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—— tert-butyl N-[(2S)-1-[[(2S)-3,3-dimethyl-1-oxo-1-[(2S)-2-[(2-phenylethylamino)methyl]pyrrolidin-1-yl]butan-2-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate 915237-04-6 C28H46N4O4
tert-butyl N-[(2S)-1-[[(2S)-3,3-dimethyl-1-oxo-1-[(2S)-2-[(2-phenylethylamino)methyl]pyrrolidin-1-yl]butan-2-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate
—— Tert-butyl 3-[7-[bis(2-trimethylsilylethoxymethyl)amino]-3-(1-methylpyrazol-4-yl)-6-thiophen-2-ylpyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carboxylate 934297-30-0 C36H57N7O4SSi2
Tert-butyl 3-[7-[bis(2-trimethylsilylethoxymethyl)amino]-3-(1-methylpyrazol-4-yl)-6-thiophen-2-ylpyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carboxylate
—— Tert-butyl 3-(6-bromo-7-chloropyrazolo[1,5-a]pyrimidin-5-yl)piperidine-1-carboxylate 934297-15-1 C16H20BrClN4O2
Tert-butyl 3-(6-bromo-7-chloropyrazolo[1,5-a]pyrimidin-5-yl)piperidine-1-carboxylate
—— tert-butyl N-[(2S)-1-[[5-methyl-4-phenyl-1-(2-trimethylsilylethoxymethyl)imidazol-2-yl]methyl-propan-2-ylamino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]-1-oxopropan-2-yl]carbamate 864825-61-6 C38H58N4O5Si
tert-butyl N-[(2S)-1-[[5-methyl-4-phenyl-1-(2-trimethylsilylethoxymethyl)imidazol-2-yl]methyl-propan-2-ylamino]-3-[4-[(2-methylpropan-2-yl)oxy]phenyl]-1-oxopropan-2-yl]carbamate
—— tert-butyl 4-[(2S)-4-[6-amino-3-chloro-5-(5-methyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]-2-ethylpiperazin-1-yl]piperidine-1-carboxylate 907207-93-6 C23H35ClN8O3
tert-butyl 4-[(2S)-4-[6-amino-3-chloro-5-(5-methyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl]-2-ethylpiperazin-1-yl]piperidine-1-carboxylate
—— tert-butyl N-[(2S)-1-[(benzotriazole-1-carbothioylamino)methyl-methylamino]-1-oxo-3-phenylpropan-2-yl]carbamate 1005383-61-8 C23H28N6O3S
tert-butyl N-[(2S)-1-[(benzotriazole-1-carbothioylamino)methyl-methylamino]-1-oxo-3-phenylpropan-2-yl]carbamate
—— tert-butyl (3S)-4-[1-[(4-chlorophenyl)methyl]-4-methylpiperidin-4-yl]-3-methylpiperazine-1-carboxylate 906559-55-5 C23H36ClN3O2
tert-butyl (3S)-4-[1-[(4-chlorophenyl)methyl]-4-methylpiperidin-4-yl]-3-methylpiperazine-1-carboxylate
—— tert-butyl (1S)-1-[methyl-[(1S)-1-phenylethyl]amino]spiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxylate 878167-42-1 C27H36N2O2
tert-butyl (1S)-1-[methyl-[(1S)-1-phenylethyl]amino]spiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxylate
—— tert-butyl N-[6-[4-(2-aminopropan-2-yl)phenyl]-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-4-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 1236410-05-1 C27H37N5O6
tert-butyl N-[6-[4-(2-aminopropan-2-yl)phenyl]-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-4-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— Tert-butyl 6-[1-tri(propan-2-yl)silylpyrrol-3-yl]-2,3-dihydroindole-1-carboxylate 1049001-58-2 C26H40N2O2Si
Tert-butyl 6-[1-tri(propan-2-yl)silylpyrrol-3-yl]-2,3-dihydroindole-1-carboxylate
—— Toluene-4-sulfonic acid 2-[2-(N-methyl-N-BOC-aminooxy)-ethoxy]-ethyl ester 1034710-22-9 C17H27NO7S
Toluene-4-sulfonic acid 2-[2-(N-methyl-N-BOC-aminooxy)-ethoxy]-ethyl ester
