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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-(propan-2-ylsulfonimidoyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C27H34N6O5S
tert-butyl 5-(cyanomethyl)-5-[4-oxo-3-[4-(propan-2-ylsulfonimidoyl)anilino]-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl 4-(cyanomethyl)-3-fluoro-4-[3-[3-methyl-4-(thiomorpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate —— C30H36FN7O4S
tert-butyl 4-(cyanomethyl)-3-fluoro-4-[3-[3-methyl-4-(thiomorpholine-4-carbonyl)anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]piperidine-1-carboxylate
—— tert-butyl 3-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-3-(cyanomethyl)azetidine-1-carboxylate —— C16H20N6O3
tert-butyl 3-(3-amino-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl)-3-(cyanomethyl)azetidine-1-carboxylate
—— tert-butyl N-[2-[[3-(4,4-dimethylcyclohexen-1-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]carbamate —— C25H42N4O3
tert-butyl N-[2-[[3-(4,4-dimethylcyclohexen-1-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]carbamate
—— tert-butyl 3-[(E)-3-oxo-3-(2-oxo-4-phenyl-1,3-oxazolidin-3-yl)prop-1-enyl]indole-1-carboxylate —— C25H24N2O5
tert-butyl 3-[(E)-3-oxo-3-(2-oxo-4-phenyl-1,3-oxazolidin-3-yl)prop-1-enyl]indole-1-carboxylate
—— tert-butyl 3-[(2S,3R)-3-bromo-4-oxo-4-(2-oxo-4-phenyl-1,3-oxazolidin-3-yl)butan-2-yl]indole-1-carboxylate —— C26H27BrN2O5
tert-butyl 3-[(2S,3R)-3-bromo-4-oxo-4-(2-oxo-4-phenyl-1,3-oxazolidin-3-yl)butan-2-yl]indole-1-carboxylate
—— tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-[methyl(2,2,2-trifluoroethyl)carbamoyl]anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate —— C29H33F3N6O5
tert-butyl 5-(cyanomethyl)-5-[3-[3-methyl-4-[methyl(2,2,2-trifluoroethyl)carbamoyl]anilino]-4-oxo-2H-pyrazolo[4,3-c]pyridin-1-yl]oxane-2-carboxylate
—— tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-3-piperidin-4-ylpyrazol-4-yl]methyl]amino]ethyl]carbamate —— C23H41N5O3
tert-butyl N-methyl-N-[2-[methyl-[[1-[(2R)-oxan-2-yl]-3-piperidin-4-ylpyrazol-4-yl]methyl]amino]ethyl]carbamate
—— tert-butyl methyl(2-(methyl((5-((tetrahydro-2H-pyran-4-yl)oxy)-1-tosyl-1H-indazol-3-yl)methyl)amino)ethyl)carbamate —— C29H40N4O6S
tert-butyl methyl(2-(methyl((5-((tetrahydro-2H-pyran-4-yl)oxy)-1-tosyl-1H-indazol-3-yl)methyl)amino)ethyl)carbamate
—— tert-butyl N-[2-[[3-(1,4-dioxaspiro[4.5]dec-7-en-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate —— C26H42N4O5
tert-butyl N-[2-[[3-(1,4-dioxaspiro[4.5]dec-7-en-8-yl)-1-[(2R)-oxan-2-yl]pyrazol-4-yl]methyl-methylamino]ethyl]-N-methylcarbamate
—— tert-butyl methyl(2-(methyl((5-((tetrahydrofuran-3-yl)oxy)-1-tosyl-1H-indazol-3-yl)methyl)amino)ethyl)carbamate —— C28H38N4O6S
tert-butyl methyl(2-(methyl((5-((tetrahydrofuran-3-yl)oxy)-1-tosyl-1H-indazol-3-yl)methyl)amino)ethyl)carbamate
—— tert-butyl N-(propan-2-ylsulfonylmethyl)carbamate —— C9H19NO4S
tert-butyl N-(propan-2-ylsulfonylmethyl)carbamate
—— tert-butyl 4-methylpiperidine-1-carboxylate;N-ethylethanamine —— C15H32N2O2
tert-butyl 4-methylpiperidine-1-carboxylate;N-ethylethanamine
—— Tert-butyl 4-[3-[7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate —— C24H32N4O3
Tert-butyl 4-[3-[7-(hydroxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate
—— tert-butyl-[5-fluoro-2-[[(E)-3-(1-methylpyrazol-4-yl)prop-2-enoyl]amino]phenyl]carbamic acid —— C18H21FN4O3
tert-butyl-[5-fluoro-2-[[(E)-3-(1-methylpyrazol-4-yl)prop-2-enoyl]amino]phenyl]carbamic acid
—— Tert-butyl-dimethyl-[7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[4.5]dec-7-en-10-yl]oxysilane —— C22H41BO3Si
Tert-butyl-dimethyl-[7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[4.5]dec-7-en-10-yl]oxysilane
—— tert-butyl N-methyl-N-[2-[methyl([[1-(oxan-2-yl)-3-(4-oxocyclohexyl)-1H-pyrazol-4-yl]methyl])amino]ethyl]carbamate —— C24H40N4O4
tert-butyl N-methyl-N-[2-[methyl([[1-(oxan-2-yl)-3-(4-oxocyclohexyl)-1H-pyrazol-4-yl]methyl])amino]ethyl]carbamate
—— Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate —— C42H70BN3O9Si
Tert-butyl 3-[2-[[2-[3-[tert-butyl(dimethyl)silyl]oxy-4-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate
