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—— methyl 3-[[7-[(1R)-1-[acetyl(methyl)amino]ethyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C21H25N3O5S
methyl 3-[[7-[(1R)-1-[acetyl(methyl)amino]ethyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— methyl 3-(3,5-dimethylisoxazol-4-yl)-5-(cis-2,6-dimethylmorpholine-4-carbonyl)-7-(trifluoromethyl)-9H-carbazole-1-carboxylate —— C27H26F3N3O5
methyl 3-(3,5-dimethylisoxazol-4-yl)-5-(cis-2,6-dimethylmorpholine-4-carbonyl)-7-(trifluoromethyl)-9H-carbazole-1-carboxylate
—— Methyl 5-(3,5-dimethyl-1,2-oxazol-4-yl)-2-(3-methylsulfonylanilino)benzoate —— C20H20N2O5S
Methyl 5-(3,5-dimethyl-1,2-oxazol-4-yl)-2-(3-methylsulfonylanilino)benzoate
—— Methyl 2-methyl-4-(6-methylpyrimidin-4-yl)pyrazole-3-carboxylate —— C11H12N4O2
Methyl 2-methyl-4-(6-methylpyrimidin-4-yl)pyrazole-3-carboxylate
—— methyl 3-[[(5S)-7-[(3-fluorophenyl)methoxymethyl]-5-methyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C25H25FN2O5S
methyl 3-[[(5S)-7-[(3-fluorophenyl)methoxymethyl]-5-methyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— Methyl 2-methyl-4-(2,5,6-trimethylpyrimidin-4-yl)pyrazole-3-carboxylate —— C13H16N4O2
Methyl 2-methyl-4-(2,5,6-trimethylpyrimidin-4-yl)pyrazole-3-carboxylate
—— methyl 4-(5-cyclopropyl-4-(difluoromethyl)thiazol-2-yl)-1-methyl-1H-pyrazol-5-carboxylate —— C13H13F2N3O2S
methyl 4-(5-cyclopropyl-4-(difluoromethyl)thiazol-2-yl)-1-methyl-1H-pyrazol-5-carboxylate
—— methyl N-[(2S)-1-[(2S,4S)-4-cyano-2-[5-[6-[4-[2-[(2S)-1-[(2R)-2-(methoxycarbonylamino)-2-(2-methoxyphenyl)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C49H51N9O7
methyl N-[(2S)-1-[(2S,4S)-4-cyano-2-[5-[6-[4-[2-[(2S)-1-[(2R)-2-(methoxycarbonylamino)-2-(2-methoxyphenyl)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl (8S,11S,14S)-14-[[(2S)-2-[[(2R)-2-[[(2R)-3-butoxy-2-[[4-(4-butylphenyl)benzoyl]-methylamino]propanoyl]amino]propanoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]-methylamino]-3,18-dimethoxy-11-methyl-10,13-dioxo-9,12-diazatricyclo[13.3.1.12,6]icosa-1(18),2,4,6(20),15(19),16-hexaene-8-carboxylate —— C63H85N7O13
methyl (8S,11S,14S)-14-[[(2S)-2-[[(2R)-2-[[(2R)-3-butoxy-2-[[4-(4-butylphenyl)benzoyl]-methylamino]propanoyl]amino]propanoyl]amino]-6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoyl]-methylamino]-3,18-dimethoxy-11-methyl-10,13-dioxo-9,12-diazatricyclo[13.3.1.12,6]icosa-1(18),2,4,6(20),15(19),16-hexaene-8-carboxylate
—— Methyl 4-(3-methoxypyrazin-2-yl)-2-methylpyrazole-3-carboxylate —— C11H12N4O3
Methyl 4-(3-methoxypyrazin-2-yl)-2-methylpyrazole-3-carboxylate
—— Methyl 4-(5-chloropyrimidin-4-yl)-2-methylpyrazole-3-carboxylate —— C10H9ClN4O2
Methyl 4-(5-chloropyrimidin-4-yl)-2-methylpyrazole-3-carboxylate
—— methyl N-[(2S)-1-[(2S,6S)-2-ethyl-6-[5-[4-[6-[2-[(6S)-5-[(2S)-2-(methoxycarbonylamino)butanoyl]-5-azaspiro[2.4]heptan-6-yl]-1H-imidazol-5-yl]naphthalen-2-yl]phenyl]-1H-imidazol-2-yl]piperidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C48H58N8O6
methyl N-[(2S)-1-[(2S,6S)-2-ethyl-6-[5-[4-[6-[2-[(6S)-5-[(2S)-2-(methoxycarbonylamino)butanoyl]-5-azaspiro[2.4]heptan-6-yl]-1H-imidazol-5-yl]naphthalen-2-yl]phenyl]-1H-imidazol-2-yl]piperidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S,4S)-2-[5-(4-bromophenyl)-1H-imidazol-2-yl]-4-pyrazin-2-yloxypyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate —— C24H29BrN6O4
methyl N-[(2S)-1-[(2S,4S)-2-[5-(4-bromophenyl)-1H-imidazol-2-yl]-4-pyrazin-2-yloxypyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate
—— methyl (2R)-5-[5-[[2-[3,5-bis(trifluoromethyl)phenyl]-2-methylpropanoyl]amino]-4-(4-fluoro-2-methylphenyl)pyridin-2-yl]-1-phosphanylpyrrolidine-2-carboxylate —— C30H29F7N3O3P
methyl (2R)-5-[5-[[2-[3,5-bis(trifluoromethyl)phenyl]-2-methylpropanoyl]amino]-4-(4-fluoro-2-methylphenyl)pyridin-2-yl]-1-phosphanylpyrrolidine-2-carboxylate
—— methyl 3-[[7-[(1S)-1-[(3-fluorophenyl)methoxy]ethyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C25H25FN2O5S
methyl 3-[[7-[(1S)-1-[(3-fluorophenyl)methoxy]ethyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[4-[(E)-2-[[[(2S)-4-acetyl-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]piperazin-2-yl]-aminomethylidene]amino]ethenyl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C44H55N9O7
methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[4-[(E)-2-[[[(2S)-4-acetyl-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]piperazin-2-yl]-aminomethylidene]amino]ethenyl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S,6S)-2-ethyl-6-[5-[4-[6-[2-[(6S)-5-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-5-azaspiro[2.4]heptan-6-yl]-1H-imidazol-5-yl]naphthalen-2-yl]phenyl]-1H-imidazol-2-yl]piperidin-1-yl]-1-oxopropan-2-yl]carbamate —— C47H56N8O6
methyl N-[(2S)-1-[(2S,6S)-2-ethyl-6-[5-[4-[6-[2-[(6S)-5-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-5-azaspiro[2.4]heptan-6-yl]-1H-imidazol-5-yl]naphthalen-2-yl]phenyl]-1H-imidazol-2-yl]piperidin-1-yl]-1-oxopropan-2-yl]carbamate
—— methyl 3-[[7-[2-[(3-fluorophenyl)methoxy]propan-2-yl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C26H27FN2O5S
methyl 3-[[7-[2-[(3-fluorophenyl)methoxy]propan-2-yl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— methyl 2-bromo-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-7-carboxylate —— C9H11BrN2O2
methyl 2-bromo-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-7-carboxylate
—— methyl 3-[[7-[(3-fluorophenyl)methoxymethyl]-5-methyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C25H25FN2O5S
methyl 3-[[7-[(3-fluorophenyl)methoxymethyl]-5-methyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— Methyl 2-methyl-4-(5-methylpyridazin-3-yl)pyrazole-3-carboxylate —— C11H12N4O2
Methyl 2-methyl-4-(5-methylpyridazin-3-yl)pyrazole-3-carboxylate
—— Methyl 2-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)pyrazole-3-carboxylate —— C9H10N4O2S
Methyl 2-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)pyrazole-3-carboxylate
—— methyl 3-[[7-[2-[acetyl(methyl)amino]propan-2-yl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C22H27N3O5S
methyl 3-[[7-[2-[acetyl(methyl)amino]propan-2-yl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— methyl 4-(5-acetyl-2-methylthiazol-4-yl)-1-methyl-1H-pyrazol-5-carboxylate —— C12H13N3O3S
methyl 4-(5-acetyl-2-methylthiazol-4-yl)-1-methyl-1H-pyrazol-5-carboxylate
—— methyl N-[(2S)-3-methyl-1-oxo-1-[(2S)-4-oxo-2-(5-phenyl-1H-imidazol-2-yl)pyrrolidin-1-yl]butan-2-yl]carbamate —— C20H24N4O4
methyl N-[(2S)-3-methyl-1-oxo-1-[(2S)-4-oxo-2-(5-phenyl-1H-imidazol-2-yl)pyrrolidin-1-yl]butan-2-yl]carbamate
—— methyl 4-(3,5-dimethyl-1,2,4-triazol-1-yl)-6-[(1R)-2-(1-methylbenzimidazol-2-yl)cyclopropyl]pyrimidine-2-carboxylate —— C21H21N7O2
methyl 4-(3,5-dimethyl-1,2,4-triazol-1-yl)-6-[(1R)-2-(1-methylbenzimidazol-2-yl)cyclopropyl]pyrimidine-2-carboxylate
—— Methyl 3-[[7-[(3-fluorophenyl)methoxymethyl]-5,5-dimethyl-2,3-dihydro-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate —— C26H27FN2O5S
Methyl 3-[[7-[(3-fluorophenyl)methoxymethyl]-5,5-dimethyl-2,3-dihydro-1,4-benzoxazepine-4-carbonyl]amino]thiophene-2-carboxylate
—— Methyl 2-methyl-4-(1-methylimidazol-4-yl)pyrazole-3-carboxylate —— C10H12N4O2
Methyl 2-methyl-4-(1-methylimidazol-4-yl)pyrazole-3-carboxylate
—— Methyl 4-(5,6-dimethylpyrimidin-4-yl)-2-methylpyrazole-3-carboxylate —— C12H14N4O2
Methyl 4-(5,6-dimethylpyrimidin-4-yl)-2-methylpyrazole-3-carboxylate
—— Methyl 2-(4-formyl-2,5-dimethyl-3-nitrophenyl)-2-[(2-methylpropan-2-yl)oxy]acetate —— C16H21NO6
Methyl 2-(4-formyl-2,5-dimethyl-3-nitrophenyl)-2-[(2-methylpropan-2-yl)oxy]acetate
—— Methyl 5-butoxy-2,3-dihydro-1,4-benzodioxine-7-carboxylate —— C14H18O5
Methyl 5-butoxy-2,3-dihydro-1,4-benzodioxine-7-carboxylate
—— methyl (2S)-2-[2,5-dimethyl-3-nitro-4-(trifluoromethylsulfonyloxy)phenyl]-2-propan-2-yloxyacetate —— C15H18F3NO8S
methyl (2S)-2-[2,5-dimethyl-3-nitro-4-(trifluoromethylsulfonyloxy)phenyl]-2-propan-2-yloxyacetate
—— methyl (2S)-3-[3-[5-[(1S)-1-[[2-[[(2R)-2-[[(2R)-3-butoxy-2-[methyl(tetradecylcarbamoyl)amino]propanoyl]amino]propanoyl]amino]acetyl]-methylamino]-2-oxo-2-[[(2S)-3-oxobutan-2-yl]amino]ethyl]-2-methoxyphenyl]-4-methoxyphenyl]-2-methylpropanoate —— C54H86N6O11
methyl (2S)-3-[3-[5-[(1S)-1-[[2-[[(2R)-2-[[(2R)-3-butoxy-2-[methyl(tetradecylcarbamoyl)amino]propanoyl]amino]propanoyl]amino]acetyl]-methylamino]-2-oxo-2-[[(2S)-3-oxobutan-2-yl]amino]ethyl]-2-methoxyphenyl]-4-methoxyphenyl]-2-methylpropanoate
—— methyl 5-[[(3E)-3-(carbamothioylhydrazinylidene)-2-oxoindol-1-yl]methyl]furan-2-carboxylate —— C16H14N4O4S
methyl 5-[[(3E)-3-(carbamothioylhydrazinylidene)-2-oxoindol-1-yl]methyl]furan-2-carboxylate
—— methyl N-[(2S)-1-[(2S)-2-[5-[7-[5-[(1R,3S,4S)-2-[(2S)-2-(methoxycarbonylamino)propanoyl]-2-azabicyclo[2.2.1]heptan-3-yl]-1H-pyrrol-2-yl]-9,10-dihydrophenanthren-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamate —— C41H47N7O6
methyl N-[(2S)-1-[(2S)-2-[5-[7-[5-[(1R,3S,4S)-2-[(2S)-2-(methoxycarbonylamino)propanoyl]-2-azabicyclo[2.2.1]heptan-3-yl]-1H-pyrrol-2-yl]-9,10-dihydrophenanthren-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamate
—— methyl N-[(2S)-1-[(6S)-6-[5-[6-[4-[2-[(2S)-3-[4-methoxy-2-(methoxycarbonylamino)butanoyl]-1,3-thiazolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]-5-azaspiro[2.4]heptan-5-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C45H52N8O7S
methyl N-[(2S)-1-[(6S)-6-[5-[6-[4-[2-[(2S)-3-[4-methoxy-2-(methoxycarbonylamino)butanoyl]-1,3-thiazolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]-5-azaspiro[2.4]heptan-5-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S,4S)-2-[5-(4-bromophenyl)-1H-imidazol-2-yl]-4-(difluoromethoxymethyl)pyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate —— C22H29BrF2N4O4
