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中文名称 英文名称 CAS号 化学式
—— US9434719, 440 as TFA salt —— C19H15F5N6O2S
—— US9434719, 428 as TFA salt —— C20H18F4N6O2S
—— US9434719, 314 as TFA salt —— C19H19F5N4O4
—— US9434719, 464 as TFA salt —— C22H19F5N6O2
—— US9434719, 272 as TFA salt —— C17H17BrF2N4O3
—— US9434719, 286 as TFA salt —— C17H17Cl2FN4O3
—— US9434719, 280 as TFA salt —— C16H16BrF2N5O3
—— US9434719, 261 as TFA salt —— C20H25FN4O3
—— US9434719, 318 as TFA salt —— C16H18BrN5O3
—— US9434719, 462 as TFA salt —— C22H18F6N6O2
—— US9434719, 220 as TFA salt —— C20H20Cl2N6O3
—— US9434719, 438 as TFA salt —— C19H16ClF2N5O2S
—— US9434719, 247 as TFA salt —— C20H19F3N6O3S
—— US9434719, 277 as TFA salt —— C17H17ClF2N4O3
—— US9434719, 279 as TFA salt —— C16H16BrF2N5O3
—— US9434719, 241 as TFA salt —— C20H22ClN7O3
—— US9434719, 218 as TFA salt —— C20H19ClFN5O4
—— US9434719, 434 as TFA salt —— C20H18F4N6O2
—— US9434719, 325 as TFA salt —— C23H20F5N5O3
—— US9434719, 264 as TFA salt —— C20H20F2N6O3
—— US9434719, 245 as TFA salt —— C20H21F5N4O4
—— US9434719, 442 as TFA salt —— C22H19F4N5O2
—— US9434719, 209 as TFA salt —— C21H22ClFN6O3
—— US9434719, 234 as TFA salt —— C19H19ClN6O3S
—— US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)thiazol-4-yl)-5-fluorobenzonitrile —— C29H31FN8O2S
—— US9670204, 162 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile —— C30H33FN8O2S
—— US9670204, 67 N-(6-(1-(chloromethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C25H25ClFN5O2S2
—— US9670204, 182 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-thiomorpholine1,1-dioxide —— C23H24FN5O2S2
—— US9670204, 75 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-ylsulfonyl)propan-1-ol —— C27H30FN5O3S2
—— US9670204, 151 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)-5-(hydroxymethyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)-1-(pyrrolidin-1-yl)ethanone —— C31H37FN6O2S
—— US9670204, 49 (4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)(1-(methylsulfonyl)pyrrolidin-3-yl)methanone —— C29H34FN7O3S2
—— US9670204, 108 ethyl2-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-5,6-dihydropyridin-1(2H)-yl)acetate —— C28H30FN5O2S
—— US9670204, 130 3-(dimethylamino)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperidin-1-yl)propan-1-one —— C29H35FN6OS
—— US9670204, 203 (S)-1-(4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)piperazin-1-yl)-2-hydroxypropan-1-one —— C26H29FN6O2S
—— US9670204, 159 1-(2-((2-ethyl-6-(1-(2-(3-hydroxyazetidin-1-yl)-2-oxoethyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl)-2,2,2-trifluoroethanone —— C31H32F4N6O3S
—— US9670204, 189 N-(2-ethyl-6-(1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)imidazo[1,2-a]pyridin-3-yl)-3-(4-fluorophenyl)-N-methyl-1,2,4-oxadiazol-5-amine —— C24H25FN6O3S
—— US9670204, 149 (2-((6-(1-(3-(dimethylamino)propyl-sulfonyl)piperidin-4-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)(methyl)amino)-4-(4-fluorophenyl)thiazol-5-yl) —— C30H39FN6O3S2
—— US9670204, 207 2-(2-ethyl-4-((4-(4-chlorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-1-[1,2]thiazinane-1,1-dioxide —— C23H24ClN5O2S2
—— US9670204, 97 2-(2-((2-ethyl-6-(1-(methylsulfonyl)piperidin-4-yl)imidazo[1,2-a]pyridin-3-yl)(methyl)amino)-5-methylthiazol-4-yl)-5-fluorobenzonitrile —— C27H29FN6O2S2
—— US9670204, 57 N-(2-ethyl-6-(4-(3-(pyrrolidin-1-yl)propylsulfonyl)piperazin-1-yl)imidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine —— C30H38FN7O2S2
—— US9670204, 208 4-(2-ethyl-3-((4-(4-fluorophenyl)thiazol-2-yl)(methyl)amino)imidazo[1,2-a]pyridin-6-yl)-N-(thiophen-2-yl)-5,6-dihydropyridine-1(2H)-carboxamide —— C29H27FN6OS2
—— Unk-N(Tfa)4Abz-hTyr-OH —— C26H22F3N7O6
—— Unk-N(Tfa)4Abz-Tyr-OBn —— C32H26F3N7O6
—— Unk-N(Tfa)4Abz-N(Me)Tyr-OH —— C26H22F3N7O6
—— US9611261, Example 276 —— C18H15Cl2FN4O2
—— US9611261, Example 341 —— C20H15ClF3N5O
—— Undecane-1,8,10-triol —— C11H24O3
—— US9624241, Example 103 —— C24H25N5O2
—— US9624241, Example 89 —— C21H20N4O4
—— undecan-6-yl (10R,15S)-12-[4-(4-fluorophenyl)-4-oxobutyl]-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-triene-4-carboxylate —— C35H48FN3O3