1,2,4-oxadiazol-5-amine
—— US9670204, 149 (2-((6-(1-(3-(dimethylamino)propyl-sulfonyl)piperidin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl) —— C30H39FN6O3S2
US9670204, 149 (2-((6-(1-(3-(dimethylamino)propyl-sulfonyl)piperidin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl)
—— US9670204, 207 2-(2-ethyl-4-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-1-[1,2]thiazinane-1,1-dioxide —— C23H24ClN5O2S2
US9670204, 207 2-(2-ethyl-4-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-1-[1,2]thiazinane-1,1-dioxide
—— US9670204, 97 2-(2-((2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile —— C27H29FN6O2S2
US9670204, 97 2-(2-((2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile
—— US9670204, 57 N-(2-ethyl-6-(4-(3-(pyrrolidin-1-yl)propylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C30H38FN7O2S2
US9670204, 57 N-(2-ethyl-6-(4-(3-(pyrrolidin-1-yl)propylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine
—— US9670204, 208 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-N-(thiophen-2-yl)-5,6-dihydropyridine-1(2H)-carboxamide —— C29H27FN6OS2
US9670204, 208 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-N-(thiophen-2-yl)-5,6-dihydropyridine-1(2H)-carboxamide
—— Unk-N(Tfa)4Abz-hTyr-OH —— C26H22F3N7O6
Unk-N(Tfa)4Abz-hTyr-OH
—— Unk-N(Tfa)4Abz-Tyr-OBn —— C32H26F3N7O6
Unk-N(Tfa)4Abz-Tyr-OBn
—— Unk-N(Tfa)4Abz-N(Me)Tyr-OH —— C26H22F3N7O6
Unk-N(Tfa)4Abz-N(Me)Tyr-OH
—— US9611261, Example 276 —— C18H15Cl2FN4O2
US9611261, Example 276
—— US9611261, Example 341 —— C20H15ClF3N5O
US9611261, Example 341
—— Undecane-1,8,10-triol —— C11H24O3
Undecane-1,8,10-triol
—— US9624241, Example 103 —— C24H25N5O2
US9624241, Example 103
—— US9624241, Example 89 —— C21H20N4O4
US9624241, Example 89
—— undecan-6-yl (10R,15S)-12-[4-(4-fluorophenyl)-4-oxobutyl]-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-triene-4-carboxylate —— C35H48FN3O3
undecan-6-yl (10R,15S)-12-[4-(4-fluorophenyl)-4-oxobutyl]-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-triene-4-carboxylate
—— US9617282, Example 219 —— C23H27N7O4S
US9617282, Example 219
—— US9617282, Example 192 —— C21H22N6O3S
US9617282, Example 192
—— US9617282, Example 222 —— C19H21N7O3S
US9617282, Example 222
—— US9617282, Example 207 —— C19H19N5O4S
US9617282, Example 207
—— US9617282, Example 45 —— C18H19N7O3S
US9617282, Example 45
—— US9617282, Example 59 —— C19H24N4O3
US9617282, Example 59
—— US9617282, Example 217 —— C20H22N6O3S
US9617282, Example 217
—— US9617282, Example 170 —— C25H29N7O4S
US9617282, Example 170
—— US9617282, Example 202 —— C18H19N7O4
US9617282, Example 202
—— US9617282, Example 50 —— C20H23N5O3
US9617282, Example 50
—— US9617282, Example 20 —— C23H25N5O3S
US9617282, Example 20
—— US9617282, Example 215 —— C20H22N6O3S
US9617282, Example 215
—— US9617282, Example 203 —— C20H20N6O4
US9617282, Example 203
—— US9617282, Example 169 —— C24H29N7O3S
US9617282, Example 169