methyl N-[(2S)-1-[(2S,4S)-2-[5-(4-bromophenyl)-1H-imidazol-2-yl]-4-(difluoromethoxymethyl)pyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate
—— methyl 4-(3,5-dimethyl-1,2,4-triazol-1-yl)-6-[(2R)-2-(1-methylbenzimidazol-2-yl)cyclopropyl]pyrimidine-2-carboxylate —— C21H21N7O2
methyl 4-(3,5-dimethyl-1,2,4-triazol-1-yl)-6-[(2R)-2-(1-methylbenzimidazol-2-yl)cyclopropyl]pyrimidine-2-carboxylate
—— methyl N-[(1S)-2-[(2S)-2-[5-[6-[4-[2-[(2S,4S)-4-(difluoromethoxy)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxo-1-phenylethyl]carbamate —— C48H50F2N8O7
methyl N-[(1S)-2-[(2S)-2-[5-[6-[4-[2-[(2S,4S)-4-(difluoromethoxy)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxo-1-phenylethyl]carbamate
—— methyl N-[1-[(2S)-2-[5-[6-[4-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-4-methylidenepyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C45H52N8O6
methyl N-[1-[(2S)-2-[5-[6-[4-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-4-methylidenepyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]naphthalen-2-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl (5E)-5-[(3-chloroanilino)methylidene]-2-methyl-4-phenylpyrrole-3-carboxylate —— C20H17ClN2O2
methyl (5E)-5-[(3-chloroanilino)methylidene]-2-methyl-4-phenylpyrrole-3-carboxylate
—— methyl N'-[[(E)-(5-bromo-3-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]carbamimidothioate —— C9H9BrN4O3S
methyl N'-[[(E)-(5-bromo-3-nitro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]carbamimidothioate
—— methyl N-[(2S)-1-[(2R)-2-[5-[4-[4-(2-aminoacetyl)phenyl]phenyl]-1H-imidazol-2-yl]cyclopentyl]-3-methyl-1-oxobutan-2-yl]carbamate —— C29H34N4O4
methyl N-[(2S)-1-[(2R)-2-[5-[4-[4-(2-aminoacetyl)phenyl]phenyl]-1H-imidazol-2-yl]cyclopentyl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl 5-[5-chloro-6-[1-[(4-methylphenyl)carbamoyl]-3,6-dihydro-2H-pyridin-4-yl]pyridin-3-yl]-1,3-oxazole-4-carboxylate —— C23H21ClN4O4
methyl 5-[5-chloro-6-[1-[(4-methylphenyl)carbamoyl]-3,6-dihydro-2H-pyridin-4-yl]pyridin-3-yl]-1,3-oxazole-4-carboxylate
—— Methyl 2-[4-(4-cyanophenyl)-1-[3-(fluoromethyl)phenyl]-2,5-dioxo-4,6,7,8-tetrahydroquinazolin-3-yl]propanoate —— C26H24FN3O4
Methyl 2-[4-(4-cyanophenyl)-1-[3-(fluoromethyl)phenyl]-2,5-dioxo-4,6,7,8-tetrahydroquinazolin-3-yl]propanoate
—— methyl (2S)-5-(4-methylphenyl)-2-[(2-methylpropan-2-yl)oxycarbonylamino]pent-4-ynoate —— C18H23NO4
methyl (2S)-5-(4-methylphenyl)-2-[(2-methylpropan-2-yl)oxycarbonylamino]pent-4-ynoate
—— Methyl 2-[3-amino-4-(cyclohexylcarbamoylamino)-2,5-dimethylphenyl]-2-[(2-methylpropan-2-yl)oxy]acetate —— C22H35N3O4
Methyl 2-[3-amino-4-(cyclohexylcarbamoylamino)-2,5-dimethylphenyl]-2-[(2-methylpropan-2-yl)oxy]acetate
—— methyl 2-(3,4-dihydro-2H-chromen-6-yl)-3-methylbenzoate —— C18H18O3
methyl 2-(3,4-dihydro-2H-chromen-6-yl)-3-methylbenzoate
—— Methyl 2-[(2-methylpropan-2-yl)oxy]-2-(2,4,5-trimethyl-3-nitrophenyl)acetate —— C16H23NO5
Methyl 2-[(2-methylpropan-2-yl)oxy]-2-(2,4,5-trimethyl-3-nitrophenyl)acetate
—— methyl 2-[4-(cyclohexylcarbamoylamino)-2-(3,4-dihydro-2H-chromen-6-yl)-5-(methanesulfonamido)-3,6-dimethylphenyl]-2-[(2-methylpropan-2-yl)oxy]acetate —— C32H45N3O7S
methyl 2-[4-(cyclohexylcarbamoylamino)-2-(3,4-dihydro-2H-chromen-6-yl)-5-(methanesulfonamido)-3,6-dimethylphenyl]-2-[(2-methylpropan-2-yl)oxy]acetate