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—— methyl (6S)-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-7-(3-methylsulfanylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate —— C25H26N4O5S
methyl (6S)-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-7-(3-methylsulfanylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate
—— methyl 3-[[(7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C24H25N3O3S
methyl 3-[[(7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— methyl (6R)-7-[(2,5-dimethoxyphenyl)methyl]-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate —— C27H30N4O7
methyl (6R)-7-[(2,5-dimethoxyphenyl)methyl]-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate
—— methyl (6S)-7-(4-acetamidophenyl)-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate —— C26H27N5O6
methyl (6S)-7-(4-acetamidophenyl)-6-[(2-methoxyphenyl)methylcarbamoyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate
—— methyl (6R)-6-(benzylcarbamoyl)-6-methyl-7-(3-methylsulfanylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate —— C24H24N4O4S
methyl (6R)-6-(benzylcarbamoyl)-6-methyl-7-(3-methylsulfanylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1-carboxylate
—— methyl 4-chloro-2-[[(7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C24H24ClN3O3S
methyl 4-chloro-2-[[(7R)-7-methyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— methyl (2Z)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[1-phenyl-3-(4-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C37H35N5O6S2
methyl (2Z)-5-(4-methoxyphenyl)-7-methyl-3-oxo-2-[[1-phenyl-3-(4-piperidin-1-ylsulfonylphenyl)pyrazol-4-yl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (4Z)-4-[(3-methoxy-4-prop-2-enoxyphenyl)methylidene]-2-methyl-1-naphthalen-1-yl-5-oxopyrrole-3-carboxylate —— C28H25NO5
methyl (4Z)-4-[(3-methoxy-4-prop-2-enoxyphenyl)methylidene]-2-methyl-1-naphthalen-1-yl-5-oxopyrrole-3-carboxylate
—— methyl 2-chloro-5-[[(Z)-2-(5-chloro-1,3-benzoxazol-2-yl)-3-oxoprop-1-enyl]amino]benzoate —— C18H12Cl2N2O4
methyl 2-chloro-5-[[(Z)-2-(5-chloro-1,3-benzoxazol-2-yl)-3-oxoprop-1-enyl]amino]benzoate
—— methyl 4-chloro-2-[[(7R)-7-ethyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C25H26ClN3O3S
methyl 4-chloro-2-[[(7R)-7-ethyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— methyl 4-[[(7R)-7-propan-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C26H29N3O3S
methyl 4-[[(7R)-7-propan-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— methyl (4Z)-1-benzyl-4-(2-fluorobenzylidene)-2-methyl-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate —— C21H18FNO3
methyl (4Z)-1-benzyl-4-(2-fluorobenzylidene)-2-methyl-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
—— methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(4-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O7S
methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(4-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(3-bromo-4-hydroxy-5-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H25BrN2O8S
methyl 2-[(3E)-2-(3-bromo-4-hydroxy-5-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(3-hydroxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H24N2O7S
methyl 2-[(3E)-2-(3-hydroxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H26N2O8S
methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(3-ethoxy-4-phenylmethoxyphenyl)-3-[hydroxy-(4-methoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(3E)-2-(3-ethoxy-4-phenylmethoxyphenyl)-3-[hydroxy-(4-methoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(2-fluorophenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H23FN2O6S
methyl 2-[(3E)-2-(2-fluorophenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[[3-[(3S)-1-[(4-chlorophenyl)carbamoyl]piperidin-3-yl]benzoyl]amino]benzoate —— C27H26ClN3O4
methyl 2-[[3-[(3S)-1-[(4-chlorophenyl)carbamoyl]piperidin-3-yl]benzoyl]amino]benzoate
—— methyl 2-[(3Z)-2-oxo-3-[[2-[[(E)-3-phenylprop-2-enoyl]amino]acetyl]hydrazinylidene]indol-1-yl]acetate —— C22H20N4O5
methyl 2-[(3Z)-2-oxo-3-[[2-[[(E)-3-phenylprop-2-enoyl]amino]acetyl]hydrazinylidene]indol-1-yl]acetate
—— methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(3-methoxy-4-phenylmethoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C34H32N2O8S
methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(3-methoxy-4-phenylmethoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(4-propan-2-ylphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H30N2O6S
methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(4-propan-2-ylphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-[4-(dimethylamino)phenyl]-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H29N3O6S
methyl 2-[(3E)-2-[4-(dimethylamino)phenyl]-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-3-[(4-butoxyphenyl)-hydroxymethylidene]-2-(4-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H25N3O8S
