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—— US9670204, 173 2-(5-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-1,2,4-thiadiazol-3-yl)-5-fluorobenzonitrile —— C29H31FN8O2S
US9670204, 173 2-(5-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-1,2,4-thiadiazol-3-yl)-5-fluorobenzonitrile
—— US9796708, Example 906 —— C26H23FN4O3
US9796708, Example 906
—— US9796708, Example 948 —— C24H23FN4O2
US9796708, Example 948
—— US9796708, Example 347 —— C25H23F3N4
US9796708, Example 347
—— US9796708, Example 436 —— C25H23FN4O
US9796708, Example 436
—— US9670204, 158 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(2,2,2-trifluoroacetoyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide —— C29H31F4N7O2S
US9670204, 158 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(2,2,2-trifluoroacetoyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide
—— US9670204, 63 tert-butyl4-(3-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)-3-oxopiperazine-1-carboxylate —— C28H31ClN6O3S
US9670204, 63 tert-butyl4-(3-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)-3-oxopiperazine-1-carboxylate
—— US9796708, Example 1267 —— C28H30F2N4O3
US9796708, Example 1267
—— US9796708, Example 1350 —— C27H28FN3O3
US9796708, Example 1350
—— US9796708, Example 600 —— C22H27FN4O5S
US9796708, Example 600
—— US9796708, Example 868 —— C24H25FN4O5S
US9796708, Example 868
—— US9796708, Example 346 —— C24H28F2N4O
US9796708, Example 346
—— US9670204, 54 N-(2-ethyl-6-(4-(methylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C24H27FN6O2S2
US9670204, 54 N-(2-ethyl-6-(4-(methylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine
—— US9796708, Example 932 —— C27H28FN5O4S
US9796708, Example 932
—— US9796708, Example 1161 —— C24H26FN3O3
US9796708, Example 1161
—— US9670204, 228 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-oxoacetate —— C27H29FN6O3S
US9670204, 228 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-oxoacetate
—— US9796708, Example 1364 —— C29H30FN3O3
US9796708, Example 1364
—— US9796708, Example 964 —— C21H22FN3O
US9796708, Example 964
—— US9796708, Example 851 —— C23H25FN4O3
US9796708, Example 851
—— US9796708, Example 355 —— C26H24FN5
US9796708, Example 355
—— US9670204, 191 2-(4-(2-ethyl-3-((3-(4-fluorophenyl)-1,2,4-thiadiazol-5-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N,N-dimethylacetamide —— C27H32FN7OS
US9670204, 191 2-(4-(2-ethyl-3-((3-(4-fluorophenyl)-1,2,4-thiadiazol-5-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N,N-dimethylacetamide
—— US9796708, Example 831 —— C19H18FN3O
US9796708, Example 831
—— US9796708, Example 408 —— C25H21F3N4
US9796708, Example 408
—— US9796708, Example 1067 —— C21H19FN6O
US9796708, Example 1067
—— US9796708, Example 657 —— C18H15ClFN3
US9796708, Example 657
—— US9670204, 163 2-(4-(3-((4-(2-cyano-4-fluorophenyl)-5-methylthiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N-methylacetamide —— C28H31FN8OS
US9670204, 163 2-(4-(3-((4-(2-cyano-4-fluorophenyl)-5-methylthiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N-methylacetamide
—— US9796708, Example 1074 —— C22H25FN4O4S
US9796708, Example 1074
—— US9796708, Example 764 —— C25H27FN4O3
US9796708, Example 764
—— US9796708, Example 1153 —— C23H23FN4O2
US9796708, Example 1153
—— US9796708, Example 599 —— C24H25FN4O2
US9796708, Example 599
—— US9796708, Example 1326 —— C19H18FN5O
US9796708, Example 1326
—— US9796708, Example 1300 —— C26H28F2N4O3
US9796708, Example 1300
—— US9670204, 171 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N,N-dimethylacetamide —— C29H32FN7OS
US9670204, 171 2-(4-(3-((4-(2-cyano-4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-N,N-dimethylacetamide
—— US9796708, Example 587 —— C20H23FN4O2S
US9796708, Example 587
—— US9670204, 126 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-2-(pyrrolidin-1-yl)ethanone —— C30H35FN6OS
US9670204, 126 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-2-(pyrrolidin-1-yl)ethanone
—— US9796708, Example 539 —— C25H20F3N3O
US9796708, Example 539
—— US9796708, Example 556 —— C25H30N4O2
US9796708, Example 556
—— US9670204, 99 4-(2-chloro-4-fluorophenyl)-N-(2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)-N-methylthiazol-2-amine —— C25H27ClFN5O2S2
US9670204, 99 4-(2-chloro-4-fluorophenyl)-N-(2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)-N-methylthiazol-2-amine
—— US9796708, Example 738 —— C24H28N4O3
US9796708, Example 738
—— US9796708, Example 965 —— C23H26FN5O5S
US9796708, Example 965
—— US9670204, 140 2-(4-(3-((5-cyano-4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide —— C28H31FN8OS
US9670204, 140 2-(4-(3-((5-cyano-4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)-2-ethylimidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-N,N-dimethylacetamide
—— US9796708, Example 382 —— C25H21F2N3O
US9796708, Example 382
—— US9796708, Example 574 —— C28H27FN4O2
US9796708, Example 574
—— US9796708, Example 1359 —— C27H27F2N3O3
US9796708, Example 1359
—— US9670204, 154 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one —— C28H32FN5O2S
US9670204, 154 1-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one
—— US9796708, Example 417 —— C27H25F3N4O2
US9796708, Example 417
—— US9796708, Example 356 —— C26H27FN4O2S
US9796708, Example 356
—— US9796708, Example 1298 —— C26H28F2N4O3
US9796708, Example 1298
—— US9796708, Example 992 —— C25H30FN3O3
US9796708, Example 992
—— US9796708, Example 686 —— C21H21FN4O3S
US9796708, Example 686