—— tert-butyl 5-((tert-butyldimethylsilyl)oxy)tetrahydro-2H-pyran-2-carboxylate —— C16H32O4Si
tert-butyl 5-((tert-butyldimethylsilyl)oxy)tetrahydro-2H-pyran-2-carboxylate
—— Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.3.1]nona-1(8),5(9),6-trien-9-yl]oxy]silane —— C21H28N2OSi
Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.3.1]nona-1(8),5(9),6-trien-9-yl]oxy]silane
—— tert-butyl 3-(2-(((R)-1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-2,2-dimethylbut-3-en-1-yl)carbamoyl)phenyl)pyrrolidine-1-carboxylate —— C38H42F2N4O3
tert-butyl 3-(2-(((R)-1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-2,2-dimethylbut-3-en-1-yl)carbamoyl)phenyl)pyrrolidine-1-carboxylate
—— Tert-butyl 6-[[(5-amino-6-chloroquinoline-8-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexane-1-carboxylate —— C21H25ClN4O3
Tert-butyl 6-[[(5-amino-6-chloroquinoline-8-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexane-1-carboxylate
—— tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2R)-4-[6-(2,5-dioxopyrrol-1-yl)hexanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C47H57F3N6O8
tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2R)-4-[6-(2,5-dioxopyrrol-1-yl)hexanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2R)-4-[3-(2,5-dioxopyrrol-1-yl)propanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C44H51F3N6O8
tert-butyl (3R,4R)-3-[[[(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2R)-4-[3-(2,5-dioxopyrrol-1-yl)propanoyl]morpholine-2-carbonyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[(1R)-4-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethylamino]-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-oxobutyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C43H59F3N8O8
tert-butyl 3-[[[(1R)-4-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethylamino]-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-oxobutyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[2-[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-4-hydroxy-2,2-dimethylbutyl]carbamoyl]phenoxy]azetidine-1-carboxylate —— C37H42F2N4O5
tert-butyl 3-[2-[[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-4-hydroxy-2,2-dimethylbutyl]carbamoyl]phenoxy]azetidine-1-carboxylate
—— tert-butyl N-[1-(thiophen-2-ylamino)propan-2-yl]carbamate —— C12H20N2O2S
tert-butyl N-[1-(thiophen-2-ylamino)propan-2-yl]carbamate
—— tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C36H46F3N5O5
tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[(2S)-2-acetyloxypropanoyl]-[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethylbut-3-enyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C37H45F3N4O5
tert-butyl 3-[[[(2S)-2-acetyloxypropanoyl]-[(1R)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethylbut-3-enyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-methylsulfonyloxypyrrolidine-1-carboxylate —— C36H46F2N4O8S
tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[(2S)-2-hydroxypropanoyl]amino]methyl]-4-methylsulfonyloxypyrrolidine-1-carboxylate
—— tert-butyl 3-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-1,2-dihydroxyethyl]pyrrolidine-1-carboxylate —— C17H35NO5Si
tert-butyl 3-[(2R)-2-[tert-butyl(dimethyl)silyl]oxy-1,2-dihydroxyethyl]pyrrolidine-1-carboxylate
—— tert-butyl 3-[[[(1S)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2-[tert-butyl(dimethyl)silyl]oxy-2-methylpropyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C40H58F3N5O5Si
tert-butyl 3-[[[(1S)-1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2-[tert-butyl(dimethyl)silyl]oxy-2-methylpropyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.3.1]nona-1(8),5(9),6-trien-8-yl]oxy]silane —— C21H28N2OSi
Trimethyl-[[3-(2-pyrrolidin-1-ylphenyl)-2-azabicyclo[3.3.1]nona-1(8),5(9),6-trien-8-yl]oxy]silane
—— tert-butyl 4-[4-(4-hydroxypyrido[3,4-d]pyrimidin-2-yl)oxypyridin-2-yl]piperazine-1-carboxylate —— C21H24N6O4
tert-butyl 4-[4-(4-hydroxypyrido[3,4-d]pyrimidin-2-yl)oxypyridin-2-yl]piperazine-1-carboxylate
—— Tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(2-hydroxyethylcarbamoyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C35H44F3N5O5
Tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-(2-hydroxyethylcarbamoyl)amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— Tert-butyl 3-[2-[[1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-4-[2-(2,5-dioxopyrrol-1-yl)ethylamino]-2,2-dimethyl-4-oxobutyl]carbamoyl]phenoxy]azetidine-1-carboxylate —— C43H46F2N6O7
Tert-butyl 3-[2-[[1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-4-[2-(2,5-dioxopyrrol-1-yl)ethylamino]-2,2-dimethyl-4-oxobutyl]carbamoyl]phenoxy]azetidine-1-carboxylate
—— tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-[1-[tert-butyl(dimethyl)silyl]oxycyclopropyl]methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C40H56F3N5O5Si
tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-[1-[tert-butyl(dimethyl)silyl]oxycyclopropyl]methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— Tert-butyl 3-[2-[[1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-oxo-4-(pentylamino)butyl]carbamoyl]phenoxy]azetidine-1-carboxylate —— C42H51F2N5O5
Tert-butyl 3-[2-[[1-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-2,2-dimethyl-4-oxo-4-(pentylamino)butyl]carbamoyl]phenoxy]azetidine-1-carboxylate
—— Tert-butyl 3-[2-[(2-chloroacetyl)amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate —— C26H37BClNO6
Tert-butyl 3-[2-[(2-chloroacetyl)amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]-2-methoxybenzoate
—— Tert-butyl 2-methoxy-3-[2-[[2-[4-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate —— C36H56BN3O8
Tert-butyl 2-methoxy-3-[2-[[2-[4-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]acetyl]amino]-2-(2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl)ethyl]benzoate
—— Tert-butyl 4-cyano-4-methylsulfonylpiperidine-1-carboxylate —— C12H20N2O4S
Tert-butyl 4-cyano-4-methylsulfonylpiperidine-1-carboxylate
—— tert-butyl 3-[[[(2S)-1-azidopropan-2-yl]carbamoyl-[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate —— C36H45F3N8O4
tert-butyl 3-[[[(2S)-1-azidopropan-2-yl]carbamoyl-[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]amino]methyl]-4-fluoropyrrolidine-1-carboxylate
—— tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]pyrrolidine-1-carboxylate —— C36H47F2N5O5
tert-butyl 3-[[[[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(oxan-4-yl)methyl]-[[(2S)-1-hydroxypropan-2-yl]carbamoyl]amino]methyl]pyrrolidine-1-carboxylate
—— tert-butyl 2-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)-4-morpholino-5,6-dihydropyrido[3,4-d]pyrimidine-7(8H)-carboxylate —— C31H34F3N5O4
tert-butyl 2-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)-4-morpholino-5,6-dihydropyrido[3,4-d]pyrimidine-7(8H)-carboxylate
—— tert-butyl N-methyl-N-[2-[methyl-[[3-[1-(3-methylbutanoyl)piperidin-4-yl]-5-[(2R)-oxan-2-yl]-1H-pyrazol-4-yl]methyl]amino]ethyl]carbamate —— C28H49N5O4
tert-butyl N-methyl-N-[2-[methyl-[[3-[1-(3-methylbutanoyl)piperidin-4-yl]-5-[(2R)-oxan-2-yl]-1H-pyrazol-4-yl]methyl]amino]ethyl]carbamate
—— Tert-butyl 4-[3-[3-fluoro-7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate —— C25H33FN4O3
Tert-butyl 4-[3-[3-fluoro-7-(methoxymethyl)pyrido[3,4-b]indol-9-yl]propyl]piperazine-1-carboxylate
—— Tert-butyl 4-[4-[5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]-3-cyanobenzoyl]-1,4-diazepane-1-carboxylate 1232417-90-1 C30H30N8O4
Tert-butyl 4-[4-[5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]-3-cyanobenzoyl]-1,4-diazepane-1-carboxylate
—— Tert-butyl 2-methyl-4-phenyl-5-sulfanylpentanoate —— C16H24O2S
Tert-butyl 2-methyl-4-phenyl-5-sulfanylpentanoate
—— tert-butyl N-[1-[4-[5-[3-amino-6-(4-propan-2-ylsulfonylphenyl)pyrazin-2-yl]-1,3,4-oxadiazol-2-yl]phenyl]ethyl]carbamate —— C28H32N6O5S
tert-butyl N-[1-[4-[5-[3-amino-6-(4-propan-2-ylsulfonylphenyl)pyrazin-2-yl]-1,3,4-oxadiazol-2-yl]phenyl]ethyl]carbamate
—— tert-butyl N-[(2S)-1-[[(2S)-5-(carbamoylamino)-1-[4-(isothiocyanatomethyl)anilino]-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate —— C24H36N6O5S
tert-butyl N-[(2S)-1-[[(2S)-5-(carbamoylamino)-1-[4-(isothiocyanatomethyl)anilino]-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate