中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3-cyano-4-methylsulfonylphenyl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H31FN4O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[3-[[dimethyl(oxo)-lambda6-sulfanylidene]amino]phenyl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H35FN4O4S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(2,4-dimethylpyrazol-3-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H32FN5O3 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C26H29FN4O3S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[2-[4-(2-amino-4-fluorophenyl)-3-(hydroxymethyl)phenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H33FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(2-oxo-1,3-dihydroindol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H31FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-fluoro-4-(2-oxo-1,3-dihydroindol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H31FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-cyano-6-oxo-3-(trifluoromethyl)-5H-phenanthridin-8-yl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H28F3N5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[(8R,9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-8-yl]-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H39FN4O4 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(3-methyl-2-oxo-1,3-benzoxazol-5-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C30H31FN4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-phenylpiperazin-1-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H38FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(2-methoxyethyl)pyrrolidin-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H39FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(3-cyano-9-fluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H28FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-naphthalen-2-ylethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C25H29N3O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H29F4N5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(oxolan-3-yl)-3,6-dihydro-2H-pyridin-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H39FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(oxan-4-ylcarbamoyl)thiophen-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H37FN4O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[4-(1-benzyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl)-2-fluorophenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C34H44FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[3-(oxolan-3-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H42FN5O4 |
|
—— |
Trifluoro-(1,1,2,2,2-pentafluoroethoxy)-(1,1,2,2,2-pentafluoroethyl)-lambda5-phosphane |
—— |
C4F13OP |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-[4-(methanesulfonamido)phenyl]phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C29H33FN4O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(propylcarbamoyl)thiophen-3-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H35FN4O4S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[5-(oxolan-3-yl)-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-1-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H42FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(2,9-difluoro-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H28F2N4O4 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(5-methoxycarbonylthiophen-3-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C28H30FN3O5S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[2-[4-(3-carbamoylphenyl)-2-fluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H31FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(2-fluoro-4-pyrazol-1-ylphenyl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C24H28FN5O3 |
|
—— |
tert-butyl 3-[2-cyano-2-[[(1R,3S,4S)-2-[(2-methylpropan-2-yl)oxycarbonyl]-2-azabicyclo[2.2.1]heptane-3-carbonyl]amino]ethyl]carbazole-9-carboxylate |
—— |
C32H38N4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-morpholin-4-yl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H34FN5O4S |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[4-(1-ethylpyrazol-4-yl)-2-fluorophenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C27H32FN5O3 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(1-methylindazol-5-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C30H32FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(1-ethylpyrazol-4-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H32FN5O3 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methyl-1-oxo-3H-isoindol-5-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C31H33FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-2-[4-[(Z)-1-amino-3-(oxan-4-ylmethylimino)prop-1-en-2-yl]-2,3-difluorophenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H39F2N5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-(2-methoxy-6-oxo-5H-phenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H32N4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(2-methoxyethyl)-2-oxo-3H-indol-6-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C32H37FN4O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(2-methylindazol-3-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H32FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[4-(6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carbonyl)furan-2-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C32H35FN6O5 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[2-fluoro-4-(2-oxo-1,3-dihydroindol-5-yl)phenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C30H31FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-[1-(oxolan-2-ylmethyl)pyrazol-4-yl]phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H36FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(3,3-dimethyl-1-oxo-2-benzofuran-5-yl)-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C31H34FN3O5 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[1-cyano-2-[2-[(2-methylpropan-2-yl)oxycarbonylamino]-6-oxo-5H-phenanthridin-8-yl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C33H39N5O6 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-(9-fluoro-5-methyl-6-oxophenanthridin-8-yl)ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C29H31FN4O4 |
|
—— |
tert-butyl (1R,2R,4S,5S,7S)-7-[[(1S)-1-cyano-2-[4-(5-cyanothiophen-2-yl)-2-fluorophenyl]ethyl]carbamoyl]-6-azatricyclo[3.2.1.02,4]octane-6-carboxylate |
—— |
C27H27FN4O3S |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[(2S)-2,4-dimethylpiperazin-1-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C27H38FN5O3 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-[1-(2,2-difluoroethyl)-6-oxopyridin-3-yl]-2-fluorophenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H31F3N4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-(2-fluoro-4-piperidin-3-ylphenyl)-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H37FN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[2-[2-chloro-4-(1-methyl-2-oxo-3H-indol-6-yl)phenyl]-1-cyanoethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C30H33ClN4O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(2S)-1-amino-3-[2-fluoro-4-(5-methyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-1-yl)phenyl]-1-oxopropan-2-yl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C28H40FN5O4 |
|
—— |
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[2-fluoro-4-(4-methyl-2-oxopiperazin-1-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate |
—— |
C26H34FN5O4 |
|