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中文名称 英文名称 CAS号 化学式 结构式图片
—— TH-1120 1196071-94-9 C17H20Cl2N2O5S2
TH-1120
—— tert-butyl ((3R,5S)-5-methyl-1-(3-nitropyridin-4-yl)piperidin-3-yl)carbamate 1405128-35-9 C16H26N4O2
tert-butyl ((3R,5S)-5-methyl-1-(3-nitropyridin-4-yl)piperidin-3-yl)carbamate
—— tert-butyl 4-((4-(6-chloro-2-methylpyridin-3-yl)-2,6-difluorophenoxy)methyl)piperidine-1-carboxylate 1204130-08-4 C23H27ClF2N2O3
tert-butyl 4-((4-(6-chloro-2-methylpyridin-3-yl)-2,6-difluorophenoxy)methyl)piperidine-1-carboxylate
—— tert-butyl 4-(3-(2-tert-butoxy-2-oxoethyl)-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]pyridin-1-yl)piperidine-1-carboxylate 1222162-01-7 C22H32N4O5
tert-butyl 4-(3-(2-tert-butoxy-2-oxoethyl)-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]pyridin-1-yl)piperidine-1-carboxylate
—— tert-butyl [(3R,4R)-1-(3-aminopyridin-4-yl)-4-fluoropiperidin-3-yl]carbamate 1052713-69-5 C15H23FN4O2
tert-butyl [(3R,4R)-1-(3-aminopyridin-4-yl)-4-fluoropiperidin-3-yl]carbamate
—— tert-butyl (6S)-3-{(1E)-3-[(1R)-2,3-dihydro-1H-inden-1-yl(3-fluoro-2,2-dimethylpropanoyl)amino]prop-1-en-1-yl}-2'-oxo-5,7-dihydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-1'(2'H)-carboxylate 1338777-94-8 C36H39FN4O4
tert-butyl (6S)-3-{(1E)-3-[(1R)-2,3-dihydro-1H-inden-1-yl(3-fluoro-2,2-dimethylpropanoyl)amino]prop-1-en-1-yl}-2'-oxo-5,7-dihydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-1'(2'H)-carboxylate
—— tert-butyl [(1R,2S)-2-azido-6,6-difluoro-2-methylcyclohexyl]carbamate 1207557-31-0 C12H20F2N4O2
tert-butyl [(1R,2S)-2-azido-6,6-difluoro-2-methylcyclohexyl]carbamate
—— tert-butyl 3,3-dimethyl-4-oxo-5-(2,2,2-trifluoro-acetyl)-piperidine-1-carboxylate 1159010-26-0 C14H20F3NO4
tert-butyl 3,3-dimethyl-4-oxo-5-(2,2,2-trifluoro-acetyl)-piperidine-1-carboxylate
—— tert-butyl 1-(5-(4-(chloromethyl)-1-(4-chlorophenyl)-1H-pyrazole-3-carboxamido)pyridin-2-yl)pyrrolidin-3-yl(methyl)carbamate 1224172-23-9 C26H30Cl2N6O3
tert-butyl 1-(5-(4-(chloromethyl)-1-(4-chlorophenyl)-1H-pyrazole-3-carboxamido)pyridin-2-yl)pyrrolidin-3-yl(methyl)carbamate
—— tert-butyl 1,7,7-trimethyl-1,4,6,7-tetrahydro-pyrazolo[4,3-c]pyridine-5-carboxylate 1159009-95-6 C14H23N3O2
tert-butyl 1,7,7-trimethyl-1,4,6,7-tetrahydro-pyrazolo[4,3-c]pyridine-5-carboxylate
—— tert-butyl 6-chloro-5-methyl-pyrimidine-4-carboxylate 1159010-93-1 C10H13ClN2O2
tert-butyl 6-chloro-5-methyl-pyrimidine-4-carboxylate
—— tert-butyl 7,7-dimethyl-3-trifluoromethyl-1,4,6,7-tetrahydro-pyrazolo[4,3-c]pyridine-5-carboxylate 1159010-27-1 C14H20F3N3O2
tert-butyl 7,7-dimethyl-3-trifluoromethyl-1,4,6,7-tetrahydro-pyrazolo[4,3-c]pyridine-5-carboxylate
—— tert-Butyl 4-hydroxy-4-(morpholinomethyl)piperidine-1-carboxylate 885617-46-9 C15H28N2O4
tert-Butyl 4-hydroxy-4-(morpholinomethyl)piperidine-1-carboxylate
—— Thieno[2,3-d]pyrimidine-6-carboxamide, 4-[[4-fluoro-2-(3-piperidinyloxy)phenyl]amino]-5-methyl-N-[(4-methyl-2-morpholinyl)methyl]- 1332710-01-6 C25H31FN6O3S
Thieno[2,3-d]pyrimidine-6-carboxamide, 4-[[4-fluoro-2-(3-piperidinyloxy)phenyl]amino]-5-methyl-N-[(4-methyl-2-morpholinyl)methyl]-
—— tert-butyl 1,3-diphenyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxylate 1202800-58-5 C23H25N3O2
tert-butyl 1,3-diphenyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxylate
—— tert-butyl N-[2-[(1S)-1-(chloromethyl)-9-methyl-5-phenylmethoxy-1,2-dihydrobenzo[e]indole-3-carbonyl]-1H-pyrrolo[2,3-c]pyridin-5-yl]carbamate 1227962-40-4 C34H33ClN4O4
tert-butyl N-[2-[(1S)-1-(chloromethyl)-9-methyl-5-phenylmethoxy-1,2-dihydrobenzo[e]indole-3-carbonyl]-1H-pyrrolo[2,3-c]pyridin-5-yl]carbamate
—— tert-butyl 3-(5-methyl-1,2,4-oxadiazol-3-yl)pyrrolidine-1-carboxylate 1225218-59-6 C12H19N3O3
tert-butyl 3-(5-methyl-1,2,4-oxadiazol-3-yl)pyrrolidine-1-carboxylate
—— tert-butyl 3-(1H-pyrazol-3-yl)pyrrolidine-1-carboxylate 1225218-81-4 C12H19N3O2
tert-butyl 3-(1H-pyrazol-3-yl)pyrrolidine-1-carboxylate
—— Tert-butyl 3-(1-methyltetrazol-5-yl)pyrrolidine-1-carboxylate 1225218-84-7 C11H19N5O2
Tert-butyl 3-(1-methyltetrazol-5-yl)pyrrolidine-1-carboxylate
—— Thiazol-5-ylmethyl 2-[1-(6-fluoroquinolin-2-yl)piperidin-4-yl]ethylcarbamate 1206673-14-4 C21H23FN4O2S
Thiazol-5-ylmethyl 2-[1-(6-fluoroquinolin-2-yl)piperidin-4-yl]ethylcarbamate
—— tert-butyl (5R)-5-(5-bromo-1H-imidazol-2-yl)-3,3-dimethyl-1,3-azasilolidine-1-carboxylate 1334314-09-8 C13H22BrN3O2Si
tert-butyl (5R)-5-(5-bromo-1H-imidazol-2-yl)-3,3-dimethyl-1,3-azasilolidine-1-carboxylate
—— thiopropionic acid S-(2-((5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-ylsulfanylmethyl)-hydroxyphosphinoyloxy)ethyl) ester 1224724-32-6 C25H24ClN2O4PS2
thiopropionic acid S-(2-((5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-ylsulfanylmethyl)-hydroxyphosphinoyloxy)ethyl) ester
—— triazolo[4,5-b]pyridin-3-yl 4-[4-fluoro-2-[(3R)-oxolan-3-yl]oxyanilino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylate 1332713-18-4 C23H18FN7O4S
triazolo[4,5-b]pyridin-3-yl 4-[4-fluoro-2-[(3R)-oxolan-3-yl]oxyanilino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylate
—— Tert-butyl 4-(1,2,4-triazol-4-ylmethyl)piperidine-1-carboxylate 1225218-70-1 C13H22N4O2
Tert-butyl 4-(1,2,4-triazol-4-ylmethyl)piperidine-1-carboxylate
—— tert-butyl 3-(4H-1,2,4-triazol-4-ylmethyl)pyrrolidine-1-carboxylate 1225218-68-7 C12H20N4O2
tert-butyl 3-(4H-1,2,4-triazol-4-ylmethyl)pyrrolidine-1-carboxylate
—— tert-butyl N-[(2S)-1-(dimethylamino)-3-(3-nitrophenyl)-1-oxopropan-2-yl]carbamate 1009093-51-9 C16H23N3O5
tert-butyl N-[(2S)-1-(dimethylamino)-3-(3-nitrophenyl)-1-oxopropan-2-yl]carbamate
—— tert-butyl 3-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)pyrrolidine-1-carboxylate 1225218-57-4 C11H17N3O4
tert-butyl 3-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)pyrrolidine-1-carboxylate
—— tert-butyl N-[4-(3-aminophenyl)-1,4-dimethyl-6-oxo-5H-pyrimidin-2-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 1221447-95-5 C22H32N4O5
tert-butyl N-[4-(3-aminophenyl)-1,4-dimethyl-6-oxo-5H-pyrimidin-2-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— tert-butyl 4-((2,6-difluoro-4-(1-methylsulfonyl-piperidin-4-yl)phenoxy)methyl)piperidine-1-carboxylate 1134109-19-5 C23H34F2N2O5S
tert-butyl 4-((2,6-difluoro-4-(1-methylsulfonyl-piperidin-4-yl)phenoxy)methyl)piperidine-1-carboxylate
—— tert-butyl 2-methoxy-3-pyridin-2-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate 1202800-48-3 C17H22N4O3
tert-butyl 2-methoxy-3-pyridin-2-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate
—— tert-butyl 2-(hydroxymethyl)thiomorpholine-4-carboxylate 911223-24-0 C10H19NO3S
tert-butyl 2-(hydroxymethyl)thiomorpholine-4-carboxylate
—— tert-butyl 3-pyridin-2-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate 1202800-43-8 C16H20N4O2
tert-butyl 3-pyridin-2-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate
—— tert-butyl N-[(2S)-3-(3-aminophenyl)-1-(dimethylamino)-1-oxopropan-2-yl]carbamate 1009093-52-0 C16H25N3O3
tert-butyl N-[(2S)-3-(3-aminophenyl)-1-(dimethylamino)-1-oxopropan-2-yl]carbamate
—— tert-butyl 3-phenyl-2-(trifluoromethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate 1202800-53-0 C18H20F3N3O2
tert-butyl 3-phenyl-2-(trifluoromethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-7-carboxylate
—— tert-butyl (3R)-3-[5-(4-bromophenyl)-1H-imidazol-2-yl]thiomorpholine-4-carboxylate 1228968-54-4 C18H22BrN3O2S
tert-butyl (3R)-3-[5-(4-bromophenyl)-1H-imidazol-2-yl]thiomorpholine-4-carboxylate
—— tert-butyl 4-[[[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-5-oxopentanoyl]amino]methyl]benzoate 1334496-39-7 C30H34N4O7
tert-butyl 4-[[[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-5-oxopentanoyl]amino]methyl]benzoate
—— thiopropionic acid S-(2-((5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-ylsulfanylmethyl)-(2-propionylsulfanylethoxy)phosphinoyloxy)ethyl) ester 1224724-33-7 C30H32ClN2O5PS3
thiopropionic acid S-(2-((5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-ylsulfanylmethyl)-(2-propionylsulfanylethoxy)phosphinoyloxy)ethyl) ester
—— tetrabenzyl 2-(2-hydroxyethoxy)propane-1,3-diyl bis(phosphate) 1220703-33-2 C33H38O10P2
tetrabenzyl 2-(2-hydroxyethoxy)propane-1,3-diyl bis(phosphate)
—— tert-butyl (5R)-5-formyl-3,3-dimethyl-1,3-azasilolidine-1-carboxylate 1334314-07-6 C11H21NO3Si
tert-butyl (5R)-5-formyl-3,3-dimethyl-1,3-azasilolidine-1-carboxylate
—— tert-butyl (5R)-5-(7-bromo-3H-benzo[e]benzimidazol-2-yl)-3,3-dimethyl-1,3-azasilolidine-1-carboxylate 1334313-78-8 C21H26BrN3O2Si
tert-butyl (5R)-5-(7-bromo-3H-benzo[e]benzimidazol-2-yl)-3,3-dimethyl-1,3-azasilolidine-1-carboxylate
—— tert-butyl (5R)-3,3-dimethyl-5-[5-[4-[2-[(2S)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-2-yl]-3H-benzo[e]benzimidazol-7-yl]phenyl]-1H-imidazol-2-yl]-1,3-azasilolidine-1-carboxylate 1334313-79-9 C39H48N6O4Si
tert-butyl (5R)-3,3-dimethyl-5-[5-[4-[2-[(2S)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-2-yl]-3H-benzo[e]benzimidazol-7-yl]phenyl]-1H-imidazol-2-yl]-1,3-azasilolidine-1-carboxylate
—— tert-butyl N-(1-pyrido[2,3-d]pyrimidin-2-ylcyclopropyl)carbamate 1159733-81-9 C15H18N4O2
tert-butyl N-(1-pyrido[2,3-d]pyrimidin-2-ylcyclopropyl)carbamate
—— tert-butyl 3-(4-chloro-phenyl)-5-phenyl-isothiazole-4-carboxylate 1101130-07-7 C20H18ClNO2S
tert-butyl 3-(4-chloro-phenyl)-5-phenyl-isothiazole-4-carboxylate
—— tert-butyl 2-((3-mercaptopyridin-2-yl)methylthio)ethylcarbamate 1147849-82-8 C13H20N2O2S2
tert-butyl 2-((3-mercaptopyridin-2-yl)methylthio)ethylcarbamate
—— type I 1231708-06-7 C39H52O12
type I
—— tert-butyl [(1R)-2-(3-amino-4-nitrophenoxy)-1-phenylethyl]carbamate 1228657-10-0 C19H23N3O5
tert-butyl [(1R)-2-(3-amino-4-nitrophenoxy)-1-phenylethyl]carbamate
—— tert-butyl 5-bromo-3-(4-chloro-phenyl)-isothiazole-4-carboxylate 1101130-06-6 C14H13BrClNO2S
tert-butyl 5-bromo-3-(4-chloro-phenyl)-isothiazole-4-carboxylate
—— tert-butyl 3-(4-chloro-phenyl)-isothiazole-4-carboxylate 1101130-05-5 C14H14ClNO2S
tert-butyl 3-(4-chloro-phenyl)-isothiazole-4-carboxylate
—— tert-butyl 2-[2-[2-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]-4-methoxyphenoxy]ethoxy]-4-methyl-N-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]anilino]acetate 1070770-90-9 C40H60N2O11
tert-butyl 2-[2-[2-[2-[bis[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]amino]-4-methoxyphenoxy]ethoxy]-4-methyl-N-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]anilino]acetate
—— Tert-butyl 4-[[5-[[3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-9-yl]oxy]pentanoylamino]methyl]benzoate 1335095-54-9 C40H50FN5O6
Tert-butyl 4-[[5-[[3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-9-yl]oxy]pentanoylamino]methyl]benzoate