methyl 2-[(3E)-3-[(4-butoxyphenyl)-hydroxymethylidene]-2-(4-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-[3-methoxy-4-(3-methylbutoxy)phenyl]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H36N2O8S
methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-[3-methoxy-4-(3-methylbutoxy)phenyl]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(4-butoxy-3-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H34N2O8S
methyl 2-[(3E)-2-(4-butoxy-3-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(Z)-[1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C23H26FN3O5
methyl 4-[(Z)-[1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 2-[(3E)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O8S
methyl 2-[(3E)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[[3-[(3R)-1-[(4-chlorophenyl)carbamoyl]piperidin-3-yl]benzoyl]amino]benzoate —— C27H26ClN3O4
methyl 2-[[3-[(3R)-1-[(4-chlorophenyl)carbamoyl]piperidin-3-yl]benzoyl]amino]benzoate
—— methyl 2-[(3E)-3-[hydroxy(pyridin-4-yl)methylidene]-2-(3-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C23H19N3O6S
methyl 2-[(3E)-3-[hydroxy(pyridin-4-yl)methylidene]-2-(3-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-pyridin-4-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H23N3O6S
methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-pyridin-4-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O7S
methyl 2-[(3E)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 7-(4-chlorophenyl)-5-methylidene-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C14H13ClN4O2
methyl 7-(4-chlorophenyl)-5-methylidene-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— methyl 2-[[(E)-3-naphthalen-1-ylprop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H21NO3S
methyl 2-[[(E)-3-naphthalen-1-ylprop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H28N2O7S
methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl (2Z)-2-[[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H27ClN4O5S
methyl (2Z)-2-[[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[(Z)-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)hydrazinylidene]methyl]benzoate —— C17H16N4O2S
methyl 4-[(Z)-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)hydrazinylidene]methyl]benzoate
—— methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H23N3O6S
methyl 2-[(4E)-4-[hydroxy-(3-propoxyphenyl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(4-ethylphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O6S
methyl 2-[(3E)-2-(4-ethylphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H30N2O8S
methyl 2-[(3E)-2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3Z)-3-[[2-[(2,2-diphenylacetyl)amino]acetyl]hydrazinylidene]-2-oxoindol-1-yl]acetate —— C27H24N4O5
methyl 2-[(3Z)-3-[[2-[(2,2-diphenylacetyl)amino]acetyl]hydrazinylidene]-2-oxoindol-1-yl]acetate
—— methyl 2-[(3E)-2-(4-hydroxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H24N2O7S
methyl 2-[(3E)-2-(4-hydroxyphenyl)-3-[hydroxy-(3-propoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(3-methoxy-4-pentoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H36N2O8S
methyl 2-[(3E)-3-[hydroxy-(3-propoxyphenyl)methylidene]-2-(3-methoxy-4-pentoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— morpholin-4-yl-[(3R)-1-(2,8,10-triazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-7-yl)piperidin-3-yl]methanone —— C20H23N5O2
morpholin-4-yl-[(3R)-1-(2,8,10-triazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-7-yl)piperidin-3-yl]methanone
—— methyl (2Z)-5-(4-methoxyphenyl)-7-methyl-2-[[3-(4-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H33N5O7S2
methyl (2Z)-5-(4-methoxyphenyl)-7-methyl-2-[[3-(4-morpholin-4-ylsulfonylphenyl)-1-phenylpyrazol-4-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 2-[(3Z)-3-[[(Z)-2-benzamido-3-(3,4-dimethoxyphenyl)prop-2-enoyl]hydrazinylidene]-2-oxoindol-1-yl]acetate —— C29H26N4O7
methyl 2-[(3Z)-3-[[(Z)-2-benzamido-3-(3,4-dimethoxyphenyl)prop-2-enoyl]hydrazinylidene]-2-oxoindol-1-yl]acetate
—— methyl 6-[[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]hexanoate —— C19H27NO6
methyl 6-[[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]hexanoate
—— methyl 2-[4-[(Z)-methoxyiminomethyl]-2-methyl-5-(trifluoromethyl)pyrazol-3-yl]sulfanylbenzoate —— C15H14F3N3O3S
methyl 2-[4-[(Z)-methoxyiminomethyl]-2-methyl-5-(trifluoromethyl)pyrazol-3-yl]sulfanylbenzoate
—— methyl 2-[(4E)-4-[hydroxy(pyridin-4-yl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C21H16N4O5S
methyl 2-[(4E)-4-[hydroxy(pyridin-4-yl)methylidene]-2,3-dioxo-5-pyridin-3-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl (4Z)-4-[4-(dimethylamino)benzylidene]-2-methyl-1-(4-methylbenzyl)-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate —— C24H26N2O3
methyl (4Z)-4-[4-(dimethylamino)benzylidene]-2-methyl-1-(4-methylbenzyl)-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate