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—— US9796708, Example 891 —— C23H25FN4O5S
US9796708, Example 891
—— US9796708, Example 360 —— C26H26FN3O
US9796708, Example 360
—— US9670204, 225 tert-butyl4-(3-((3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazine-1-carboxylate —— C27H32ClN7O2S
US9670204, 225 tert-butyl4-(3-((3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazine-1-carboxylate
—— US9796708, Example 616 —— C23H26FN3O2
US9796708, Example 616
—— US9670204, 178 2-(1-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)azetidin-3-ylamino)-1-(3-hydroxyazetidin-1-yl)ethanone —— C27H30FN7O2S
US9670204, 178 2-(1-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)azetidin-3-ylamino)-1-(3-hydroxyazetidin-1-yl)ethanone
—— US9796708, Example 1011 —— C26H29FN4O4
US9796708, Example 1011
—— US9670204, 196 (R)-5-((4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)methyl)oxazolidin-2-one —— C28H31FN6O2S
US9670204, 196 (R)-5-((4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)methyl)oxazolidin-2-one
—— US9670204, 223 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone —— C30H35FN6O2S
US9670204, 223 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone
—— US9670204, 53 4-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)butan-1-one —— C29H36FN7OS
US9670204, 53 4-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)butan-1-one
—— US9796708, Example 960 —— C24H24FN3O4
US9796708, Example 960
—— US9796708, Example 744 —— C24H27FN4O4S
US9796708, Example 744
—— US9796708, Example 509 —— C28H27F3N4O2
US9796708, Example 509
—— US9670204, 112 (S)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone —— C30H35FN6O2S
US9670204, 112 (S)-2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-hydroxypyrrolidin-1-yl)ethanone
—— US9796708, Example 342 —— C25H29FN6O2
US9796708, Example 342
—— US9796708, Example 617 —— C23H26N4O3
US9796708, Example 617
—— US9796708, Example 1157 —— C27H30FN3O3
US9796708, Example 1157
—— US9670204, 152 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-(hydroxymethyl)azetidin-1-yl)ethanone —— C31H37FN6O3S
US9670204, 152 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(3-(hydroxymethyl)azetidin-1-yl)ethanone
—— US9796708, Example 840 —— C21H23FN4O3S
US9796708, Example 840
—— US9796708, Example 870 —— C22H19FN4O3
US9796708, Example 870
—— US9796708, Example 661 —— C21H22FN3O5S2
US9796708, Example 661
—— US9670204, 221 4-(4-chlorophenyl)-N-(6-(3,6-dihydro-2H-pyran-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-N-methylthiazol-2-amine —— C24H23ClN4OS
US9670204, 221 4-(4-chlorophenyl)-N-(6-(3,6-dihydro-2H-pyran-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-N-methylthiazol-2-amine
—— US9796708, Example 871 —— C21H20FN3O3
US9796708, Example 871
—— US9796708, Example 1118 —— C20H20FN3O2
US9796708, Example 1118
—— US9670204, 169 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N-methylacetamide —— C27H29FN8OS
US9670204, 169 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N-methylacetamide
—— US9670204, 168 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide —— C28H31FN8OS
US9670204, 168 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide
—— US9796708, Example 1037 —— C20H19F2N3O
US9796708, Example 1037
—— US9796708, Example 353 —— C25H24ClFN4
US9796708, Example 353
—— US9796708, Example 826 —— C22H24N4O3S
US9796708, Example 826
—— US9796708, Example 665 —— C19H17ClFN3O
US9796708, Example 665
—— US9796708, Example 641 —— C20H20FN3O
US9796708, Example 641
—— US9796708, Example 407 —— C24H26F2N4O
US9796708, Example 407
—— US9796708, Example 1235 —— C20H20FN3O
US9796708, Example 1235
—— US9796708, Example 437 —— C27H23FN4O
US9796708, Example 437
—— US9670204, 155 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide —— C28H34FN7O2S
US9670204, 155 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide
—— US9796708, Example 1158 —— C21H20FN3O3
US9796708, Example 1158
—— US9796708, Example 633 —— C22H23F2N3O
US9796708, Example 633
—— US9796708, Example 345 —— C25H24F2N4
US9796708, Example 345
—— US9796708, Example 1082 —— C22H24FN3O3
US9796708, Example 1082
—— US9796708, Example 1151 —— C23H22FN3O2
US9796708, Example 1151
—— US9796708, Example 1010 —— C24H28FN3O3
US9796708, Example 1010
—— US9796708, Example 1133 —— C27H33FN4O2
US9796708, Example 1133
—— US9796708, Example 903 —— C20H19FN4O2
US9796708, Example 903
—— US9670204, 164 2-(2-((2-ethyl-6-(4-(2-(3-fluoroazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile —— C29H30F2N8OS
US9670204, 164 2-(2-((2-ethyl-6-(4-(2-(3-fluoroazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile
—— US9796708, Example 734 —— C21H22FN3O3S
US9796708, Example 734
—— US9796708, Example 804 —— C22H20F4N4O5S
US9796708, Example 804
—— US9796708, Example 1111 —— C22H16F2N6O2
US9796708, Example 1111
—— US9796708, Example 656 —— C20H18N4O
US9796708, Example 656
—— US9796708, Example 941 —— C25H26BFN4O4
US9796708, Example 941
—— US9434719, 401 as TFA salt —— C20H20F2N6O2
US9434719, 401 as TFA salt
—— US9650358, Example 43 —— C26H22ClFN6
US9650358, Example 43