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中文名称 英文名称 CAS号 化学式
—— US9670204, 133 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-2-(3-fluoroazetidin-1-yl)ethanone —— C29H32F2N6OS
—— US9796708, Example 824 —— C20H18FN3O5S
—— US9796708, Example 856 —— C21H20FN3O2
—— US9796708, Example 601 —— C19H19ClFN3O
—— US9796708, Example 597 —— C24H26FN3O3
—— US9796708, Example 1119 —— C20H20FN3O2
—— US9670204, 200 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)propane-1,2-dione —— C26H27FN6O2S
—— US9670204, 129 2-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)ethanone —— C28H33FN6OS
—— US9670204, 111 (R)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone —— C30H35FN6O2S
—— US9796708, Example 706 —— C19H18ClN3O
—— US9718825, Example 563 —— C18H12Cl2N4O2S
—— US9718825, Example 534 —— C19H15Cl2N5O3S
—— US9796708, Example 1269 —— C29H32F2N4O3
—— US9796708, Example 557 —— C24H28N4O2
—— US9718825, Example 448 —— C20H15ClF2N6O2S
—— US9796708, Example 813 —— C20H19FN4O2
—— US9796708, Example 621 —— C19H17BrFN3O
—— US9670204, 201 5-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazine-1-carbonyl)pyrrolidin-2-one —— C28H30FN7O2S
—— US9718825, Example 546 —— C23H21Cl2N7O3S
—— US9796708, Example 721 —— C20H20FN3O
—— US9796708, Example 433 —— C25H26FN3O2
—— US9796708, Example 1054 —— C21H22FN3O
—— US9796708, Example 729 —— C21H22N4O2
—— US9670204, 122 5-((4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)methyl)oxazolidin-2-one —— C28H31FN6O2S
—— US9670204, 119 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N-(2-hydroxyethyl)-N-methylacetamide —— C29H35FN6O2S
—— US9670204, 215 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one —— C27H30FN5OS
—— US9670204, 59 methyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-ylsulfonyl)acetate —— C26H29FN6O4S2
—— US9796708, Example 1064 —— C27H31FN4O2
—— US9670204, 144 2-((2-ethyl-6-(1-(2-(3-(hydroxymethyl)azetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazole-5-carbonitrile —— C31H34FN7O2S
—— US9670204, 121 N-(cyanomethyl)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N-methylacetamide —— C29H32FN7OS
—— US9796708, Example 628 —— C22H21N5O
—— US9796708, Example 921 —— C20H20FN3O3S
—— US9796708, Example 814 —— C23H23FN4O3
—— US9796708, Example 874 —— C22H22FN3O3
—— US9796708, Example 630 —— C19H19N3O
—— US9670204, 190 2-(4-(2-ethyl-3-((3-(4-fluorophenyl)-1,2,4-thiadiazol-5-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-yl)-N,N-dimethylacetamide —— C27H30FN7OS
—— US9796708, Example 909 —— C25H21FN4O3
—— US9796708, Example 898 —— C19H19FN4
—— US9670204, 197 (S)-5-((4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)methyl)oxazolidin-2-one —— C28H31FN6O2S
—— US9796708, Example 592 —— C27H24F2N4O
—— US9670204, 134 1-(3-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)azetidin-1-yl)ethanone —— C29H33FN6OS
—— US9670204, 172 2-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile —— C31H34FN7O2S
—— US9670204, 156 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxyazetidin-1-yl)ethanone —— C30H35FN6O3S
—— US9796708, Example 658 —— C19H18FN3O
—— US9796708, Example 1249 —— C24H21FN4O3
—— US9670204, 170 2-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile —— C30H32FN7O2S
—— US9670204, 167 2-(2-((6-(4-(2-(azetidin-1-yl)-2-oxoethyl)piperazin-1-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile —— C29H31FN8OS
—— US9796708, Example 439 —— C24H26FN3O2
—— US9670204, 44 tert-butyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazine-1-carbonyl)pyrrolidine-1-carboxylate —— C33H40FN7O3S
—— US9670204, 56 N-(6-(4-(3-(dimethylamino)propyl-sulfonyl)piperazin-1-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C28H36FN7O2S2