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—— methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decane-8-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C35H45N3O9
methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decane-8-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,4S)-6-[cyclohexyl(methyl)carbamoyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H42N2O9S
methyl 4-[(2S,4S)-6-[cyclohexyl(methyl)carbamoyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-6-(benzylcarbamoyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C26H31NO6
methyl 4-[(2S,3S,4R)-6-(benzylcarbamoyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3R)-1-(2,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C14H17NO3
methyl (3R)-1-(2,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,4S)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C35H48N2O13S
methyl 4-[(2S,4S)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3R)-1-(3-methoxycarbonylphenyl)-5-oxopyrrolidine-3-carboxylate —— C14H15NO5
methyl (3R)-1-(3-methoxycarbonylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3R)-1-(2,4-dimethoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C14H17NO5
methyl (3R)-1-(2,4-dimethoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,3R,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]carbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C36H40N2O8S
methyl 4-[(2S,3R,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]carbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3S)-1-(4-bromo-3-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C13H14BrNO3
methyl (3S)-1-(4-bromo-3-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3R)-1-(3,5-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H11Cl2NO3
methyl (3R)-1-(3,5-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2R,4R)-6-[(2-aminophenyl)carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C24H28N2O7
methyl 4-[(2R,4R)-6-[(2-aminophenyl)carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3S)-1-(3-amino-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C13H16N2O3
methyl (3S)-1-(3-amino-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3S)-1-(2,3-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H11Cl2NO3
methyl (3S)-1-(2,3-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,3R,4R)-6-[2,2-dimethoxyethyl(methyl)carbamoyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C27H41NO10
methyl 4-[(2S,3R,4R)-6-[2,2-dimethoxyethyl(methyl)carbamoyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C22H29NO7
methyl 4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-(azocane-1-carbonyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C25H35NO6
methyl 4-[(2R,4R)-6-(azocane-1-carbonyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3S)-5-oxo-1-(4-sulfamoylphenyl)pyrrolidine-3-carboxylate —— C12H14N2O5S
methyl (3S)-5-oxo-1-(4-sulfamoylphenyl)pyrrolidine-3-carboxylate
—— methyl 4-[(2S,3S,4R)-6-[(1R)-1-[[(2R,3R,11bS)-3-ethyl-9,10-dimethoxy-2,3,4,6,7,11b-hexahydro-1H-benzo[a]quinolizin-2-yl]methyl]-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C48H62N2O10
methyl 4-[(2S,3S,4R)-6-[(1R)-1-[[(2R,3R,11bS)-3-ethyl-9,10-dimethoxy-2,3,4,6,7,11b-hexahydro-1H-benzo[a]quinolizin-2-yl]methyl]-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carbonyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,4S)-6-[2,2-dimethoxyethyl(methyl)carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C23H33NO8
methyl 4-[(2S,4S)-6-[2,2-dimethoxyethyl(methyl)carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3S)-1-(4-bromo-2,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C14H16BrNO3
methyl (3S)-1-(4-bromo-2,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3S)-1-(2,5-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H11Cl2NO3
methyl (3S)-1-(2,5-dichlorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3S)-1-(3-chloro-4-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H11ClFNO3
methyl (3S)-1-(3-chloro-4-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2R,4R)-6-(benzylcarbamoyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C25H29NO7
methyl 4-[(2R,4R)-6-(benzylcarbamoyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,3R,4S)-6-(benzylcarbamoyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C26H31NO6
methyl 4-[(2R,3R,4S)-6-(benzylcarbamoyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-(benzylcarbamoyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H36N2O9S
methyl 4-[(2R,4R)-6-(benzylcarbamoyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-6-(azocane-1-carbonyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C29H43NO8
methyl 4-[(2S,3S,4R)-6-(azocane-1-carbonyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3R)-1-(3-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H12FNO3
methyl (3R)-1-(3-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl (3S)-1-naphthalen-2-yl-5-oxopyrrolidine-3-carboxylate —— C16H15NO3
methyl (3S)-1-naphthalen-2-yl-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C28H41NO10
methyl 4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3R)-1-(4-bromo-2-chlorophenyl)-5-oxopyrrolidine-3-carboxylate —— C12H11BrClNO3
methyl (3R)-1-(4-bromo-2-chlorophenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-[4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C31H37N3O7
methyl 4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-[4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C30H37N3O8
methyl 4-[(2S,3S,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl (3S)-1-(4-methoxycarbonyl-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C15H17NO5
methyl (3S)-1-(4-methoxycarbonyl-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H49NO12
methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,4S)-6-(azocane-1-carbonyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H42N2O9S
methyl 4-[(2S,4S)-6-(azocane-1-carbonyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]carbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C36H40N2O8S
methyl 4-[(2S,3S,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]carbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C30H29N3O6
methyl 4-[(2R,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C33H36N4O9S
methyl 4-[(2R,4R)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-6-[2-[(5-nitropyridin-2-yl)amino]ethylcarbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H37N5O11S
methyl 4-[(2R,4R)-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-6-[2-[(5-nitropyridin-2-yl)amino]ethylcarbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,4S)-6-(azocane-1-carbonyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C25H35NO7
methyl 4-[(2S,4S)-6-(azocane-1-carbonyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,3S,4S)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C30H37N3O8
methyl 4-[(2R,3S,4S)-6-(1H-benzimidazol-2-ylmethylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C25H35NO6
methyl 4-[(2R,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-[(2-aminophenyl)carbamoyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C31H35N3O9S
methyl 4-[(2R,4R)-6-[(2-aminophenyl)carbamoyl]-2-[2-[2-hydroxyethyl-(4-methoxyphenyl)sulfonylamino]ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-6-(benzylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C29H37NO8
methyl 4-[(2S,3S,4R)-6-(benzylcarbamoyl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3S,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C29H43NO8
methyl 4-[(2S,3S,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3R,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C32H49NO12
methyl 4-[(2S,3R,4R)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-6-[2-[(5-nitropyridin-2-yl)amino]ethylcarbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C29H30N4O8
methyl 4-[(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-6-[2-[(5-nitropyridin-2-yl)amino]ethylcarbamoyl]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate —— C25H35NO7
methyl 4-[(2R,4R)-6-[cyclohexyl(methyl)carbamoyl]-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C29H43NO10
methyl 4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]benzoate
—— methyl 4-[(2R,3R,4S)-6-[cyclohexyl(methyl)carbamoyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate —— C26H37NO6
methyl 4-[(2R,3R,4S)-6-[cyclohexyl(methyl)carbamoyl]-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]benzoate