—— tert-butyl N-[2-(2-(18F)fluoranylethoxy)ethoxy]-N-methylcarbamate 1034710-43-4 C10H20FNO4
tert-butyl N-[2-(2-(18F)fluoranylethoxy)ethoxy]-N-methylcarbamate
—— tert-Butyl 1,3-thiazol-4-yl[(2,4,5-trifluorophenyl)sulfonyl]carbamate 1235406-62-8 C14H13F3N2O4S2
tert-Butyl 1,3-thiazol-4-yl[(2,4,5-trifluorophenyl)sulfonyl]carbamate
—— tert-butyl N-[3-[methyl-(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]propyl]-N-[4-[(2-methylpropan-2-yl)oxycarbonyl-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]amino]butyl]carbamate 1104804-44-5 C32H53N7O9
tert-butyl N-[3-[methyl-(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]propyl]-N-[4-[(2-methylpropan-2-yl)oxycarbonyl-[3-[(2-methylpropan-2-yl)oxycarbonylamino]propyl]amino]butyl]carbamate
—— tert-butyl {2-[4-(4-amino-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl)phenyl]-2-methylpropyl}carbamate 1236408-37-9 C23H31N5O4
tert-butyl {2-[4-(4-amino-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl)phenyl]-2-methylpropyl}carbamate
—— tert-butyl N-[6-[4-(2-acetamidopropan-2-yl)phenyl]-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-4-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 1236410-06-2 C29H39N5O7
tert-butyl N-[6-[4-(2-acetamidopropan-2-yl)phenyl]-2-methoxy-5-oxo-7,8-dihydropyrido[4,3-d]pyrimidin-4-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— tert-butyl 4-(5-chloro-4-fluoro-2-hydroxyphenyl)-1H-pyrazole-1-carboxylate 1235407-14-3 C14H14ClFN2O3
tert-butyl 4-(5-chloro-4-fluoro-2-hydroxyphenyl)-1H-pyrazole-1-carboxylate
—— tert-butyl (3S)-3-[(1-methylpiperidin-4-yl)-phenylmethoxycarbonylamino]piperidine-1-carboxylate 1107638-92-5 C24H37N3O4
tert-butyl (3S)-3-[(1-methylpiperidin-4-yl)-phenylmethoxycarbonylamino]piperidine-1-carboxylate
—— tert-butyl N-[(2R)-1-[2-(ethylcarbamothioyl)hydrazinyl]-1-oxo-3-pyridin-3-ylpropan-2-yl]carbamate 944705-72-0 C16H25N5O3S
tert-butyl N-[(2R)-1-[2-(ethylcarbamothioyl)hydrazinyl]-1-oxo-3-pyridin-3-ylpropan-2-yl]carbamate
—— tert-butyl (2S,4R)-2-{[(1R,13E,15S)-4,4-dioxido-2-oxo-4-thia-3-azaspiro(bicyclo[13.1.0]hexadecane-5,1'-cyclopropane]-13-en-1-yl]carbamoyl}-4-({2-[2-(isopropylamino)-1,3-thiazol-4-yl]-7-methoxyquinolin-4-yl}oxy)pyrrolidine-1-carboxylate 1013924-96-3 C42H56N6O8S2
tert-butyl (2S,4R)-2-{[(1R,13E,15S)-4,4-dioxido-2-oxo-4-thia-3-azaspiro(bicyclo[13.1.0]hexadecane-5,1'-cyclopropane]-13-en-1-yl]carbamoyl}-4-({2-[2-(isopropylamino)-1,3-thiazol-4-yl]-7-methoxyquinolin-4-yl}oxy)pyrrolidine-1-carboxylate
—— tert-Butyl N-[2-(ethanesulfonyl)phenyl]carbamate 1365272-94-1 C13H19NO4S
tert-Butyl N-[2-(ethanesulfonyl)phenyl]carbamate
—— Tert-butyl 3-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2-methoxyphenyl]methyl-methylamino]propanoate 1111235-47-2 C37H50N6O7S
Tert-butyl 3-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2-methoxyphenyl]methyl-methylamino]propanoate
—— Tert-butyl 2-[2-[2-[methyl(pyridin-2-yl)amino]ethoxy]-5-nitrophenoxy]acetate 1111238-52-8 C20H25N3O6
Tert-butyl 2-[2-[2-[methyl(pyridin-2-yl)amino]ethoxy]-5-nitrophenoxy]acetate
—— tert-butyl N-[3-[7-(benzenesulfonyl)-4-[3-(hydroxymethyl)-4,5-dimethoxyanilino]pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate 1111236-60-2 C30H37N5O7S
tert-butyl N-[3-[7-(benzenesulfonyl)-4-[3-(hydroxymethyl)-4,5-dimethoxyanilino]pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate
—— Tert-butyl 4-(4-pyridin-4-yl-1,3-thiazol-2-yl)piperazine-1-carboxylate 668484-52-4 C17H22N4O2S
Tert-butyl 4-(4-pyridin-4-yl-1,3-thiazol-2-yl)piperazine-1-carboxylate
—— trans-2-benzyl-7-chloro-8-methyl-2,3,4,4a,6,10b-hexahydro-1H-isochromeno[4,3-c]pyridine 1135492-29-3 C20H22ClNO
trans-2-benzyl-7-chloro-8-methyl-2,3,4,4a,6,10b-hexahydro-1H-isochromeno[4,3-c]pyridine
—— tert-butyl N-[3-[7-(benzenesulfonyl)-4-(3-formyl-4,5-dimethoxyanilino)pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate 1111236-62-4 C30H35N5O7S
tert-butyl N-[3-[7-(benzenesulfonyl)-4-(3-formyl-4,5-dimethoxyanilino)pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate
—— tert-butyl 3-((1S)-1-azido-2-{[tert-butyl(dimethyl)silyl]oxy}ethyl)-5-(trifluoromethyl)benzoate 1237536-03-6 C20H30F3N3O3Si
tert-butyl 3-((1S)-1-azido-2-{[tert-butyl(dimethyl)silyl]oxy}ethyl)-5-(trifluoromethyl)benzoate
—— tert-butyl N-[3-[7-(benzenesulfonyl)-4-[3-(hydroxymethyl)-4-methoxyanilino]pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate 1111235-42-7 C29H35N5O6S
tert-butyl N-[3-[7-(benzenesulfonyl)-4-[3-(hydroxymethyl)-4-methoxyanilino]pyrrolo[2,3-d]pyrimidin-5-yl]propyl]-N-methylcarbamate
—— tert-butyl 3-[(1R)-1,2-dihydroxyethyl]-5-(trifluoromethyl)benzoate 1237536-01-4 C14H17F3O4
tert-butyl 3-[(1R)-1,2-dihydroxyethyl]-5-(trifluoromethyl)benzoate
—— tert-butyl 2-(2-methoxy-N-methyl-5-nitroanilino)acetate 1111238-24-4 C14H20N2O5
tert-butyl 2-(2-methoxy-N-methyl-5-nitroanilino)acetate
—— tert-butyl N-[(2S)-1-[[(2S)-1-[(2S)-4-[2-[[4-[[2-[(3S)-4-[(2S)-3,3-dimethyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperazin-1-yl]-2-oxoethyl]carbamoyl]benzoyl]amino]acetyl]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperazin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate 1088500-42-8 C72H102N12O14
tert-butyl N-[(2S)-1-[[(2S)-1-[(2S)-4-[2-[[4-[[2-[(3S)-4-[(2S)-3,3-dimethyl-2-[[(2S)-2-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propanoyl]amino]butanoyl]-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperazin-1-yl]-2-oxoethyl]carbamoyl]benzoyl]amino]acetyl]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]piperazin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]-N-methylcarbamate
—— Tert-butyl 2-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2,3-dimethoxyphenyl]methyl-methylamino]acetate 1111236-64-6 C37H50N6O8S
Tert-butyl 2-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2,3-dimethoxyphenyl]methyl-methylamino]acetate
—— tert-butyl 4-(1-([6-(trifluoromethyl)pyridin-2-yl]sulfonyl)ethyl)piperidine-1-carboxylate 1138331-87-9 C18H25F3N2O4S
tert-butyl 4-(1-([6-(trifluoromethyl)pyridin-2-yl]sulfonyl)ethyl)piperidine-1-carboxylate
—— tert-butyl (6-methoxybenzo[d]thiazol-2-yl)carbamate 1338645-97-8 C13H16N2O3S
tert-butyl (6-methoxybenzo[d]thiazol-2-yl)carbamate
—— Tert-butyl 4-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2-methoxyphenyl]methyl-methylamino]butanoate 1111235-55-2 C38H52N6O7S
Tert-butyl 4-[[5-[[7-(benzenesulfonyl)-5-[3-[methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propyl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2-methoxyphenyl]methyl-methylamino]butanoate
—— tert-butyl N-(3-pyrrolidin-1-ylphenyl)carbamate 1258532-12-5 C15H22N2O2
tert-butyl N-(3-pyrrolidin-1-ylphenyl)carbamate
—— tert-butyl 5-(2,2-dimethylbutyl)-2-{2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethyl}-1H-imidazole-1-carboxylate 1021938-85-1 C28H43BN2O4
tert-butyl 5-(2,2-dimethylbutyl)-2-{2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethyl}-1H-imidazole-1-carboxylate
—— tert-butyl 6-(8-(benzo[d]thiazol-2-yl((2-(trimethylsilyl)ethoxy)methyl)carbamoyl)-3,4-dihydroisoquinolin-2(lH)-yl)-3-(3-phenoxypropyl)picolinate 1235036-71-1 C42H50N4O5SSi
tert-butyl 6-(8-(benzo[d]thiazol-2-yl((2-(trimethylsilyl)ethoxy)methyl)carbamoyl)-3,4-dihydroisoquinolin-2(lH)-yl)-3-(3-phenoxypropyl)picolinate
—— tert-butyl [4-(4-fluorophenyl)-2,2-dimethyl-2H-chromen-7-yl]carbamate 1110662-48-0 C22H24FNO3
tert-butyl [4-(4-fluorophenyl)-2,2-dimethyl-2H-chromen-7-yl]carbamate
—— tert-butyl 6-(4-chlorophenyl)-1-methyl-7-oxa-3-azabicyclo[4.1.0]heptane-3-carboxylate 1108154-58-0 C17H22ClNO3
tert-butyl 6-(4-chlorophenyl)-1-methyl-7-oxa-3-azabicyclo[4.1.0]heptane-3-carboxylate
—— tert-butyl (2S)-3-(4-aminophenyl)-2-[[2-(diethylamino)-5-(2,2,2-trifluoroethyl)pyrimidin-4-yl]amino]propanoate 873686-86-3 C23H32F3N5O2
tert-butyl (2S)-3-(4-aminophenyl)-2-[[2-(diethylamino)-5-(2,2,2-trifluoroethyl)pyrimidin-4-yl]amino]propanoate
—— tert-butyl N-([1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)carbamate 1038516-66-3 C12H16N4O2
tert-butyl N-([1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)carbamate
—— tert-butyl 5-amino-3-(4-(benzyloxy)phenyl)-4-cyano-1H-pyrazole-1-carboxylate 1235034-93-1 C22H22N4O3
tert-butyl 5-amino-3-(4-(benzyloxy)phenyl)-4-cyano-1H-pyrazole-1-carboxylate
—— tert-butyl 3-(2-(l,3-dioxolan-2-yl)ethyl)-6-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(lH)-yl)picolinate 1235036-24-4 C32H34N4O5S
tert-butyl 3-(2-(l,3-dioxolan-2-yl)ethyl)-6-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(lH)-yl)picolinate
—— tert-butyl (4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl)carbamate 1266335-77-6 C14H18N4O2
tert-butyl (4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl)carbamate
—— tert-butyl 4-(1-methyl-1-([6-(trifluoromethyl)pyridin-2-yl]sulfonyl)ethyl)piperidine-1-carboxylate 1138331-88-0 C19H27F3N2O4S
tert-butyl 4-(1-methyl-1-([6-(trifluoromethyl)pyridin-2-yl]sulfonyl)ethyl)piperidine-1-carboxylate
—— tert-butyl N-[4-bromo-2-(trifluoromethyl)phenyl]carbamate 1393442-28-8 C12H13BrF3NO2
tert-butyl N-[4-bromo-2-(trifluoromethyl)phenyl]carbamate
—— t-butyl {4-[3-(3,5-dichlorophenyl)-3-(trifluoromethyl)pyrrolidin-1-yl]-2-(trifluoromethyl)benzyl}carbamate 1221694-10-5 C24H24Cl2F6N2O2
t-butyl {4-[3-(3,5-dichlorophenyl)-3-(trifluoromethyl)pyrrolidin-1-yl]-2-(trifluoromethyl)benzyl}carbamate
—— tert-butyl 3-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)azetidine-1-carboxylate 1138331-93-7 C18H24F3NO4S
tert-butyl 3-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)azetidine-1-carboxylate